Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Inhibition |
= |
70 |
% |
PubChem BioAssay data set |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Inhibition |
= |
94 |
% |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
15776.11 |
nM |
PubChem BioAssay data set |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
67095.43 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
91 |
% |
PubChem BioAssay data set |
NPT2046 |
Cell Line |
EVSA-T |
Homo sapiens |
IC50 |
= |
152104.99 |
nM |
PubChem BioAssay data set |
NPT1708 |
Individual Protein |
Serine/threonine-protein kinase 16 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1945 |
Cell Line |
CHP-126 |
Homo sapiens |
IC50 |
= |
1177183.5 |
nM |
12828470 |
NPT321 |
Protein Family |
cAMP-dependent protein kinase (PKA) |
Homo sapiens |
IC50 |
> |
1000000 |
nM |
15270579 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
13789.44 |
nM |
24411199 |
NPT2172 |
Cell Line |
SIMA |
Homo sapiens |
IC50 |
= |
3053925.22 |
nM |
25913865 |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
46011.53 |
nM |
24128145 |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
98232.98 |
nM |
23691978 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
9677274 |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757718 |
NPT1560 |
Protein Complex |
Cyclin-dependent kinase 4/cyclin D1 |
Homo sapiens |
IC50 |
= |
14210 |
nM |
10924160 |
NPT3356 |
Individual Protein |
Tyrosine-protein kinase receptor Tie-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10924160 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
IC50 |
= |
118844.75 |
nM |
PubChem BioAssay data set |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Activity |
= |
100 |
% |
25437304 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
361473.6 |
nM |
22934600 |
NPT1673 |
Individual Protein |
CaM kinase I gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23547843 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
42000 |
nM |
PubChem BioAssay data set |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1810 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
PubChem BioAssay data set |
NPT2085 |
Cell Line |
Kasumi 1 |
|
IC50 |
= |
3862743.65 |
nM |
PubChem BioAssay data set |
NPT3352 |
Individual Protein |
Dual specificity testis-specific protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
7264681 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
TGI |
> |
100000 |
nM |
16378367 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
> |
100000 |
nM |
25737008 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
TGI |
> |
100000 |
nM |
25737008 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
TGI |
> |
100000 |
nM |
25737008 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
> |
100000 |
nM |
25737008 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
TGI |
> |
100000 |
nM |
20804165 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23891163 |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
16824.65 |
nM |
9873651 |
NPT3932 |
Individual Protein |
Dual specificity protein kinase CLK1 |
Mus musculus |
IC50 |
= |
4300 |
nM |
12880316 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
21705225 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
19459643 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
23057874 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3981.07 |
nM |
11170665 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
GI50 |
= |
3250 |
nM |
16289636 |
NPT2087 |
Cell Line |
L-540 |
Homo sapiens |
IC50 |
= |
155761.97 |
nM |
20420415 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
19815.27 |
nM |
23215246 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23215246 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
21677.04 |
nM |
23215246 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
9457.85 |
nM |
PubChem BioAssay data set |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Kd |
> |
10000 |
nM |
20718449 |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17844993 |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19700322 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12220 |
nM |
25798528 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
15470 |
nM |
25798528 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
11630 |
nM |
25798528 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
25798528 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
53826.98 |
nM |
20594848 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
12699389 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
12699389 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
10.1016/0960-894X(95)00424-R |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
10.1016/0960-894X(95)00424-R |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
19900 |
nM |
10.1016/0960-894X(95)00424-R |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
19900 |
nM |
10.1016/0960-894X(95)00424-R |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
IC50 |
= |
6900 |
nM |
12542359 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
22400 |
nM |
DrugMatrix in vitro pharmacology data |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LC50 |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
LC50 |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
TGI |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
TGI |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
TGI |
= |
79432.82 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3338 |
Individual Protein |
Myosin IIIA |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
7560060 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
DrugMatrix in vivo data: Pathology |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
5010 |
nM |
23131412 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
24920381 |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
1831458.64 |
nM |
25728027 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000 |
nM |
18341287 |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18973387 |
NPT3322 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18547115 |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
16441076 |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Kd |
> |
10000 |
nM |
10579872 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
19150 |
|
22280481 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26026364 |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
772001.89 |
nM |
18817444 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
92.6 |
% |
20058933 |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25934225 |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
12617583 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
25118.86 |
nM |
16989519 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
16989519 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
31622.78 |
nM |
11374975 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
12193038 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
IC50 |
= |
650 |
nM |
15104506 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3981.1 |
nM |
7760068 |
NPT3369 |
Individual Protein |
Interferon-induced, double-stranded RNA-activated protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
1517739 |
NPT3340 |
Individual Protein |
Serine/threonine-protein kinase Nek1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25667960 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21131198 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
569912.59 |
nM |
24411199 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Kd |
= |
260 |
nM |
15104484 |
NPT3328 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 11 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8558523 |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
15000 |
nM |
PubChem BioAssay data set |
NPT1560 |
Protein Complex |
Cyclin-dependent kinase 4/cyclin D1 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
PubChem BioAssay data set |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
950 |
nM |
PubChem BioAssay data set |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
25900 |
nM |
PubChem BioAssay data set |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18461966 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
170 |
nM |
22292922 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11277744 |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
65621.74 |
nM |
22209731 |
NPT2094 |
Cell Line |
SKM-1 |
Homo sapiens |
IC50 |
= |
917722.45 |
nM |
19105653 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
50933.09 |
nM |
16441083 |
NPT3281 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Inhibition |
= |
41 |
% |
PubChem BioAssay data set |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Inhibition |
= |
26 |
% |
PubChem BioAssay data set |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
Inhibition |
= |
57 |
% |
PubChem BioAssay data set |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Inhibition |
= |
10 |
% |
PubChem BioAssay data set |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22472691 |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
113128.24 |
nM |
24479418 |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
= |
50118.7 |
nM |
20022253 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
19319.68 |
nM |
PubChem BioAssay data set |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18298075 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20000 |
nM |
23347584 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
8800 |
nM |
18396905 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Activity |
= |
71 |
% |
17559265 |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
228842.04 |
nM |
24273638 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
1080 |
nM |
26052978 |
NPT3109 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25066952 |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17696332 |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
657700.07 |
nM |
PubChem BioAssay data set |
NPT1981 |
Cell Line |
NCI-H1882 |
Homo sapiens |
IC50 |
= |
40599.79 |
nM |
18077363 |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Kd |
= |
1200 |
nM |
17850214 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1560 |
Protein Complex |
Cyclin-dependent kinase 4/cyclin D1 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
PubChem BioAssay data set |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
1559987.36 |
nM |
PubChem BioAssay data set |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
24154.61 |
nM |
23398362 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
363635.14 |
nM |
23398362 |
NPT1927 |
Cell Line |
ARH-77 |
Homo sapiens |
IC50 |
= |
96021.87 |
nM |
23398362 |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
9974.95 |
nM |
23398362 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
86238.96 |
nM |
PubChem BioAssay data set |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
8912.5 |
nM |
23634759 |
NPT3249 |
Individual Protein |
Tyrosine- and threonine-specific cdc2-inhibitory kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
9083483 |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
IC50 |
= |
800 |
nM |
PubChem BioAssay data set |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
IC50 |
= |
230 |
nM |
PubChem BioAssay data set |
NPT2213 |
Individual Protein |
Cyclin-dependent kinase 4 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
PubChem BioAssay data set |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
101747.68 |
nM |
PubChem BioAssay data set |
NPT2143 |
Cell Line |
ST486 |
Homo sapiens |
IC50 |
= |
10350.98 |
nM |
24725159 |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Kd |
> |
10000 |
nM |
26090896 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Kd |
> |
10000 |
nM |
22642560 |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
197264.41 |
nM |
22587572 |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
245147.48 |
nM |
22545792 |
NPT3233 |
Individual Protein |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
Kd |
> |
10000 |
nM |
25176187 |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
238629.47 |
nM |
24095094 |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Kd |
= |
4500 |
nM |
24095094 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
57569.45 |
nM |
23303337 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
TGI |
> |
100000 |
nM |
24893224 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24893224 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
24893224 |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24893224 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Activity |
= |
89 |
% |
24893224 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
LC50 |
= |
100000 |
nM |
24370114 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
24370114 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
LC50 |
= |
100000 |
nM |
24370114 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
100000 |
nM |
24370114 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
24370114 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
25871261 |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
187061.23 |
nM |
12398531 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
17500 |
nM |
20000781 |
NPT1948 |
Cell Line |
A253 cell line |
|
IC50 |
= |
271299.4 |
nM |
17378609 |
NPT2146 |
Cell Line |
YT |
Homo sapiens |
IC50 |
= |
536409.57 |
nM |
11325232 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
57.1 |
% |
20801038 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Activity |
= |
89 |
% |
12502331 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
IC50 |
= |
3000 |
nM |
12502331 |
NPT3323 |
Individual Protein |
Cell division cycle 2-like protein kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11754602 |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
215862.58 |
nM |
15387665 |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8984155 |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
91329.79 |
nM |
7908950 |
NPT3918 |
Individual Protein |
Synapsin-1 |
Bos taurus |
IC50 |
= |
1000 |
nM |
20061160 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
1069 |
nM |
19729316 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
TGI |
= |
39800 |
nM |
19729316 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
39800 |
nM |
19674905 |
NPT1986 |
Cell Line |
RPMI 8402 |
Homo sapiens |
IC50 |
= |
13626.18 |
nM |
11277769 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
105590.46 |
nM |
7964780 |
NPT2030 |
Cell Line |
U-698-M |
Homo sapiens |
IC50 |
= |
1257210.93 |
nM |
16499337 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
87 |
% |
18610999 |
NPT2041 |
Cell Line |
P31-FUJ |
Homo sapiens |
IC50 |
= |
3063548 |
nM |
18610999 |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
18320.78 |
nM |
10869203 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Inhibition |
= |
87 |
% |
21419633 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
7800 |
nM |
25647077 |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
2690 |
nM |
19919060 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3980 |
nM |
23268606 |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15267244 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
126376.05 |
nM |
21043460 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
0.6 |
nM |
10395496 |
NPT2213 |
Individual Protein |
Cyclin-dependent kinase 4 |
Homo sapiens |
IC50 |
= |
100 |
nM |
10395496 |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
102847.78 |
nM |
24144848 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
7000 |
nM |
21028898 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
1041.8 |
nM |
20961068 |
NPT3342 |
Individual Protein |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16872140 |
NPT2064 |
Cell Line |
UACC-812 |
Homo sapiens |
IC50 |
= |
711871.91 |
nM |
20499851 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
TGI |
= |
50118.72 |
nM |
22545792 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
22545792 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
22545792 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
TGI |
= |
50118.72 |
nM |
20000780 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
TGI |
= |
50118.72 |
nM |
20028081 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
TGI |
= |
50118.72 |
nM |
20028081 |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
392068.67 |
nM |
15974618 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
10715.19 |
nM |
19739599 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
6151085 |
|
10464018 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
6863365 |
|
11412985 |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Activity |
= |
87 |
% |
18001087 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
12500 |
nM |
17970595 |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
18053715 |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
29958.23 |
nM |
16933872 |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
68047.3 |
nM |
12762807 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Activity |
= |
99 |
% |
19674906 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
11324 |
nM |
19113968 |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
17417907 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
24079846 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Activity |
= |
88 |
% |
25981689 |
NPT1910 |
Cell Line |
ECC4 |
Homo sapiens |
IC50 |
= |
381103.5 |
nM |
11975486 |
NPT1572 |
Protein Family |
Glycogen synthase kinase-3 |
Homo sapiens |
IC50 |
= |
60000 |
nM |
21612217 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
230 |
nM |
21807523 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
16300 |
nM |
23869482 |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
115394.77 |
nM |
19555121 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
11858761 |
NPT3306 |
Individual Protein |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
15006398 |
NPT2009 |
Cell Line |
NCI-H2081 |
Homo sapiens |
IC50 |
= |
291494.17 |
nM |
2985785 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
8072.35 |
nM |
15863306 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
42002.75 |
nM |
16366608 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
18068979 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
18068979 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
11600 |
nM |
17438054 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Activity |
= |
95 |
% |
17438054 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7600 |
nM |
19285414 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
EC50 |
= |
151 |
nM |
16792425 |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Kd |
> |
10000 |
nM |
16441071 |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Kd |
= |
2300 |
nM |
19403314 |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
31139.75 |
nM |
18268091 |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
12861.34 |
nM |
18378710 |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
21093117 |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
87895.71 |
nM |
20566771 |
NPT2203 |
Cell Line |
GDM-1 |
Homo sapiens |
IC50 |
= |
117740.38 |
nM |
21397998 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Inhibition |
= |
10 |
% |
21429630 |
NPT3168 |
Individual Protein |
Casein kinase I alpha |
Homo sapiens |
Inhibition |
= |
1 |
% |
21429630 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Inhibition |
= |
25 |
% |
21429630 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Inhibition |
= |
13 |
% |
21429630 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Inhibition |
= |
85 |
% |
21641797 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
Inhibition |
= |
95 |
% |
21641799 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Inhibition |
= |
87 |
% |
21546135 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Inhibition |
= |
28 |
% |
21665469 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Inhibition |
= |
38 |
% |
21419633 |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
535327.66 |
nM |
21824772 |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
73389.58 |
nM |
21741732 |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
1593659.14 |
nM |
21855181 |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1974 |
Cell Line |
IST-SL2 |
Homo sapiens |
IC50 |
= |
24534.35 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
94354.13 |
nM |
22088956 |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Kd |
= |
1800 |
nM |
22440626 |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12065443 |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
167901.08 |
nM |
10.1007/s00044-013-0488-5 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
10.1007/s00044-012-0385-3 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
36327.57 |
nM |
23237840 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3162.3 |
nM |
23567963 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
160 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
67643.75 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
160 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
700 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3371 |
Individual Protein |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5623.4 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
81901.8 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
TGI |
> |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
17000 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
27914.44 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
36324.56 |
nM |
DrugMatrix in vivo data: Pathology |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
795144.61 |
nM |
24107081 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Kd |
> |
10000 |
nM |
24246731 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
82413.81 |
nM |
24463437 |
NPT1921 |
Cell Line |
COR-L279 |
Homo sapiens |
IC50 |
= |
12290.71 |
nM |
24448419 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
140 |
nM |
24878195 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Activity |
= |
80 |
% |
25129868 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Activity |
= |
92 |
% |
25218911 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
16380 |
nM |
25593095 |
NPT1929 |
Cell Line |
CPC-N |
Homo sapiens |
IC50 |
= |
307404.66 |
nM |
25740159 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Activity |
= |
92 |
% |
26254943 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
50104.81 |
nM |
26900657 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
31600 |
nM |
26948407 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
TGI |
= |
31600 |
nM |
26948407 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
TGI |
= |
31600 |
nM |
26948407 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
TGI |
= |
31600 |
nM |
26948407 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
31600 |
nM |
26948407 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
31600 |
nM |
26948407 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
31600 |
nM |
26948407 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
87 |
% |
27338658 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
24300 |
nM |
15161186 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
> |
100000 |
nM |
15857140 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
TGI |
> |
100000 |
nM |
15857140 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
TGI |
> |
100000 |
nM |
16884291 |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
253600.45 |
nM |
17107790 |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
574588.42 |
nM |
17477518 |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18370373 |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
55603.6 |
nM |
19093884 |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18954984 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
288118.25 |
nM |
20036560 |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
3731800.11 |
nM |
20055418 |
NPT1944 |
Cell Line |
D-247MG |
Homo sapiens |
IC50 |
= |
12351.58 |
nM |
16921367 |
NPT2110 |
Cell Line |
SCLC-21H |
Homo sapiens |
IC50 |
= |
325330.31 |
nM |
20637529 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Ki |
= |
790 |
nM |
19966789 |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
21200.8 |
nM |
19966789 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
187904.9 |
nM |
PubChem BioAssay data set |
NPT3265 |
Individual Protein |
Casein kinase I isoform alpha-like |
Homo sapiens |
Kd |
> |
10000 |
nM |
21080629 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
21135175 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
21712146 |
NPT1985 |
Cell Line |
OPM-2 |
Homo sapiens |
IC50 |
= |
37294.95 |
nM |
PubChem BioAssay data set |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
22435669 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
= |
3200 |
nM |
23252603 |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
23252603 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
4653.5 |
nM |
10.6019/CHEMBL1201861 |
NPT3120 |
Individual Protein |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
5.26 |
% |
10.6019/CHEMBL1201861 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
220 |
nM |
10.6019/CHEMBL1201861 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
480 |
nM |
10.6019/CHEMBL1201861 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.6019/CHEMBL1201861 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
19952.62 |
nM |
10.6019/CHEMBL1201861 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.6019/CHEMBL1201861 |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
1151643.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Activity |
= |
97 |
% |
23591111 |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23786452 |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
97742.94 |
nM |
24015327 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24015327 |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Activity |
= |
84 |
% |
24328302 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
PubChem BioAssay data set |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Inhibition |
= |
41 |
% |
24694055 |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
48620.15 |
nM |
25563890 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25462271 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
GI50 |
= |
13900 |
nM |
25176189 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
15500 |
nM |
25176189 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
22600 |
nM |
25176189 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
25200 |
nM |
25176189 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
32210.69 |
nM |
25238284 |
NPT2196 |
Cell Line |
NB1 |
Homo sapiens |
IC50 |
= |
12330.75 |
nM |
25218912 |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Kd |
> |
10000 |
nM |
25221651 |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
31013.48 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
54640 |
nM |
10.1039/C4MD00211C |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
55010 |
nM |
10.1039/C4MD00211C |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Inhibition |
= |
20 |
% |
10.1039/C4MD00211C |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
125195.19 |
nM |
Patent: US8871728 B2 |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.1039/C5MD00247H |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Kd |
> |
10000 |
nM |
26890114 |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
26890114 |
NPT1982 |
Cell Line |
NCI-H1963 |
Homo sapiens |
IC50 |
= |
56454.89 |
nM |
10.1039/C5MD00451A |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
69210.81 |
nM |
10654414 |
NPT2183 |
Cell Line |
NCI-H1694 |
Homo sapiens |
IC50 |
= |
119199.31 |
nM |
10654414 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
29376.5 |
nM |
26465675 |
NPT3335 |
Individual Protein |
Serine/threonine-protein kinase DCLK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.1016/S0040-4020(00)00994-7 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
IC50 |
= |
18000 |
nM |
16180824 |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
47044.83 |
nM |
20729083 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15000 |
nM |
12350160 |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
10000 |
nM |
12762820 |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
63409.27 |
nM |
8496706 |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
78078.44 |
nM |
16933872 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
39719.15 |
nM |
PubChem BioAssay data set |
NPT623 |
Cell Line |
NALM-6 |
Homo sapiens |
IC50 |
= |
77040.4 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
27925.44 |
nM |
PubChem BioAssay data set |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23354071 |
NPT3319 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22892213 |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
1512148.85 |
nM |
18314958 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20159656 |
NPT1983 |
Cell Line |
NCI-H64 |
Homo sapiens |
IC50 |
= |
33859.72 |
nM |
20159656 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20159656 |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
26684850 |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Activity |
= |
73 |
% |
18280170 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
22400 |
nM |
22409377 |
NPT2011 |
Cell Line |
NCI-H719 |
Homo sapiens |
IC50 |
= |
576484.82 |
nM |
7130986 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
5780.96 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
2880 |
nM |
25739048 |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25735399 |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
74627.49 |
nM |
12639558 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
158 |
nM |
22831798 |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26218649 |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19193024 |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
33493.62 |
nM |
19193024 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12398532 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
16933891 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25556102 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25556102 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Activity |
= |
90 |
% |
11520227 |
NPT3260 |
Individual Protein |
Phosphatidylinositol-5-phosphate 4-kinase type-2 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
16372404 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
93 |
% |
20701299 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Activity |
= |
94 |
% |
16933872 |
NPT3355 |
Individual Protein |
TGF-beta receptor type II |
Homo sapiens |
Kd |
> |
10000 |
nM |
541686 |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
9460.82 |
nM |
21377877 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Activity |
= |
89 |
% |
24992702 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
3700 |
nM |
12502331 |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Activity |
= |
75 |
% |
21381696 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
22545792 |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
3236014 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
15165148 |
NPT1923 |
Cell Line |
DMS-153 |
Homo sapiens |
IC50 |
= |
65496.58 |
nM |
15165148 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
15165148 |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Kd |
= |
3300 |
nM |
17266369 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45500 |
nM |
17266369 |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
134636.02 |
nM |
21726077 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
25118.86 |
nM |
23770448 |
NPT2013 |
Cell Line |
SK-MM-2 |
Homo sapiens |
IC50 |
= |
817603.91 |
nM |
PubChem BioAssay data set |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
4600 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
20000 |
nM |
PubChem BioAssay data set |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
17500572 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
LC50 |
= |
100000 |
nM |
17500572 |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22591513 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
160 |
nM |
22209731 |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
450 |
nM |
22209731 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19928832 |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
25437914 |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
21338.95 |
nM |
25556102 |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
501318.19 |
nM |
25556102 |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Activity |
= |
90 |
% |
11720542 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23282042 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23282042 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23282042 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23189988 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23189988 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
14510614 |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12088422 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
16330.52 |
nM |
12088422 |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Kd |
> |
10000 |
nM |
4020828 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10753475 |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12477351 |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
704500.47 |
nM |
7853002 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Kd |
= |
3400 |
nM |
18450456 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
21144756 |
NPT1189 |
Cell Line |
DG-75 |
Homo sapiens |
IC50 |
= |
42654.59 |
nM |
21356592 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
520 |
nM |
21774499 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
37011.99 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2047 |
Cell Line |
HC-1 |
Homo sapiens |
IC50 |
= |
64145.7 |
nM |
DrugMatrix in vitro pharmacology data |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
GI50 |
= |
5400 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2115 |
Cell Line |
HCC2157 |
Homo sapiens |
IC50 |
= |
194528.37 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21920638 |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
3603147.33 |
nM |
22850214 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
124538.39 |
nM |
14706813 |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.1007/s00044-011-9832-9 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45500 |
nM |
10.1007/s00044-012-0142-7 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Activity |
= |
83 |
% |
23547728 |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
2125913.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
10.6019/CHEMBL1201861 |
NPT4601 |
Cell Line |
EHEB |
Homo sapiens |
IC50 |
= |
79182.87 |
nM |
10.6019/CHEMBL1201861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12300 |
nM |
10.6019/CHEMBL1201861 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20480 |
nM |
10.6019/CHEMBL1201861 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
9620 |
nM |
10.6019/CHEMBL1201861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14140 |
nM |
10.6019/CHEMBL1201861 |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Kd |
> |
10000 |
nM |
23916255 |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
111724.94 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2200 |
Cell Line |
RPMI-6666 |
Homo sapiens |
IC50 |
= |
13912.09 |
nM |
DrugMatrix in vivo data: Pathology |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
24871162 |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26132075 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
26176165 |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
592673.7 |
nM |
24087924 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
FC |
= |
0.797 |
|
19606850 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
11641.26 |
nM |
11170658 |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
1903177.24 |
nM |
12747783 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
17561406 |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
157184.3 |
nM |
18522867 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.033 |
% |
21885167 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
6.98 |
% |
21885167 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.386 |
% |
21885167 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
30568 |
|
21999614 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
24350 |
|
22421020 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
3945095 |
|
22421020 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
3926015 |
|
22421020 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
3146605 |
|
22421020 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
8258813 |
|
24936232 |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
271582.51 |
nM |
10.1039/C0MD00022A |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
128960.48 |
nM |
26209834 |
NPT2193 |
Cell Line |
IM-9 |
Homo sapiens |
IC50 |
= |
4134790.74 |
nM |
26922225 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26789378 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
167435.8 |
nM |
14695799 |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Kd |
> |
10000 |
nM |
14695799 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Kd |
= |
2900 |
nM |
23434422 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
5010 |
nM |
2853205 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
5010 |
nM |
2853205 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
13645.83 |
nM |
16933872 |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
86404.61 |
nM |
9873511 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
25527.01 |
nM |
22705001 |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Kd |
> |
10000 |
nM |
21377877 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3000 |
nM |
12570374 |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Kd |
> |
10000 |
nM |
19530698 |
NPT3209 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24388833 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12250 |
nM |
15656657 |
NPT3168 |
Individual Protein |
Casein kinase I alpha |
Homo sapiens |
IC50 |
= |
4000 |
nM |
22642560 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45500 |
nM |
PubChem BioAssay data set |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
2627163.43 |
nM |
PubChem BioAssay data set |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT2198 |
Cell Line |
NCI-H524 |
Homo sapiens |
IC50 |
= |
61357.78 |
nM |
15165133 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Kd |
> |
10000 |
nM |
9548870 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
7528785 |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
486181.98 |
nM |
PubChem BioAssay data set |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Activity |
= |
97 |
% |
PubChem BioAssay data set |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Activity |
= |
83 |
% |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
1.5 |
|
15620238 |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
34942.19 |
nM |
18341287 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
18341287 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
19600 |
nM |
18341287 |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
999510.84 |
nM |
23501115 |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
28907.96 |
nM |
PubChem BioAssay data set |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19674905 |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
3271124.21 |
nM |
19674905 |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
> |
10000 |
nM |
12880316 |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
541947.97 |
nM |
23145909 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
2970349.79 |
nM |
20590100 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
540 |
nM |
18855442 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
16472241 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Inhibition |
= |
29 |
% |
PubChem BioAssay data set |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
940 |
nM |
PubChem BioAssay data set |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
1770 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
31622.78 |
nM |
15646539 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
TGI |
= |
31622.78 |
nM |
15646539 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
TGI |
= |
31622.78 |
nM |
15646539 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
25464882 |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
994666 |
nM |
24927053 |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
37185.65 |
nM |
25707014 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
31105.92 |
nM |
22834923 |
NPT3268 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22834923 |
NPT2105 |
Cell Line |
NCI-H1436 |
Homo sapiens |
IC50 |
= |
534165.12 |
nM |
23282083 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
IC50 |
> |
100000 |
nM |
23079524 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
23305920 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16872140 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Inhibition |
= |
63 |
% |
12036352 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
100000 |
nM |
24485783 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
100000 |
nM |
24485783 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
TGI |
= |
100000 |
nM |
24485783 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
100000 |
nM |
24582402 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
100000 |
nM |
24582402 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
TGI |
= |
100000 |
nM |
24582402 |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
185096.81 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
PubChem BioAssay data set |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
100 |
nM |
PubChem BioAssay data set |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
800 |
nM |
PubChem BioAssay data set |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
500 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
38.6 |
% |
12828470 |
NPT2033 |
Cell Line |
JIYOYE |
Homo sapiens |
IC50 |
= |
8502.64 |
nM |
PubChem BioAssay data set |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Activity |
= |
88 |
% |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
4897.79 |
nM |
PubChem BioAssay data set |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
4450 |
nM |
PubChem BioAssay data set |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
23354072 |
NPT3302 |
Individual Protein |
Ankyrin repeat and protein kinase domain-containing protein 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11325240 |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
283583.33 |
nM |
11325240 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Kd |
= |
1900 |
nM |
8254344 |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
71418 |
nM |
18198839 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23252848 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
TGI |
> |
100000 |
nM |
23316950 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
23316950 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23316950 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
TGI |
> |
100000 |
nM |
23316950 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23316950 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23316950 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23368966 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
> |
100000 |
nM |
23368966 |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25679337 |
NPT2142 |
Cell Line |
REH |
Homo sapiens |
IC50 |
= |
1288588.87 |
nM |
11063609 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Activity |
= |
79 |
% |
18616221 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18616221 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
39800 |
nM |
26836364 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16724849 |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25629304 |
NPT1908 |
Cell Line |
EC-GI-10 |
Homo sapiens |
IC50 |
= |
3488600.74 |
nM |
8699187 |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
163948.44 |
nM |
16441065 |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Kd |
= |
700 |
nM |
15332848 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
27986.86 |
nM |
16872140 |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Activity |
= |
85 |
% |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
TGI |
> |
100000 |
nM |
18179176 |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
231382.23 |
nM |
23395661 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
500 |
nM |
18396905 |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19919060 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
46.75 |
% |
18771321 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
40.69 |
% |
18771321 |
NPT3368 |
Individual Protein |
cGMP-dependent protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25136754 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
TGI |
= |
100000 |
nM |
15332839 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
IC50 |
= |
33890.81 |
nM |
14695798 |
NPT3460 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 3 |
Homo sapiens |
Activity |
= |
97 |
% |
20961068 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45500 |
nM |
23454511 |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
21067210 |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Kd |
> |
10000 |
nM |
21067210 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
10096858 |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
237377.57 |
nM |
9358635 |
NPT1968 |
Cell Line |
OMC-1 |
Homo sapiens |
IC50 |
= |
1803656.01 |
nM |
19572738 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
25338277 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
24712.2 |
nM |
25338277 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
15800 |
nM |
25419616 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
15800 |
nM |
25419616 |
NPT2145 |
Cell Line |
TE-15 |
Homo sapiens |
IC50 |
= |
878570.36 |
nM |
23806110 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
IC50 |
> |
100000 |
nM |
11000039 |
NPT3278 |
Individual Protein |
LIM domain kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15974607 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
23964644 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
76 |
% |
4031900 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26483136 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Ki |
= |
250 |
nM |
20363142 |
NPT3300 |
Individual Protein |
Serine/threonine-protein kinase 32B |
Homo sapiens |
Kd |
> |
10000 |
nM |
11473423 |
NPT2171 |
Cell Line |
SIG-M5 |
Homo sapiens |
IC50 |
= |
31683.34 |
nM |
18419154 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
3237831.19 |
nM |
22413887 |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26287401 |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
174048.85 |
nM |
26287401 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
24900 |
nM |
10820113 |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10820113 |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
560842.99 |
nM |
15104487 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
823093.66 |
nM |
24645629 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
12542361 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
19627125 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
19627125 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
10075797 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
10075797 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
9214739 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
9461655 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
7775983 |
NPT3250 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18303848 |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
1846263.23 |
nM |
12713401 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Activity |
= |
92 |
% |
23675610 |
NPT2129 |
Cell Line |
SNU-C1 |
Homo sapiens |
IC50 |
= |
521320.49 |
nM |
23675610 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
4 |
% |
9435889 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
13645.83 |
nM |
15050613 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
7.3 |
% |
10.1016/S0960-894X(01)80759-9 |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
99493.17 |
nM |
16039849 |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
15648.22 |
nM |
12747785 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Activity |
= |
106 |
% |
19716307 |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
48493.71 |
nM |
15332848 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
130531.16 |
nM |
18598080 |
NPT3815 |
Individual Protein |
Tyrosine-protein kinase LCK |
Mus musculus |
Activity |
= |
76 |
% |
PubChem BioAssay data set |
NPT3334 |
Individual Protein |
Citron Rho-interacting kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
17067151 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
7943.28 |
nM |
12193039 |
NPT2079 |
Cell Line |
EW-12 |
Homo sapiens |
IC50 |
= |
3183581.18 |
nM |
22704889 |
NPT2186 |
Cell Line |
RL |
Homo sapiens |
IC50 |
= |
3550039.47 |
nM |
16309322 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50000 |
nM |
22545792 |
NPT2147 |
Cell Line |
LB647-SCLC |
Homo sapiens |
IC50 |
= |
66308.76 |
nM |
10650093 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Inhibition |
= |
19 |
% |
10650082 |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
12398532 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19943620 |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20155971 |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
312627.38 |
nM |
20825224 |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
2516947.16 |
nM |
22801644 |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
255825.87 |
nM |
20627740 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6.56 |
% |
16643031 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
13.2 |
% |
16643031 |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
> |
10000 |
nM |
24547740 |
NPT3210 |
Individual Protein |
BMP-2-inducible protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
12662110 |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15711537 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
106625.21 |
nM |
18578517 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
31753.5 |
nM |
18183025 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
> |
100000 |
nM |
17850214 |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
158950.05 |
nM |
18183025 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
64120.96 |
nM |
18183025 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17850214 |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10998351 |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Kd |
= |
470 |
nM |
PubChem BioAssay data set |
NPT2054 |
Cell Line |
LU-165 |
Homo sapiens |
IC50 |
= |
514066.17 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
450 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
22024.8 |
nM |
23398362 |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
310350.41 |
nM |
23398362 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
2694 |
nM |
23398362 |
NPT3348 |
Individual Protein |
NUAK family SNF1-like kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
15800 |
nM |
23398362 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
15800 |
nM |
23398362 |
NPT2035 |
Cell Line |
NCCIT |
Homo sapiens |
IC50 |
= |
7554.82 |
nM |
23398362 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
707.95 |
nM |
PubChem BioAssay data set |
NPT1953 |
Cell Line |
D-336MG |
Homo sapiens |
IC50 |
= |
543555.6 |
nM |
18077363 |
NPT3258 |
Individual Protein |
Mixed lineage kinase 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15270558 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
19278239 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
18163584 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
11277747 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
11277747 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
7400820 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
7400820 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
12932143 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22429052 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
23395661 |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Activity |
= |
80 |
% |
24484201 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
6165.95 |
nM |
26042639 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
IC50 |
= |
5000 |
nM |
19159272 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
220 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
20493686 |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
54319.87 |
nM |
25466192 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
24168147 |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
1095906.33 |
nM |
14510607 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
73 |
% |
25237727 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
48900 |
nM |
25237727 |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25237727 |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
26808.23 |
nM |
23079524 |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
22220686 |
NPT2733 |
Individual Protein |
Protein kinase Pfmrk |
Plasmodium falciparum |
IC50 |
> |
1000000 |
nM |
24582402 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
33000 |
nM |
24582402 |
NPT3238 |
Individual Protein |
Dual specificity protein kinase TTK |
Homo sapiens |
Kd |
= |
2100 |
nM |
7807120 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
20000 |
nM |
14738378 |
NPT3360 |
Individual Protein |
Tubulin alpha-1 chain |
Rattus norvegicus |
Kd |
> |
10000 |
nM |
12182864 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12608854 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12608854 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12608854 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12608854 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12608854 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
18293907 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
19853459 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
19853459 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
19853459 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
19853459 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
19775092 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
19775092 |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
258377.84 |
nM |
12088422 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
19689125 |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
182814.32 |
nM |
PubChem BioAssay data set |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
787988.9 |
nM |
23701598 |
NPT3298 |
Individual Protein |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
Kd |
> |
10000 |
nM |
23755851 |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
17015.23 |
nM |
14584959 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
26259802 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
24387703 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
3210015 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
930 |
nM |
PubChem BioAssay data set |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
72108.79 |
nM |
20045651 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
20045651 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
8691203 |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
158401.98 |
nM |
8691203 |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
762104.74 |
nM |
8691203 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Activity |
= |
90 |
% |
8691203 |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Kd |
> |
10000 |
nM |
20634065 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
21053938 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
60 |
|
22652254 |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
335973.74 |
nM |
22652254 |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
= |
50118.7 |
nM |
12662101 |
NPT2075 |
Cell Line |
NCI-H2196 |
Homo sapiens |
IC50 |
= |
155583.88 |
nM |
23046382 |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Kd |
= |
2100 |
nM |
23046382 |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
85068.26 |
nM |
PubChem BioAssay data set |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23634786 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
9722490 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
50000 |
nM |
1336040 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Activity |
= |
97 |
% |
16562846 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
1602301 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
24328269 |
NPT2179 |
Cell Line |
LC-1F |
Homo sapiens |
IC50 |
= |
41570.47 |
nM |
13678412 |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
ID50 |
= |
0.65 |
nM |
25739048 |
NPT3289 |
Individual Protein |
Serine/threonine-protein kinase RIO3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25739048 |
NPT3362 |
Individual Protein |
Mitogen-activated protein kinase 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19904995 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
25856683 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Activity |
= |
85 |
% |
17618015 |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
719245.68 |
nM |
25136754 |
NPT3294 |
Individual Protein |
Activin receptor type-2A |
Homo sapiens |
Kd |
> |
10000 |
nM |
20570625 |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Kd |
= |
1100 |
nM |
1593279 |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
21060.03 |
nM |
11858752 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20800 |
nM |
23022281 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
14400 |
nM |
17609121 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
66314.86 |
nM |
9748371 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
22409377 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
25710081 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
26105195 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
IC50 |
= |
520 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
6300 |
nM |
20363129 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
6300 |
nM |
20363129 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
6300 |
nM |
21504848 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11100 |
nM |
8350092 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
40000 |
nM |
8350092 |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
7807122 |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757713 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
19906.73 |
nM |
15165148 |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
37671.17 |
nM |
12477351 |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
35086.06 |
nM |
20185316 |
NPT2104 |
Cell Line |
NCI-H1417 |
Homo sapiens |
IC50 |
= |
831094.08 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
24603.68 |
nM |
PubChem BioAssay data set |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
29011.29 |
nM |
DrugMatrix in vitro pharmacology data |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
17782.8 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Activity |
= |
83 |
% |
DrugMatrix in vitro pharmacology data |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Kd |
= |
990 |
nM |
PubChem BioAssay data set |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
26042639 |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
1116559.1 |
nM |
11929285 |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15217281 |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
2492757.98 |
nM |
9090867 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
207660.6 |
nM |
17567069 |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
10479316 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
GI50 |
= |
16300 |
nM |
17502410 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
17638695 |
NPT3311 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17923492 |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
262492.63 |
nM |
18056272 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
14400 |
nM |
18056275 |
NPT929 |
Cell Line |
BC1 cell line |
|
IC50 |
= |
19119.83 |
nM |
20439614 |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
26864.62 |
nM |
20439614 |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
39584.24 |
nM |
20439614 |
NPT2125 |
Cell Line |
NCI-H1522 |
Homo sapiens |
IC50 |
= |
124614.88 |
nM |
20439614 |
NPT3261 |
Individual Protein |
cAMP-dependent protein kinase beta-1 catalytic subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
19075048 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
20000 |
nM |
19114678 |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
19114678 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
IC50 |
= |
520 |
nM |
19114678 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
4600 |
nM |
19114678 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19114678 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17400 |
nM |
19307369 |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19273669 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
19738019 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
19738019 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6000 |
nM |
19738019 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
270 |
nM |
20547801 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
220 |
nM |
20547801 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5011.9 |
nM |
20014752 |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
2421 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Activity |
= |
74 |
% |
DrugMatrix in vitro pharmacology data |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1906 |
Cell Line |
EB-3 |
Homo sapiens |
IC50 |
= |
23183.11 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Activity |
= |
86 |
% |
22194678 |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
42667.14 |
nM |
27387357 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
10.1016/S0960-894X(97)00178-9 |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16539393 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
42756.29 |
nM |
17438052 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Activity |
= |
78 |
% |
17438047 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18524583 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
19307360 |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
23517.86 |
nM |
21145140 |
NPT2023 |
Cell Line |
NB7 |
Homo sapiens |
IC50 |
= |
489817.07 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1598 |
Individual Protein |
Casein kinase II alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
DrugMatrix in vitro pharmacology data |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT385 |
Cell Line |
SR |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
TGI |
= |
100000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
Potency |
|
35481.3 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Kd |
> |
10000 |
nM |
22533850 |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
143212.28 |
nM |
25847765 |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
259090.91 |
nM |
25946116 |
NPT2061 |
Cell Line |
NCI-H889 |
Homo sapiens |
IC50 |
= |
885930.05 |
nM |
15711537 |
NPT2076 |
Cell Line |
NCI-H2227 |
Homo sapiens |
IC50 |
= |
2388232.9 |
nM |
15711537 |
NPT3345 |
Individual Protein |
Cyclin-dependent kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16698266 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
> |
100000 |
nM |
19128055 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
TGI |
> |
100000 |
nM |
19128055 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
79400 |
nM |
19128055 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
99400 |
nM |
19128055 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
TGI |
= |
79400 |
nM |
19128055 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
LC50 |
= |
79400 |
nM |
19128055 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
TGI |
= |
79400 |
nM |
19128055 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
TGI |
= |
79400 |
nM |
19128055 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
19128055 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
19128055 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
IC50 |
= |
34000 |
nM |
19128055 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25000 |
nM |
19128055 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
23280.91 |
nM |
19128055 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
19128055 |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Kd |
> |
10000 |
nM |
19128055 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
13995.87 |
nM |
19128055 |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Activity |
= |
80 |
% |
19128055 |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
13837.88 |
nM |
17850214 |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
69677.19 |
nM |
18183025 |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
146076.73 |
nM |
18183025 |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
199.5 |
nM |
18183025 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
5093.31 |
nM |
18183025 |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
11562.35 |
nM |
18183025 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
33596.87 |
nM |
16680159 |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15958589 |
NPT3305 |
Individual Protein |
Chaperone activity of bc1 complex-like, mitochondrial |
Homo sapiens |
Kd |
> |
10000 |
nM |
21440449 |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Kd |
> |
10000 |
nM |
21417417 |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
69546.74 |
nM |
21080703 |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Kd |
> |
10000 |
nM |
21944287 |
NPT3341 |
Individual Protein |
Serine/threonine-protein kinase Nek5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21982796 |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Activity |
= |
90 |
% |
PubChem BioAssay data set |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
650 |
nM |
10.6019/CHEMBL1201861 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
0.11 |
|
10.6019/CHEMBL1201861 |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24681986 |
NPT3343 |
Individual Protein |
Uncharacterized aarF domain-containing protein kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18077363 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
700 |
nM |
26741853 |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
2033588 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
6400 |
nM |
17150358 |
NPT3288 |
Individual Protein |
Interleukin-1 receptor-associated kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3228 |
Individual Protein |
Adaptor-associated kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
16800 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
19300 |
nM |
DrugMatrix in vitro pharmacology data |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
19900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2151 |
Cell Line |
NCI-H345 |
Homo sapiens |
IC50 |
= |
38910.65 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
1380352.25 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
200 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
48921.16 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2058 |
Cell Line |
NCI-H128 |
Homo sapiens |
IC50 |
= |
3515053.41 |
nM |
24183741 |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
24079882 |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
293211.15 |
nM |
22050318 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8450319 |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
272690.38 |
nM |
21616566 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
IC50 |
> |
10000 |
nM |
12762787 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
705405.63 |
nM |
19105653 |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
18768.84 |
nM |
15104491 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
22387.2 |
nM |
25695368 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
17782.8 |
nM |
16989516 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757708 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
1993318.27 |
nM |
12398536 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
IC50 |
> |
25000 |
nM |
18656986 |
NPT3310 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15921411 |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
4414875.88 |
nM |
8882436 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
86297.85 |
nM |
23252848 |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
557476.86 |
nM |
15844938 |
NPT6579 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Mus musculus |
IC50 |
= |
5000 |
nM |
19453174 |
NPT6579 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Mus musculus |
Inhibition |
= |
63 |
% |
19453174 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22483395 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22483395 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22483395 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
23886345 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22694318 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
15497936 |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
28796.91 |
nM |
15270566 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
12823.31 |
nM |
19691312 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
18989978 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
17498.47 |
nM |
18989978 |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
19938815 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
28000 |
nM |
20041704 |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
351370.07 |
nM |
10579870 |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19778068 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23451797 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
30900 |
nM |
15026054 |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
530972.91 |
nM |
16038541 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
19998.62 |
nM |
25127165 |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT2093 |
Cell Line |
PF-382 |
Homo sapiens |
IC50 |
= |
50966.93 |
nM |
16724853 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
TGI |
= |
100000 |
nM |
17685651 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25000 |
nM |
22703109 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
3199666.93 |
nM |
22703109 |
NPT1942 |
Cell Line |
CESS |
Homo sapiens |
IC50 |
= |
20854.94 |
nM |
22703109 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
22703109 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
170 |
nM |
1875335 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
3959031 |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
256416.74 |
nM |
3339605 |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
42892.97 |
nM |
18070958 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Kd |
> |
10000 |
nM |
18070958 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
25442.53 |
nM |
20100877 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
18955522 |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19223615 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Activity |
= |
81 |
% |
19223615 |
NPT3325 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Gallus gallus |
Kd |
> |
10000 |
nM |
19223615 |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19581457 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
24600 |
nM |
19581457 |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
12600.71 |
nM |
19581457 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
100000 |
nM |
19581457 |
NPT2090 |
Cell Line |
SNU-16 |
Homo sapiens |
IC50 |
= |
117136.98 |
nM |
19581457 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
13152.25 |
nM |
19581457 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
TGI |
> |
100000 |
nM |
18625771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
20585132 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
60000 |
nM |
20585132 |
NPT2194 |
Cell Line |
IMR-5 |
Homo sapiens |
IC50 |
= |
35313.88 |
nM |
18625771 |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18573937 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
793 |
nM |
16472241 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
34000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
450 |
nM |
DrugMatrix in vitro pharmacology data |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
40000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11100 |
nM |
DrugMatrix in vitro pharmacology data |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
32000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
18200 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1977 |
Cell Line |
LOUCY |
Homo sapiens |
IC50 |
= |
32125.3 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2095 |
Cell Line |
TALL-1 |
Homo sapiens |
IC50 |
= |
69736.44 |
nM |
21624500 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23644202 |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
> |
10000 |
nM |
24513185 |
NPT2077 |
Cell Line |
SCC-3 |
Homo sapiens |
IC50 |
= |
14295.59 |
nM |
24727243 |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
72450.97 |
nM |
16132 |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
487530.57 |
nM |
211235 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
25937011 |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
18494522 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10560729 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9000 |
nM |
20218657 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20155971 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8840 |
nM |
17346076 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
IC50 |
= |
12680 |
nM |
17346076 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
Activity |
>= |
60 |
% |
17346076 |
NPT2 |
Others |
Unspecified |
|
Activity |
>= |
60 |
% |
17346076 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19500 |
nM |
17346076 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
17346076 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
17930 |
nM |
17346076 |
NPT1985 |
Cell Line |
OPM-2 |
Homo sapiens |
IC50 |
= |
18460 |
nM |
21894898 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
Activity |
= |
50 |
% |
21894898 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
17358082 |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
124527.68 |
nM |
22671987 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19783432 |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Kd |
= |
1400 |
nM |
17343407 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
TGI |
= |
31622.78 |
nM |
10785421 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
20304655 |
NPT1936 |
Cell Line |
BC-3 |
Homo sapiens |
IC50 |
= |
18030.54 |
nM |
19757855 |
NPT796 |
Individual Protein |
Peripheral myelin protein 22 |
Homo sapiens |
Potency |
= |
37933 |
nM |
15026054 |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14640515 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
1310157.97 |
nM |
25918997 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
14575447 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
12713393 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
16038534 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
15568769 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
15568769 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
19319.68 |
nM |
16933872 |
NPT2163 |
Cell Line |
KMOE-2 |
Homo sapiens |
IC50 |
= |
171934.05 |
nM |
23245401 |
NPT3257 |
Individual Protein |
Serine/threonine-protein kinase 32C |
Homo sapiens |
Kd |
> |
10000 |
nM |
20619938 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
7.13 |
% |
8350094 |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19489596 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
11170670 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
LC50 |
> |
100000 |
nM |
1800632 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
LC50 |
> |
100000 |
nM |
1800632 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
1800632 |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
1424380.13 |
nM |
17512741 |
NPT583 |
Individual Protein |
Inositol monophosphatase 1 |
Rattus norvegicus |
Potency |
= |
2818.4 |
nM |
21970540 |
NPT3238 |
Individual Protein |
Dual specificity protein kinase TTK |
Homo sapiens |
Kd |
= |
1600 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
73 |
% |
15974612 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Activity |
= |
73 |
% |
15679321 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
IC50 |
= |
700 |
nM |
12444688 |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
700000 |
nM |
12762792 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
700 |
nM |
12762792 |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
650 |
nM |
12762792 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
48083.93 |
nM |
12662097 |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22316191 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
270 |
nM |
12444693 |
NPT3251 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25899335 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5000 |
nM |
19585998 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
19585998 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
FC |
= |
4 |
|
20189404 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
25730346 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
12662099 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10924178 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
1955885 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
1955885 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
15848.93 |
nM |
1955885 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
15848.93 |
nM |
1955885 |
NPT3255 |
Individual Protein |
Myosin light chain kinase family member 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16499324 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Activity |
= |
96 |
% |
22316191 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
180 |
nM |
25127165 |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
263426.13 |
nM |
18824363 |
NPT1949 |
Cell Line |
BL-41 |
Homo sapiens |
IC50 |
= |
25959.74 |
nM |
9677265 |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17892263 |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Activity |
= |
40 |
% |
25646964 |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
247038.2 |
nM |
1955885 |
NPT3314 |
Individual Protein |
Bone morphogenetic protein receptor type-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15497933 |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Kd |
> |
10000 |
nM |
16441074 |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
3345314.54 |
nM |
11908979 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
7900 |
nM |
11908979 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
700 |
nM |
11908979 |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Activity |
= |
88 |
% |
11908979 |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11908979 |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Kd |
> |
10000 |
nM |
11908979 |
NPT2083 |
Cell Line |
KARPAS-422 |
Homo sapiens |
IC50 |
= |
9963.36 |
nM |
24844534 |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
12662097 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
34.5 |
% |
13678412 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
1.1 |
% |
13678412 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
64.5 |
% |
13678412 |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Kd |
> |
10000 |
nM |
19105653 |
NPT1995 |
Cell Line |
NB17 |
Homo sapiens |
IC50 |
= |
163480.55 |
nM |
19105653 |
NPT3256 |
Individual Protein |
Serine/threonine-protein kinase WEE1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22168134 |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
> |
10000 |
nM |
20361780 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
1799649.14 |
nM |
7798959 |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18440233 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
16368.17 |
nM |
10785435 |
NPT2102 |
Cell Line |
MC-CAR |
Homo sapiens |
IC50 |
= |
489089.26 |
nM |
9784163 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
80 |
|
14510607 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
32912.91 |
nM |
1593285 |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
3699829.44 |
nM |
20100662 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
17000 |
nM |
18687007 |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24417634 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Activity |
= |
87 |
% |
11277748 |
NPT1907 |
Cell Line |
EB2 |
Homo sapiens |
IC50 |
= |
1284013.5 |
nM |
18336005 |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
44969.75 |
nM |
PubChem BioAssay data set |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
553126.65 |
nM |
16933888 |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22704889 |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
24381.87 |
nM |
18183025 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
18183025 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
100000 |
nM |
18183025 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
LC50 |
= |
100000 |
nM |
18183025 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
FC |
= |
2 |
|
17850214 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2 |
|
17850214 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
160 |
nM |
18183025 |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Activity |
= |
84 |
% |
18183025 |
NPT3295 |
Individual Protein |
Activin receptor type-2B |
Homo sapiens |
Kd |
> |
10000 |
nM |
18183025 |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Activity |
= |
90 |
% |
18183025 |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
93498.84 |
nM |
22037378 |
NPT2103 |
Cell Line |
MONO-MAC-6 |
Homo sapiens |
IC50 |
= |
38247.72 |
nM |
22037378 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
6966.27 |
nM |
22037378 |
NPT2167 |
Cell Line |
LB996-RCC |
Homo sapiens |
IC50 |
= |
59920.46 |
nM |
22037378 |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
215710.45 |
nM |
22037378 |
NPT3313 |
Individual Protein |
Bone morphogenetic protein receptor type-1A |
Homo sapiens |
Kd |
> |
10000 |
nM |
22037378 |
NPT1918 |
Cell Line |
DMS-79 |
Homo sapiens |
IC50 |
= |
89108.79 |
nM |
22037378 |
NPT3337 |
Individual Protein |
Serine/threonine-protein kinase DCLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
977399.04 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
10349.96 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3297 |
Individual Protein |
Non-receptor tyrosine-protein kinase TNK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1160 |
Cell Line |
BJ |
Homo sapiens |
Activity |
= |
106.3 |
% |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
TGI |
= |
100000 |
nM |
23398362 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
490 |
nM |
23398362 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
111476.52 |
nM |
23398362 |
NPT2037 |
Cell Line |
NCI-H2107 |
Homo sapiens |
IC50 |
= |
109311.87 |
nM |
22703163 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
79400 |
nM |
26035018 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
79400 |
nM |
25466198 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
63100 |
nM |
25466198 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
TGI |
= |
63100 |
nM |
25466198 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
TGI |
= |
63100 |
nM |
25466198 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
TGI |
= |
63100 |
nM |
25466198 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
63100 |
nM |
25466198 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
78300 |
nM |
25466198 |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Kd |
> |
10000 |
nM |
25700232 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
26331986 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
22704889 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
23611151 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
23611151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
25000 |
nM |
14695801 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20000 |
nM |
14695801 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
15387655 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
15387655 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
650 |
nM |
15387655 |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
652087.01 |
nM |
21666868 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
TGI |
> |
100000 |
nM |
10691710 |
NPT3224 |
Individual Protein |
Phosphorylase kinase gamma subunit 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22409377 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
20596.2 |
nM |
11754614 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
2640897.23 |
nM |
22694318 |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14640511 |
NPT625 |
Tissue |
Liver |
Mus musculus |
Activity |
= |
67 |
% |
10691721 |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
5761.16 |
nM |
19524436 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Activity |
= |
96 |
% |
24175613 |
NPT3307 |
Individual Protein |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18694644 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2180 |
nM |
12762801 |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
350 |
nM |
22500574 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
87 |
% |
22500574 |
NPT3361 |
Individual Protein |
Mitogen-activated protein kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25798528 |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
32474.53 |
nM |
26000707 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
19186.69 |
nM |
12105963 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
12105963 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
12105963 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
12105963 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
5395.11 |
nM |
19117486 |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
1780897.98 |
nM |
PubChem BioAssay data set |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
12502308 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19715320 |
NPT1951 |
Cell Line |
CMK |
Homo sapiens |
IC50 |
= |
207544.75 |
nM |
19715320 |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
422989.77 |
nM |
23978065 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19618920 |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
18980381 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
460315.44 |
nM |
12502328 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
73.12 |
% |
12502328 |
NPT2081 |
Cell Line |
HCC1599 |
Homo sapiens |
IC50 |
= |
14597.5 |
nM |
8254346 |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22671987 |
NPT3321 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8158164 |
NPT1717 |
Individual Protein |
Serine/threonine-protein kinase 25 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16378367 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
450 |
nM |
19105653 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
700 |
nM |
16989525 |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
79665.77 |
nM |
10346943 |
NPT464 |
Cell Line |
Daudi |
Homo sapiens |
IC50 |
= |
3151547.87 |
nM |
16252909 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
15000 |
nM |
12662094 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
9871565 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22400 |
nM |
23320609 |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24063567 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Inhibition |
= |
40 |
% |
17988094 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Activity |
= |
104 |
% |
22245048 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Activity |
= |
83 |
% |
23350733 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
TGI |
= |
12589.25 |
nM |
24328302 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
24328302 |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
22758788 |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Activity |
= |
90 |
% |
18288804 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14420 |
nM |
11929285 |
NPT2010 |
Cell Line |
NCI-H716 |
Homo sapiens |
IC50 |
= |
4070874.01 |
nM |
26327273 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10096852 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
26052978 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
26052978 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
26052978 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
16180824 |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
320 |
nM |
10869229 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
25100 |
nM |
19845338 |
NPT3220 |
Individual Protein |
Ephrin type-A receptor 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26295746 |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
23190013 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
11455.13 |
nM |
PubChem BioAssay data set |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
1143513.71 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
25100 |
nM |
10560729 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
529923.15 |
nM |
25871540 |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
466316.23 |
nM |
11087610 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
10000 |
nM |
24842703 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
52077.03 |
nM |
21377877 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
LC50 |
> |
100000 |
nM |
17315955 |
NPT3243 |
Individual Protein |
myosin light chain kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18640035 |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
64020.73 |
nM |
8759172 |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17985844 |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
947719.91 |
nM |
PubChem BioAssay data set |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Kd |
= |
2900 |
nM |
20934335 |
NPT2113 |
Cell Line |
EW-24 |
Homo sapiens |
IC50 |
= |
1192057.4 |
nM |
20923180 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20923180 |
NPT3301 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19072209 |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
140782.48 |
nM |
22612410 |
NPT1980 |
Cell Line |
NB14 |
Homo sapiens |
IC50 |
= |
2022490.6 |
nM |
26048785 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
PubChem BioAssay data set |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Kd |
> |
10000 |
nM |
22850207 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
24359277 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
24359277 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
TGI |
> |
100000 |
nM |
1791472 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
TGI |
> |
100000 |
nM |
1791472 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
> |
100000 |
nM |
1791472 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
1791472 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
1791472 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
LC50 |
> |
100000 |
nM |
1791472 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
1336040 |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
22230050 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
52966.34 |
nM |
3373220 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
19098.53 |
nM |
3373220 |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22100311 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11575963 |
NPT1925 |
Cell Line |
CAL-148 |
Homo sapiens |
IC50 |
= |
181377.41 |
nM |
26083682 |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18808182 |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
914521.52 |
nM |
19374389 |
NPT1656 |
Individual Protein |
Protein kinase N1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
9548870 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
6481359 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
6481359 |
NPT2187 |
Cell Line |
RL95-2 |
Homo sapiens |
IC50 |
= |
82234.34 |
nM |
6481359 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
6481359 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
810 |
nM |
7515410 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
IC50 |
= |
360 |
nM |
88001 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
IC50 |
= |
100 |
nM |
88001 |
NPT2 |
Others |
Unspecified |
|
Activity |
>= |
60 |
% |
88001 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
15838.22 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
35156.04 |
nM |
PubChem BioAssay data set |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
27861.21 |
nM |
19653666 |
NPT1692 |
Individual Protein |
Mitogen-activated protein kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11975483 |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11975483 |
NPT1671 |
Individual Protein |
AMP-activated protein kinase, alpha-2 subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
23795891 |
NPT3339 |
Individual Protein |
Myosin-IIIB |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Activity |
= |
94 |
% |
PubChem BioAssay data set |
NPT2038 |
Cell Line |
NCI-H748 |
Homo sapiens |
IC50 |
= |
263974.37 |
nM |
PubChem BioAssay data set |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
160 |
nM |
12350153 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
25000 |
nM |
20521771 |
NPT3813 |
Individual Protein |
Tyrosine-protein kinase SRC |
Gallus gallus |
Activity |
= |
89 |
% |
17253849 |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
700 |
nM |
20614907 |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
290923.4 |
nM |
2128517 |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
1751971.49 |
nM |
26316467 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20614907 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Activity |
= |
82 |
% |
23006147 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
TGI |
= |
63095.73 |
nM |
20521782 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
TGI |
= |
63095.73 |
nM |
18808182 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
TGI |
= |
63095.73 |
nM |
18808182 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
63095.73 |
nM |
18808182 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
TGI |
= |
63095.73 |
nM |
18808182 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
18808182 |
NPT3304 |
Individual Protein |
Serine/threonine-protein kinase receptor R3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20307086 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50 |
= |
130000 |
nM |
23891163 |
NPT3108 |
Protein Family |
Casein kinase I |
Homo sapiens |
IC50 |
= |
17000 |
nM |
23891163 |
NPT321 |
Protein Family |
cAMP-dependent protein kinase (PKA) |
Homo sapiens |
IC50 |
> |
1000000 |
nM |
23891163 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
1000000 |
nM |
23891163 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
IC50 |
= |
229043.51 |
nM |
9651160 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19628311 |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
25652.88 |
nM |
PubChem BioAssay data set |
NPT84 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
Rattus norvegicus |
IC50 |
= |
11000 |
nM |
12502326 |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
29948.34 |
nM |
19361168 |
NPT3252 |
Individual Protein |
Serine/threonine-protein kinase PFTAIRE-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25856683 |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757722 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26147490 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1000000 |
nM |
16499322 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
IC50 |
= |
34000 |
nM |
16499322 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
16499322 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
160 |
nM |
9134742 |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Kd |
> |
10000 |
nM |
18260638 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
22512738 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
Patent: US9114126 B2 |
NPT2157 |
Cell Line |
SUP-T1 |
Homo sapiens |
IC50 |
= |
4498219.81 |
nM |
21332115 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Kd |
> |
10000 |
nM |
2045820 |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19746919 |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
164277.16 |
nM |
20624681 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Activity |
= |
84 |
% |
20624681 |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Kd |
> |
10000 |
nM |
19081726 |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Kd |
> |
10000 |
nM |
24601675 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
280 |
nM |
19902967 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
350 |
nM |
26854381 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
5050 |
nM |
17958396 |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
1502931.78 |
nM |
17958396 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
9871657 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
15848.93 |
nM |
9871657 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17609121 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17609121 |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
923655.35 |
nM |
23634786 |
NPT3264 |
Individual Protein |
Serine/threonine-protein kinase RIO1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18630962 |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
18630962 |
NPT1999 |
Cell Line |
TUR |
Homo sapiens |
IC50 |
= |
2055521.78 |
nM |
10869208 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
28000 |
nM |
12880316 |
NPT1969 |
Cell Line |
TGW |
Homo sapiens |
IC50 |
= |
17812.38 |
nM |
21865038 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18293903 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
907720.04 |
nM |
PubChem BioAssay data set |
NPT2136 |
Cell Line |
MDA-MB-134-VI |
Homo sapiens |
IC50 |
= |
220192.9 |
nM |
20112996 |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20329738 |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15125956 |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
2016726 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Activity |
= |
87 |
% |
2016726 |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
1325586.13 |
nM |
15808482 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
20200 |
nM |
17261619 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Activity |
= |
83 |
% |
17239490 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
0.1 |
% |
17923494 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
55.9 |
% |
17923494 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
50.9 |
% |
17923494 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
44 |
% |
17938181 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
48 |
% |
17938181 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
1.1 |
% |
17938181 |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
17967918 |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Activity |
= |
93 |
% |
20070106 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
370 |
nM |
20171758 |
NPT2156 |
Cell Line |
SU-DHL-1 |
Homo sapiens |
IC50 |
= |
162830.54 |
nM |
18347108 |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
74334.93 |
nM |
20038624 |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
268865.97 |
nM |
18591277 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
5260.17 |
nM |
18779359 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
131690.04 |
nM |
18644957 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
20350950 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18710917 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
18710917 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
29623.86 |
nM |
18710917 |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
34252.45 |
nM |
18725450 |
NPT1560 |
Protein Complex |
Cyclin-dependent kinase 4/cyclin D1 |
Homo sapiens |
IC50 |
= |
27000 |
nM |
18474583 |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
18299417 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
24300 |
nM |
18391041 |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
37706.93 |
nM |
18443122 |
NPT1994 |
Cell Line |
MHH-CALL-2 |
Homo sapiens |
IC50 |
= |
322126.72 |
nM |
19124664 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Activity |
= |
76 |
% |
19651906 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Activity |
= |
91 |
% |
19651906 |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
70477.75 |
nM |
19546358 |
NPT1950 |
Cell Line |
BL-70 |
Homo sapiens |
IC50 |
= |
20327.36 |
nM |
18625769 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
16100 |
nM |
18625769 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
18625769 |
NPT3253 |
Individual Protein |
Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
20625154 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
IC50 |
= |
130000 |
nM |
20660668 |
NPT2059 |
Cell Line |
NCI-H2141 |
Homo sapiens |
IC50 |
= |
34653.34 |
nM |
19188393 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
20805391 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21443195 |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
37.7 |
nM |
21543140 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
21981980 |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2158 |
Cell Line |
TE-441-T |
Homo sapiens |
IC50 |
= |
36114.81 |
nM |
22194678 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
88 |
% |
22931300 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1007/s00044-010-9338-x |
NPT2131 |
Cell Line |
WSU-NHL |
Homo sapiens |
IC50 |
= |
2563674.86 |
nM |
10.1007/s00044-009-9206-8 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
16865.53 |
nM |
23414843 |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
81680.39 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
TGI |
= |
100000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12300 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
27200 |
nM |
Open TG-GATES in vivo data: Pathology |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Activity |
= |
71 |
% |
DrugMatrix in vivo data: Biochemistry |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
85282.14 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
TGI |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
TGI |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
TGI |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
TGI |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
50100 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
42278.68 |
nM |
DrugMatrix in vivo data: Hematology |
NPT2184 |
Cell Line |
NCI-H510A |
Homo sapiens |
IC50 |
= |
30032.86 |
nM |
DrugMatrix in vivo data: Hematology |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25050881 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
26288696 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
26288696 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3981.07 |
nM |
26465972 |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
630305.11 |
nM |
10425145 |
NPT2060 |
Cell Line |
NCI-H2171 |
Homo sapiens |
IC50 |
= |
159236.9 |
nM |
10869194 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
6309.6 |
nM |
20427099 |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Activity |
= |
82 |
% |
17417907 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
13273.94 |
nM |
17665952 |
NPT2195 |
Cell Line |
LC4-1 |
Homo sapiens |
IC50 |
= |
18873.45 |
nM |
18494522 |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18280170 |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
50928.62 |
nM |
PubChem BioAssay data set |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
123979.1 |
nM |
PubChem BioAssay data set |
NPT2124 |
Cell Line |
MRK-nu-1 |
Homo sapiens |
IC50 |
= |
7129.69 |
nM |
9677282 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
20681570 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5000 |
nM |
24079882 |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
28973.31 |
nM |
17346076 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
17346076 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22779787 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22779787 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
427385.75 |
nM |
12398543 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Activity |
= |
90 |
% |
23002419 |
NPT2691 |
Individual Protein |
Voltage-gated L-type calcium channel alpha-1C subunit |
Homo sapiens |
IC50 |
= |
23400 |
nM |
24387347 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
IC50 |
= |
3100 |
nM |
21131198 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
12800 |
nM |
16989519 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
12600 |
nM |
16989519 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
16989519 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
12600 |
nM |
20704304 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
20704304 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
12600 |
nM |
22272829 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
22272829 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
22272829 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
12600 |
nM |
22272829 |
NPT2164 |
Cell Line |
KMS-12-PE |
Homo sapiens |
IC50 |
= |
1386464.14 |
nM |
26200131 |
NPT3350 |
Individual Protein |
Tyrosine-protein kinase Srms |
Homo sapiens |
Kd |
> |
10000 |
nM |
24928403 |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Kd |
> |
10000 |
nM |
21377877 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
31622.78 |
nM |
9249977 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
9249977 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
9249977 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
TGI |
= |
39810.72 |
nM |
9249977 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
165626.13 |
nM |
9249977 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
42000 |
nM |
17488128 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25856683 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5623.4 |
nM |
25856683 |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
20035.63 |
nM |
17910513 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
24387703 |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15387655 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Kd |
= |
2000 |
nM |
15043411 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
13489.63 |
nM |
26854381 |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.1021/np50041a029 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
280 |
nM |
10.1016/S0261-2194(02)00175-8 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10000 |
nM |
12617583 |
NPT1909 |
Cell Line |
ECC12 |
Homo sapiens |
IC50 |
= |
288995.18 |
nM |
10.1016/j.jssas.2011.10.002 |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
292958.51 |
nM |
25237727 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
IC50 |
= |
210 |
nM |
19848434 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
280 |
nM |
19848434 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
30100 |
nM |
20402524 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14700 |
nM |
20402524 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
20402524 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
9770 |
nM |
20402524 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
16800 |
nM |
19072548 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17800 |
nM |
19245261 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14700 |
nM |
19245261 |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
470292.57 |
nM |
11858752 |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
848063.91 |
nM |
26231157 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
46700 |
nM |
PubChem BioAssay data set |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15387642 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
35700 |
nM |
19995673 |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
489497.82 |
nM |
9514014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
28600 |
nM |
11170665 |
NPT3241 |
Individual Protein |
Serine/threonine-protein kinase NEK9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18479163 |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
93717.13 |
nM |
18442289 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17190444 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
5000 |
nM |
17190444 |
NPT3230 |
Individual Protein |
Serine/threonine-protein kinase 17B |
Homo sapiens |
Kd |
> |
10000 |
nM |
19818612 |
NPT1917 |
Cell Line |
CA46 |
Homo sapiens |
IC50 |
= |
92430.78 |
nM |
17844994 |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
742149.72 |
nM |
17844994 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12300 |
nM |
23964704 |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
113370.14 |
nM |
19627125 |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
16360.13 |
nM |
16643030 |
NPT3308 |
Individual Protein |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23013356 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
15497945 |
NPT6206 |
Individual Protein |
Voltage-gated N-type calcium channel alpha-1B subunit |
Homo sapiens |
EC50 |
= |
27580 |
nM |
12828469 |
NPT4155 |
Protein Complex |
CDK6/cyclin D1 |
Homo sapiens |
IC50 |
= |
23500 |
nM |
17958396 |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25856683 |