Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT2246 |
Cell Line |
T-cells |
|
IC50 |
= |
3820.0 |
nM |
PMID[509245] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8540.0 |
nM |
PMID[509262] |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
8030.0 |
nM |
PMID[509262] |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
7240.0 |
nM |
PMID[509262] |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
9100.0 |
nM |
PMID[509262] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
9660.0 |
nM |
PMID[509262] |
NPT859 |
Cell Line |
HFF |
Homo sapiens |
TD50 |
>= |
320.0 |
uM |
PMID[509263] |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
562.3 |
nM |
PMID[509268] |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
n.a. |
3219.7 |
nM |
PMID[509268] |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
n.a. |
33498.3 |
nM |
PMID[509268] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
> |
100000.0 |
nM |
PMID[509278] |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
IC50 |
> |
133000.0 |
nM |
PMID[509290] |
NPT1249 |
Individual Protein |
Canalicular multispecific organic anion transporter 2 |
Homo sapiens |
IC50 |
> |
133000.0 |
nM |
PMID[509290] |
NPT1028 |
Individual Protein |
Multidrug resistance-associated protein 4 |
Homo sapiens |
IC50 |
> |
133000.0 |
nM |
PMID[509290] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
50.0 |
% |
PMID[509294] |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
> |
100000.0 |
nM |
PMID[509300] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4.55 |
nM |
PMID[509231] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.42 |
nM |
PMID[509231] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
6.02 |
mg.kg-1 |
PMID[509231] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.0003008 |
ug.mL-1 |
PMID[509232] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.0008689 |
ug.mL-1 |
PMID[509232] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.34 |
nM |
PMID[509233] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1.92 |
nM |
PMID[509233] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4.49 |
nM |
PMID[509233] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2.34 |
nM |
PMID[509233] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
5.4 |
nM |
PMID[509234] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
351.0 |
nM |
PMID[509235] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
5.4 |
nM |
PMID[509236] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
3.36 |
n.a. |
PMID[509236] |
NPT27 |
Others |
Unspecified |
|
T1/2 |
< |
2.0 |
hr |
PMID[509236] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6.5 |
nM |
PMID[509237] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
9.2 |
nM |
PMID[509237] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
7.94 |
nM |
PMID[509237] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
6.02 |
mg.kg-1 |
PMID[509237] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
0.5 |
mg kg-1 5day-1 |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
1.1 |
mg kg-1 5day-1 |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
3.1 |
mg kg-1 5day-1 |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
5.0 |
mg kg-1 5day-1 |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
No. of mice survived |
= |
10.0 |
n.a. |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
No. of mice survived |
= |
4.0 |
n.a. |
PMID[509238] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
3.15 |
mg.kg-1 |
PMID[509239] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
0.3 |
mg.kg-1 |
PMID[509240] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
0.5 |
mg kg-1 |
PMID[509240] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.5 |
nM |
PMID[509241] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Parasitemia |
= |
0.0 |
% |
PMID[509241] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Parasitemia |
= |
32.0 |
% |
PMID[509241] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
5.0 |
% |
PMID[509241] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
3.36 |
n.a. |
PMID[509241] |
NPT27 |
Others |
Unspecified |
|
Solubility |
= |
4700.0 |
ug.mL-1 |
PMID[509241] |
NPT35 |
Others |
n.a. |
|
Solubility |
= |
256.0 |
ug.mL-1 |
PMID[509241] |
NPT35 |
Others |
n.a. |
|
Solubility |
= |
63.4 |
ug.mL-1 |
PMID[509241] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
T1/2 |
= |
52.2 |
n.a. |
PMID[509241] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
114.1 |
ml min-1 kg-1 |
PMID[509241] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
8.4 |
l kg-1 |
PMID[509241] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
F |
= |
1.4 |
% |
PMID[509241] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
25.0 |
nM |
PMID[509242] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
14.0 |
nM |
PMID[509243] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
0.00074 |
ug.mL-1 |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
9.1 |
day |
PMID[509244] |
NPT27 |
Others |
Unspecified |
|
T1/2 |
= |
0.8667 |
hr |
PMID[509244] |
NPT27 |
Others |
Unspecified |
|
Vd |
= |
8.0 |
L.kg-1 |
PMID[509244] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
114.0 |
mL.min-1.kg-1 |
PMID[509244] |
NPT27 |
Others |
Unspecified |
|
F |
= |
1.4 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
2.0 |
(mg/kg)/day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
4.3 |
(mg/kg)/day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
2.7 |
(mg/kg)/day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
6.2 |
(mg/kg)/day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
3.1 |
(mg/kg)/day |
PMID[509244] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
0.0012 |
ug.mL-1 |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED90 |
= |
5.0 |
1/mg.1/kg.1/day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Reduction |
= |
99.95 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Reduction |
> |
99.99 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Reduction |
= |
14.7 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Reduction |
= |
98.0 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Reduction |
= |
99.78 |
% |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
79.0 |
day |
PMID[509244] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
CC50 |
= |
89600.0 |
nM |
PMID[509245] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1780.0 |
nM |
PMID[509245] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Selectivity index |
= |
23.0 |
n.a. |
PMID[509245] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Selectivity index |
= |
48.0 |
n.a. |
PMID[509245] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.00074 |
ug.mL-1 |
PMID[509246] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.0012 |
ug.mL-1 |
PMID[509246] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
98.0 |
% |
PMID[509246] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
99.78 |
% |
PMID[509246] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
7.9 |
day |
PMID[509246] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
9.1 |
day |
PMID[509246] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
3.3 |
n.a. |
PMID[509246] |
NPT2248 |
Organism |
Plasmodium vinckei petteri |
Plasmodium vinckei petteri |
ED50 |
= |
0.3 |
mg/kg/day |
PMID[509247] |
NPT2248 |
Organism |
Plasmodium vinckei petteri |
Plasmodium vinckei petteri |
ED90 |
= |
0.7 |
mg/kg/day |
PMID[509247] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.2 |
nM |
PMID[509248] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2.8 |
nM |
PMID[509249] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.2 |
nM |
PMID[509251] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
14300.0 |
nM |
PMID[509252] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC80 |
> |
125.0 |
uM |
PMID[509252] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1.26 |
nM |
PMID[509253] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.53 |
nM |
PMID[509254] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.45 |
nM |
PMID[509255] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
1.26 |
nM |
PMID[509255] |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
IC50 |
= |
0.6 |
ug.mL-1 |
PMID[509256] |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
25.0 |
ug.mL-1 |
PMID[509256] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
11.0 |
day |
PMID[509257] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
9.8 |
day |
PMID[509257] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
12.4 |
day |
PMID[509257] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
99.4 |
% |
PMID[509257] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
98.7 |
% |
PMID[509257] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
99.8 |
% |
PMID[509257] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
14300.0 |
nM |
PMID[509259] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC80 |
> |
125.0 |
uM |
PMID[509259] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
26.7 |
% |
PMID[509259] |
NPT610 |
Others |
Molecular identity unknown |
|
Activity |
= |
63.0 |
% |
PMID[509259] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.53 |
nM |
PMID[509260] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2.11 |
nM |
PMID[509260] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
3.4 |
nM |
PMID[509261] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4.2 |
nM |
PMID[509261] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
Ratio IC50 |
= |
2.41 |
n.a. |
PMID[509261] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Inhibition |
= |
100.0 |
% |
PMID[509261] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
ED50 |
= |
5.88 |
mg.kg-1 |
PMID[509261] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
ED90 |
= |
10.57 |
mg/kg |
PMID[509261] |
NPT486 |
Organism |
Toxoplasma gondii |
Toxoplasma gondii |
IC50 |
= |
310.0 |
nM |
PMID[509263] |
NPT27 |
Others |
Unspecified |
|
TI |
= |
1814.0 |
n.a. |
PMID[509263] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Cmax |
= |
0.034 |
ug.mL-1 |
PMID[509264] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
AUC |
= |
168.0 |
ng.hr.mL-1 |
PMID[509264] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
T1/2 |
= |
3.9 |
hr |
PMID[509264] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Cmax |
= |
0.119 |
ug.mL-1 |
PMID[509264] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
AUC |
= |
382.0 |
ng.hr.mL-1 |
PMID[509264] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
T1/2 |
= |
1.9 |
hr |
PMID[509264] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1000000.0 |
nM |
PMID[509265] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Inhibition |
> |
90.0 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
81.0 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
97.0 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
99.0 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
6.2 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
6.9 |
day |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
> |
7.6 |
day |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
99.7 |
% |
PMID[509266] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Survival |
= |
13.2 |
day |
PMID[509266] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
24.0 |
% |
PMID[509267] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
2.5 |
nM |
PMID[509267] |
NPT2 |
Others |
Unspecified |
|
deltaA |
= |
0.18 |
n.a. |
PMID[509267] |
NPT27 |
Others |
Unspecified |
|
Activity |
= |
0.007 |
/hr |
PMID[509270] |
NPT27 |
Others |
Unspecified |
|
Activity |
= |
0.002 |
/hr |
PMID[509270] |
NPT35 |
Others |
n.a. |
|
Activity |
= |
0.002 |
/hr |
PMID[509270] |
NPT2254 |
Organism |
Schistosoma mansoni |
Schistosoma mansoni |
Activity |
= |
100.0 |
% |
PMID[509271] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
n.a. |
4.8 |
nM |
PMID[509268] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
70.8 |
nM |
PMID[509268] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
63.1 |
nM |
PMID[509268] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
ED50 |
= |
3.1 |
mg.kg-1 |
PMID[509274] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
ED90 |
= |
5.8 |
mg kg-1 |
PMID[509274] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.0004 |
ug.mL-1 |
PMID[509275] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
> |
99.9 |
% |
PMID[509276] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
MST |
= |
19.0 |
day |
PMID[509276] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
MST |
= |
38.5 |
day |
PMID[509276] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
MST |
= |
40.0 |
day |
PMID[509276] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
T1/2 |
= |
1.0 |
hr |
PMID[509277] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
30000.0 |
nM |
PMID[509278] |
NPT3148 |
Organism |
Cytomegalovirus |
Cytomegalovirus |
EC50 |
= |
5300.0 |
nM |
PMID[509278] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Inhibition |
= |
50.0 |
% |
PMID[509279] |
NPT475 |
Organism |
Plasmodium yoelii |
Plasmodium yoelii |
IC50 |
< |
1000.0 |
nM |
PMID[509279] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (moderate) |
= |
1.0 |
n.a. |
PMID[509280] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (moderate) |
= |
17.0 |
% |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (acute) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (acute) |
= |
0.0 |
% |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (cytolytic) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (choleostasis) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (severe hepatitis) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (chronic liver disease) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (cirrhosis) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (granulomatous hepatitis) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (association with vascular disease) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (steatosis) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (malignant tumour) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (benign tumour) |
= |
0.0 |
n.a. |
PMID[509280] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
F |
= |
1.4 |
% |
PMID[509281] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
4.0 |
n.a. |
PMID[509281] |
NPT475 |
Organism |
Plasmodium yoelii |
Plasmodium yoelii |
ED50 |
= |
6.0 |
mg.kg-1 |
PMID[509281] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Survival |
= |
20.8 |
day |
PMID[509282] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
> |
99.9 |
% |
PMID[509282] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
> |
64000.0 |
nM |
PMID[509283] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
IC50 |
= |
3.0 |
nM |
PMID[509284] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
27.5 |
% |
PMID[509284] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
33.3 |
% |
PMID[509284] |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
Activity |
= |
48.0 |
% |
PMID[509284] |
NPT2258 |
Organism |
Plasmodium falciparum NF54 |
Plasmodium falciparum NF54 |
IC50 |
= |
5.77 |
nM |
PMID[509286] |
NPT485 |
Organism |
Plasmodium falciparum (isolate K1 / Thailand) |
Plasmodium falciparum K1 |
IC50 |
= |
7.26 |
nM |
PMID[509286] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4.5 |
nM |
PMID[509286] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.3 |
n.a. |
PMID[509286] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.8 |
n.a. |
PMID[509286] |
NPT35 |
Others |
n.a. |
|
Tm |
= |
186.0 |
degrees C |
PMID[509287] |
NPT35 |
Others |
n.a. |
|
T |
= |
131.8 |
degrees C |
PMID[509287] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.8 |
nM |
PMID[509287] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.3 |
nM |
PMID[509287] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.6 |
n.a. |
PMID[509287] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
100000.0 |
nM |
PMID[509287] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
26316.0 |
n.a. |
PMID[509287] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
59.5 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
41000.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
393.83 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
87.83 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
163.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
28170000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
100.83 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
733.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
398.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
2.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1526.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
501.5 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
9.5 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
107.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
6.44 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
143.4 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
1.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
59200.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
16.8 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BASO |
= |
0.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
138.5 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
13978.67 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
391.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1608.5 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BASOLE |
= |
0.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
1.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5800000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
36.22 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
136500.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
16120.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
86.67 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
23.58 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
377200.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
62.52 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
2.5 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
9.83 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
= |
0.0 |
/100WBC |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1214170.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
54.83 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
42800.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
363.17 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
96.83 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
156.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
26170000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
102.67 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
636.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
594.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1823.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
656.5 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
9.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
117.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.92 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
142.62 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
1.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
58500.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
18.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
183.33 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
14952.83 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
238.5 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1642.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5890000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
36.13 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
133700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
17020.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
87.17 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
22.73 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
370200.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
61.45 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
1.5 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
10.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1183500.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
66.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
41700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
405.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
88.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
25670000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
103.0 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
703.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
249.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
2.1 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1553.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
155.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
116.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
6.23 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
145.23 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
2.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
58000.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
14.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
0.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
14690.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
490.33 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1319.67 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
0.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5700000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
36.23 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
136300.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
16500.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
88.67 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
23.93 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
376700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
63.6 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
3.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
8.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1120000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
52.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
43700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
430.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
101.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
176.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
23330000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
105.67 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
586.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
552.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
1.6 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1600.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
887.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
8.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
117.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
6.02 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
144.53 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
59300.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
18.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
153.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
12396.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
197.67 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1920.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5880000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
36.63 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
134700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
14670.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
84.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
22.93 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
368000.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
62.33 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
1.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
13.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1198670.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
46.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
41300.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
349.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
77.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
160.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
27000000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
103.33 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
666.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
259.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
2.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1446.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
331.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
100.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
6.54 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
142.23 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
56300.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
11.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
390.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
14550.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
453.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1407.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
2.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5210000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
33.1 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
126000.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
16800.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
24.23 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
380700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
63.67 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
2.67 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1173000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
55.33 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
43000.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
329.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
100.0 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
25000000.0 |
nM |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
516.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
790.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1716.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
649.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
9.67 |
U.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
123.7 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.73 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
143.53 |
mEq.L-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
17.3 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
257.33 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
17040.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
413.67 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
1822.33 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
1.33 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
6130000.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
135700.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
19530.0 |
cells.uL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
87.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
22.17 |
pg |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
370300.0 |
ug.mL-1 |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
59.77 |
fL |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
2.0 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
9.67 |
% |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
= |
0.33 |
/100WBC |
PMID[509288] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1300330.0 |
cells.uL-1 |
PMID[509288] |
NPT1173 |
Organism |
Candida albicans SC5314 |
Candida albicans SC5314 |
FICI |
= |
0.112 |
n.a. |
PMID[509289] |
NPT713 |
Individual Protein |
Bile salt export pump |
Homo sapiens |
IC50 |
> |
133000.0 |
nM |
PMID[509290] |
NPT475 |
Organism |
Plasmodium yoelii |
Plasmodium yoelii |
Activity |
= |
0.0 |
% |
PMID[509291] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
20.0 |
nM |
PMID[509292] |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
64000.0 |
nM |
PMID[509292] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
8.42 |
% |
PMID[509293] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.55 |
% |
PMID[509294] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
3.43 |
% |
PMID[509295] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
23.59 |
% |
PMID[509296] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
-0.09 |
% |
PMID[509297] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
0.34 |
% |
PMID[509298] |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Inhibition |
= |
19.11 |
% |
PMID[509299] |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
Inhibition |
= |
6.04 |
% |
PMID[509299] |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
Inhibition |
= |
13.66 |
% |
PMID[509299] |
NPT173 |
Organism |
Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
= |
9.17 |
% |
PMID[509299] |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
= |
12.03 |
% |
PMID[509299] |
NPT747 |
Organism |
Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
= |
30.63 |
% |
PMID[509299] |
NPT2922 |
Organism |
Staphylococcus aureus subsp. aureus |
Staphylococcus aureus subsp. aureus |
Inhibition |
= |
8.78 |
% |
PMID[509299] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.8 |
nM |
PMID[509300] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2.3 |
nM |
PMID[509300] |
NPT633 |
Organism |
Leishmania donovani |
Leishmania donovani |
IC50 |
= |
42290.0 |
nM |
PMID[509300] |
NPT633 |
Organism |
Leishmania donovani |
Leishmania donovani |
IC50 |
= |
90930.0 |
nM |
PMID[509300] |
NPT841 |
Organism |
Leishmania major |
Leishmania major |
IC50 |
= |
22540.0 |
nM |
PMID[509300] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.0 |
n.a. |
PMID[509300] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.0 |
n.a. |
PMID[509300] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
4.0 |
n.a. |
PMID[509300] |