*Note: the InCHIKey will be temporarily assigned as the "Common Name" if no IUPAC name or alternative short name is available.
**Note: the Chemical Classification was calculated by NPClassifier Version 1.5. Reference: PMID:34662515.
Organism ID | Organism Name | Taxonomy Level | Family | SuperKingdom | Isolation Part | Collection Location | Collection Time | Reference |
---|
☑ Note for Reference:
In addition to directly collecting NP source organism data from primary literature (where reference will provided as NCBI PMID or DOI links), NPASS also integrated them from below databases:
☉ UNPD: Universal Natural Products Database [PMID: 23638153].
☉ StreptomeDB: a database of streptomycetes natural products [PMID: 33051671].
☉ TM-MC: a database of medicinal materials and chemical compounds in Northeast Asian traditional medicine [PMID: 26156871].
☉ TCM@Taiwan: a Traditional Chinese Medicine database [PMID: 21253603].
☉ TCMID: a Traditional Chinese Medicine database [PMID: 29106634].
☉ TCMSP: The traditional Chinese medicine systems pharmacology database and analysis platform [PMID: 24735618].
☉ HerDing: a herb recommendation system to treat diseases using genes and chemicals [PMID: 26980517].
☉ MetaboLights: a metabolomics database [PMID: 27010336].
☉ FooDB: a database of constituents, chemistry and biology of food species [www.foodb.ca].
Organism ID | NP ID | Organism Material Preparation | Organism Part | NP Quantity (Standard) | NP Quantity (Minimum) | NP Quantity (Maximum) | Quantity Unit | Reference |
---|
☑ Note for Reference:
In addition to directly collecting NP quantitative data from primary literature (where reference will provided as NCBI PMID or DOI links), NPASS also integrated NP quantitative records for specific NP domains (e.g., NPS from foods or herbs) from domain-specific databases. These databases include:
☉ DUKE: Dr. Duke's Phytochemical and Ethnobotanical Databases.
☉ PHENOL EXPLORER: is the first comprehensive database on polyphenol content in foods [PMID: 24103452], its homepage can be accessed at here.
☉ FooDB: a database of constituents, chemistry and biology of food species [www.foodb.ca].
Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT4977 | Individual Protein | Human immunodeficiency virus type 1 REV | Human immunodeficiency virus 1 | Kd | = | 180.0 | nM | PMID[547890] |
NPT4978 | Individual Protein | Phosphatidylcholine-retinol O-acyltransferase | Homo sapiens | IC50 | = | 14900.0 | nM | PMID[547891] |
NPT150 | Individual Protein | Anthrax lethal factor | Bacillus anthracis | Ki | = | 500.0 | nM | PMID[547906] |
NPT50 | Individual Protein | Tyrosyl-DNA phosphodiesterase 1 | Homo sapiens | IC50 | = | 8000000.0 | nM | PMID[547961] |
NPT472 | Individual Protein | Vanilloid receptor | Homo sapiens | IC50 | = | 400.0 | nM | PMID[547969] |
NPT4999 | Individual Protein | Menin | Homo sapiens | Tm | = | 42.5 | degrees C | PMID[547970] |
NPT4999 | Individual Protein | Menin | Homo sapiens | Tm | = | 43.81 | degrees C | PMID[547970] |
NPT4999 | Individual Protein | Menin | Homo sapiens | Tm | = | 45.19 | degrees C | PMID[547970] |
NPT4999 | Individual Protein | Menin | Homo sapiens | Kd | = | 15600.0 | nM | PMID[547970] |
NPT1886 | Cell Line | J774 | Mus musculus | Activity | = | 87.3 | % | PMID[547982] |
NPT1886 | Cell Line | J774 | Mus musculus | Activity | = | 69.8 | % | PMID[547982] |
NPT317 | Uncleic Acid | Nucleic Acid | MIC | = | 1000.0 | nM | PMID[547885] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 410.0 | nM | PMID[547886] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 380.0 | nM | PMID[547886] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 4340.0 | nM | PMID[547886] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 470.0 | nM | PMID[547886] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 91.0 | nM | PMID[547886] | |
NPT27 | Others | Unspecified | C50 | = | 0.34 | uM | PMID[547887] | |
NPT27 | Others | Unspecified | Uptake at C50 | = | 1.6 | n.a. | PMID[547887] | |
NPT27 | Others | Unspecified | Kill at C50 | = | 82.0 | % | PMID[547887] | |
NPT27 | Others | Unspecified | LD90 | = | 0.46 | uM | PMID[547887] | |
NPT2 | Others | Unspecified | K | = | 3.4 | M-1 | PMID[547888] | |
NPT2 | Others | Unspecified | Ki | = | 13500.0 | nM | PMID[547888] | |
NPT2 | Others | Unspecified | K | = | 8.0 | M-2 | PMID[547888] | |
NPT2 | Others | Unspecified | K | n.a. | 4.0 | M-1 | PMID[547888] | |
NPT24 | Organism | Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | K | = | 120000.0 | M-1 | PMID[547889] |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 920.0 | nM | PMID[547892] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 440.0 | nM | PMID[547893] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 380.0 | nM | PMID[547893] | |
NPT317 | Uncleic Acid | Nucleic Acid | tRNA peak exclusion | = | 77.8 | % | PMID[547894] | |
NPT317 | Uncleic Acid | Nucleic Acid | DNA peak exclusion | = | 100.0 | % | PMID[547894] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 140.0 | nM | PMID[547895] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 120.0 | nM | PMID[547895] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 160.0 | nM | PMID[547895] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 3970.0 | nM | PMID[547895] | |
NPT2 | Others | Unspecified | Kd | = | 350.0 | nM | PMID[547896] | |
NPT2 | Others | Unspecified | IC50 | = | 50.0 | nM | PMID[547897] | |
NPT2 | Others | Unspecified | Inhibition | = | 76.0 | % | PMID[547897] | |
NPT2 | Others | Unspecified | IC50 | = | 9.0 | nM | PMID[547897] | |
NPT2 | Others | Unspecified | Inhibition | = | 100.0 | % | PMID[547897] | |
NPT2 | Others | Unspecified | Denaturation rate constant | = | 0.095 | min-1 | PMID[547897] | |
NPT4383 | Uncleic Acid | Ribosomal RNA A-site | Kd | = | 19.0 | nM | PMID[547898] | |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | Incidence | = | 22.0 | % | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | Incidence | = | 98.0 | % | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | No. of tumors | = | 0.5 | n.a. | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | No. of tumors | = | 3.0 | n.a. | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | Incidence | = | 25.0 | % | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | Incidence | = | 80.0 | % | PMID[547899] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | No. of tumors | = | 1.13 | n.a. | PMID[547899] |
NPT27 | Others | Unspecified | K2 | = | 0.018 | min-1 | PMID[547900] | |
NPT27 | Others | Unspecified | K2 | = | 0.062 | min-1 | PMID[547900] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2000.0 | nM | PMID[547901] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 3000.0 | nM | PMID[547901] |
NPT4383 | Uncleic Acid | Ribosomal RNA A-site | Activity | = | -474.3 | n.a. | PMID[547901] | |
NPT35 | Others | n.a. | Kd | = | 100.0 | nM | PMID[547902] | |
NPT35 | Others | n.a. | Kd | = | 1000.0 | nM | PMID[547903] | |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | Kd | = | 8500.0 | nM | PMID[547904] |
NPT317 | Uncleic Acid | Nucleic Acid | Frel | = | 0.46 | n.a. | PMID[547904] | |
NPT2 | Others | Unspecified | IC50 | = | 7000.0 | nM | PMID[547905] | |
NPT2 | Others | Unspecified | IC50 | = | 35000.0 | nM | PMID[547905] | |
NPT4979 | Uncleic Acid | Rev responsive element (RRE) RNA | Kd | = | 180.0 | nM | PMID[547907] | |
NPT4979 | Uncleic Acid | Rev responsive element (RRE) RNA | Kd | = | 370.0 | nM | PMID[547907] | |
NPT4979 | Uncleic Acid | Rev responsive element (RRE) RNA | Ratio | = | 2.1 | n.a. | PMID[547907] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | IZ | = | 15.0 | mm | PMID[547908] |
NPT19 | Organism | Escherichia coli | Escherichia coli | IZ | = | 18.0 | mm | PMID[547908] |
NPT19 | Organism | Escherichia coli | Escherichia coli | IZ | = | 12.0 | mm | PMID[547908] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 0.5 | ug.mL-1 | PMID[547909] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 64.0 | ug.mL-1 | PMID[547909] |
NPT1521 | Organism | Stenotrophomonas maltophilia | Stenotrophomonas maltophilia | MIC | = | 512.0 | ug.mL-1 | PMID[547909] |
NPT1521 | Organism | Stenotrophomonas maltophilia | Stenotrophomonas maltophilia | MIC | = | 64.0 | ug.mL-1 | PMID[547909] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 250.0 | ug.mL-1 | PMID[547910] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC | = | 250.0 | ug.mL-1 | PMID[547910] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC | = | 125.0 | ug.mL-1 | PMID[547910] |
NPT2901 | Organism | Bifidobacterium thermophilum | Bifidobacterium thermophilum | MIC | = | 250.0 | ug.mL-1 | PMID[547910] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 125.0 | ug.mL-1 | PMID[547910] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC | = | 500.0 | ug.mL-1 | PMID[547910] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 62.5 | ug.mL-1 | PMID[547910] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 500.0 | ug.mL-1 | PMID[547910] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC | = | 62.5 | ug.mL-1 | PMID[547910] |
NPT2901 | Organism | Bifidobacterium thermophilum | Bifidobacterium thermophilum | MIC | = | 125.0 | ug.mL-1 | PMID[547910] |
NPT2901 | Organism | Bifidobacterium thermophilum | Bifidobacterium thermophilum | MIC | = | 500.0 | ug.mL-1 | PMID[547910] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 128.0 | ug.mL-1 | PMID[547911] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 12.0 | ug.mL-1 | PMID[547911] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 96.0 | ug.mL-1 | PMID[547911] |
NPT26263 | SINGLE PROTEIN | Aminoglycoside 3'-phosphotransferase type IIb | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | Km | = | 17500.0 | nM | PMID[547911] |
NPT26263 | SINGLE PROTEIN | Aminoglycoside 3'-phosphotransferase type IIb | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | Kcat/Km | = | 120000.0 | /M/s | PMID[547911] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547912] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 0.12 | ug.mL-1 | PMID[547912] |
NPT938 | Organism | Cavia porcellus | Cavia porcellus | Activity | = | 0.0 | % | PMID[547913] |
NPT938 | Organism | Cavia porcellus | Cavia porcellus | Activity | = | 100.0 | % | PMID[547913] |
NPT938 | Organism | Cavia porcellus | Cavia porcellus | Activity | = | 50.0 | % | PMID[547913] |
NPT2 | Others | Unspecified | Kd | = | 308.0 | nM | PMID[547914] | |
NPT2 | Others | Unspecified | Kd | = | 313.0 | nM | PMID[547914] | |
NPT2 | Others | Unspecified | Kd | = | 320.0 | nM | PMID[547914] | |
NPT2 | Others | Unspecified | Kd | = | 6300.0 | nM | PMID[547914] | |
NPT2 | Others | Unspecified | Kd | = | 2300.0 | nM | PMID[547914] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547915] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | >= | 32.0 | ug.mL-1 | PMID[547915] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | >= | 32.0 | ug.mL-1 | PMID[547915] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 16.0 | ug.mL-1 | PMID[547915] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 8.0 | ug.mL-1 | PMID[547915] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 0.5 | ug.mL-1 | PMID[547915] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | IZ | = | 9.0 | mm | PMID[547916] |
NPT2 | Others | Unspecified | Kd | = | 8000.0 | nM | PMID[547917] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 384.0 | ug.mL-1 | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 96.0 | ug.mL-1 | PMID[547918] |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | MIC | = | 1.5 | ug.mL-1 | PMID[547918] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 384.0 | ug.mL-1 | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 6.0 | ug.mL-1 | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | > | 384.0 | ug.mL-1 | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | Ratio | > | 64.0 | n.a. | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | Ratio | = | 16.0 | n.a. | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 48.0 | ug.mL-1 | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | Ratio | = | 8.0 | n.a. | PMID[547918] |
NPT19 | Organism | Escherichia coli | Escherichia coli | IC50 | = | 10500.0 | nM | PMID[547918] |
NPT2 | Others | Unspecified | Kcat | = | 2.4 | /s | PMID[547918] | |
NPT2 | Others | Unspecified | Kcat/Km | = | 42.0 | 10'-4/M/s | PMID[547918] | |
NPT2 | Others | Unspecified | Km | = | 5700.0 | nM | PMID[547918] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 24.0 | ug.mL-1 | PMID[547918] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 2.0 | ug.mL-1 | PMID[547919] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 256.0 | ug.mL-1 | PMID[547919] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC | = | 1.0 | ug.mL-1 | PMID[547919] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC | = | 0.5 | ug.mL-1 | PMID[547919] |
NPT1118 | Organism | Streptococcus pneumoniae | Streptococcus pneumoniae | MIC | = | 64.0 | ug.mL-1 | PMID[547919] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 8.0 | ug.mL-1 | PMID[547919] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547919] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 512.0 | ug.mL-1 | PMID[547919] |
NPT20 | Organism | Candida albicans | Candida albicans | MIC | >= | 512.0 | ug.mL-1 | PMID[547919] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547920] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547920] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | >= | 2000.0 | ug.mL-1 | PMID[547920] |
NPT2 | Others | Unspecified | Km | = | 6000.0 | nM | PMID[547920] | |
NPT2 | Others | Unspecified | Vmax | = | 3.22 | umol/min/mg | PMID[547920] | |
NPT2 | Others | Unspecified | Kcat | = | 1.61 | /s | PMID[547920] | |
NPT2 | Others | Unspecified | Kcat/Km | = | 26.8 | 10'4/M/s | PMID[547920] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 64.0 | ug.mL-1 | PMID[547920] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 8.0 | ug.mL-1 | PMID[547920] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 4.0 | ug.mL-1 | PMID[547920] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 16.0 | ug.mL-1 | PMID[547920] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 125.0 | ug.mL-1 | PMID[547920] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547920] |
NPT175 | Organism | Enterococcus faecalis | Enterococcus faecalis | MIC | = | 64.0 | ug.mL-1 | PMID[547920] |
NPT175 | Organism | Enterococcus faecalis | Enterococcus faecalis | MIC | >= | 250.0 | ug.mL-1 | PMID[547920] |
NPT2 | Others | Unspecified | Tm | = | 65.8 | degrees C | PMID[547921] | |
NPT2 | Others | Unspecified | Tm | = | 64.7 | degrees C | PMID[547921] | |
NPT2 | Others | Unspecified | Tm | = | 62.9 | degrees C | PMID[547921] | |
NPT2 | Others | Unspecified | Ka | = | 7.0 | 10'4/M | PMID[547921] | |
NPT2 | Others | Unspecified | Ka | = | 2.6 | 10'7/M | PMID[547921] | |
NPT2 | Others | Unspecified | Ka | = | 9.9 | 10'6/M | PMID[547921] | |
NPT2 | Others | Unspecified | IC50 | = | 11000.0 | nM | PMID[547922] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 60.0 | nM | PMID[547923] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | > | 256.0 | ug.mL-1 | PMID[547924] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 64.0 | ug.mL-1 | PMID[547924] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 0.13 | ug.mL-1 | PMID[547924] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 0.25 | ug.mL-1 | PMID[547924] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | IC50 | = | 0.6 | ug.mL-1 | PMID[547925] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 2.0 | ug.mL-1 | PMID[547926] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547926] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 128.0 | ug.mL-1 | PMID[547926] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 32.0 | ug.mL-1 | PMID[547926] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 128.0 | ug.mL-1 | PMID[547926] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | = | 0.5 | ug.mL-1 | PMID[547926] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | > | 128.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 128.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 32.0 | ug.mL-1 | PMID[547926] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 16.0 | ug.mL-1 | PMID[547926] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2.0 | ug.mL-1 | PMID[547926] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547926] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 32.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | Inhibition | = | 40.0 | % | PMID[547926] |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 1550.0 | nM | PMID[547926] | |
NPT1548 | Organism | Pseudomonas aeruginosa PAO1 | Pseudomonas aeruginosa PAO1 | MIC | = | 4.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 8.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 4.0 | ug.mL-1 | PMID[547926] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 2.0 | ug.mL-1 | PMID[547926] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547927] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547927] |
NPT317 | Uncleic Acid | Nucleic Acid | Delta Tm | = | 0.0 | degrees C | PMID[547928] | |
NPT605 | Organism | Homo sapiens | Homo sapiens | Activity | = | 0.0 | % | PMID[547929] |
NPT1118 | Organism | Streptococcus pneumoniae | Streptococcus pneumoniae | MIC | = | 1.0 | ug.mL-1 | PMID[547930] |
NPT747 | Organism | Acinetobacter baumannii | Acinetobacter baumannii | MIC | = | 64.0 | ug.mL-1 | PMID[547930] |
NPT1521 | Organism | Stenotrophomonas maltophilia | Stenotrophomonas maltophilia | MIC | > | 512.0 | ug.mL-1 | PMID[547930] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 512.0 | ug.mL-1 | PMID[547930] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 8.0 | ug.mL-1 | PMID[547930] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547930] |
NPT1118 | Organism | Streptococcus pneumoniae | Streptococcus pneumoniae | MIC | = | 32.0 | ug.mL-1 | PMID[547930] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC | = | 0.5 | ug.mL-1 | PMID[547930] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC | = | 0.25 | ug.mL-1 | PMID[547930] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 256.0 | ug.mL-1 | PMID[547930] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547930] |
NPT35 | Others | n.a. | Kd | = | 2600.0 | nM | PMID[547931] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 10.0 | % | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 6.0 | % | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | FC | = | 1.5 | n.a. | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | FC | = | 3.0 | n.a. | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 70.3 | % | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 52.0 | % | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 0.31 | /s | PMID[547933] | |
NPT317 | Uncleic Acid | Nucleic Acid | Activity | = | 0.06 | /s | PMID[547933] | |
NPT2 | Others | Unspecified | Kcat/Km | = | 1.5 | 10'5/s/M | PMID[547934] | |
NPT2 | Others | Unspecified | Kcat | = | 1.59 | /s | PMID[547934] | |
NPT2 | Others | Unspecified | Km | = | 10600.0 | nM | PMID[547934] | |
NPT2905 | Organism | Nocardia farcinica | Nocardia farcinica | MIC | > | 1024.0 | ug.mL-1 | PMID[547935] |
NPT2905 | Organism | Nocardia farcinica | Nocardia farcinica | MIC | = | 16.0 | ug.mL-1 | PMID[547935] |
NPT4981 | Organism | Clostridium sordellii | Clostridium sordellii | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1824 | Organism | Clostridium sporogenes | Clostridium sporogenes | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4835 | Organism | Clostridium tertium | Clostridium tertium | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4831 | Organism | Actinomyces meyeri | Actinomyces meyeri | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1129 | Organism | Actinomyces viscosus | Actinomyces viscosus | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4982 | Organism | Collinsella aerofaciens | Collinsella aerofaciens | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4836 | Organism | Eggerthella lenta | Eggerthella lenta | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4983 | Organism | Eubacterium limosum | Eubacterium limosum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4128 | Organism | Lactobacillus fermentum | Lactobacillus fermentum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1825 | Organism | Lactobacillus plantarum | Lactobacillus plantarum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT3593 | Organism | Lactobacillus sp. | Lactobacillus sp. | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT167 | Organism | Propionibacterium acnes | Propionibacterium acnes | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4819 | Organism | Anaerococcus prevotii | Anaerococcus prevotii | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4984 | Organism | Anaerococcus tetradius | Anaerococcus tetradius | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4817 | Organism | Finegoldia magna | Finegoldia magna | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4818 | Organism | Peptoniphilus asaccharolyticus | Peptoniphilus asaccharolyticus | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4821 | Organism | Peptostreptococcus anaerobius | Peptostreptococcus anaerobius | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4820 | Organism | Peptostreptococcus micros | Parvimonas micra | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 4.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4985 | Organism | Clostridium acetobutylicum | Clostridium acetobutylicum | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4986 | Organism | Clostridium bifermentans | Clostridium bifermentans | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4987 | Organism | Clostridium butyricum | Clostridium butyricum | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4988 | Organism | Clostridium cadaveris | Clostridium cadaveris | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4833 | Organism | Clostridium paraputrificum | Clostridium paraputrificum | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4989 | Organism | Clostridium ramosum | Clostridium ramosum | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4834 | Organism | Clostridium septicum | Clostridium septicum | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4981 | Organism | Clostridium sordellii | Clostridium sordellii | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT1824 | Organism | Clostridium sporogenes | Clostridium sporogenes | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4835 | Organism | Clostridium tertium | Clostridium tertium | MIC | = | 1.0 | ug.mL-1 | PMID[547936] |
NPT4831 | Organism | Actinomyces meyeri | Actinomyces meyeri | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT1129 | Organism | Actinomyces viscosus | Actinomyces viscosus | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4982 | Organism | Collinsella aerofaciens | Collinsella aerofaciens | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4836 | Organism | Eggerthella lenta | Eggerthella lenta | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4983 | Organism | Eubacterium limosum | Eubacterium limosum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4128 | Organism | Lactobacillus fermentum | Lactobacillus fermentum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT1825 | Organism | Lactobacillus plantarum | Lactobacillus plantarum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT3593 | Organism | Lactobacillus sp. | Lactobacillus sp. | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT167 | Organism | Propionibacterium acnes | Propionibacterium acnes | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4819 | Organism | Anaerococcus prevotii | Anaerococcus prevotii | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4984 | Organism | Anaerococcus tetradius | Anaerococcus tetradius | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4817 | Organism | Finegoldia magna | Finegoldia magna | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4818 | Organism | Peptoniphilus asaccharolyticus | Peptoniphilus asaccharolyticus | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4821 | Organism | Peptostreptococcus anaerobius | Peptostreptococcus anaerobius | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4820 | Organism | Peptostreptococcus micros | Parvimonas micra | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT1092 | Organism | Bacteroides fragilis | Bacteroides fragilis | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4810 | Organism | Bacteroides distasonis | Parabacteroides distasonis | MIC50 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4812 | Organism | Parabacteroides merdae | Parabacteroides merdae | MIC50 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4811 | Organism | Bacteroides ovatus | Bacteroides ovatus | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT3572 | Organism | Bacteroides thetaiotaomicron | Bacteroides thetaiotaomicron | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1092 | Organism | Bacteroides fragilis | Bacteroides fragilis | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4810 | Organism | Bacteroides distasonis | Parabacteroides distasonis | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4810 | Organism | Bacteroides distasonis | Parabacteroides distasonis | MIC | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4812 | Organism | Parabacteroides merdae | Parabacteroides merdae | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4812 | Organism | Parabacteroides merdae | Parabacteroides merdae | MIC | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4811 | Organism | Bacteroides ovatus | Bacteroides ovatus | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT3572 | Organism | Bacteroides thetaiotaomicron | Bacteroides thetaiotaomicron | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4809 | Organism | Bacteroides caccae | Bacteroides caccae | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4813 | Organism | Bacteroides stercoris | Bacteroides stercoris | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4807 | Organism | Bacteroides uniformis | Bacteroides uniformis | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4809 | Organism | Bacteroides caccae | Bacteroides caccae | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4813 | Organism | Bacteroides stercoris | Bacteroides stercoris | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4807 | Organism | Bacteroides uniformis | Bacteroides uniformis | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT1484 | Organism | Fusobacterium nucleatum | Fusobacterium nucleatum | MIC50 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4825 | Organism | Fusobacterium mortiferum | Fusobacterium mortiferum | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4828 | Organism | Fusobacterium necrophorum | Fusobacterium necrophorum | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4826 | Organism | Fusobacterium varium | Fusobacterium varium | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4990 | Organism | Fusobacterium sp. | Fusobacterium sp. | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4827 | Organism | Porphyromonas asaccharolytica | Porphyromonas asaccharolytica | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4991 | Organism | Porphyromonas somerae | Porphyromonas somerae | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4824 | Organism | Prevotella bivia | Prevotella bivia | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4992 | Organism | Prevotella corporis | Prevotella corporis | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4993 | Organism | Prevotella disiens | Prevotella disiens | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT1128 | Organism | Prevotella intermedia | Prevotella intermedia | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4429 | Organism | Prevotella loescheii | Prevotella loescheii | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4829 | Organism | Prevotella melaninogenica | Prevotella melaninogenica | MIC50 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT4994 | Organism | Clostridium clostridioforme | Clostridium clostridioforme | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT2940 | Organism | Clostridium difficile | Clostridium difficile | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT1484 | Organism | Fusobacterium nucleatum | Fusobacterium nucleatum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4825 | Organism | Fusobacterium mortiferum | Fusobacterium mortiferum | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4828 | Organism | Fusobacterium necrophorum | Fusobacterium necrophorum | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4826 | Organism | Fusobacterium varium | Fusobacterium varium | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4990 | Organism | Fusobacterium sp. | Fusobacterium sp. | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4827 | Organism | Porphyromonas asaccharolytica | Porphyromonas asaccharolytica | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4991 | Organism | Porphyromonas somerae | Porphyromonas somerae | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4824 | Organism | Prevotella bivia | Prevotella bivia | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4992 | Organism | Prevotella corporis | Prevotella corporis | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4993 | Organism | Prevotella disiens | Prevotella disiens | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1128 | Organism | Prevotella intermedia | Prevotella intermedia | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4429 | Organism | Prevotella loescheii | Prevotella loescheii | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4829 | Organism | Prevotella melaninogenica | Prevotella melaninogenica | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4994 | Organism | Clostridium clostridioforme | Clostridium clostridioforme | MIC90 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT2940 | Organism | Clostridium difficile | Clostridium difficile | MIC90 | = | 512.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 32.0 | ug.mL-1 | PMID[547936] |
NPT1484 | Organism | Fusobacterium nucleatum | Fusobacterium nucleatum | MIC | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4825 | Organism | Fusobacterium mortiferum | Fusobacterium mortiferum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4828 | Organism | Fusobacterium necrophorum | Fusobacterium necrophorum | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4826 | Organism | Fusobacterium varium | Fusobacterium varium | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT4990 | Organism | Fusobacterium sp. | Fusobacterium sp. | MIC | = | 2.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4827 | Organism | Porphyromonas asaccharolytica | Porphyromonas asaccharolytica | MIC | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4991 | Organism | Porphyromonas somerae | Porphyromonas somerae | MIC | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4824 | Organism | Prevotella bivia | Prevotella bivia | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT4992 | Organism | Prevotella corporis | Prevotella corporis | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT4993 | Organism | Prevotella disiens | Prevotella disiens | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT1128 | Organism | Prevotella intermedia | Prevotella intermedia | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT4429 | Organism | Prevotella loescheii | Prevotella loescheii | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT4829 | Organism | Prevotella melaninogenica | Prevotella melaninogenica | MIC | = | 8.0 | ug.mL-1 | PMID[547936] |
NPT4994 | Organism | Clostridium clostridioforme | Clostridium clostridioforme | MIC | = | 32.0 | ug.mL-1 | PMID[547936] |
NPT2940 | Organism | Clostridium difficile | Clostridium difficile | MIC | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | = | 64.0 | ug.mL-1 | PMID[547936] |
NPT4995 | Organism | Clostridium innocuum | Clostridium innocuum | MIC50 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1359 | Organism | Clostridium perfringens | Clostridium perfringens | MIC50 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4985 | Organism | Clostridium acetobutylicum | Clostridium acetobutylicum | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4986 | Organism | Clostridium bifermentans | Clostridium bifermentans | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4987 | Organism | Clostridium butyricum | Clostridium butyricum | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4988 | Organism | Clostridium cadaveris | Clostridium cadaveris | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4833 | Organism | Clostridium paraputrificum | Clostridium paraputrificum | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4989 | Organism | Clostridium ramosum | Clostridium ramosum | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4834 | Organism | Clostridium septicum | Clostridium septicum | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4981 | Organism | Clostridium sordellii | Clostridium sordellii | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT1824 | Organism | Clostridium sporogenes | Clostridium sporogenes | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4835 | Organism | Clostridium tertium | Clostridium tertium | MIC50 | = | 256.0 | ug.mL-1 | PMID[547936] |
NPT4831 | Organism | Actinomyces meyeri | Actinomyces meyeri | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT1129 | Organism | Actinomyces viscosus | Actinomyces viscosus | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT2900 | Organism | Bifidobacterium longum | Bifidobacterium longum | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4982 | Organism | Collinsella aerofaciens | Collinsella aerofaciens | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4836 | Organism | Eggerthella lenta | Eggerthella lenta | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4983 | Organism | Eubacterium limosum | Eubacterium limosum | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4128 | Organism | Lactobacillus fermentum | Lactobacillus fermentum | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT1825 | Organism | Lactobacillus plantarum | Lactobacillus plantarum | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT3593 | Organism | Lactobacillus sp. | Lactobacillus sp. | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT167 | Organism | Propionibacterium acnes | Propionibacterium acnes | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4819 | Organism | Anaerococcus prevotii | Anaerococcus prevotii | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4984 | Organism | Anaerococcus tetradius | Anaerococcus tetradius | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4817 | Organism | Finegoldia magna | Finegoldia magna | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4818 | Organism | Peptoniphilus asaccharolyticus | Peptoniphilus asaccharolyticus | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4821 | Organism | Peptostreptococcus anaerobius | Peptostreptococcus anaerobius | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4820 | Organism | Peptostreptococcus micros | Parvimonas micra | MIC50 | = | 128.0 | ug.mL-1 | PMID[547936] |
NPT4995 | Organism | Clostridium innocuum | Clostridium innocuum | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1359 | Organism | Clostridium perfringens | Clostridium perfringens | MIC90 | > | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4985 | Organism | Clostridium acetobutylicum | Clostridium acetobutylicum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4986 | Organism | Clostridium bifermentans | Clostridium bifermentans | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4987 | Organism | Clostridium butyricum | Clostridium butyricum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4988 | Organism | Clostridium cadaveris | Clostridium cadaveris | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4833 | Organism | Clostridium paraputrificum | Clostridium paraputrificum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4989 | Organism | Clostridium ramosum | Clostridium ramosum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT4834 | Organism | Clostridium septicum | Clostridium septicum | MIC90 | = | 1024.0 | ug.mL-1 | PMID[547936] |
NPT1101 | Organism | Staphylococcus aureus subsp. aureus RN4220 | Staphylococcus aureus subsp. aureus RN4220 | MIC | = | 2.0 | ug.mL-1 | PMID[547938] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 4.0 | ug.mL-1 | PMID[547938] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 2.0 | ug.mL-1 | PMID[547938] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547939] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 3.0 | ug.mL-1 | PMID[547939] |
NPT2908 | Organism | Streptomyces coelicolor | Streptomyces coelicolor | MIC | = | 0.3 | ug.mL-1 | PMID[547940] |
NPT2908 | Organism | Streptomyces coelicolor | Streptomyces coelicolor | MIC | = | 0.8 | ug.mL-1 | PMID[547940] |
NPT2908 | Organism | Streptomyces coelicolor | Streptomyces coelicolor | MIC | = | 0.5 | ug.mL-1 | PMID[547940] |
NPT2908 | Organism | Streptomyces coelicolor | Streptomyces coelicolor | MIC | = | 0.2 | ug.mL-1 | PMID[547940] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | Activity | = | 8.0 | ug ml-1 | PMID[547941] |
NPT2909 | Organism | Shigella flexneri | Shigella flexneri | Activity | = | 8.0 | ug ml-1 | PMID[547941] |
NPT2911 | Organism | Pseudomonas putida | Pseudomonas putida | Activity | = | 8.0 | ug ml-1 | PMID[547941] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | Activity | = | 8.0 | ug ml-1 | PMID[547941] |
NPT317 | Uncleic Acid | Nucleic Acid | EC50 | = | 7.0 | nM | PMID[547942] | |
NPT25608 | PROTEIN NUCLEIC-ACID COMPLEX | Bacterial 70S ribosome | Bacteria | IC50 | = | 32.0 | nM | PMID[547942] |
NPT4795 | Subcellular | Ribosome | IC50 | = | 252000.0 | nM | PMID[547942] | |
NPT175 | Organism | Enterococcus faecalis | Enterococcus faecalis | MIC | = | 125.0 | ug.mL-1 | PMID[547943] |
NPT175 | Organism | Enterococcus faecalis | Enterococcus faecalis | MIC | = | 16.0 | ug.mL-1 | PMID[547943] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547943] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 125.0 | ug.mL-1 | PMID[547943] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 2.0 | ug.mL-1 | PMID[547943] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547943] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547943] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 8.0 | ug.mL-1 | PMID[547944] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2.0 | ug.mL-1 | PMID[547944] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547944] |
NPT2 | Others | Unspecified | IC50 | = | 7.9 | nM | PMID[547945] | |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC50 | = | 2.0 | ug.mL-1 | PMID[547946] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC90 | = | 32.0 | ug.mL-1 | PMID[547946] |
NPT27 | Others | Unspecified | log10(%HIA +10) | = | 1.041 | n.a. | PMID[547947] | |
NPT1101 | Organism | Staphylococcus aureus subsp. aureus RN4220 | Staphylococcus aureus subsp. aureus RN4220 | MIC | <= | 1.0 | ug.mL-1 | PMID[547948] |
NPT1101 | Organism | Staphylococcus aureus subsp. aureus RN4220 | Staphylococcus aureus subsp. aureus RN4220 | MIC | = | 64.0 | ug.mL-1 | PMID[547948] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 128.0 | ug.mL-1 | PMID[547950] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | <= | 1.0 | ug.mL-1 | PMID[547950] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 32.0 | ug.mL-1 | PMID[547950] |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 1500.0 | nM | PMID[547953] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 1100.0 | nM | PMID[547953] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | < | 1000.0 | nM | PMID[547954] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 417.0 | nM | PMID[547954] | |
NPT317 | Uncleic Acid | Nucleic Acid | Tm | = | 69.1 | degrees C | PMID[547954] | |
NPT317 | Uncleic Acid | Nucleic Acid | Delta Tm | = | 0.2 | degrees C | PMID[547954] | |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_bilirubinemia | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_cholecystitis | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_cholelithiasis | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_cirrhosis | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_elevated liver function tests | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_hepatic failure | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_hepatic necrosis | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_hepatitis | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_hepatomegaly | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_jaundice | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_liver disease | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_liver fatty | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_liver function tests abnormal | = | 0.0 | n.a. | PMID[547957] |
NPT20596 | PHENOTYPE | Hepatotoxicity | n.a. | HepSE_Combined Scores | = | 0.0 | n.a. | PMID[547957] |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 6000.0 | nM | PMID[547958] | |
NPT317 | Uncleic Acid | Nucleic Acid | Tm | = | 50.0 | degrees C | PMID[547958] | |
NPT317 | Uncleic Acid | Nucleic Acid | Tm | > | 70.0 | degrees C | PMID[547958] | |
NPT317 | Uncleic Acid | Nucleic Acid | Inhibition | = | 10.0 | % | PMID[547958] | |
NPT317 | Uncleic Acid | Nucleic Acid | Kd | = | 11000.0 | nM | PMID[547959] | |
NPT317 | Uncleic Acid | Nucleic Acid | Tm | = | 48.0 | degrees C | PMID[547959] | |
NPT317 | Uncleic Acid | Nucleic Acid | Tm | > | 70.0 | degrees C | PMID[547959] | |
NPT317 | Uncleic Acid | Nucleic Acid | Inhibition | = | 10.0 | % | PMID[547959] | |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 0.5 | ug.mL-1 | PMID[547960] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 64.0 | ug.mL-1 | PMID[547960] |
NPT4996 | Organism | Chryseobacterium meningosepticum | Elizabethkingia meningoseptica | MIC | = | 12.5 | ug.mL-1 | PMID[547962] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 6.25 | ug.mL-1 | PMID[547962] |
NPT4997 | Organism | Klebsiella oxytoca | Klebsiella oxytoca | MIC | = | 6.25 | ug.mL-1 | PMID[547962] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 3.13 | ug.mL-1 | PMID[547962] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 25.0 | ug.mL-1 | PMID[547962] |
NPT4998 | Organism | Staphylococcus xylosus | Staphylococcus xylosus | MIC | = | 0.2 | ug.mL-1 | PMID[547962] |
NPT4805 | Organism | Rhodococcus equi | Rhodococcus equi | MIC | = | 1.56 | ug.mL-1 | PMID[547962] |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | MIC | = | 0.78 | ug.mL-1 | PMID[547962] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 18.75 | ug.mL-1 | PMID[547963] |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | MIC | = | 18.75 | ug.mL-1 | PMID[547963] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 18.75 | ug.mL-1 | PMID[547963] |
NPT2 | Others | Unspecified | Kd | = | 1270.0 | nM | PMID[547964] | |
NPT2 | Others | Unspecified | Kd | = | 1148.0 | nM | PMID[547964] | |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1100.0 | nM | PMID[547964] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4400.0 | nM | PMID[547964] |
NPT19 | Organism | Escherichia coli | Escherichia coli | IZ | = | 26.12 | mm | PMID[547965] |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | IZ | = | 26.12 | mm | PMID[547965] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | IZ | = | 25.78 | mm | PMID[547965] |
NPT766 | Organism | Proteus vulgaris | Proteus vulgaris | IZ | = | 25.29 | mm | PMID[547965] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 1.0 | ug.mL-1 | PMID[547966] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547966] |
NPT317 | Uncleic Acid | Nucleic Acid | Delta Tm | = | 2.0 | degrees C | PMID[547967] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 1474.0 | nM | PMID[547967] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2.0 | ug.mL-1 | PMID[547966] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 16.0 | ug.mL-1 | PMID[547966] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 32.0 | ug.mL-1 | PMID[547966] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 128.0 | ug.mL-1 | PMID[547966] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547966] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | > | 128.0 | ug.mL-1 | PMID[547966] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | = | 0.5 | ug.mL-1 | PMID[547966] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 128.0 | ug.mL-1 | PMID[547966] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 128.0 | ug.mL-1 | PMID[547966] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 32.0 | ug.mL-1 | PMID[547966] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547966] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 2.0 | ug.mL-1 | PMID[547966] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC95 | = | 15.62 | uM | PMID[547968] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC95 | = | 7.81 | uM | PMID[547968] |
NPT2 | Others | Unspecified | Ki | = | 18800.0 | nM | PMID[547970] | |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT729 | Organism | Micrococcus luteus | Micrococcus luteus | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT4619 | Organism | Raoultella planticola | Raoultella planticola | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 12.5 | ug.mL-1 | PMID[547971] |
NPT2 | Others | Unspecified | Tm | = | 64.2 | degrees C | PMID[547972] | |
NPT1276 | Organism | Gibberella zeae | Gibberella zeae | MIC | = | 62.5 | ug.mL-1 | PMID[547973] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547973] |
NPT175 | Organism | Enterococcus faecalis | Enterococcus faecalis | MIC | >= | 250.0 | ug.mL-1 | PMID[547973] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547973] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 125.0 | ug.mL-1 | PMID[547973] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547973] |
NPT317 | Uncleic Acid | Nucleic Acid | K | = | 1.6 | 10'7/M | PMID[547974] | |
NPT317 | Uncleic Acid | Nucleic Acid | K | = | 3.0 | 10'7/M | PMID[547974] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 192000.0 | nM | PMID[547974] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 684000.0 | nM | PMID[547974] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 150000.0 | nM | PMID[547974] | |
NPT317 | Uncleic Acid | Nucleic Acid | IC50 | = | 378000.0 | nM | PMID[547974] | |
NPT27 | Others | Unspecified | Delta Tm | = | 1.0 | degrees C | PMID[547974] | |
NPT27 | Others | Unspecified | Delta Tm | = | 0.5 | degrees C | PMID[547974] | |
NPT27 | Others | Unspecified | Delta Tm | = | 0.0 | degrees C | PMID[547974] | |
NPT27 | Others | Unspecified | Delta Tm | = | 0.2 | degrees C | PMID[547974] | |
NPT2 | Others | Unspecified | Inhibition | = | 60.0 | % | PMID[547975] | |
NPT2 | Others | Unspecified | IC50 | = | 88200.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | IC50 | = | 93700.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | IC50 | = | 143000.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | IC50 | = | 76700.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Kd | = | 11600.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Kd | = | 1880.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Kd | = | 15200.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Kd | = | 11700.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Ratio | = | 1.0 | n.a. | PMID[547975] | |
NPT2 | Others | Unspecified | Kd | = | 11300.0 | nM | PMID[547975] | |
NPT2 | Others | Unspecified | Activity | = | 70.0 | % | PMID[547975] | |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 240000.0 | nM | PMID[547976] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1000.0 | nM | PMID[547976] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | Ratio | = | 240.0 | n.a. | PMID[547976] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 1.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 0.5 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | > | 128.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 64.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 128.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 32.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 2.0 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | < | 0.25 | ug.mL-1 | PMID[547977] |
NPT20529 | NON-MOLECULAR | NON-PROTEIN TARGET | n.a. | MIC | = | 4.0 | ug.mL-1 | PMID[547977] |
NPT32 | Organism | Mus musculus | Mus musculus | Activity | = | 87.3 | % | PMID[547977] |
NPT32 | Organism | Mus musculus | Mus musculus | Activity | = | 69.8 | % | PMID[547977] |
NPT2 | Others | Unspecified | Inhibition | = | 20.4 | % | PMID[547978] | |
NPT2 | Others | Unspecified | Delta Tm | = | 10.8 | degrees C | PMID[547978] | |
NPT2 | Others | Unspecified | Delta Tm | = | 10.5 | degrees C | PMID[547978] | |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 33.2 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 37400.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 318.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 78.6 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 60.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 108.4 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 630.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 251.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 1.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1256.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 120.6 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 5.92 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 146.8 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 1.6 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 60600.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASOLE | = | 0.32 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.58 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 7260000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 46.94 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 149000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 8690.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 81.52 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 20.58 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 318000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 64.68 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 2.16 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 13.88 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1531200.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 28.6 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 39400.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 254.6 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 67.8 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 104.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 104.6 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 576.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 224.8 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 4.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1406.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 106.6 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 6.58 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 148.6 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 2.4 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 66400.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASOLE | = | 0.42 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 8060000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 48.44 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 163400.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 13040.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 85.12 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 20.26 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 337400.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 60.1 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 1.44 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 11.28 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1226000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 29.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 336.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 73.8 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 66.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 109.6 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 606.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 307.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 2.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1286.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 138.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 6.96 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 151.8 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 62200.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASOLE | = | 0.36 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.6 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 7450000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 49.44 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 156000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 6840.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 82.08 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 20.94 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 315800.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 66.34 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 1.68 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 14.3 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1274600.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 26.9 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 38500.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 200.9 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 62.4 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 110.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 107.1 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 545.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 177.2 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 3.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1352.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 111.6 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 6.5 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 151.5 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 2.2 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 65200.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASOLE | = | 0.48 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.51 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 8010000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 48.92 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 158800.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 12820.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 83.46 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 19.85 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 324700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 61.12 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 1.54 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 12.95 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1208100.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 76.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 39300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 317.17 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 81.17 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 123.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 31170000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 98.33 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 671.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 312.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 1.9 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1655.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 94.5 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LIPASE | = | 9.83 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 101.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 5.16 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 143.02 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 2.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 58800.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | URATE | = | 6.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASO | = | 0.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOS | = | 33.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 9048.5 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 80.17 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 1521.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BASOLE | = | 0.0 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.17 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 5460000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 32.87 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 129500.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 10680.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 86.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 23.72 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 394000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 60.18 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 0.83 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 12.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBCNUC | = | 0.0 | /100WBC | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1211330.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 93.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 41700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 402.5 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 122.83 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 147.5 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 26400000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 575.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 305.17 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 2.1 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1420.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 83.5 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LIPASE | = | 85.83 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 81.8 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 2.5 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 56300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | URATE | = | 8.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOS | = | 14.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 9629.83 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 72.5 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 1049.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 5360000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 33.82 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 134800.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 10770.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 90.17 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 25.28 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 399200.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 63.3 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 0.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 9.0 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBCNUC | = | 0.17 | /100WBC | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1275330.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 98.5 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 5.46 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 144.0 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 81.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 41000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 367.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 87.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 116.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 33330000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 97.0 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 896.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 277.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1563.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 107.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LIPASE | = | 10.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 108.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 5.83 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 143.17 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 1.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 59700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | URATE | = | 4.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOS | = | 0.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 8427.33 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 92.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 980.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.0 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 33.8 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 134000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 9500.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 88.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 24.57 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 396300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 61.9 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 1.0 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 10.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1108330.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 68.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 40300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 434.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 94.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 120.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 26330000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 104.0 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 746.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 481.67 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 2.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 224.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 105.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 6.71 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 148.83 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BILI | = | 1.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 60300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | URATE | = | 11.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 7805.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 76.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 785.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 5670000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 34.13 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 133000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 8670.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 89.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 23.47 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 389700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 60.2 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 9.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1077000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 85.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 40700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 386.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 105.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 150.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 32330000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 99.33 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 743.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 327.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 1.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1436.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 167.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 103.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | POTASSIUM | = | 5.99 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 145.3 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 60700.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 7138.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 0.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 362.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 5490000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 34.47 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 137000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 7500.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 94.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 25.0 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 397300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 62.97 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONOLE | = | 0.0 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 5.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBCNUC | = | 0.33 | /100WBC | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1072670.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALT | = | 68.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALB | = | 43300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | ALP | = | 349.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | AST | = | 98.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | BUN | = | 166.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CO2 | = | 24670000.0 | nM | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHLORIDE | = | 103.33 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CHOL | = | 683.3 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CK | = | 235.33 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | CREAT | = | 2.2 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | GLUC | = | 1520.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LDH | = | 230.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LIPASE | = | 10.0 | U.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PHOS | = | 108.7 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | SODIUM | = | 149.37 | mEq.L-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PROT | = | 63000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | URATE | = | 15.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOS | = | 26.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYM | = | 7627.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MONO | = | 51.67 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTSG | = | 528.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | EOSLE | = | 0.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | RBC | = | 5340000.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HCT | = | 34.2 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | HGB | = | 135300.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | WBC | = | 8230.0 | cells.uL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | LYMLE | = | 92.67 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCH | = | 25.57 | pg | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCHC | = | 396000.0 | ug.mL-1 | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | MCV | = | 64.43 | fL | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | NEUTLE | = | 6.33 | % | PMID[547979] |
NPT29 | Organism | Rattus norvegicus | Rattus norvegicus | PLAT | = | 1152670.0 | cells.uL-1 | PMID[547979] |
NPT713 | Individual Protein | Bile salt export pump | Homo sapiens | IC50 | > | 135000.0 | nM | PMID[547980] |
NPT32 | Organism | Mus musculus | Mus musculus | LD50 | = | 24.0 | mg.kg-1 | PMID[547981] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 0.5 | ug.mL-1 | PMID[547982] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1.0 | ug.mL-1 | PMID[547982] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 128.0 | ug.mL-1 | PMID[547982] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 64.0 | ug.mL-1 | PMID[547982] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 128.0 | ug.mL-1 | PMID[547982] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 32.0 | ug.mL-1 | PMID[547982] |
NPT18 | Organism | Pseudomonas aeruginosa | Pseudomonas aeruginosa | MIC | = | 2.0 | ug.mL-1 | PMID[547982] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | < | 0.25 | ug.mL-1 | PMID[547982] |
NPT2898 | Organism | Acinetobacter lwoffii | Acinetobacter lwoffii | MIC | = | 64.0 | ug.mL-1 | PMID[547982] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2.0 | ug.mL-1 | PMID[547982] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 4.0 | ug.mL-1 | PMID[547982] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 1.0 | ug.mL-1 | PMID[547982] |
NPT173 | Organism | Klebsiella pneumoniae | Klebsiella pneumoniae | MIC | = | 4.0 | ug.mL-1 | PMID[547982] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 2.0 | ug.mL-1 | PMID[547983] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 2.0 | ug.mL-1 | PMID[547983] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 256.0 | ug.mL-1 | PMID[547983] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 256.0 | ug.mL-1 | PMID[547983] |
NPT4383 | Uncleic Acid | Ribosomal RNA A-site | IC50 | = | 76.0 | nM | PMID[547984] | |
NPT4383 | Uncleic Acid | Ribosomal RNA A-site | IC50 | = | 87.0 | nM | PMID[547984] | |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 400000.0 | nM | PMID[547984] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 1560.0 | nM | PMID[547984] |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 3130.0 | nM | PMID[547984] |
NPT602 | Organism | Mycobacterium smegmatis | Mycobacterium smegmatis | MIC | = | 780.0 | nM | PMID[547984] |
NPT1550 | Organism | Bacillus anthracis | Bacillus anthracis | MIC | = | 1560.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 400000.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 200000.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 100000.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 400000.0 | nM | PMID[547984] |
NPT17 | Organism | Staphylococcus epidermidis | Staphylococcus epidermidis | MIC | = | 1560.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1560.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 6300.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 3200.0 | nM | PMID[547984] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 1600.0 | nM | PMID[547984] |
NPT4383 | Uncleic Acid | Ribosomal RNA A-site | IC50 | = | 139.0 | nM | PMID[547984] | |
NPT27 | Others | Unspecified | Activity | = | 50.0 | % | PMID[547984] | |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Kd | = | 100.0 | nM | PMID[547985] |
NPT2 | Others | Unspecified | Kd | = | 1.0 | nM | PMID[547986] | |
NPT2 | Others | Unspecified | Kd | = | 1100.0 | nM | PMID[547986] | |
NPT2 | Others | Unspecified | Kd | = | 100.0 | nM | PMID[547986] | |
NPT2 | Others | Unspecified | Ratio IC50 | = | 200.0 | n.a. | PMID[547986] | |
NPT2 | Others | Unspecified | Selectivity ratio | = | 1100.0 | n.a. | PMID[547986] | |
NPT2 | Others | Unspecified | Ratio IC50 | = | 20.0 | n.a. | PMID[547986] | |
NPT2 | Others | Unspecified | Selectivity ratio | = | 100.0 | n.a. | PMID[547986] | |
NPT2 | Others | Unspecified | Kd | = | 5.0 | nM | PMID[547986] | |
NPT2 | Others | Unspecified | Inhibition | = | 20.0 | % | PMID[547986] | |
NPT2 | Others | Unspecified | Kd | = | 779000.0 | nM | PMID[547988] | |
NPT20556 | SINGLE PROTEIN | Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Inhibition | = | 13.52 | % | PMID[547989] |
NPT20555 | ORGANISM | SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | Inhibition | = | -0.07 | % | PMID[547990] |
NPT27 | Others | Unspecified | Inhibition | = | 20.0 | % | PMID[547991] | |
NPT20555 | ORGANISM | SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | IC50 | > | 20000.0 | nM | PMID[547992] |
NPT20555 | ORGANISM | SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | IC50 | > | 19952.62 | nM | PMID[547992] |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | > | 50.0 | ug.mL-1 | PMID[547993] |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Kd | = | 1390.0 | nM | PMID[547994] |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Kd | = | 1415.0 | nM | PMID[547994] |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Ratio | = | 1.0 | n.a. | PMID[547994] |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Kd | = | 1950.0 | nM | PMID[547994] |
NPT536 | Uncleic Acid | microRNA 21 | Homo sapiens | Ratio | = | 1.4 | n.a. | PMID[547994] |
☑ Note for Activity Records:
☉ The quantitative biological activities were primarily integrated from ChEMBL (Version-30) database and were also directly collected from PubMed literature. PubMed PMID was provided as the reference link for each activity record.
Top-200 similar NPs were calculated against the active-NP-set (includes 4,3285 NPs with experimentally-derived bioactivity available in NPASS)
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC176381 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
1.0 | High Similarity | NPC195969 |
0.9759 | High Similarity | NPC214376 |
0.9759 | High Similarity | NPC314408 |
0.9759 | High Similarity | NPC477060 |
0.9759 | High Similarity | NPC123746 |
0.9759 | High Similarity | NPC43850 |
0.9759 | High Similarity | NPC314007 |
0.9651 | High Similarity | NPC315334 |
0.9639 | High Similarity | NPC313552 |
0.9157 | High Similarity | NPC263058 |
0.9036 | High Similarity | NPC315969 |
0.9 | High Similarity | NPC330590 |
0.8617 | High Similarity | NPC315036 |
0.8571 | High Similarity | NPC318258 |
0.8421 | Intermediate Similarity | NPC471628 |
0.8421 | Intermediate Similarity | NPC56298 |
0.7864 | Intermediate Similarity | NPC57436 |
0.7864 | Intermediate Similarity | NPC121479 |
0.7717 | Intermediate Similarity | NPC306838 |
0.7624 | Intermediate Similarity | NPC221148 |
0.7447 | Intermediate Similarity | NPC470282 |
0.7416 | Intermediate Similarity | NPC316807 |
0.7349 | Intermediate Similarity | NPC322801 |
0.7349 | Intermediate Similarity | NPC129100 |
0.7349 | Intermediate Similarity | NPC291650 |
0.7333 | Intermediate Similarity | NPC70574 |
0.7333 | Intermediate Similarity | NPC100204 |
0.7333 | Intermediate Similarity | NPC83248 |
0.7315 | Intermediate Similarity | NPC241597 |
0.7283 | Intermediate Similarity | NPC165119 |
0.7222 | Intermediate Similarity | NPC98750 |
0.7174 | Intermediate Similarity | NPC36927 |
0.7174 | Intermediate Similarity | NPC271772 |
0.7105 | Intermediate Similarity | NPC94319 |
0.697 | Remote Similarity | NPC328646 |
0.6882 | Remote Similarity | NPC471420 |
0.6771 | Remote Similarity | NPC192025 |
0.6771 | Remote Similarity | NPC125253 |
0.6771 | Remote Similarity | NPC253975 |
0.6701 | Remote Similarity | NPC83839 |
0.6667 | Remote Similarity | NPC150557 |
0.6667 | Remote Similarity | NPC470284 |
0.6606 | Remote Similarity | NPC317534 |
0.6517 | Remote Similarity | NPC327486 |
0.6517 | Remote Similarity | NPC223174 |
0.6517 | Remote Similarity | NPC327753 |
0.6346 | Remote Similarity | NPC470283 |
0.6311 | Remote Similarity | NPC208537 |
0.6311 | Remote Similarity | NPC270005 |
0.631 | Remote Similarity | NPC34877 |
0.631 | Remote Similarity | NPC290179 |
0.6293 | Remote Similarity | NPC313813 |
0.625 | Remote Similarity | NPC20035 |
0.6211 | Remote Similarity | NPC314772 |
0.6211 | Remote Similarity | NPC314968 |
0.6161 | Remote Similarity | NPC59589 |
0.6147 | Remote Similarity | NPC188453 |
0.6147 | Remote Similarity | NPC42320 |
0.6118 | Remote Similarity | NPC317023 |
0.61 | Remote Similarity | NPC476523 |
0.6092 | Remote Similarity | NPC17455 |
0.6036 | Remote Similarity | NPC314413 |
0.6036 | Remote Similarity | NPC239705 |
0.6036 | Remote Similarity | NPC314398 |
0.6022 | Remote Similarity | NPC474468 |
0.6 | Remote Similarity | NPC244539 |
0.6 | Remote Similarity | NPC472025 |
0.5982 | Remote Similarity | NPC62845 |
0.5982 | Remote Similarity | NPC166242 |
0.5982 | Remote Similarity | NPC322449 |
0.5982 | Remote Similarity | NPC189854 |
0.5982 | Remote Similarity | NPC92874 |
0.5938 | Remote Similarity | NPC313762 |
0.5929 | Remote Similarity | NPC10897 |
0.5929 | Remote Similarity | NPC325900 |
0.5904 | Remote Similarity | NPC67660 |
0.5904 | Remote Similarity | NPC130683 |
0.5904 | Remote Similarity | NPC145112 |
0.5904 | Remote Similarity | NPC157514 |
0.5904 | Remote Similarity | NPC323361 |
0.5904 | Remote Similarity | NPC269166 |
0.5904 | Remote Similarity | NPC242073 |
0.5904 | Remote Similarity | NPC246558 |
0.5904 | Remote Similarity | NPC107914 |
0.5904 | Remote Similarity | NPC58629 |
0.5904 | Remote Similarity | NPC165198 |
0.5904 | Remote Similarity | NPC89145 |
0.5897 | Remote Similarity | NPC314306 |
0.5887 | Remote Similarity | NPC68327 |
0.5833 | Remote Similarity | NPC303727 |
0.5795 | Remote Similarity | NPC477757 |
0.5795 | Remote Similarity | NPC472026 |
0.5795 | Remote Similarity | NPC477755 |
0.5795 | Remote Similarity | NPC477750 |
0.5795 | Remote Similarity | NPC477762 |
0.5795 | Remote Similarity | NPC477753 |
0.5795 | Remote Similarity | NPC477763 |
0.5778 | Remote Similarity | NPC6848 |
0.5745 | Remote Similarity | NPC476694 |
0.5745 | Remote Similarity | NPC28959 |
0.5745 | Remote Similarity | NPC476695 |
0.5745 | Remote Similarity | NPC137554 |
0.5745 | Remote Similarity | NPC255535 |
0.5745 | Remote Similarity | NPC299603 |
0.5745 | Remote Similarity | NPC476696 |
0.5745 | Remote Similarity | NPC285014 |
0.5726 | Remote Similarity | NPC139857 |
0.5714 | Remote Similarity | NPC315980 |
0.5701 | Remote Similarity | NPC61894 |
0.5701 | Remote Similarity | NPC475603 |
0.5663 | Remote Similarity | NPC326533 |
0.5652 | Remote Similarity | NPC475918 |
0.5638 | Remote Similarity | NPC475694 |
0.5638 | Remote Similarity | NPC473710 |
0.5635 | Remote Similarity | NPC75839 |
0.5632 | Remote Similarity | NPC219040 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC176381 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
1.0 | High Similarity | NPD5795 | Approved |
1.0 | High Similarity | NPD5797 | Approved |
1.0 | High Similarity | NPD5794 | Approved |
1.0 | High Similarity | NPD5796 | Clinical (unspecified phase) |
1.0 | High Similarity | NPD5798 | Approved |
0.9759 | High Similarity | NPD3203 | Approved |
0.9759 | High Similarity | NPD3207 | Approved |
0.9759 | High Similarity | NPD3209 | Approved |
0.9759 | High Similarity | NPD2698 | Approved |
0.9759 | High Similarity | NPD3201 | Approved |
0.9759 | High Similarity | NPD3202 | Approved |
0.9759 | High Similarity | NPD3208 | Approved |
0.9639 | High Similarity | NPD3200 | Clinical (unspecified phase) |
0.9 | High Similarity | NPD5377 | Approved |
0.9 | High Similarity | NPD5381 | Approved |
0.9 | High Similarity | NPD5378 | Approved |
0.8602 | High Similarity | NPD4282 | Approved |
0.8421 | Intermediate Similarity | NPD4835 | Approved |
0.8421 | Intermediate Similarity | NPD4837 | Approved |
0.8421 | Intermediate Similarity | NPD4838 | Approved |
0.8421 | Intermediate Similarity | NPD4836 | Approved |
0.8182 | Intermediate Similarity | NPD5376 | Approved |
0.7864 | Intermediate Similarity | NPD35 | Approved |
0.7864 | Intermediate Similarity | NPD4833 | Approved |
0.7624 | Intermediate Similarity | NPD1450 | Approved |
0.7624 | Intermediate Similarity | NPD1449 | Approved |
0.7349 | Intermediate Similarity | NPD9033 | Approved |
0.7349 | Intermediate Similarity | NPD9030 | Approved |
0.7349 | Intermediate Similarity | NPD9031 | Approved |
0.7349 | Intermediate Similarity | NPD9032 | Approved |
0.7315 | Intermediate Similarity | NPD3731 | Phase 3 |
0.729 | Intermediate Similarity | NPD2690 | Discontinued |
0.7212 | Intermediate Similarity | NPD2700 | Approved |
0.72 | Intermediate Similarity | NPD6428 | Approved |
0.7182 | Intermediate Similarity | NPD4832 | Approved |
0.7182 | Intermediate Similarity | NPD4831 | Approved |
0.7182 | Intermediate Similarity | NPD4830 | Approved |
0.7105 | Intermediate Similarity | NPD4826 | Approved |
0.7105 | Intermediate Similarity | NPD4828 | Approved |
0.7105 | Intermediate Similarity | NPD4827 | Approved |
0.7045 | Intermediate Similarity | NPD67 | Phase 2 |
0.7045 | Intermediate Similarity | NPD9034 | Approved |
0.6957 | Remote Similarity | NPD6436 | Phase 3 |
0.6792 | Remote Similarity | NPD8045 | Clinical (unspecified phase) |
0.6637 | Remote Similarity | NPD3204 | Clinical (unspecified phase) |
0.66 | Remote Similarity | NPD3716 | Discontinued |
0.6517 | Remote Similarity | NPD9445 | Approved |
0.6486 | Remote Similarity | NPD6941 | Approved |
0.6476 | Remote Similarity | NPD881 | Approved |
0.6239 | Remote Similarity | NPD7141 | Clinical (unspecified phase) |
0.6239 | Remote Similarity | NPD7140 | Approved |
0.6239 | Remote Similarity | NPD7139 | Approved |
0.6211 | Remote Similarity | NPD9435 | Approved |
0.6211 | Remote Similarity | NPD9434 | Approved |
0.614 | Remote Similarity | NPD8087 | Discontinued |
0.6095 | Remote Similarity | NPD1447 | Phase 3 |
0.6095 | Remote Similarity | NPD1446 | Phase 3 |
0.6078 | Remote Similarity | NPD4759 | Clinical (unspecified phase) |
0.5977 | Remote Similarity | NPD6123 | Approved |
0.5963 | Remote Similarity | NPD2255 | Approved |
0.595 | Remote Similarity | NPD8346 | Approved |
0.595 | Remote Similarity | NPD8347 | Approved |
0.595 | Remote Similarity | NPD8345 | Approved |
0.5904 | Remote Similarity | NPD895 | Approved |
0.5904 | Remote Similarity | NPD892 | Phase 3 |
0.5904 | Remote Similarity | NPD893 | Approved |
0.5904 | Remote Similarity | NPD887 | Approved |
0.5904 | Remote Similarity | NPD890 | Clinical (unspecified phase) |
0.5904 | Remote Similarity | NPD891 | Phase 3 |
0.5904 | Remote Similarity | NPD889 | Approved |
0.5904 | Remote Similarity | NPD894 | Approved |
0.5904 | Remote Similarity | NPD888 | Phase 3 |
0.5897 | Remote Similarity | NPD6430 | Approved |
0.5897 | Remote Similarity | NPD6429 | Approved |
0.5826 | Remote Similarity | NPD8174 | Phase 2 |
0.5783 | Remote Similarity | NPD2269 | Approved |
0.5778 | Remote Similarity | NPD1457 | Discontinued |
0.5773 | Remote Similarity | NPD372 | Clinical (unspecified phase) |
0.576 | Remote Similarity | NPD591 | Approved |
0.576 | Remote Similarity | NPD577 | Phase 3 |
0.5739 | Remote Similarity | NPD8307 | Discontinued |
0.5728 | Remote Similarity | NPD394 | Phase 3 |
0.5663 | Remote Similarity | NPD905 | Approved |
0.5663 | Remote Similarity | NPD904 | Phase 3 |
0.5631 | Remote Similarity | NPD361 | Discontinued |
0.5625 | Remote Similarity | NPD389 | Phase 3 |
0.5603 | Remote Similarity | NPD8140 | Approved |
Bioactivity similarity was calculated based on bioactivity descriptors of compounds. The bioactivity descriptors were calculated by a recently developed AI algorithm Chemical Checker (CC) [Nature Biotechnology, 38:1087–1096, 2020; Nature Communications, 12:3932, 2021], which evaluated bioactivity similarities at five levels:
☉ A: chemistry similarity;
☉ B: biological targets similarity;
☉ C: networks similarity;
☉ D: cell-based bioactivity similarity;
☉ E: similarity based on clinical data.
Those 5 categories of CC bioactivity descriptors were calculated and then subjected to manifold projection using UMAP algorithm, to project all NPs on a 2-Dimensional space. The current NP was highlighted with a small circle in the 2-D map. Below figures: left-to-right, A-to-E.