Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Residual Activity |
= |
61 |
% |
19689125 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
11520227 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
11520227 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10583.9 |
nM |
12880316 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
12880316 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Activity |
= |
63 |
% |
15387639 |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
79 |
% |
18157122 |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
91 |
% |
PubChem BioAssay data set |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PubChem BioAssay data set |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1708 |
Individual Protein |
Serine/threonine-protein kinase 16 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
75 |
% |
20430633 |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
98 |
% |
19818612 |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
= |
10000 |
nM |
18803421 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
22418279 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
23691978 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
13 |
nM |
23734701 |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11374948 |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
100 |
% |
22537362 |
NPT3356 |
Individual Protein |
Tyrosine-protein kinase receptor Tie-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10924160 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Activity |
= |
89 |
% |
25437304 |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
97 |
% |
21044847 |
NPT1673 |
Individual Protein |
CaM kinase I gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
64 |
% |
PubChem BioAssay data set |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23547843 |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
7769392 |
NPT3352 |
Individual Protein |
Dual specificity testis-specific protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
7264681 |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Residual Activity |
= |
107 |
% |
15679329 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3162.3 |
nM |
20361780 |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
84 |
% |
8277313 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
47 |
% |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
AC50 |
= |
10000 |
nM |
23327668 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23215246 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
50 |
nM |
23215246 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Inhibition |
= |
79 |
% |
22342628 |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
113 |
% |
18952424 |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
127 |
% |
21131198 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Kd |
> |
10000 |
nM |
23286240 |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
17877337 |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19700322 |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
117 |
% |
22758788 |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Activity |
= |
90 |
% |
PubChem BioAssay data set |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
12662101 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
80 |
% |
9051910 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
99 |
% |
19734910 |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
DrugMatrix in vitro pharmacology data |
NPT3338 |
Individual Protein |
Myosin IIIA |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
97 |
% |
DrugMatrix in vitro pharmacology data |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1900 |
nM |
7910522 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
122 |
% |
8960059 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
47.3 |
nM |
21452899 |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Residual Activity |
= |
111 |
% |
DrugMatrix in vivo data: Pathology |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
104 |
% |
22328583 |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
112 |
% |
26383126 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
100 |
% |
19105653 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
10 |
% |
16203143 |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
86 |
% |
19285413 |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
81 |
% |
19743809 |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
116 |
% |
22280816 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000 |
nM |
18341287 |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15270579 |
NPT3322 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18547115 |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
16441076 |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Kd |
> |
10000 |
nM |
15387639 |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
15844941 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
36 |
% |
11678655 |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
76 |
% |
19327990 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2000 |
nM |
26026364 |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
103 |
% |
15026054 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
100 |
% |
20675131 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
73.1 |
nM |
25406853 |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
111 |
% |
25978520 |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
12617583 |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
79 |
% |
12617583 |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
123 |
% |
12617583 |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
17547458 |
NPT3319 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25659770 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
= |
51 |
nM |
11720520 |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
100 |
% |
23327668 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
23819871 |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
110 |
% |
23819871 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26706176 |
NPT3369 |
Individual Protein |
Interferon-induced, double-stranded RNA-activated protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
1517739 |
NPT3340 |
Individual Protein |
Serine/threonine-protein kinase Nek1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25667960 |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
45 |
% |
21131198 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
112 |
% |
10514320 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
6309.6 |
nM |
9917297 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
25554367 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Kd |
= |
59 |
nM |
15104484 |
NPT3328 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 11 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8558523 |
NPT56 |
Individual Protein |
Beta-lactamase AmpC |
Escherichia coli K-12 |
Potency |
= |
7079.5 |
nM |
PubChem BioAssay data set |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Kd |
= |
950 |
nM |
PubChem BioAssay data set |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
111 |
% |
PubChem BioAssay data set |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11277744 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
47 |
% |
22209731 |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
19105653 |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
18177008 |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
98 |
% |
24262380 |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
59 |
% |
PubChem BioAssay data set |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Activity |
= |
7 |
% |
24582402 |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22472691 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
19178292 |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
36 |
% |
18298075 |
NPT3335 |
Individual Protein |
Serine/threonine-protein kinase DCLK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18298075 |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18298075 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
23350733 |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
41 |
% |
17665952 |
NPT3109 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25066952 |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17696332 |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
10.1007/s00044-013-0466-y |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
57 |
% |
23806014 |
NPT3295 |
Individual Protein |
Activin receptor type-2B |
Homo sapiens |
Kd |
= |
4800 |
nM |
15711537 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
45 |
% |
15711537 |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18844338 |
NPT3460 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 3 |
Homo sapiens |
Activity |
= |
96 |
% |
PubChem BioAssay data set |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
112 |
% |
PubChem BioAssay data set |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
= |
2400 |
nM |
PubChem BioAssay data set |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PubChem BioAssay data set |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21945458 |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
PubChem BioAssay data set |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
23398362 |
NPT9 |
Individual Protein |
DNA polymerase eta |
Homo sapiens |
Potency |
|
22387.2 |
nM |
23398362 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
23398362 |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
Activity |
= |
30 |
day |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
PubChem BioAssay data set |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Kd |
> |
10000 |
nM |
26090896 |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
22694270 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Kd |
> |
10000 |
nM |
22671987 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
83 |
% |
22079755 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
123 |
% |
22871217 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24893224 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
24893224 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Activity |
= |
83 |
% |
24893224 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
25871540 |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
10000 |
nM |
12398531 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
20575589 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
-2 |
% |
25765759 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
2 |
% |
20801038 |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
93 |
% |
26123643 |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
12 |
% |
22418278 |
NPT3323 |
Individual Protein |
Cell division cycle 2-like protein kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11754602 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
91 |
% |
19874044 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
45 |
% |
20061160 |
NPT4095 |
Protein Complex |
Mammalian target of Rapamycin (mTORC1) |
Homo sapiens |
Residual Activity |
= |
123 |
% |
23376010 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
85 |
% |
26147490 |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
80 |
% |
16933872 |
NPT3220 |
Individual Protein |
Ephrin type-A receptor 6 |
Homo sapiens |
Kd |
= |
2200 |
nM |
19344127 |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
19284743 |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23006147 |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
114 |
% |
20420415 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
19 |
% |
10924160 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
20499922 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
12589.3 |
nM |
10691710 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
68 |
% |
12502308 |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
40 |
% |
24195466 |
NPT3342 |
Individual Protein |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
Kd |
= |
1100 |
nM |
26046820 |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
65 |
% |
26048790 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
7 |
% |
26317881 |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
18177012 |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
82 |
% |
15974618 |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
120 |
% |
15620243 |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
19265396 |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
3336016 |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Activity |
= |
66 |
% |
18001087 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
23999046 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
89 |
% |
8676127 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Activity |
= |
86 |
% |
19674906 |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
16513346 |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
20726569 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
101 |
% |
18494522 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
21612217 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
108 |
% |
21807523 |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
21925888 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
20035556 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26000707 |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19456120 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7079.5 |
nM |
19318257 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
= |
120 |
nM |
10571160 |
NPT3306 |
Individual Protein |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
Kd |
= |
640 |
nM |
15006398 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
108 |
% |
9871552 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
123 |
% |
7310807 |
NPT3454 |
Individual Protein |
PAS domain-containing serine/threonine-protein kinase |
Homo sapiens |
Residual Activity |
= |
92 |
% |
3127589 |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
14125.4 |
nM |
12392731 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Inhibition |
= |
20 |
% |
17438054 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Activity |
= |
86 |
% |
17438054 |
NPT3249 |
Individual Protein |
Tyrosine- and threonine-specific cdc2-inhibitory kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
17067151 |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Kd |
> |
10000 |
nM |
15730240 |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Kd |
> |
10000 |
nM |
19081718 |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
19403314 |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
108 |
% |
19093848 |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
65 |
% |
19524330 |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
5 |
% |
20516287 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
18426954 |
NPT3454 |
Individual Protein |
PAS domain-containing serine/threonine-protein kinase |
Homo sapiens |
Residual Activity |
= |
34 |
% |
20566771 |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Ki |
= |
2511.89 |
nM |
16472241 |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
21429630 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
DrugMatrix in vitro pharmacology data |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
DrugMatrix in vitro pharmacology data |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22440626 |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
23151429 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Potency |
= |
2592.9 |
nM |
23140987 |
NPT532 |
Individual Protein |
Lysine-specific demethylase 4A |
Homo sapiens |
Potency |
|
50118.7 |
nM |
23391589 |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
91 |
% |
23823011 |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
82 |
% |
Open TG-GATES in vivo data: Biochemistry |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Ki |
= |
2511.89 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3371 |
Individual Protein |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
11220.2 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
126 |
% |
Open TG-GATES in vivo data: Biochemistry |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
78 |
% |
Open TG-GATES in vivo data: Hematology |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
77 |
% |
Open TG-GATES in vivo data: Hematology |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Activity |
= |
104 |
% |
Open TG-GATES in vivo data: Pathology |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
88 |
% |
Open TG-GATES in vivo data: Organ Weight |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
91 |
% |
Open TG-GATES in vivo data: Organ Weight |
NPT484 |
Individual Protein |
Luciferin 4-monooxygenase |
Photinus pyralis |
Potency |
= |
1258.9 |
nM |
DrugMatrix in vivo data: Pathology |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
89 |
% |
DrugMatrix in vivo data: Hematology |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
57 |
% |
24224794 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Kd |
> |
10000 |
nM |
24246731 |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
24388809 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
24412719 |
NPT3209 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24268596 |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
24631185 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
24967731 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Activity |
= |
84 |
% |
25372601 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
9 |
nM |
10.1039/C4MD00303A |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
76 |
% |
21980963 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Potency |
|
10000 |
nM |
4851320 |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
4851320 |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
22418278 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
24 |
% |
PubChem BioAssay data set |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
73 |
% |
17107790 |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
19093884 |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18954984 |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
12589.3 |
nM |
19084294 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
101 |
% |
20017493 |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
13 |
% |
19966789 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
28183.8 |
nM |
21080647 |
NPT3311 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22036991 |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
55 |
% |
22877635 |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
23252603 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Inhibition |
= |
97 |
% |
23252603 |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
23252603 |
NPT3120 |
Individual Protein |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Ki |
= |
63.1 |
nM |
10.6019/CHEMBL1201861 |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
12589.3 |
nM |
10.6019/CHEMBL1201861 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
92 |
% |
10.6019/CHEMBL1201861 |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
FC |
= |
4.2 |
|
10.6019/CHEMBL1201861 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
49 |
% |
23538115 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Activity |
= |
71 |
% |
23601706 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Activity |
= |
122 |
% |
23644210 |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23786452 |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
76 |
% |
24015327 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24015327 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Inhibition |
= |
8 |
% |
23906422 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Inhibition |
= |
39 |
% |
23860593 |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
57 |
% |
24074025 |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
102 |
% |
PubChem BioAssay data set |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
81 |
% |
PubChem BioAssay data set |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
794.3 |
nM |
24742384 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25462271 |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
44668.4 |
nM |
25311567 |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Kd |
> |
10000 |
nM |
25221651 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
113 |
% |
25734520 |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
83 |
% |
25906087 |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
26100440 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
10.1039/C5MD00247H |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.1039/C5MD00247H |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Kd |
> |
10000 |
nM |
26890114 |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
26890114 |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
101 |
% |
26443078 |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Residual Activity |
= |
83 |
% |
26890116 |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
27186676 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
1 |
% |
11170656 |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
= |
3000 |
nM |
18611050 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
122 |
% |
23869482 |
NPT1139 |
Individual Protein |
Arachidonate 15-lipoxygenase, type II |
Homo sapiens |
Potency |
|
7943.3 |
nM |
25651042 |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Ki |
= |
1000 |
nM |
26420067 |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26465675 |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
79 |
% |
20729083 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Ki |
= |
5.012 |
nM |
15921411 |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Residual Activity |
= |
68 |
% |
16933872 |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
10346942 |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
12 |
% |
24387661 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
98 |
% |
24387661 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Activity |
= |
83 |
% |
PubChem BioAssay data set |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23354071 |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
34 |
% |
26394152 |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
20624681 |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
92 |
% |
19762244 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20159656 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20159656 |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
26684850 |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
99 |
% |
7853002 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25739048 |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25735399 |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19193024 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20718475 |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
90 |
% |
20718475 |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
112 |
% |
19555084 |
NPT3260 |
Individual Protein |
Phosphatidylinositol-5-phosphate 4-kinase type-2 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
16372404 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
75 |
% |
20701299 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
102 |
% |
20704304 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Activity |
= |
5 |
% |
16933872 |
NPT3355 |
Individual Protein |
TGF-beta receptor type II |
Homo sapiens |
Kd |
> |
10000 |
nM |
15921416 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
69 |
% |
11975502 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Activity |
= |
69 |
% |
24992702 |
NPT800 |
Individual Protein |
M-phase phosphoprotein 8 |
Homo sapiens |
Potency |
|
31622.8 |
nM |
12502331 |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14695800 |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
81 |
% |
7769392 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Activity |
= |
3 |
% |
11141109 |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
84 |
% |
17343407 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
25537529 |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
135 |
% |
25537529 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
34 |
% |
25630222 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
18077363 |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
15104491 |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
20598551 |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
9392880 |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
66 |
% |
22119124 |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
794.3 |
nM |
19013823 |
NPT4 |
Individual Protein |
Large T antigen |
Simian virus 40 |
IC50 |
|
4870 |
nM |
22239601 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19928832 |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
17346076 |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Activity |
= |
87 |
% |
11720542 |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12088422 |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Kd |
= |
1900 |
nM |
15012986 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
= |
9400 |
nM |
4020828 |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
98 |
% |
11858989 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1400 |
nM |
10753475 |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12477351 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
125 |
% |
15369401 |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
77 |
% |
16759114 |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
16870428 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
107 |
% |
18164197 |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18457386 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16774.4 |
nM |
8277312 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
21144756 |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
77 |
% |
21663319 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1900 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
DrugMatrix in vitro pharmacology data |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
126 |
% |
22194678 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11220.2 |
nM |
8621716 |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
49 |
% |
8862725 |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
109 |
% |
23072299 |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
92 |
% |
23072299 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Activity |
= |
85 |
% |
23214452 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Activity |
= |
92 |
% |
10.6019/CHEMBL1201861 |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
45 |
% |
10.6019/CHEMBL1201861 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
10.6019/CHEMBL1201861 |
NPT3294 |
Individual Protein |
Activin receptor type-2A |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
64800 |
nM |
23916255 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
8.04 |
|
24074257 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
3006 |
nM |
23708010 |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
83 |
% |
DrugMatrix in vivo data: Pathology |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
111 |
% |
DrugMatrix in vivo data: Pathology |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
24333581 |
NPT58 |
Individual Protein |
Bloom syndrome protein |
Homo sapiens |
Potency |
= |
50118.7 |
nM |
15646539 |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26132075 |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
93 |
% |
14613317 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
17630726 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
17582659 |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
21885167 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26789378 |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Kd |
> |
10000 |
nM |
14695799 |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
90 |
% |
11549443 |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15787429 |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Ki |
> |
10000 |
nM |
25237727 |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Kd |
> |
10000 |
nM |
21377877 |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
10 |
% |
20483615 |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
Activity |
= |
30 |
day |
17854154 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
17190457 |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11374954 |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
14 |
% |
26034885 |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
26000707 |
NPT135 |
Individual Protein |
Chromobox protein homolog 1 |
Homo sapiens |
Potency |
|
56234.1 |
nM |
22642560 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
= |
210 |
nM |
PubChem BioAssay data set |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Kd |
> |
10000 |
nM |
9548870 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
= |
170 |
nM |
7528785 |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
98 |
% |
PubChem BioAssay data set |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
19 |
% |
PubChem BioAssay data set |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
PubChem BioAssay data set |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
PubChem BioAssay data set |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
1522422 |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
18598078 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
101 |
% |
22330636 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17571903 |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
113 |
% |
17428663 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Activity |
= |
78 |
% |
PubChem BioAssay data set |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Activity |
= |
91 |
% |
10.1007/s00044-008-9111-6 |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
10869194 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
20596.2 |
nM |
23190013 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
11 |
% |
11520232 |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
100 |
% |
18336006 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Inhibition |
= |
13 |
% |
18341287 |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
17665951 |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
136 |
% |
20349977 |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
55 |
% |
25970729 |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
= |
3100 |
nM |
12880316 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Ki |
= |
1258.93 |
nM |
25856683 |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
76 |
% |
25856683 |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
59 |
% |
25856683 |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
16 |
% |
22647719 |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
88 |
% |
21036050 |
NPT3252 |
Individual Protein |
Serine/threonine-protein kinase PFTAIRE-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
80 |
% |
15646539 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
95 |
% |
PubChem BioAssay data set |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
= |
270 |
nM |
PubChem BioAssay data set |
NPT3310 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25173852 |
NPT3268 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22834923 |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
68 |
% |
25238443 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
9358638 |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
11 |
% |
10075755 |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
16872140 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
88 |
% |
24582402 |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
19191549 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
11220.2 |
nM |
19097799 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
141 |
% |
PubChem BioAssay data set |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
63 |
% |
PubChem BioAssay data set |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
PubChem BioAssay data set |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Kd |
= |
1700 |
nM |
23354072 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22264149 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8254344 |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
121 |
% |
8350085 |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25621853 |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
115 |
% |
25211145 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
910 |
nM |
18616221 |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
27 |
% |
25259516 |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25629304 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
8699187 |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
37 |
% |
8699187 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
8699187 |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Activity |
= |
92 |
% |
PubChem BioAssay data set |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
26226070 |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
18500841 |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Kd |
> |
10000 |
nM |
21067210 |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
69 |
% |
16499325 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
26151487 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Ki |
= |
501.19 |
nM |
26225905 |
NPT3168 |
Individual Protein |
Casein kinase I alpha |
Homo sapiens |
Ki |
= |
1000 |
nM |
26225905 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
4600 |
nM |
15974618 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
105 |
% |
22530813 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2300 |
nM |
22530813 |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
110 |
% |
14643343 |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
15104512 |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Kd |
> |
10000 |
nM |
23376010 |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
22934671 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
25338277 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
37847 |
nM |
21273070 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
78 |
% |
18986200 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
23964644 |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
20801664 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
27 |
% |
18271521 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26483136 |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
70 |
% |
15497941 |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
101 |
% |
23234407 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
21534539 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
12088430 |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Residual Activity |
= |
89 |
% |
22413887 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
1 |
% |
25682561 |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10820113 |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14640522 |
NPT3250 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18303848 |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
23046382 |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
23046382 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Activity |
= |
103 |
% |
23675610 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
82 |
% |
9435889 |
NPT3305 |
Individual Protein |
Chaperone activity of bc1 complex-like, mitochondrial |
Homo sapiens |
Kd |
> |
10000 |
nM |
15050613 |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
92 |
% |
15050621 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
12589.3 |
nM |
10.1016/S0960-894X(01)80759-9 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
15771418 |
NPT63 |
Individual Protein |
Bromodomain adjacent to zinc finger domain protein 2B |
Homo sapiens |
Potency |
|
79432.8 |
nM |
17485662 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
13115.4 |
nM |
PubChem BioAssay data set |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Activity |
= |
107 |
% |
23354071 |
NPT3815 |
Individual Protein |
Tyrosine-protein kinase LCK |
Mus musculus |
Activity |
= |
44 |
% |
PubChem BioAssay data set |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
58 |
% |
15974607 |
NPT3334 |
Individual Protein |
Citron Rho-interacting kinase |
Homo sapiens |
Kd |
= |
510 |
nM |
17067151 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Inhibition |
= |
39 |
% |
22552195 |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
56 |
% |
22703109 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5623.4 |
nM |
22545792 |
NPT154 |
Individual Protein |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
12444692 |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
21353549 |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
52 |
% |
20825224 |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
8098735 |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11754618 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15067.2 |
nM |
9917283 |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
21428459 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
93 |
% |
19307359 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
19307359 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
30 |
nM |
23013356 |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
114 |
% |
20627740 |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
29 |
% |
16643031 |
NPT3238 |
Individual Protein |
Dual specificity protein kinase TTK |
Homo sapiens |
Kd |
= |
4500 |
nM |
12444694 |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
4800 |
nM |
14510605 |
NPT3210 |
Individual Protein |
BMP-2-inducible protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
12662110 |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
103 |
% |
22552195 |
NPT3255 |
Individual Protein |
Myosin light chain kinase family member 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15711537 |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15711537 |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
99 |
% |
18183025 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
= |
120 |
nM |
18183025 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
67 |
% |
18183025 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
28 |
% |
17850214 |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
27 |
% |
18183025 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17850214 |
NPT3281 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10998351 |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
= |
3200 |
nM |
PubChem BioAssay data set |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
121 |
% |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
19952.6 |
nM |
22831798 |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
23398362 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
2310 |
nM |
23398362 |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
80 |
% |
23398362 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
23398362 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT3348 |
Individual Protein |
NUAK family SNF1-like kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23398362 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
169.71 |
% |
23398362 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
91.14 |
% |
23398362 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
160.87 |
% |
23398362 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
151.97 |
% |
23398362 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29092.9 |
nM |
23398362 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
127 |
% |
23398362 |
NPT1417 |
Individual Protein |
Transcriptional regulator ERG |
Homo sapiens |
Potency |
|
50118.7 |
nM |
23398362 |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
96 |
% |
24930833 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
83 |
% |
18077363 |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
10.1016/0960-894X(95)00257-T |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
113 |
% |
13678412 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
AC50 |
= |
5011.87 |
nM |
19943624 |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Activity |
= |
94 |
% |
15270558 |
NPT3258 |
Individual Protein |
Mixed lineage kinase 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15270558 |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
109 |
% |
18177012 |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
105 |
% |
22429052 |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Activity |
= |
95 |
% |
19514743 |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
83 |
% |
20493686 |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
108 |
% |
12617583 |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
110 |
% |
10978207 |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25237727 |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Potency |
|
17290.6 |
nM |
25237727 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
46 |
% |
25763602 |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
10924166 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
8.66 |
nM |
16203143 |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
1431942 |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
76 |
% |
15217282 |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
= |
63095.7 |
nM |
18281952 |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
104 |
% |
12880316 |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
86 |
% |
8904842 |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
170 |
nM |
21741249 |
NPT3360 |
Individual Protein |
Tubulin alpha-1 chain |
Rattus norvegicus |
Kd |
= |
4900 |
nM |
12182864 |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
97 |
% |
15921436 |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
= |
350 |
nM |
20598551 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
21856049 |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
10978206 |
NPT3298 |
Individual Protein |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
Kd |
> |
10000 |
nM |
25275213 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
18348535 |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
6513.1 |
nM |
16724845 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
= |
32 |
nM |
25124114 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
112 |
% |
8691207 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Ki |
= |
251.19 |
nM |
24460410 |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
13678412 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
13678412 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
24460410 |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
113 |
% |
8691203 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Activity |
= |
83 |
% |
8691203 |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
8691203 |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
8691203 |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Kd |
> |
10000 |
nM |
20634065 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
75 |
% |
PubChem BioAssay data set |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
122 |
% |
22652254 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
1122 |
nM |
12662101 |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
12880316 |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
PubChem BioAssay data set |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
9722490 |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Activity |
= |
103 |
% |
16562846 |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
92 |
% |
24328302 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
15497961 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
91 |
% |
20363129 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Inhibition |
= |
93 |
% |
20363129 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
100 |
nM |
26327273 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
50 |
nM |
26327273 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Inhibition |
= |
95 |
% |
23356964 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Inhibition |
= |
37 |
% |
23356964 |
NPT3289 |
Individual Protein |
Serine/threonine-protein kinase RIO3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25739048 |
NPT3362 |
Individual Protein |
Mitogen-activated protein kinase 7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19904995 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Activity |
= |
98 |
% |
17618015 |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Activity |
= |
109 |
% |
10.3390/70200112 |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
81 |
% |
20189813 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
15387645 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
91 |
% |
22264170 |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
22264170 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
22901896 |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
24 |
% |
14695791 |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
22472691 |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Kd |
> |
10000 |
nM |
1593279 |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
63095.7 |
nM |
23830699 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
11975483 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
-1 |
% |
15787428 |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Activity |
= |
97 |
% |
19344127 |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
23327905 |
NPT3300 |
Individual Protein |
Serine/threonine-protein kinase 32B |
Homo sapiens |
Kd |
= |
4900 |
nM |
22834923 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Activity |
= |
65 |
% |
25856683 |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757713 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
70.2 |
% |
2869146 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
67 |
% |
16510283 |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
17407813 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
20185316 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
20185316 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
12589.25 |
nM |
20185316 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
20185316 |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
108 |
% |
PubChem BioAssay data set |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
21495717 |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Kd |
= |
9600 |
nM |
PubChem BioAssay data set |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
Residual Activity |
= |
101 |
% |
DrugMatrix in vitro pharmacology data |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
44 |
% |
DrugMatrix in vitro pharmacology data |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Activity |
= |
92 |
% |
DrugMatrix in vitro pharmacology data |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
109 |
% |
DrugMatrix in vitro pharmacology data |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
115 |
% |
23964704 |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
14640511 |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
109 |
% |
19874044 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Activity |
= |
89 |
% |
10.1016/0960-894X(96)00418-0 |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
97 |
% |
19947605 |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
93 |
% |
20558071 |
NPT2816 |
Individual Protein |
Bromodomain-containing protein 4 |
Homo sapiens |
IC50 |
= |
2500 |
nM |
18411318 |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
20145081 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
18411316 |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
109 |
% |
18426954 |
NPT3261 |
Individual Protein |
cAMP-dependent protein kinase beta-1 catalytic subunit |
Homo sapiens |
Kd |
= |
530 |
nM |
19075048 |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
19114678 |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Kd |
> |
10000 |
nM |
19114678 |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
Activity |
= |
30 |
day |
19114678 |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
106 |
% |
19114678 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
= |
42 |
nM |
19114678 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
90 |
% |
19273669 |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19273669 |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
80 |
% |
19721064 |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Kd |
= |
4200 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
DrugMatrix in vitro pharmacology data |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
15646539 |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
12852755 |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
59 |
% |
16213713 |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16539393 |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
17438052 |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
17488817 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Activity |
= |
87 |
% |
17438047 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18524583 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
95 |
% |
19457674 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1598 |
Individual Protein |
Casein kinase II alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
100 |
% |
DrugMatrix in vitro pharmacology data |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
= |
3100 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9200 |
nM |
22194678 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
98 |
% |
22352809 |
NPT3278 |
Individual Protein |
LIM domain kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22858097 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Kd |
> |
10000 |
nM |
22533850 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
95 |
% |
23434030 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
AC50 |
= |
501.19 |
nM |
24177359 |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
25847765 |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
68 |
% |
12036347 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
127 |
% |
15711537 |
NPT3345 |
Individual Protein |
Cyclin-dependent kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17064068 |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
17064068 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
100 |
nM |
19128055 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
50 |
nM |
19128055 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
26 |
% |
19128055 |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Kd |
> |
10000 |
nM |
19128055 |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
19128055 |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Activity |
= |
93 |
% |
19128055 |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
87 |
% |
19128055 |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
18183025 |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
97 |
% |
18183025 |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15958589 |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Kd |
> |
10000 |
nM |
21417417 |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Kd |
> |
10000 |
nM |
21944287 |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
843.7 |
nM |
21982796 |
NPT3341 |
Individual Protein |
Serine/threonine-protein kinase Nek5 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21982796 |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
88 |
% |
21982796 |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
105 |
% |
10.6019/CHEMBL1201861 |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
58 |
% |
10.6019/CHEMBL1201861 |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
111 |
% |
10.6019/CHEMBL1201861 |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
10.6019/CHEMBL1201861 |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Kd |
> |
10000 |
nM |
10.6019/CHEMBL1201861 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
66 |
% |
10.6019/CHEMBL1201861 |
NPT3361 |
Individual Protein |
Mitogen-activated protein kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23829517 |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
8 |
% |
23829517 |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18077363 |
NPT3343 |
Individual Protein |
Uncharacterized aarF domain-containing protein kinase 4 |
Homo sapiens |
Kd |
= |
4900 |
nM |
18077363 |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
69 |
% |
26142492 |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
7307.8 |
nM |
4032421 |
NPT1814 |
Individual Protein |
Glucagon receptor |
Homo sapiens |
IC50 |
= |
80.17 |
nM |
16472241 |
NPT3288 |
Individual Protein |
Interleukin-1 receptor-associated kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3228 |
Individual Protein |
Adaptor-associated kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
123 |
% |
DrugMatrix in vivo data: Hematology |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
53 |
% |
10.6019/CHEMBL3433997 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
94 |
% |
11784156 |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
43 |
% |
26331426 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8450319 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
108 |
% |
15921415 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Activity |
= |
61 |
% |
19105653 |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
51 |
% |
22686608 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
21873059 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
98 |
% |
14611848 |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18288806 |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000 |
nM |
10757708 |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
10691710 |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
20050684 |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
91 |
% |
21982797 |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24216090 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
= |
3300 |
nM |
18989978 |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
84 |
% |
1294697 |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19778068 |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23451797 |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
24099364 |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
104 |
% |
11908979 |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
15026054 |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
115 |
% |
15043420 |
NPT8 |
Individual Protein |
DNA polymerase iota |
Homo sapiens |
Potency |
|
1584.9 |
nM |
15332845 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
12 |
% |
16933872 |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
78 |
% |
16933872 |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
16038541 |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
86 |
% |
PubChem BioAssay data set |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
8786369 |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
0 |
% |
13678412 |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
40 |
% |
13678412 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
14.3 |
nM |
16134928 |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
122 |
% |
6834379 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
3339605 |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
74 |
% |
17513021 |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
118 |
% |
17938185 |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
100 |
% |
17938185 |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19805556 |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Activity |
= |
42 |
% |
20667728 |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
20100877 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
36.8 |
% |
20100877 |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
18694944 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
18955522 |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
= |
6000 |
nM |
18955522 |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19223615 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Activity |
= |
70 |
% |
19223615 |
NPT3325 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Gallus gallus |
Kd |
> |
10000 |
nM |
19223615 |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
49 |
% |
19223615 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
8912.5 |
nM |
19223619 |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
121 |
% |
19528279 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
163.6 |
nM |
19528279 |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19581457 |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
118 |
% |
19581457 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
123 |
% |
19581457 |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
105 |
% |
19581457 |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
100 |
% |
19581457 |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
106 |
% |
18625771 |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20625154 |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
-1 |
% |
16472241 |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
108 |
% |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
96 |
% |
DrugMatrix in vitro pharmacology data |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
22194678 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Kd |
= |
2700 |
nM |
22691154 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
210 |
nM |
22217866 |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
10.1007/s00044-012-0429-8 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23644202 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
77 |
% |
DrugMatrix in vivo data: Hematology |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
112 |
% |
23571415 |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
110 |
% |
24513185 |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
= |
6800 |
nM |
24530492 |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
15646539 |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
25801157 |
NPT3233 |
Individual Protein |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
Kd |
> |
10000 |
nM |
18973388 |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
90 |
% |
18494522 |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
18387711 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
AC50 |
= |
15848.93 |
nM |
18611050 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2600 |
nM |
10560729 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5011.9 |
nM |
19425589 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20155971 |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
113 |
% |
19591451 |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
18715034 |
NPT1671 |
Individual Protein |
AMP-activated protein kinase, alpha-2 subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
23985009 |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Residual Activity |
= |
77 |
% |
23977995 |
NPT3339 |
Individual Protein |
Myosin-IIIB |
Homo sapiens |
Kd |
> |
10000 |
nM |
12762791 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1700 |
nM |
19783432 |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14640515 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
4.55 |
% |
19425589 |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
106 |
% |
19425589 |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
26 |
% |
12880304 |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
19193025 |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Residual Activity |
= |
98 |
% |
18610999 |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
124 |
% |
16971124 |
NPT4094 |
Individual Protein |
Serine/threonine-protein kinase WNK3 |
Homo sapiens |
Residual Activity |
= |
75 |
% |
15921404 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
7 |
% |
15921404 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
19658408 |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
16933872 |
NPT3257 |
Individual Protein |
Serine/threonine-protein kinase 32C |
Homo sapiens |
Kd |
> |
10000 |
nM |
20619938 |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
8350094 |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19489596 |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
19489596 |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
105 |
% |
17618015 |
NPT443 |
Individual Protein |
Histone acetyltransferase GCN5 |
Homo sapiens |
Potency |
|
631 |
nM |
12502331 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Activity |
= |
73 |
% |
21084196 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
300 |
nM |
12662097 |
NPT486 |
Organism |
Toxoplasma gondii |
Toxoplasma gondii |
IC50 |
= |
1000 |
nM |
12662097 |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
IC50 |
= |
5000 |
nM |
12662097 |
NPT4094 |
Individual Protein |
Serine/threonine-protein kinase WNK3 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
20932756 |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
16643037 |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
43 |
% |
17993275 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Potency |
= |
5011.9 |
nM |
11473423 |
NPT3251 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
25899335 |
NPT796 |
Individual Protein |
Peripheral myelin protein 22 |
Homo sapiens |
Potency |
= |
26854.5 |
nM |
8229009 |
NPT3304 |
Individual Protein |
Serine/threonine-protein kinase receptor R3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21420296 |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
112 |
% |
24613627 |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
= |
3800 |
nM |
21155593 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Inhibition |
= |
88 |
% |
10650082 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
66 |
% |
10579864 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Inhibition |
= |
92 |
% |
10579864 |
NPT1443 |
Individual Protein |
Pyruvate dehydrogenase kinase isoform 1 |
Homo sapiens |
Inhibition |
= |
87 |
% |
10579864 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Inhibition |
= |
53 |
% |
10579864 |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Inhibition |
= |
98 |
% |
16499330 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Inhibition |
= |
75 |
% |
15787444 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Inhibition |
= |
61 |
% |
15787444 |
NPT1610 |
Individual Protein |
Rho-associated protein kinase 2 |
Rattus norvegicus |
Inhibition |
= |
61 |
% |
15787444 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
94 |
% |
15787444 |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
122 |
% |
18579374 |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Ki |
= |
794.33 |
nM |
23394318 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
45 |
% |
18288809 |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Activity |
= |
99 |
% |
10869195 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
111 |
% |
23489626 |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
112 |
% |
12662097 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
125892.5 |
nM |
3965717 |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
44668.4 |
nM |
19388705 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
18327911 |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17892263 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
95 |
% |
18977148 |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Activity |
= |
106 |
% |
25646964 |
NPT3265 |
Individual Protein |
Casein kinase I isoform alpha-like |
Homo sapiens |
Kd |
= |
1900 |
nM |
15497933 |
NPT3314 |
Individual Protein |
Bone morphogenetic protein receptor type-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15497933 |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Kd |
> |
10000 |
nM |
21419633 |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
91 |
% |
11908979 |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
11908979 |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Activity |
= |
70 |
% |
11908979 |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Kd |
> |
10000 |
nM |
11908979 |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
11374948 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
19 |
% |
17604394 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Activity |
= |
87 |
% |
20923180 |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Kd |
> |
10000 |
nM |
19105653 |
NPT3256 |
Individual Protein |
Serine/threonine-protein kinase WEE1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22206869 |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
18557621 |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
= |
53 |
nM |
22250891 |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
109 |
% |
8277314 |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
41 |
% |
PubChem BioAssay data set |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18440233 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5011.9 |
nM |
PubChem BioAssay data set |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
24479418 |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
92 |
% |
17822299 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
18288806 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
3548.1 |
nM |
15104514 |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Kd |
> |
10000 |
nM |
23434420 |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24417634 |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
95 |
% |
24417634 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Activity |
= |
49 |
% |
12398531 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
55 |
% |
18336005 |
NPT3368 |
Individual Protein |
cGMP-dependent protein kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15711537 |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
18578517 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Activity |
= |
89 |
% |
18183025 |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Activity |
= |
93 |
% |
18183025 |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Residual Activity |
= |
104 |
% |
18183025 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
18183025 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Activity |
= |
82 |
% |
18183025 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
107 |
% |
22037378 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
14125.4 |
nM |
22037378 |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
22037378 |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
22037378 |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
124 |
% |
22037378 |
NPT3313 |
Individual Protein |
Bone morphogenetic protein receptor type-1A |
Homo sapiens |
Kd |
> |
10000 |
nM |
22037378 |
NPT3337 |
Individual Protein |
Serine/threonine-protein kinase DCLK3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
DrugMatrix in vitro pharmacology data |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
16000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Kd |
= |
28 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
72 |
% |
DrugMatrix in vitro pharmacology data |
NPT3297 |
Individual Protein |
Non-receptor tyrosine-protein kinase TNK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
23398362 |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
76 |
% |
23398362 |
NPT58 |
Individual Protein |
Bloom syndrome protein |
Homo sapiens |
Potency |
= |
50118.7 |
nM |
23398362 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
23398362 |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
49 |
% |
23398362 |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
18077363 |
NPT4095 |
Protein Complex |
Mammalian target of Rapamycin (mTORC1) |
Homo sapiens |
Residual Activity |
= |
90 |
% |
18077363 |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
22703163 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
25700232 |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Kd |
> |
10000 |
nM |
25700232 |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
15848.93 |
nM |
25700232 |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Activity |
= |
76 |
% |
10425121 |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Kd |
> |
10000 |
nM |
10425121 |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24035339 |
NPT794 |
Individual Protein |
Endonuclease 4 |
Escherichia coli K-12 |
Potency |
= |
25118.9 |
nM |
24900585 |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
20575572 |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
14125.4 |
nM |
22409377 |
NPT3224 |
Individual Protein |
Phosphorylase kinase gamma subunit 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22409377 |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Activity |
= |
113 |
% |
18321710 |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
29081 |
nM |
17320402 |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
19691309 |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Kd |
> |
10000 |
nM |
14640511 |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
20 |
% |
21090801 |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
11170656 |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
9599274 |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
19952.6 |
nM |
24725159 |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
Residual Activity |
= |
92 |
% |
15787464 |
NPT3307 |
Individual Protein |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18694644 |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
12 |
% |
22500574 |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22500574 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
26000707 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
79 |
% |
10.1016/S0960-894X(01)81072-6 |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
106 |
% |
12105963 |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
109 |
% |
19117486 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
99 |
% |
19022675 |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
66 |
% |
16643023 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
88 |
% |
PubChem BioAssay data set |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
= |
650 |
nM |
22280363 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19715320 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
22748705 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Kd |
> |
10000 |
nM |
11087594 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
98 |
% |
23327905 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20540535 |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
16643037 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
10417.9 |
nM |
23013292 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
113 |
% |
23013292 |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
106 |
% |
22304344 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
74 |
% |
23376010 |
NPT3321 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
8158164 |
NPT1717 |
Individual Protein |
Serine/threonine-protein kinase 25 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11908966 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
72 |
% |
20735051 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Activity |
= |
84 |
% |
22245048 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
92 |
% |
11262075 |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
794.3 |
nM |
23350733 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Activity |
= |
91 |
% |
23350733 |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Kd |
> |
10000 |
nM |
22758788 |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Activity |
= |
86 |
% |
PubChem BioAssay data set |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Activity |
= |
84 |
% |
PubChem BioAssay data set |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
10096852 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Inhibition |
= |
63 |
% |
PubChem BioAssay data set |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
PubChem BioAssay data set |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
16180824 |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
23190013 |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
9873651 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
25 |
% |
25871540 |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
109 |
% |
16562826 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
108 |
% |
PubChem BioAssay data set |
NPT3308 |
Individual Protein |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
Kd |
= |
1700 |
nM |
PubChem BioAssay data set |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
69 |
% |
24963714 |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
19739600 |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18640035 |
NPT3243 |
Individual Protein |
myosin light chain kinase 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18640035 |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
113 |
% |
25894905 |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
69 |
% |
26000707 |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18288805 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Residual Activity |
= |
42 |
% |
24617951 |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20934335 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20923180 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
105.85 |
% |
12398531 |
NPT3301 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19072209 |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
41 |
% |
22206869 |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
14125.4 |
nM |
10.1039/C3MD00097D |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
PubChem BioAssay data set |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
24499261 |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
58 |
% |
24491225 |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Kd |
> |
10000 |
nM |
22850207 |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Residual Activity |
= |
97 |
% |
18729518 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
1336040 |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
22230050 |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Residual Activity |
= |
102 |
% |
15509169 |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
117 |
% |
3373220 |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22100311 |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
17782.8 |
nM |
25856683 |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11575963 |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
119 |
% |
18558743 |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
8984155 |
NPT1656 |
Individual Protein |
Protein kinase N1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20797856 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
101 |
% |
7130986 |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
88 |
% |
PubChem BioAssay data set |
NPT1692 |
Individual Protein |
Mitogen-activated protein kinase 6 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11975483 |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000 |
nM |
11975483 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
112 |
% |
PubChem BioAssay data set |
NPT3813 |
Individual Protein |
Tyrosine-protein kinase SRC |
Gallus gallus |
Activity |
= |
79 |
% |
17253849 |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
120 |
% |
19200744 |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
65 |
% |
9917310 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
31622.8 |
nM |
12141856 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Residual Activity |
= |
107 |
% |
9548870 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
12141874 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Activity |
= |
104 |
% |
23006147 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Ki |
= |
1000 |
nM |
23647487 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
24467317 |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
PubChem BioAssay data set |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
620 |
nM |
23022281 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
26147490 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
21824777 |
NPT183 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Rattus norvegicus |
Inhibition |
= |
68 |
% |
24175613 |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Ki |
= |
2511.89 |
nM |
20429578 |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Kd |
> |
10000 |
nM |
19746919 |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
19746919 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Activity |
= |
85 |
% |
20624681 |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Kd |
> |
10000 |
nM |
10654420 |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Kd |
> |
10000 |
nM |
24601675 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
1000 |
nM |
23701597 |
NPT3264 |
Individual Protein |
Serine/threonine-protein kinase RIO1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
22512738 |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
109 |
% |
23265253 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
25730346 |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
87 |
% |
PubChem BioAssay data set |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
111 |
% |
19848432 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6513.1 |
nM |
22209732 |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
83 |
% |
9358640 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14575 |
nM |
21865038 |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
18543965 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
-1 |
% |
19572738 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
IC50 |
= |
188 |
nM |
25798528 |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17547458 |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
107 |
% |
19762244 |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Kd |
= |
1600 |
nM |
15125956 |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Kd |
> |
10000 |
nM |
2016726 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29092.9 |
nM |
16949283 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Inhibition |
= |
87.2 |
% |
17194835 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Activity |
= |
81.4 |
% |
17261619 |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
108 |
% |
17261619 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
17189664 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Activity |
= |
90 |
% |
17337097 |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
17553680 |
NPT3302 |
Individual Protein |
Ankyrin repeat and protein kinase domain-containing protein 1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17724159 |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
17967918 |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
14 |
% |
19700225 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
20430485 |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
86 |
% |
19884373 |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
98 |
% |
18285488 |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
20368405 |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
10000 |
nM |
18809939 |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
92 |
% |
18809945 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Inhibition |
= |
89 |
% |
18838584 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Inhibition |
= |
3 |
% |
18710917 |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Inhibition |
= |
80 |
% |
18710917 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Inhibition |
= |
93 |
% |
18710917 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
0 |
% |
18710917 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
97 |
% |
18710917 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Inhibition |
= |
88 |
% |
18710917 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Inhibition |
= |
87 |
% |
18710917 |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000 |
nM |
18710917 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
110 |
% |
18710917 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8210 |
nM |
18725438 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
85 |
% |
18725450 |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
18474583 |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Kd |
> |
10000 |
nM |
18299417 |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
19104019 |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
65 |
% |
21049906 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
114 |
% |
19651906 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Activity |
= |
21 |
% |
19651906 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Activity |
= |
86 |
% |
19651906 |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Kd |
> |
10000 |
nM |
19721071 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
23109.3 |
nM |
20547809 |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
41 |
% |
19487444 |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
55 |
% |
18591275 |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Activity |
= |
0 |
% |
18625769 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
90 |
% |
18625769 |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
43 |
% |
18625769 |
NPT3253 |
Individual Protein |
Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha |
Homo sapiens |
Kd |
> |
10000 |
nM |
20625154 |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
32 |
% |
20713672 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Kd |
> |
10000 |
nM |
20805391 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Kd |
> |
10000 |
nM |
20014752 |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Activity |
= |
102 |
% |
21440339 |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Kd |
> |
10000 |
nM |
21981980 |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
81 |
% |
DrugMatrix in vitro pharmacology data |
NPT1814 |
Individual Protein |
Glucagon receptor |
Homo sapiens |
Inhibition |
< |
20 |
% |
DrugMatrix in vitro pharmacology data |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
80 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Kd |
> |
10000 |
nM |
DrugMatrix in vitro pharmacology data |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
85 |
% |
DrugMatrix in vitro pharmacology data |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
10.1007/s00044-012-0011-4 |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
10.1007/s00044-012-0202-z |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Activity |
= |
107 |
% |
23228471 |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Residual Activity |
= |
94 |
% |
23357308 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
117 |
% |
23454532 |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Kd |
> |
10000 |
nM |
23973821 |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
10.1007/s00044-013-0790-2 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
9.8 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
84 |
% |
Open TG-GATES in vivo data: Hematology |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
3548133.9 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
= |
150 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3448 |
Individual Protein |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
Open TG-GATES in vivo data: Organ Weight |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
= |
1600 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
24927053 |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
26034885 |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
103 |
% |
26214729 |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
115 |
% |
25682561 |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
59 |
% |
23691978 |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
54 |
% |
23571415 |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
18280170 |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
23127886 |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
99 |
% |
22071302 |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Residual Activity |
= |
95 |
% |
20614907 |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Ki |
= |
2511.89 |
nM |
10691716 |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
17190454 |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
14738381 |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
105 |
% |
19879673 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Inhibition |
= |
93.4 |
% |
24963714 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
19450986 |
NPT3350 |
Individual Protein |
Tyrosine-protein kinase Srms |
Homo sapiens |
Kd |
> |
10000 |
nM |
22148475 |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
17698848 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
113 |
% |
9868168 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1100 |
nM |
25856683 |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
25856683 |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
98 |
% |
25856683 |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15387655 |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
93 |
% |
14695799 |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
49 |
% |
21856049 |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
83 |
% |
10617079 |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Kd |
> |
10000 |
nM |
9868148 |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
50 |
nM |
12617583 |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Residual Activity |
= |
90 |
% |
19318121 |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
108 |
% |
15921421 |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
1 |
% |
26295595 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
12589.25 |
nM |
25322455 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
7943.28 |
nM |
25322455 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
25322455 |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
400 |
nM |
22834923 |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
61 |
% |
26231157 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
88 |
% |
11858756 |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
121 |
% |
11858756 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Kd |
> |
10000 |
nM |
15387642 |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
15332856 |
NPT3241 |
Individual Protein |
Serine/threonine-protein kinase NEK9 |
Homo sapiens |
Kd |
> |
10000 |
nM |
9917295 |
NPT3230 |
Individual Protein |
Serine/threonine-protein kinase 17B |
Homo sapiens |
Kd |
> |
10000 |
nM |
19835393 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
8063 |
nM |
7097296 |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
17844994 |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Kd |
> |
10000 |
nM |
17844994 |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
101 |
% |
23964704 |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
107 |
% |
22209731 |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
19689125 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
1000 |
nM |
23013356 |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
= |
790 |
nM |
25856683 |