Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
30 |
nM |
12182872 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
50 |
% |
15177438 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
25 |
% |
8676340 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
TD50 |
= |
0.01 |
ug/ml |
8676340 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
32 |
nM |
10346933 |
NPT313 |
Cell Line |
P388CPT5 |
Mus musculus |
IC50 |
= |
2800 |
nM |
10346933 |
NPT4451 |
Individual Protein |
DNA topoisomerase I |
Mus musculus |
MIC |
= |
86 |
nM |
10346933 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
87.5 |
|
10346933 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
700 |
nM |
7707314 |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
24 |
nM |
9876111 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
57 |
nM |
9876111 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
57 |
nM |
9876111 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3.1 |
nM |
9876111 |
NPT604 |
Individual Protein |
Serum albumin |
Homo sapiens |
Activity |
= |
1.8 |
|
8289200 |
NPT604 |
Individual Protein |
Serum albumin |
Homo sapiens |
Activity |
= |
2.3 |
|
8289200 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ID50 |
< |
3.2 |
ug/ml |
12161136 |
NPT2046 |
Cell Line |
EVSA-T |
Homo sapiens |
ID50 |
< |
3.2 |
ug/ml |
12161136 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
ID50 |
< |
3.2 |
ug/ml |
12161136 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
ID50 |
< |
3.2 |
ug/ml |
12161136 |
NPT573 |
Cell Line |
M19-MEL |
Homo sapiens |
ID50 |
< |
0.013 |
ug/ml |
12161136 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ID50 |
< |
3.2 |
ug/ml |
12161136 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
ID50 |
< |
0.005 |
ug/ml |
12161136 |
NPT4452 |
Cell Line |
CCD 19Lu |
Homo sapiens |
IC50 |
= |
2 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.005 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT4453 |
Cell Line |
Lu-99 cell line |
|
IC50 |
= |
0.001 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.005 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
679 |
nM |
7853331 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
46 |
nM |
7853331 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
48 |
nM |
7853331 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
207 |
nM |
7853331 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
37 |
nM |
7853331 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
= |
41 |
nM |
7853331 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.00474 |
ug/ml |
9632364 |
NPT4454 |
Cell Line |
HOC-21 cell line |
|
IC50 |
= |
0.0147 |
ug/ml |
9632364 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
0.00463 |
ug/ml |
9632364 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Ratio |
= |
0.39 |
|
9632364 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
7 |
nM |
12565975 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
4.9 |
% |
12565975 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
12639541 |
NPT4455 |
Cell Line |
CAKI-2 |
Homo sapiens |
IC50 |
= |
3960 |
nM |
12639541 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2530 |
nM |
12639541 |
NPT4456 |
Cell Line |
HEC-1B cell line |
|
IC50 |
= |
8640 |
nM |
12639541 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
66 |
nM |
12639541 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
CC50 |
= |
820 |
nM |
1846923 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
23 |
nM |
1846923 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
127000 |
nM |
7699697 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
18 |
% |
15080977 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
19 |
% |
15080977 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
10 |
% |
15080977 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
78 |
% |
15080977 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
68 |
% |
15080977 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Inhibition |
= |
40 |
% |
15080977 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Inhibition |
= |
76 |
% |
2155323 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Inhibition |
= |
85 |
% |
2155323 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
0.02 |
ug/ml |
2155323 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
0.08 |
ug/ml |
2155323 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
> |
100000 |
nM |
9767632 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
CC50 |
= |
10 |
nM |
9767632 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
CC50 |
= |
6 |
nM |
9767632 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
9 |
nM |
14552770 |
NPT4457 |
Cell Line |
KB VCR R |
|
IC50 |
= |
9 |
nM |
14552770 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7 |
nM |
14552770 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8 |
nM |
14552770 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
7 |
nM |
14552770 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
7 |
nM |
14552770 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1016/0960-894X(95)00360-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
330000 |
nM |
10576688 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
14000000 |
nM |
10576688 |
NPT4456 |
Cell Line |
HEC-1B cell line |
|
IC50 |
= |
60 |
nM |
10576688 |
NPT4458 |
Cell Line |
Caov-3 cell line |
|
IC50 |
= |
2900000 |
nM |
10576688 |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
46000000 |
nM |
10576688 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Therapeutic index |
= |
8 |
|
7381856 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
2 |
ug/ml |
7381856 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Inhibition |
= |
100 |
% |
10.1016/0960-894X(94)00462-O |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
40 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
70 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
30 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
35 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1040 |
nM |
10411476 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
330 |
nM |
12873503 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
0.77 |
|
12873503 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
17 |
nM |
11334569 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14 |
nM |
11334569 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
17 |
nM |
11334569 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
11334569 |
NPT2058 |
Cell Line |
NCI-H128 |
Homo sapiens |
IC50 |
= |
18 |
nM |
11334569 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
11334569 |
NPT4451 |
Individual Protein |
DNA topoisomerase I |
Mus musculus |
IC50 |
= |
40000 |
nM |
11334569 |
NPT204 |
Individual Protein |
Acetylcholinesterase |
Homo sapiens |
Inhibition |
= |
23 |
% |
11334569 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.00474 |
ug/ml |
7932525 |
NPT4454 |
Cell Line |
HOC-21 cell line |
|
IC50 |
= |
0.0147 |
ug/ml |
7932525 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
0.00463 |
ug/ml |
7932525 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
15 |
nM |
11052802 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
375 |
nM |
11052802 |
NPT3804 |
Cell Line |
Human Tumor Cell lines |
|
GI50 |
= |
44 |
nM |
11052802 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
5 |
nM |
10.1016/S0960-894X(97)10181-0 |
NPT4459 |
Cell Line |
833K |
|
IC50 |
= |
10 |
nM |
10.1016/S0960-894X(97)10181-0 |
NPT2786 |
Cell Line |
DC3F |
Cricetulus griseus |
IC50 |
= |
6 |
nM |
10.1016/S0960-894X(97)10181-0 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0.001 |
nM |
10.1016/S0960-894X(97)10181-0 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
80 |
nM |
10841808 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
67 |
nM |
10841808 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
88 |
nM |
10841808 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
11563925 |
NPT4460 |
Cell Line |
L2987 |
Homo sapiens |
IC50 |
= |
400 |
nM |
11755358 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
11020283 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
11020283 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
11020283 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
11020283 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
11020283 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
11020283 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
11020283 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
11020283 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
5.4 |
nM |
10479293 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8.5 |
nM |
10479293 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
6.3 |
nM |
10479293 |
NPT4462 |
Cell Line |
NCI-H928 |
|
IC50 |
= |
7.8 |
nM |
10479293 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1016/S0960-894X(01)80589-8 |
NPT1986 |
Cell Line |
RPMI 8402 |
Homo sapiens |
IC50 |
= |
5 |
nM |
12747798 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
61000 |
nM |
12747798 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
15 |
nM |
8246238 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
MIC |
= |
10 |
nM |
8246238 |
NPT322 |
Individual Protein |
DNA topoisomerase II beta |
Homo sapiens |
MIC |
> |
100000 |
nM |
8246238 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
13 |
nM |
12620081 |
NPT4264 |
Cell Line |
Lewis lung carcinoma cell line |
|
IC50 |
= |
33 |
nM |
12620081 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
5.6 |
nM |
12620081 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
2 |
|
12620081 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
1.4 |
|
12620081 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
33 |
nM |
9207945 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.6 |
nM |
9207945 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
13 |
nM |
11384245 |
NPT4463 |
Cell Line |
LL |
|
IC50 |
= |
33 |
nM |
11384245 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
5.6 |
nM |
11384245 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
680 |
nM |
8410981 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
10.1016/S0960-894X(01)80158-X |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
100 |
% |
10.1016/S0960-894X(01)80158-X |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT4457 |
Cell Line |
KB VCR R |
|
IC50 |
= |
0.03 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.09 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
10.1016/S0960-894X(01)80158-X |
NPT91 |
Cell Line |
KB |
Homo sapiens |
TD50 |
= |
0.008 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TD50 |
= |
0.006 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TD50 |
= |
0.01 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
TD50 |
= |
0.01 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT4464 |
Cell Line |
L1210/Adr |
Mus musculus |
TD50 |
= |
0.045 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
36 |
% |
10.1016/S0960-894X(97)00398-3 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
126 |
nM |
10.1016/S0960-894X(97)00398-3 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
600 |
nM |
15026047 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
ID50 |
= |
2.8 |
nM |
11965362 |
NPT4465 |
Cell Line |
HCT-116/VM46 |
Homo sapiens |
ID50 |
= |
2.4 |
nM |
11965362 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ID50 |
= |
3.8 |
nM |
11965362 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
ID50 |
= |
3.9 |
nM |
11965362 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
CC50 |
= |
800 |
nM |
2537428 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
14 |
nM |
2537428 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
5300 |
nM |
14667232 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
13 |
% |
8355258 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
< |
0.5 |
% |
8355258 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
< |
0.2 |
% |
8355258 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
1.8 |
|
8355258 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
2.3 |
|
8355258 |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
140 |
nM |
10.1016/0960-894X(96)00132-1 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
210 |
nM |
10.1016/0960-894X(96)00132-1 |
NPT4458 |
Cell Line |
Caov-3 cell line |
|
IC50 |
= |
30 |
nM |
10.1016/0960-894X(96)00132-1 |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
1170 |
nM |
10.1016/0960-894X(96)00132-1 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
180 |
nM |
10.1016/0960-894X(96)00132-1 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
700 |
nM |
9003520 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
51 |
nM |
9003520 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
= |
53 |
nM |
9003520 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
87.8 |
nM |
9003520 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
8 |
nM |
9003520 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
210 |
nM |
10.1016/0960-894X(96)00131-X |
NPT4458 |
Cell Line |
Caov-3 cell line |
|
IC50 |
= |
30 |
nM |
10.1016/0960-894X(96)00131-X |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
1170 |
nM |
10.1016/0960-894X(96)00131-X |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
180 |
nM |
10.1016/0960-894X(96)00131-X |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
140 |
nM |
10.1016/0960-894X(96)00131-X |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
60 |
nM |
15081041 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
320 |
nM |
15081041 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
310 |
nM |
15081041 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
330 |
nM |
11052801 |
NPT4466 |
Cell Line |
Panel (56 tumour cell lines) |
|
IC50 |
= |
40 |
nM |
10714502 |
NPT4467 |
Protein Family |
Somatostatin receptor |
Homo sapiens |
IC50 |
= |
2.21 |
nM |
12617894 |
NPT517 |
Cell Line |
Panel NCI-60 (60 carcinoma cell lines) |
Homo sapiens |
GI50 |
= |
10 |
nM |
15743190 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
< |
0.005 |
ug/ml |
15225719 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
< |
0.005 |
ug/ml |
15225719 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
2.72 |
ug/ml |
15225719 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
EC50 |
= |
350 |
nM |
15454230 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
117.2 |
nM |
15454230 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1414.4 |
nM |
15454230 |
NPT1986 |
Cell Line |
RPMI 8402 |
Homo sapiens |
IC50 |
= |
6 |
nM |
15482929 |
NPT1986 |
Cell Line |
RPMI 8402 |
Homo sapiens |
IC50 |
> |
10000 |
nM |
15482929 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
10 |
nM |
15482929 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
15482929 |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
IC50 |
= |
10 |
nM |
15482929 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
20 |
nM |
15482929 |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
IC50 |
= |
20 |
nM |
15482929 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
15509164 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
15509164 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
15509164 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
15509164 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
15509164 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
15509164 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
15509164 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
15509164 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
16033260 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
30 |
nM |
16033260 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
220 |
nM |
16033260 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
20 |
nM |
16033260 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
40 |
nM |
16033260 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
300 |
nM |
15801827 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
EC50 |
= |
1.2 |
nM |
15857116 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
EC50 |
= |
0.15 |
nM |
15857116 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.84 |
nM |
15916431 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5385 |
nM |
15916431 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
98.2 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
98 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
75.8 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
75 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
60.6 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
39.1 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
83.2 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
94.7 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
76.9 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
93.5 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
98.1 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
-0.4 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
49.5 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
62 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
-11.7 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
77 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
93.1 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
5.4 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
65.8 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
93.8 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
47.8 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
95.3 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
46 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
90.6 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
94.6 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
16.2 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
7.1 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
61.9 |
% |
16413779 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Inhibition |
= |
78.5 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
-1.9 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
7.5 |
% |
16413779 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Inhibition |
= |
33.4 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
-3.8 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
-7.1 |
% |
16413779 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
-3.2 |
% |
16413779 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16442283 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
16442283 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16442283 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16442283 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
16442283 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
16442283 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16442283 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
16442283 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
0.1 |
nM |
16686539 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
18 |
nM |
16686539 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
30 |
nM |
16686539 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
52 |
nM |
16686539 |
NPT3723 |
Cell Line |
CT26 |
Mus musculus |
IC50 |
= |
34 |
nM |
16686539 |
NPT4469 |
Cell Line |
Renca |
Mus musculus |
IC50 |
= |
304 |
nM |
16686539 |
NPT4471 |
Cell Line |
Panel (12 tumour cell lines) |
Homo sapiens |
IC70 |
= |
8.6 |
nM |
16621542 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
16913702 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16913702 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16913702 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
16913702 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
16913702 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16913702 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
16913702 |
NPT517 |
Cell Line |
Panel NCI-60 (60 carcinoma cell lines) |
Homo sapiens |
Activity |
= |
0.0405 |
nM |
16750365 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
16913702 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
69 |
% |
16971123 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17402722 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
17402722 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17402722 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17402722 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
17402722 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
17402722 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17402722 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
47 |
% |
17035025 |
NPT4472 |
Individual Protein |
DNA topoisomerase I |
Leishmania donovani donovani |
Inhibition |
= |
55 |
% |
17444624 |
NPT4472 |
Individual Protein |
DNA topoisomerase I |
Leishmania donovani donovani |
Inhibition |
= |
39 |
% |
17444624 |
NPT4472 |
Individual Protein |
DNA topoisomerase I |
Leishmania donovani donovani |
Inhibition |
= |
65 |
% |
17444624 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17411092 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
291 |
nM |
17204425 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
14 |
nM |
17204425 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
6 |
nM |
17204425 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
500 |
nM |
17547457 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
3.6 |
nM |
17552563 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
4 |
nM |
17254669 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
3 |
nM |
17254669 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
IC50 |
= |
5 |
nM |
17254669 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
3 |
nM |
17254669 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
17254669 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17254669 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17254669 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17254669 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17254669 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17254669 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
4.7 |
% |
17658776 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
9.5 |
% |
17658776 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
32.9 |
% |
17658776 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
43.1 |
% |
17658776 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17676830 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
17676830 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17676830 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17676830 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
17676830 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
17676830 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
17676830 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17696418 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17676830 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
17696418 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17696418 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17696418 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
17696418 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
17696418 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17696418 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
17696418 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
77 |
% |
17194596 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
EC50 |
= |
2.1 |
nM |
17287122 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
69 |
nM |
17498951 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
IC50 |
= |
45 |
nM |
17498951 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
98 |
nM |
17498951 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
80 |
nM |
17498951 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
18 |
nM |
17498951 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
32.1 |
nM |
17624792 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
680 |
nM |
17158054 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
32 |
nM |
17158054 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
15 |
nM |
17158054 |
NPT309 |
Cell Line |
1A9 |
Homo sapiens |
ED50 |
= |
3.2 |
nM |
17350834 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
6.9 |
nM |
17350834 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.2 |
nM |
17350834 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
2 |
nM |
17350834 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
16.7 |
nM |
17350834 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
ED50 |
= |
10.9 |
nM |
17350834 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
20.9 |
nM |
17350834 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
15 |
nM |
17350834 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
17418582 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
10 |
nM |
17418582 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
2 |
nM |
17418582 |
NPT4475 |
Cell Line |
CEM/C2 |
Homo sapiens |
GI50 |
> |
1000 |
nM |
17418582 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
30 |
nM |
17418582 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
20 |
nM |
17418582 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
67 |
nM |
17827007 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
80 |
nM |
17827007 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24 |
nM |
17827007 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
75 |
nM |
17827007 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
40 |
nM |
18076140 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
63.3 |
% |
18178085 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
84.1 |
% |
18178085 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
18178085 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
18178085 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1080 |
nM |
18178085 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
4160 |
nM |
18178085 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
13 |
nM |
18178085 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
1.7 |
nM |
17962028 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1.5 |
nM |
17962028 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
1.4 |
nM |
18061452 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
180 |
nM |
18180162 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
GI50 |
= |
6000 |
nM |
18180162 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
220 |
nM |
18180162 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
GI50 |
= |
23760 |
nM |
18180162 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
90 |
nM |
18180162 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
2800 |
nM |
18180162 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
> |
200000 |
nM |
18040043 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
3150 |
nM |
18095653 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
12500 |
nM |
18095653 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
9670 |
nM |
18095653 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3120 |
nM |
18095653 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
280 |
nM |
18095653 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
180 |
nM |
18424133 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
3160 |
nM |
18424133 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8810 |
nM |
18424133 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Ratio IC50 |
= |
2.8 |
|
18424133 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
0.2 |
|
18511275 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.004 |
nM |
18511275 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10 |
nM |
18511275 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.004 |
nM |
18511275 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
= |
0.16 |
ug/ml |
11000035 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
= |
0.014 |
ug/ml |
11000035 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
> |
100 |
ug/ml |
11000035 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
= |
0.18 |
ug/ml |
11000035 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
= |
0.06 |
ug/ml |
11000035 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
90 |
% |
10691712 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3000 |
nM |
11430001 |
NPT4476 |
Individual Protein |
DNA topoisomerase |
Bos taurus |
IC50 |
= |
17000 |
nM |
11430001 |
NPT4451 |
Individual Protein |
DNA topoisomerase I |
Mus musculus |
IC50 |
= |
12000 |
nM |
11430001 |
NPT4477 |
Individual Protein |
DNA topoisomerase 1 |
Chlorocebus aethiops |
IC50 |
= |
27000 |
nM |
11430001 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
4000 |
nM |
11430001 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
17000 |
nM |
11430001 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
9000 |
nM |
11430001 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
IC50 |
> |
300000 |
nM |
11430001 |
NPT908 |
Individual Protein |
Ribonuclease pancreatic |
Bos taurus |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4478 |
Individual Protein |
Deoxyribonuclease-1 |
Bos taurus |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4479 |
Individual Protein |
Deoxyribonuclease-2-alpha |
Sus scrofa |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4480 |
Individual Protein |
DNA ligase |
Enterobacteria phage T4 |
IC50 |
> |
300000 |
nM |
11430001 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
300000 |
nM |
11430001 |
NPT4481 |
Individual Protein |
Type-2 restriction enzyme BamHI |
Bacillus amyloliquefaciens |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4482 |
Individual Protein |
Type-2 restriction enzyme EcoRI |
Escherichia coli |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4483 |
Individual Protein |
Type-2 restriction enzyme HindIII |
Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4484 |
Individual Protein |
Type-2 restriction enzyme PstI |
Providencia stuartii |
IC50 |
> |
300000 |
nM |
11430001 |
NPT4485 |
Individual Protein |
Type-2 restriction enzyme ScaI |
Streptomyces caespitosus |
IC50 |
> |
300000 |
nM |
11430001 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
IC50 |
> |
300000 |
nM |
11430001 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
= |
110 |
ug/ml |
11678653 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
= |
0.6 |
ug/ml |
11678653 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
> |
20 |
ug/ml |
11678653 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4 |
nM |
17673337 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
14 |
nM |
17673337 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
165 |
nM |
17673337 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
83 |
nM |
17673337 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
18220355 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
ED50 |
= |
0.07 |
ug/ml |
18220355 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED50 |
= |
0.19 |
ug/ml |
18220355 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81.3 |
% |
18296054 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
9 |
nM |
18676151 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC10 |
= |
0.2 |
nM |
18676151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5 |
nM |
18676151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
61000 |
nM |
18676151 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
> |
10000 |
nM |
18676151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
18676151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25 |
nM |
18676151 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26 |
nM |
18676151 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
18774864 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.08 |
ug/ml |
18774864 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
0.07 |
ug/ml |
18774864 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.19 |
ug/ml |
18774864 |
NPT3749 |
Tissue |
Hippocampus |
Rattus norvegicus |
Activity |
= |
51.6 |
% |
18676148 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
0.2 |
|
19303306 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4 |
nM |
19303306 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
19303306 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
4 |
nM |
19303306 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
> |
10000 |
nM |
19303306 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
6 |
nM |
19012996 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
14 |
nM |
19012996 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.2 |
|
19012996 |
NPT26 |
Individual Protein |
Reverse transcriptase |
Human immunodeficiency virus 1 |
IC50 |
> |
200 |
ug/ml |
1710653 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
8.7 |
ug/ml |
10.1021/np50125a006 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.6 |
ug/ml |
10.1021/np50125a006 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.9 |
ug/ml |
8882430 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
100 |
ug/ml |
8882430 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
200 |
ug/ml |
15165164 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
5 |
ug/ml |
15165164 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
8759170 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
0.01 |
ug/ml |
15270571 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
ED50 |
= |
57 |
nM |
15043407 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
ED50 |
= |
258 |
nM |
15043407 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
22 |
nM |
15043407 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
28 |
nM |
15043407 |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
ED50 |
= |
29 |
nM |
15043407 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
230 |
nM |
15043407 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.6 |
ug/ml |
9514005 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
110 |
ug/ml |
9514005 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
0.054 |
ug/ml |
9514005 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
330 |
nM |
18419110 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
6.2 |
nM |
18419110 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
1650 |
nM |
18419110 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
12 |
nM |
18419110 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
3160 |
nM |
18419110 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8810 |
nM |
18419110 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
18841903 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
18841903 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
18841903 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
330 |
nM |
19530720 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
> |
0.01 |
nM |
19026551 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
> |
0.01 |
nM |
19026551 |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
ED50 |
> |
0.01 |
nM |
19026551 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
12 |
ug/ml |
14510601 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
75 |
ug/ml |
14510601 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.6 |
ug/ml |
8254347 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
110 |
ug/ml |
8254347 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
0.054 |
ug/ml |
8254347 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
0.01 |
ug/ml |
11858737 |
NPT4486 |
Cell Line |
LX-1 |
Homo sapiens |
IC50 |
= |
120 |
nM |
11858737 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
9 |
nM |
11858737 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
4 |
nM |
11858737 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
= |
8.7 |
ug/ml |
8158166 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
> |
20 |
ug/ml |
8158166 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Activity |
= |
0.6 |
ug/ml |
8158166 |
NPT141 |
Organism |
Agrobacterium tumefaciens |
Agrobacterium tumefaciens |
Activity |
= |
-100 |
% |
10.1021/np50107a012 |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
IC50 |
= |
28.7 |
nM |
11858760 |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
28.7 |
nM |
11858760 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
86.1 |
nM |
11858760 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
28.7 |
nM |
11858760 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28.7 |
nM |
11858760 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
2.3 |
ug/ml |
7130986 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.6 |
ug/ml |
8021652 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
8.7 |
ug/ml |
8021652 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
110 |
ug/ml |
8021652 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
0.02 |
ug/ml |
8021652 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
240 |
nM |
18554906 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3280 |
nM |
18554906 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
18554906 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
130 |
nM |
18554906 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10 |
nM |
18554906 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
200 |
nM |
18554906 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
170 |
nM |
18554906 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
90 |
nM |
18554906 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3 |
nM |
18554906 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6 |
nM |
18829334 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
18829334 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
14 |
nM |
18829334 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
0.072 |
ug/ml |
19328687 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
Activity |
= |
0.089 |
ug/ml |
19328687 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
Activity |
= |
0.035 |
ug/ml |
19328687 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
0.6 |
ug/ml |
1479381 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC12 |
= |
8.7 |
ug/ml |
1479381 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
1000000 |
nM |
15974606 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
20000 |
nM |
15974606 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
130000 |
nM |
15974606 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
= |
72 |
nM |
15730238 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
EC50 |
= |
6.9 |
nM |
15730238 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
EC50 |
= |
59 |
nM |
15730238 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
0.07 |
ug/ml |
16499333 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
18630891 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
18630891 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
18630891 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
18630891 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
18630891 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
18630891 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
18630891 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
18630891 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4 |
nM |
18771930 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
4 |
nM |
18771930 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
18771930 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25 |
nM |
18771930 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26 |
nM |
18771930 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
0.2 |
|
18771930 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
18771930 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
> |
10000 |
nM |
18771930 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Activity |
= |
61.4 |
% |
18313176 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Activity |
= |
28.4 |
% |
18313176 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Activity |
= |
19.4 |
% |
18313176 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Activity |
= |
14.6 |
% |
18313176 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Activity |
= |
3.8 |
% |
18313176 |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Activity |
= |
40.5 |
% |
18313176 |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Activity |
= |
24.5 |
% |
18313176 |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Activity |
= |
10.9 |
% |
18313176 |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Activity |
= |
5.3 |
% |
18313176 |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Activity |
= |
55.1 |
% |
18313176 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
Inhibition |
= |
15.4 |
% |
18313176 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
58 |
nM |
19345580 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
89 |
nM |
19345580 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
72 |
nM |
19345580 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
86.2 |
% |
19345580 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
40 |
nM |
19203291 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
100 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
34.6 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
18 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
15.5 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
28.4 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
17.5 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
23.6 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
10.3 |
% |
19203291 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Activity |
= |
21.7 |
% |
19203291 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
19256478 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
12500 |
nM |
19256478 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
9700 |
nM |
19256478 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
19256478 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19256478 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
800 |
nM |
19585998 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
47 |
nM |
19541483 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
120 |
nM |
19541483 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
40 |
nM |
19715319 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
30 |
nM |
19715319 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
GI50 |
= |
10 |
nM |
19715319 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19715319 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
80 |
nM |
19715319 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19715319 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
100 |
nM |
19715319 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
19715319 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
700 |
nM |
19715319 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19715319 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
600 |
nM |
19715319 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
19715319 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
200 |
nM |
19715319 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
400 |
nM |
19715319 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
20 |
nM |
19715319 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
19715319 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1700 |
nM |
19715319 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
40 |
nM |
19715319 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
19715319 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
60 |
nM |
19715319 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
19715319 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
44.8 |
% |
19715319 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
84 |
% |
19715319 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
0.023 |
nM |
19743858 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
43.21 |
nM |
19743858 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2 |
nM |
19655762 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3 |
nM |
19655762 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
3 |
nM |
19655762 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
6 |
nM |
19655762 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19655762 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
38 |
nM |
19655762 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
455 |
nM |
19655762 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4 |
nM |
19299037 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
4 |
nM |
19299037 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
0.2 |
|
19299037 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
19299037 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5.379 |
nM |
20063889 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
1900 |
nM |
19664930 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
GI50 |
= |
1700 |
nM |
19664930 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
1300 |
nM |
19664930 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
460 |
nM |
19664930 |
NPT1723 |
Cell Line |
HBL-100 |
Homo sapiens |
GI50 |
= |
230 |
nM |
19664930 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
GI50 |
= |
210 |
nM |
19664930 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19783447 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19783447 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19783447 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
19783447 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
19783447 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
19783447 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
19783447 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
19783447 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
69.4 |
% |
19800803 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
41 |
% |
19954977 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
54 |
% |
19954977 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1460 |
nM |
19954977 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7420 |
nM |
19954977 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2770 |
nM |
19954977 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
19954977 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1850 |
nM |
19954977 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
860 |
nM |
20093033 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
850 |
nM |
20093033 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
920 |
nM |
20093033 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
65 |
nM |
20093033 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3570 |
nM |
20093033 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
75.5 |
% |
20093033 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
78.3 |
% |
20093033 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
Inhibition |
= |
40 |
% |
20006518 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20155916 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20155916 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20155916 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20155916 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
20155916 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
20155916 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
40 |
nM |
20155916 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
20155916 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
940 |
nM |
20188578 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
630 |
nM |
20188578 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
0.05 |
% |
20188578 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
39.5 |
% |
20188578 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
75.3 |
% |
20188578 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
640 |
nM |
20188578 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
80 |
nM |
20188578 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
80 |
nM |
19939682 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
660 |
nM |
19939682 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
19939682 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
630 |
nM |
19939682 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
760 |
nM |
19939682 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
41.2 |
% |
19939682 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
79 |
% |
19939682 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
210 |
nM |
19916529 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
280 |
nM |
19916529 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.06 |
nM |
19839614 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
60 |
nM |
19863101 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1220 |
nM |
19653666 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1220 |
nM |
19653666 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1220 |
nM |
19653666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1220 |
nM |
19653666 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
130 |
nM |
19691293 |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
160 |
nM |
19691293 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
580 |
nM |
19836231 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1070 |
nM |
19836231 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
19836231 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
680 |
nM |
19836231 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
67 |
nM |
19836231 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
67.1 |
% |
19836231 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
84.5 |
% |
19836231 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
280 |
nM |
19453174 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19702283 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
20329739 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2 |
nM |
20329739 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
1000 |
nM |
20329739 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
EC50 |
= |
160 |
nM |
20192247 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
940 |
nM |
20356735 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
590 |
nM |
20356735 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
1300 |
nM |
20438092 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
210 |
nM |
20438092 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
280 |
nM |
20438092 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
2000 |
nM |
20438092 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
GI50 |
= |
150 |
nM |
20438092 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
68.8 |
% |
20392646 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
40.3 |
% |
20392646 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
300 |
nM |
20392646 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
400 |
nM |
20392646 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
400 |
nM |
20392646 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
500 |
nM |
20392646 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
100 |
nM |
20392646 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
FC |
= |
1 |
|
20392545 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
< |
13 |
nM |
20392545 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20392545 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
< |
13 |
nM |
20392545 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
33 |
% |
20591678 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
1 |
% |
20591678 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
Activity |
= |
25 |
% |
20591678 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
570 |
nM |
20591678 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
30 |
nM |
20591678 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
190 |
nM |
20591678 |
NPT1329 |
Cell Line |
Detroit 551 |
Homo sapiens |
GI50 |
= |
990 |
nM |
20591678 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
60 |
nM |
20591678 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2 |
nM |
20590148 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
20590148 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20630766 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
20630766 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20630766 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20630766 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
20630766 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
20630766 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20630766 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
20630766 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
EC50 |
= |
60 |
nM |
20825206 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
FC |
= |
0.258 |
|
16680159 |
NPT2 |
Others |
Unspecified |
|
LD50 |
= |
20 |
nM |
20655220 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
4200 |
nM |
20619511 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14200 |
nM |
20619511 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2300 |
nM |
20619511 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
20619511 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1100 |
nM |
20619511 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
25000 |
nM |
20638158 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
> |
25000 |
nM |
20638158 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
73 |
% |
20638158 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
2200 |
nM |
20662543 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
85 |
% |
20662543 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
GI50 |
= |
6000 |
nM |
20662543 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
2800 |
nM |
20662543 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1030 |
nM |
20662543 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
220 |
nM |
20662543 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
80 |
nM |
20662543 |
NPT1329 |
Cell Line |
Detroit 551 |
Homo sapiens |
GI50 |
= |
990 |
nM |
20662543 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
90 |
nM |
20662543 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0 |
% |
20662543 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
20662543 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.83 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1.41 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1.12 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1.32 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.89 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
0.56 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
794.33 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1258.93 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1000 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
501.19 |
nM |
19734910 |
NPT1021 |
Organism |
Leishmania infantum |
Leishmania infantum |
IC50 |
= |
34400 |
nM |
18644961 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
57 |
nM |
20942490 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
3100 |
nM |
20942490 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
710 |
nM |
20942490 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21044847 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
330 |
nM |
21044847 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
16240 |
nM |
21044847 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
67 |
nM |
21074444 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
700 |
nM |
21074444 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
80 |
nM |
21074444 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21074444 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21074444 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21074444 |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
1000 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
25.1 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
5.6 |
nM |
PubChem BioAssay data set |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
= |
4466.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
134 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
794.3 |
nM |
PubChem BioAssay data set |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
3548.1 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
4466.8 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT1197 |
Individual Protein |
Huntingtin |
Homo sapiens |
Potency |
= |
5623.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
316.2 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
5 |
nM |
PubChem BioAssay data set |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Potency |
= |
12995.3 |
nM |
PubChem BioAssay data set |
NPT536 |
Uncleic Acid |
microRNA 21 |
Homo sapiens |
Potency |
= |
104 |
nM |
PubChem BioAssay data set |
NPT537 |
Individual Protein |
Ras-related protein Rab-9A |
Homo sapiens |
Potency |
= |
398.1 |
nM |
PubChem BioAssay data set |
NPT537 |
Individual Protein |
Ras-related protein Rab-9A |
Homo sapiens |
Potency |
= |
46109.1 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
35.5 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
31.6 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
28.2 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Potency |
= |
104 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
44.7 |
nM |
PubChem BioAssay data set |
NPT791 |
Individual Protein |
Cruzipain |
Trypanosoma cruzi |
Potency |
= |
3981.1 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
398.1 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
3548.1 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
1122 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
316.2 |
nM |
PubChem BioAssay data set |
NPT211 |
Individual Protein |
Hypoxia-inducible factor 1 alpha |
Homo sapiens |
Potency |
= |
79.4 |
nM |
PubChem BioAssay data set |
NPT211 |
Individual Protein |
Hypoxia-inducible factor 1 alpha |
Homo sapiens |
Potency |
= |
125.9 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
17782.8 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
8912.5 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
PubChem BioAssay data set |
NPT796 |
Individual Protein |
Peripheral myelin protein 22 |
Homo sapiens |
Potency |
= |
239.3 |
nM |
PubChem BioAssay data set |
NPT60 |
Individual Protein |
Lysosomal alpha-glucosidase |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
15.8 |
nM |
PubChem BioAssay data set |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT442 |
Individual Protein |
Ferritin light chain |
Equus caballus |
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT442 |
Individual Protein |
Ferritin light chain |
Equus caballus |
Potency |
= |
14125.4 |
nM |
PubChem BioAssay data set |
NPT4446 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
EC50 |
> |
55700 |
nM |
PubChem BioAssay data set |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Potency |
= |
46.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
1412.5 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
1000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
1122 |
nM |
PubChem BioAssay data set |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT58 |
Individual Protein |
Bloom syndrome protein |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
17782.8 |
nM |
PubChem BioAssay data set |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PubChem BioAssay data set |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
125.9 |
nM |
PubChem BioAssay data set |
NPT4487 |
Individual Protein |
Os06g0676700 protein |
Oryza sativa Japonica Group |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
4466.8 |
nM |
PubChem BioAssay data set |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
3981.1 |
nM |
PubChem BioAssay data set |
NPT583 |
Individual Protein |
Inositol monophosphatase 1 |
Rattus norvegicus |
Potency |
= |
316.2 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
3548.1 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
2238.7 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
25.1 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
199.5 |
nM |
PubChem BioAssay data set |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
251.2 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
56.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
EC50 |
< |
100 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
79.4 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
631 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
6309.6 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
501.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
22387.2 |
nM |
PubChem BioAssay data set |
NPT2944 |
Individual Protein |
Relaxin receptor 1 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
= |
316.2 |
nM |
PubChem BioAssay data set |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
Inhibition |
= |
27 |
% |
18824603 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
61 |
% |
18824603 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
11 |
nM |
21071230 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8.9 |
nM |
21071230 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
17 |
nM |
21071230 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2430 |
nM |
21115246 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
590 |
nM |
21115246 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
610 |
nM |
21115246 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21115246 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
64.3 |
% |
21115246 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
69 |
nM |
21095131 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
IC50 |
= |
45 |
nM |
21095131 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
98 |
nM |
21095131 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
18 |
nM |
21095131 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
80 |
nM |
21095131 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.06 |
nM |
20939540 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
200 |
nM |
20961093 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3600 |
nM |
20961093 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
31620 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
> |
100000 |
nM |
21115210 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
50120 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
31620 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
160 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.15 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
16.91 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
41.61 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
25.73 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
11.51 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
10.4 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
65.62 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
10.92 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
71.45 |
% |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
21.25 |
% |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
60 |
nM |
21115210 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
60 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
50 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
21115210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
21186067 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
650 |
nM |
21186067 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
21186067 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
80 |
% |
21186067 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
18 |
nM |
21353568 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
IC50 |
= |
45 |
nM |
21353568 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
69 |
nM |
21353568 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
80 |
nM |
21353568 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
98 |
nM |
21353568 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
260 |
nM |
21341674 |
NPT2 |
Others |
Unspecified |
|
Ratio |
> |
250 |
|
21341674 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
1 |
|
21341674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
300 |
nM |
21341674 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
1 |
nM |
21341674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
52 |
nM |
21341674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
57 |
nM |
21341674 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Ratio |
> |
77 |
|
21341674 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
> |
1000 |
nM |
21341674 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12 |
nM |
21341674 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
13 |
nM |
21341674 |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
7079.5 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
4609 |
nM |
PubChem BioAssay data set |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
3162.3 |
nM |
PubChem BioAssay data set |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
3548.1 |
nM |
PubChem BioAssay data set |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
28183.8 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
366.3 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
2059.6 |
nM |
PubChem BioAssay data set |
NPT443 |
Individual Protein |
Histone acetyltransferase GCN5 |
Homo sapiens |
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT800 |
Individual Protein |
M-phase phosphoprotein 8 |
Homo sapiens |
Potency |
|
100000 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
13371.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1412.5 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
8912.5 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT135 |
Individual Protein |
Chromobox protein homolog 1 |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
5323.3 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
1471.6 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
2332.3 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
2908.1 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
460.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
7307.8 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
AC50 |
= |
6309.57 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
AC50 |
= |
19952.62 |
nM |
PubChem BioAssay data set |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
1584.89 |
nM |
PubChem BioAssay data set |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
2511.89 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
96 |
% |
21334793 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
4 |
% |
21334793 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
35 |
% |
21334793 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
8 |
nM |
21388138 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
33 |
nM |
21388138 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
GI50 |
= |
47 |
nM |
21388138 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
GI50 |
= |
90 |
nM |
21388138 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
200 |
nM |
21388138 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
480 |
nM |
21388138 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
1300 |
nM |
21388138 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6000 |
nM |
21388138 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
69.15 |
% |
21419530 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1080 |
nM |
21419530 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3970 |
nM |
21419530 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
310 |
nM |
21419530 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
970 |
nM |
21419530 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
65 |
nM |
21419530 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
21513293 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
< |
40 |
nM |
21513293 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
21513293 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21599000 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
190 |
nM |
21599000 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11120 |
nM |
21599000 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
890 |
nM |
21599000 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Ratio IC50 |
= |
29.67 |
|
21599000 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
Ratio IC50 |
= |
0.08 |
|
21599000 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
Ratio IC50 |
= |
4.68 |
|
21599000 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.6 |
nM |
21410162 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
459.3 |
nM |
21410162 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Activity |
= |
60 |
% |
21620534 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.072 |
ug/ml |
21684168 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.096 |
ug/ml |
21684168 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1.54 |
ug/ml |
21684168 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
6.88 |
ug/ml |
21684168 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
400 |
nM |
21601964 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21601964 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
500 |
nM |
21601964 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
100 |
nM |
21601964 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
58 |
% |
21601964 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
20.9 |
% |
21601964 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21775156 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
91 |
nM |
21873069 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
166 |
nM |
21873069 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2544 |
nM |
21873069 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
7860 |
nM |
21873069 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21710981 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
21710981 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21710981 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21710981 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
21710981 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
21710981 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21710981 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21710981 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
95 |
% |
21710981 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
3 |
nM |
21973054 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21823606 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
21823606 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21823606 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21823606 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
21823606 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
21823606 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21823606 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
13 |
nM |
21823606 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
17.78 |
% |
21843907 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
27.06 |
% |
21843907 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
50.18 |
% |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
19.64 |
% |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
27.27 |
% |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
47.95 |
% |
21843907 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
33.78 |
% |
21843907 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
9550 |
nM |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
21843907 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
13.94 |
% |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
12.79 |
% |
21843907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
44 |
% |
21843907 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
40.88 |
% |
21843907 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
1168.9 |
nM |
PubChem BioAssay data set |
NPT8 |
Individual Protein |
DNA polymerase iota |
Homo sapiens |
Potency |
|
89125.1 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
2818.4 |
nM |
PubChem BioAssay data set |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Potency |
|
251.2 |
nM |
PubChem BioAssay data set |
NPT698 |
Individual Protein |
Regulator of G-protein signaling 4 |
Homo sapiens |
Potency |
|
2667.9 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
82 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
44.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
25.1 |
nM |
PubChem BioAssay data set |
NPT1160 |
Cell Line |
BJ |
Homo sapiens |
EC50 |
= |
7.67 |
nM |
PubChem BioAssay data set |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
Potency |
|
1778.3 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
20.6 |
nM |
PubChem BioAssay data set |
NPT291 |
Individual Protein |
Serotonin 2b (5-HT2b) receptor |
Homo sapiens |
IC50 |
= |
970 |
nM |
DrugMatrix in vitro pharmacology data |
NPT291 |
Individual Protein |
Serotonin 2b (5-HT2b) receptor |
Homo sapiens |
Ki |
= |
617 |
nM |
DrugMatrix in vitro pharmacology data |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8930 |
nM |
21983445 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
56 |
nM |
21978950 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
260 |
nM |
22044245 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
260 |
nM |
22044245 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
260 |
nM |
22044245 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
260 |
nM |
22044245 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
260 |
nM |
22044245 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
17 |
% |
22047801 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
52 |
% |
22047801 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
11 |
% |
22047801 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
17.42 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
13.42 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
18.67 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
21.21 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
17.59 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6.71 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
11.36 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
46.12 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
5.39 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3.06 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3.05 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
47.24 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
59.5 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
58.52 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
18.36 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
16.24 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.27 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
23.38 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
20.21 |
% |
22104973 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
20.25 |
% |
22104973 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
0.6 |
ug/ml |
21985060 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
7 |
% |
22123322 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
18 |
% |
22123322 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2600 |
nM |
22197145 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1800 |
nM |
22197145 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
800 |
nM |
22197145 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
22197145 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
CC50 |
= |
3 |
nM |
22047799 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
CC50 |
= |
5 |
nM |
22047799 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
CC50 |
= |
4 |
nM |
22047799 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
CC50 |
= |
70 |
nM |
22047799 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
20 |
nM |
22047799 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
CC50 |
= |
30 |
nM |
22047799 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
20 |
nM |
22047799 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
CC50 |
= |
15 |
nM |
22047799 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
CC50 |
= |
200 |
nM |
22047799 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
300 |
nM |
22047799 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
55.5 |
% |
22245048 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
27 |
% |
22305342 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
26 |
% |
22305342 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
5 |
nM |
22305342 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
59.9 |
% |
22318164 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
260 |
nM |
22318164 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1180 |
nM |
22318164 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2370 |
nM |
22318164 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3910 |
nM |
22318164 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1010 |
nM |
22318164 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8 |
nM |
22325897 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
71 |
nM |
22325897 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
600 |
nM |
22325897 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
26 |
nM |
22325897 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
1980 |
nM |
22325897 |
NPT4489 |
Individual Protein |
Heterogeneous nuclear ribonucleoprotein A1 |
Homo sapiens |
Kd |
= |
82.7 |
nM |
22071521 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
14.03 |
nM |
PubChem BioAssay data set |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
145.21 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
19.41 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
30.27 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
11.64 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
33.73 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
14.96 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
14.49 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
27.16 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
173.78 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
76.38 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
176.6 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
32.21 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
11.56 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
11.97 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
11.07 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
38.82 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
80.91 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
18.16 |
nM |
PubChem BioAssay data set |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
937.56 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
1324.34 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
36.64 |
nM |
PubChem BioAssay data set |
NPT573 |
Cell Line |
M19-MEL |
Homo sapiens |
GI50 |
|
47.97 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
22.34 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
20.65 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
159.22 |
nM |
PubChem BioAssay data set |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
GI50 |
|
48.31 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
106.66 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
33.65 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
209.41 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
26.06 |
nM |
PubChem BioAssay data set |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI50 |
|
26.67 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
114.82 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
297.85 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
18.11 |
nM |
PubChem BioAssay data set |
NPT575 |
Cell Line |
KM-20L2 |
Homo sapiens |
GI50 |
|
77.62 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
27.16 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
158.85 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
151.71 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
23.01 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
11.51 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
11.35 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
95.06 |
nM |
PubChem BioAssay data set |
NPT731 |
Cell Line |
LXFL 529 |
Homo sapiens |
GI50 |
|
372.39 |
nM |
PubChem BioAssay data set |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
GI50 |
|
20.56 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
64.42 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
22.54 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
20.18 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
15.78 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
10.64 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
65.77 |
nM |
PubChem BioAssay data set |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
GI50 |
|
25.35 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
11.8 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
184.08 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
11.53 |
nM |
PubChem BioAssay data set |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
|
816.58 |
nM |
PubChem BioAssay data set |
NPT578 |
Cell Line |
SNB-78 |
Homo sapiens |
GI50 |
|
332.66 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
21.38 |
nM |
PubChem BioAssay data set |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
GI50 |
|
242.66 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
54.33 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
17.95 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
44.87 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
227.51 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
285.76 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
25.64 |
nM |
PubChem BioAssay data set |
NPT738 |
Cell Line |
SN12K1 |
Homo sapiens |
GI50 |
|
24.49 |
nM |
PubChem BioAssay data set |
NPT732 |
Cell Line |
HOP-18 |
Homo sapiens |
GI50 |
|
122.18 |
nM |
PubChem BioAssay data set |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
6400 |
nM |
22326393 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18300 |
nM |
22326393 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15200 |
nM |
22326393 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
FC |
= |
4 |
|
22326393 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
4 |
nM |
22276775 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
20 |
nM |
22276775 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
15 |
nM |
22276775 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
22329436 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
22329436 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
22329436 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
22329436 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
22329436 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
22329436 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
22329436 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
13 |
nM |
22329436 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.6 |
nM |
22376176 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
400 |
nM |
22542106 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1570 |
nM |
22542106 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
22.9 |
nM |
22647222 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
33.8 |
nM |
22647222 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22409771 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22409771 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22409771 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22409771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
100 |
nM |
22409771 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7 |
nM |
22749423 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
5 |
nM |
22749423 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
22749423 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
63.1 |
% |
22819942 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
26.3 |
% |
22819942 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
9170 |
nM |
22819942 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
9920 |
nM |
22819942 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
9290 |
nM |
22819942 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
7940 |
nM |
22819942 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
CC50 |
= |
4 |
nM |
22884523 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
CC50 |
= |
3 |
nM |
22884523 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
CC50 |
= |
5 |
nM |
22884523 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
CC50 |
= |
4 |
nM |
22884523 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
CC50 |
= |
70 |
nM |
22884523 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
80 |
nM |
22884523 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
CC50 |
= |
50 |
nM |
22884523 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
40 |
nM |
22884523 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
CC50 |
= |
80 |
nM |
22884523 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
CC50 |
= |
200 |
nM |
22884523 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
300 |
nM |
22884523 |
NPT4490 |
Cell Line |
IMR-90 |
Homo sapiens |
IC50 |
= |
430 |
nM |
22863526 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
70 |
nM |
22863526 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2 |
nM |
22863526 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
80 |
nM |
22863526 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
3 |
nM |
22758788 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
10 |
nM |
22867707 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
150 |
nM |
22867707 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
1000 |
nM |
22867707 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
22867707 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
< |
1000 |
nM |
22867707 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
22867707 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
70 |
nM |
22867707 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
70 |
nM |
22867707 |
NPT3882 |
Cell Line |
MFE-296 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
22867707 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2610 |
nM |
23084702 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
110 |
nM |
23084702 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
43.6 |
nM |
23084702 |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
14125.4 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
8912.5 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT478 |
Individual Protein |
Ataxin-2 |
Homo sapiens |
Potency |
|
1778.3 |
nM |
PubChem BioAssay data set |
NPT478 |
Individual Protein |
Ataxin-2 |
Homo sapiens |
Potency |
|
10 |
nM |
PubChem BioAssay data set |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
400 |
nM |
23153813 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1570 |
nM |
23153813 |
NPT4491 |
Individual Protein |
DNA topoisomerase type IB small subunit |
Leishmania major |
EC50 |
= |
670 |
nM |
22932312 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
2000 |
nM |
22932312 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
620 |
nM |
22932312 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
23142674 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
70 |
nM |
23142674 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
12750 |
nM |
23142674 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
170 |
nM |
23142674 |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23142674 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT2743 |
Cell Line |
MCF-12A |
Homo sapiens |
IC50 |
< |
10 |
nM |
23142674 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
> |
95 |
% |
22698783 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
60 |
% |
22698783 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
48 |
|
22698783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.8 |
nM |
22698783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24 |
nM |
22698783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
423 |
nM |
22698783 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
8.8 |
nM |
22698783 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
3.83 |
|
23137376 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio |
= |
3.4 |
|
23137376 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17.96 |
% |
23137376 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17.56 |
% |
23137376 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Activity |
= |
23.81 |
% |
23137376 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Activity |
= |
17.61 |
% |
23137376 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
14.05 |
% |
23062825 |
NPT67 |
Individual Protein |
Cholinesterase |
Equus caballus |
Inhibition |
= |
3.9 |
% |
23062825 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
GI50 |
> |
287000 |
nM |
22867019 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
< |
3 |
nM |
22867019 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
> |
287000 |
nM |
22867019 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
220 |
nM |
22867019 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
GI50 |
= |
6290 |
nM |
22867019 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
GI50 |
> |
287000 |
nM |
22867019 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
83 |
nM |
22867019 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
33 |
nM |
22867019 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
170 |
nM |
22867019 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
46.6 |
% |
22503656 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
23.1 |
% |
22503656 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
1010 |
nM |
22503656 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1530 |
nM |
22503656 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1060 |
nM |
22503656 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1380 |
nM |
22503656 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37.1 |
nM |
23102893 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
121 |
nM |
23102893 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
28.7 |
nM |
23102893 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
15.8 |
nM |
23102893 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
3750 |
nM |
10.1007/s00044-009-9233-5 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
4950 |
nM |
10.1007/s00044-009-9233-5 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
4750 |
nM |
10.1007/s00044-009-9233-5 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
429.9 |
ug/ml |
10.1007/s00044-010-9381-7 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
58 |
ug/ml |
10.1007/s00044-010-9381-7 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.28 |
ug/ml |
10.1007/s00044-010-9381-7 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
68.6 |
% |
23354071 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
17.7 |
% |
23354071 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
51 |
% |
23419739 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
6 |
% |
23419739 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
88 |
% |
23419739 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
69 |
% |
23419739 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
50 |
nM |
23357037 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7 |
nM |
23357037 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2 |
nM |
23357037 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
231.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
89.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
37.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
79.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
18.4 |
nM |
PubChem BioAssay data set |
NPT2268 |
Cell Line |
DOK |
Homo sapiens |
IC50 |
= |
18.92 |
nM |
10.6019/CHEMBL1201861 |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
15.75 |
nM |
10.6019/CHEMBL1201861 |
NPT1184 |
Cell Line |
Daoy |
Homo sapiens |
IC50 |
= |
0.4809 |
nM |
10.6019/CHEMBL1201861 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2281.94 |
nM |
10.6019/CHEMBL1201861 |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
3.067 |
nM |
10.6019/CHEMBL1201861 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
436.37 |
nM |
10.6019/CHEMBL1201861 |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
4.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2269 |
Cell Line |
EPLC-272H |
Homo sapiens |
IC50 |
= |
72.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
1.474 |
nM |
10.6019/CHEMBL1201861 |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
0.7735 |
nM |
10.6019/CHEMBL1201861 |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
0.09574 |
nM |
10.6019/CHEMBL1201861 |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
0.9311 |
nM |
10.6019/CHEMBL1201861 |
NPT2270 |
Cell Line |
Detroit562 |
Homo sapiens |
IC50 |
= |
13.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2271 |
Cell Line |
DoTc2-4510 |
Homo sapiens |
IC50 |
= |
4.032 |
nM |
10.6019/CHEMBL1201861 |
NPT1908 |
Cell Line |
EC-GI-10 |
Homo sapiens |
IC50 |
= |
7.904 |
nM |
10.6019/CHEMBL1201861 |
NPT3465 |
Cell Line |
ECC10 |
Homo sapiens |
IC50 |
= |
3.853 |
nM |
10.6019/CHEMBL1201861 |
NPT2272 |
Cell Line |
EFM-19 |
Homo sapiens |
IC50 |
= |
126.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2273 |
Cell Line |
EFO-21 |
Homo sapiens |
IC50 |
= |
20.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2274 |
Cell Line |
EFO-27 |
Homo sapiens |
IC50 |
= |
80.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2275 |
Cell Line |
EGI-1 |
Homo sapiens |
IC50 |
= |
25.07 |
nM |
10.6019/CHEMBL1201861 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
7.077 |
nM |
10.6019/CHEMBL1201861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
0.8149 |
nM |
10.6019/CHEMBL1201861 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
116.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
6.477 |
nM |
10.6019/CHEMBL1201861 |
NPT2278 |
Cell Line |
COLO-741 |
Homo sapiens |
IC50 |
= |
109.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2279 |
Cell Line |
COLO-792 |
Homo sapiens |
IC50 |
= |
169.17 |
nM |
10.6019/CHEMBL1201861 |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
436.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
15.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2281 |
Cell Line |
ABC-1 |
Homo sapiens |
IC50 |
= |
3.468 |
nM |
10.6019/CHEMBL1201861 |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
2.438 |
nM |
10.6019/CHEMBL1201861 |
NPT2282 |
Cell Line |
C32 |
Homo sapiens |
IC50 |
= |
13.37 |
nM |
10.6019/CHEMBL1201861 |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
0.4281 |
nM |
10.6019/CHEMBL1201861 |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
269.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2283 |
Cell Line |
DK-MG |
Homo sapiens |
IC50 |
= |
84.75 |
nM |
10.6019/CHEMBL1201861 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
81.1 |
nM |
10.6019/CHEMBL1201861 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
6.663 |
nM |
10.6019/CHEMBL1201861 |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
85.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2284 |
Cell Line |
C3A |
Homo sapiens |
IC50 |
= |
56.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
41.48 |
nM |
10.6019/CHEMBL1201861 |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
11.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2285 |
Cell Line |
COR-L105 |
Homo sapiens |
IC50 |
= |
184.93 |
nM |
10.6019/CHEMBL1201861 |
NPT1918 |
Cell Line |
DMS-79 |
Homo sapiens |
IC50 |
= |
31.85 |
nM |
10.6019/CHEMBL1201861 |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
0.6022 |
nM |
10.6019/CHEMBL1201861 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
16.13 |
nM |
10.6019/CHEMBL1201861 |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
1.534 |
nM |
10.6019/CHEMBL1201861 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
IC50 |
= |
5.354 |
nM |
10.6019/CHEMBL1201861 |
NPT2286 |
Cell Line |
CAL-120 |
Homo sapiens |
IC50 |
= |
594.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
6.849 |
nM |
10.6019/CHEMBL1201861 |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
40.93 |
nM |
10.6019/CHEMBL1201861 |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
IC50 |
= |
6.072 |
nM |
10.6019/CHEMBL1201861 |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
4.408 |
nM |
10.6019/CHEMBL1201861 |
NPT2288 |
Cell Line |
AN3-CA |
Homo sapiens |
IC50 |
= |
33.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2289 |
Cell Line |
CAL-12T |
Homo sapiens |
IC50 |
= |
262.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2290 |
Cell Line |
CAL-27 |
Homo sapiens |
IC50 |
= |
2.018 |
nM |
10.6019/CHEMBL1201861 |
NPT2291 |
Cell Line |
CP50-MEL-B |
Homo sapiens |
IC50 |
= |
72.08 |
nM |
10.6019/CHEMBL1201861 |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
208.15 |
nM |
10.6019/CHEMBL1201861 |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
9.314 |
nM |
10.6019/CHEMBL1201861 |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
2.043 |
nM |
10.6019/CHEMBL1201861 |
NPT2292 |
Cell Line |
CAL-33 |
Homo sapiens |
IC50 |
= |
5.997 |
nM |
10.6019/CHEMBL1201861 |
NPT2293 |
Cell Line |
CAL-39 |
Homo sapiens |
IC50 |
= |
19.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
0.4292 |
nM |
10.6019/CHEMBL1201861 |
NPT2294 |
Cell Line |
23132-87 |
Homo sapiens |
IC50 |
= |
19.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
4.183 |
nM |
10.6019/CHEMBL1201861 |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
3.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
168.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2298 |
Cell Line |
BALL-1 |
Homo sapiens |
IC50 |
= |
108.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2299 |
Cell Line |
CAL-51 |
Homo sapiens |
IC50 |
= |
29.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2300 |
Cell Line |
CAL-54 |
Homo sapiens |
IC50 |
= |
4.758 |
nM |
10.6019/CHEMBL1201861 |
NPT2301 |
Cell Line |
CAL-62 |
Homo sapiens |
IC50 |
= |
0.9836 |
nM |
10.6019/CHEMBL1201861 |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
0.9054 |
nM |
10.6019/CHEMBL1201861 |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
35.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2302 |
Cell Line |
639-V |
Homo sapiens |
IC50 |
= |
0.1714 |
nM |
10.6019/CHEMBL1201861 |
NPT2303 |
Cell Line |
647-V |
Homo sapiens |
IC50 |
= |
0.8964 |
nM |
10.6019/CHEMBL1201861 |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
21.55 |
nM |
10.6019/CHEMBL1201861 |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
120.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2304 |
Cell Line |
CAL-72 |
Homo sapiens |
IC50 |
= |
150.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2305 |
Cell Line |
CAL-85-1 |
Homo sapiens |
IC50 |
= |
7923.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2306 |
Cell Line |
Ca-Ski |
Homo sapiens |
IC50 |
= |
4.97 |
nM |
10.6019/CHEMBL1201861 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
2.211 |
nM |
10.6019/CHEMBL1201861 |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
2.029 |
nM |
10.6019/CHEMBL1201861 |
NPT2307 |
Cell Line |
769-P |
Homo sapiens |
IC50 |
= |
25.34 |
nM |
10.6019/CHEMBL1201861 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
5.021 |
nM |
10.6019/CHEMBL1201861 |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
1.853 |
nM |
10.6019/CHEMBL1201861 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
87.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2309 |
Cell Line |
CAPAN-1 |
Homo sapiens |
IC50 |
= |
14.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2310 |
Cell Line |
CaR-1 |
Homo sapiens |
IC50 |
= |
6.427 |
nM |
10.6019/CHEMBL1201861 |
NPT2311 |
Cell Line |
Calu-3 |
Homo sapiens |
IC50 |
= |
32.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
1.502 |
nM |
10.6019/CHEMBL1201861 |
NPT2312 |
Cell Line |
8305C |
Homo sapiens |
IC50 |
= |
93.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2313 |
Cell Line |
BCPAP |
Homo sapiens |
IC50 |
= |
3.041 |
nM |
10.6019/CHEMBL1201861 |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
121.91 |
nM |
10.6019/CHEMBL1201861 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
5.547 |
nM |
10.6019/CHEMBL1201861 |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
178.95 |
nM |
10.6019/CHEMBL1201861 |
NPT1313 |
Cell Line |
Capan-2 |
Homo sapiens |
IC50 |
= |
452.29 |
nM |
10.6019/CHEMBL1201861 |
NPT1215 |
Cell Line |
8505C |
Homo sapiens |
IC50 |
= |
3.301 |
nM |
10.6019/CHEMBL1201861 |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
257.84 |
nM |
10.6019/CHEMBL1201861 |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
4.564 |
nM |
10.6019/CHEMBL1201861 |
NPT2314 |
Cell Line |
BEN |
Homo sapiens |
IC50 |
= |
107.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2315 |
Cell Line |
BFTC-905 |
Homo sapiens |
IC50 |
= |
0.1398 |
nM |
10.6019/CHEMBL1201861 |
NPT2316 |
Cell Line |
CFPAC-1 |
Homo sapiens |
IC50 |
= |
14.75 |
nM |
10.6019/CHEMBL1201861 |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
3.275 |
nM |
10.6019/CHEMBL1201861 |
NPT2317 |
Cell Line |
ChaGo-K-1 |
Homo sapiens |
IC50 |
= |
304.67 |
nM |
10.6019/CHEMBL1201861 |
NPT1944 |
Cell Line |
D-247MG |
Homo sapiens |
IC50 |
= |
39.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
12.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2319 |
Cell Line |
A204 |
Homo sapiens |
IC50 |
= |
4.525 |
nM |
10.6019/CHEMBL1201861 |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
3.599 |
nM |
10.6019/CHEMBL1201861 |
NPT2320 |
Cell Line |
BFTC-909 |
Homo sapiens |
IC50 |
= |
6.925 |
nM |
10.6019/CHEMBL1201861 |
NPT2321 |
Cell Line |
BHT-101 |
Homo sapiens |
IC50 |
= |
1.822 |
nM |
10.6019/CHEMBL1201861 |
NPT2322 |
Cell Line |
CHL-1 |
Homo sapiens |
IC50 |
= |
6.091 |
nM |
10.6019/CHEMBL1201861 |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
9.114 |
nM |
10.6019/CHEMBL1201861 |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
3.198 |
nM |
10.6019/CHEMBL1201861 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
2.902 |
nM |
10.6019/CHEMBL1201861 |
NPT2323 |
Cell Line |
BHY |
Homo sapiens |
IC50 |
= |
5.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2324 |
Cell Line |
CHP-212 |
Homo sapiens |
IC50 |
= |
1.026 |
nM |
10.6019/CHEMBL1201861 |
NPT1953 |
Cell Line |
D-336MG |
Homo sapiens |
IC50 |
= |
5.205 |
nM |
10.6019/CHEMBL1201861 |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
17.73 |
nM |
10.6019/CHEMBL1201861 |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
1.669 |
nM |
10.6019/CHEMBL1201861 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
3.688 |
nM |
10.6019/CHEMBL1201861 |
NPT2325 |
Cell Line |
BPH-1 |
Homo sapiens |
IC50 |
= |
2.082 |
nM |
10.6019/CHEMBL1201861 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
25.99 |
nM |
10.6019/CHEMBL1201861 |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
62.09 |
nM |
10.6019/CHEMBL1201861 |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
22.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2327 |
Cell Line |
D-423MG |
Homo sapiens |
IC50 |
= |
2.551 |
nM |
10.6019/CHEMBL1201861 |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
22.59 |
nM |
10.6019/CHEMBL1201861 |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
10.12 |
nM |
10.6019/CHEMBL1201861 |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
1.749 |
nM |
10.6019/CHEMBL1201861 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
1985.76 |
nM |
10.6019/CHEMBL1201861 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
17.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2328 |
Cell Line |
COLO-678 |
Homo sapiens |
IC50 |
= |
3682.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2329 |
Cell Line |
COLO-679 |
Homo sapiens |
IC50 |
= |
4791.52 |
nM |
10.6019/CHEMBL1201861 |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
291.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2330 |
Cell Line |
D-566MG |
Homo sapiens |
IC50 |
= |
0.1315 |
nM |
10.6019/CHEMBL1201861 |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
4.251 |
nM |
10.6019/CHEMBL1201861 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
1552.36 |
nM |
10.6019/CHEMBL1201861 |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
2.381 |
nM |
10.6019/CHEMBL1201861 |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
23.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2332 |
Cell Line |
COLO-680N |
Homo sapiens |
IC50 |
= |
72.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
13.82 |
nM |
10.6019/CHEMBL1201861 |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
1.161 |
nM |
10.6019/CHEMBL1201861 |
NPT2333 |
Cell Line |
DBTRG-05MG |
Homo sapiens |
IC50 |
= |
40.86 |
nM |
10.6019/CHEMBL1201861 |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
0.8157 |
nM |
10.6019/CHEMBL1201861 |
NPT2334 |
Cell Line |
NCI-H1793 |
Homo sapiens |
IC50 |
= |
27.23 |
nM |
10.6019/CHEMBL1201861 |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
253.14 |
nM |
10.6019/CHEMBL1201861 |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
1.028 |
nM |
10.6019/CHEMBL1201861 |
NPT2335 |
Cell Line |
NCI-H596 |
|
IC50 |
= |
2968.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2336 |
Cell Line |
OE19 |
Homo sapiens |
IC50 |
= |
3273.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
25.55 |
nM |
10.6019/CHEMBL1201861 |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
IC50 |
= |
4.753 |
nM |
10.6019/CHEMBL1201861 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
29.49 |
nM |
10.6019/CHEMBL1201861 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
4.713 |
nM |
10.6019/CHEMBL1201861 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
51.29 |
nM |
10.6019/CHEMBL1201861 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
37.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
3.017 |
nM |
10.6019/CHEMBL1201861 |
NPT2339 |
Cell Line |
TGBC24TKB |
Homo sapiens |
IC50 |
= |
53.71 |
nM |
10.6019/CHEMBL1201861 |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
3.365 |
nM |
10.6019/CHEMBL1201861 |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
13.52 |
nM |
10.6019/CHEMBL1201861 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
3.734 |
nM |
10.6019/CHEMBL1201861 |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
34.38 |
nM |
10.6019/CHEMBL1201861 |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
57.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2340 |
Cell Line |
KU-19-19 |
Homo sapiens |
IC50 |
= |
22.03 |
nM |
10.6019/CHEMBL1201861 |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
31.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
27.08 |
nM |
10.6019/CHEMBL1201861 |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
5270.72 |
nM |
10.6019/CHEMBL1201861 |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
28.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1980 |
Cell Line |
NB14 |
Homo sapiens |
IC50 |
= |
0.9071 |
nM |
10.6019/CHEMBL1201861 |
NPT2341 |
Cell Line |
NCI-H1975 |
Homo sapiens |
IC50 |
= |
334.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2342 |
Cell Line |
NCI-H630 |
Homo sapiens |
IC50 |
= |
282.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2343 |
Cell Line |
NCI-H650 |
Homo sapiens |
IC50 |
= |
54.96 |
nM |
10.6019/CHEMBL1201861 |
NPT1968 |
Cell Line |
OMC-1 |
Homo sapiens |
IC50 |
= |
78.21 |
nM |
10.6019/CHEMBL1201861 |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
2.406 |
nM |
10.6019/CHEMBL1201861 |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
1.725 |
nM |
10.6019/CHEMBL1201861 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
54.75 |
nM |
10.6019/CHEMBL1201861 |
NPT2344 |
Cell Line |
SK-MEL-24 |
Homo sapiens |
IC50 |
= |
38.51 |
nM |
10.6019/CHEMBL1201861 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
4.082 |
nM |
10.6019/CHEMBL1201861 |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
76.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2346 |
Cell Line |
TI-73 |
Homo sapiens |
IC50 |
= |
14.55 |
nM |
10.6019/CHEMBL1201861 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
55.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
33.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2347 |
Cell Line |
GMS-10 |
Homo sapiens |
IC50 |
= |
7.311 |
nM |
10.6019/CHEMBL1201861 |
NPT2348 |
Cell Line |
HLE |
Homo sapiens |
IC50 |
= |
5.753 |
nM |
10.6019/CHEMBL1201861 |
NPT2349 |
Cell Line |
HMV-2 cell line |
|
IC50 |
= |
8.887 |
nM |
10.6019/CHEMBL1201861 |
NPT2350 |
Cell Line |
HN |
Homo sapiens |
IC50 |
= |
1.399 |
nM |
10.6019/CHEMBL1201861 |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
2.579 |
nM |
10.6019/CHEMBL1201861 |
NPT1505 |
Cell Line |
J82 |
Homo sapiens |
IC50 |
= |
4.722 |
nM |
10.6019/CHEMBL1201861 |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
8.365 |
nM |
10.6019/CHEMBL1201861 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
3.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
7.654 |
nM |
10.6019/CHEMBL1201861 |
NPT2352 |
Cell Line |
MHH-ES-1 |
Homo sapiens |
IC50 |
= |
0.1293 |
nM |
10.6019/CHEMBL1201861 |
NPT1995 |
Cell Line |
NB17 |
Homo sapiens |
IC50 |
= |
2.175 |
nM |
10.6019/CHEMBL1201861 |
NPT2353 |
Cell Line |
NCI-H1993 |
Homo sapiens |
IC50 |
= |
9621.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2354 |
Cell Line |
NCI-H2009 |
Homo sapiens |
IC50 |
= |
68.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2355 |
Cell Line |
NCI-H2029 |
Homo sapiens |
IC50 |
= |
491.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
13.55 |
nM |
10.6019/CHEMBL1201861 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
311.44 |
nM |
10.6019/CHEMBL1201861 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
9.968 |
nM |
10.6019/CHEMBL1201861 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
956.65 |
nM |
10.6019/CHEMBL1201861 |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
0.9022 |
nM |
10.6019/CHEMBL1201861 |
NPT2357 |
Cell Line |
RT-112 |
Homo sapiens |
IC50 |
= |
14.88 |
nM |
10.6019/CHEMBL1201861 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
17.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
IC50 |
= |
329.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2359 |
Cell Line |
SK-MEL-30 |
Homo sapiens |
IC50 |
= |
2281.97 |
nM |
10.6019/CHEMBL1201861 |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
711.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2360 |
Cell Line |
SW756 |
Homo sapiens |
IC50 |
= |
4.211 |
nM |
10.6019/CHEMBL1201861 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
25.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2362 |
Cell Line |
TYK-nu |
Homo sapiens |
IC50 |
= |
4.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2363 |
Cell Line |
U-118-MG |
Homo sapiens |
IC50 |
= |
19 |
nM |
10.6019/CHEMBL1201861 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
0.7058 |
nM |
10.6019/CHEMBL1201861 |
NPT2364 |
Cell Line |
GP5d |
Homo sapiens |
IC50 |
= |
12.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2365 |
Cell Line |
HO-1-N-1 |
Homo sapiens |
IC50 |
= |
0.8385 |
nM |
10.6019/CHEMBL1201861 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
3293.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
14.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2366 |
Cell Line |
JEG-3 |
Homo sapiens |
IC50 |
= |
13.12 |
nM |
10.6019/CHEMBL1201861 |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
3634.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
8.123 |
nM |
10.6019/CHEMBL1201861 |
NPT2367 |
Cell Line |
KYSE-140 |
Homo sapiens |
IC50 |
= |
69.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
9492.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
7325.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
0.8418 |
nM |
10.6019/CHEMBL1201861 |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
1.925 |
nM |
10.6019/CHEMBL1201861 |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
182.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2368 |
Cell Line |
NCI-H2030 |
Homo sapiens |
IC50 |
= |
48.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2369 |
Cell Line |
NCI-H2052 |
Homo sapiens |
IC50 |
= |
28.34 |
nM |
10.6019/CHEMBL1201861 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
188.55 |
nM |
10.6019/CHEMBL1201861 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
IC50 |
= |
43.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2370 |
Cell Line |
RVH-421 |
Homo sapiens |
IC50 |
= |
71.47 |
nM |
10.6019/CHEMBL1201861 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
4.662 |
nM |
10.6019/CHEMBL1201861 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
10.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2371 |
Cell Line |
SW837 |
Homo sapiens |
IC50 |
= |
48.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
24.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
13.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
69.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
88.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
0.02543 |
nM |
10.6019/CHEMBL1201861 |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
0.701 |
nM |
10.6019/CHEMBL1201861 |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
1.759 |
nM |
10.6019/CHEMBL1201861 |
NPT2372 |
Cell Line |
H-EMC-SS |
Homo sapiens |
IC50 |
= |
95.58 |
nM |
10.6019/CHEMBL1201861 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
IC50 |
= |
8.787 |
nM |
10.6019/CHEMBL1201861 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
1.398 |
nM |
10.6019/CHEMBL1201861 |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
3029.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
2.504 |
nM |
10.6019/CHEMBL1201861 |
NPT2373 |
Cell Line |
KYSE-150 cell line |
|
IC50 |
= |
245.96 |
nM |
10.6019/CHEMBL1201861 |
NPT2374 |
Cell Line |
KYSE-180 |
Homo sapiens |
IC50 |
= |
13.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
58.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
2.733 |
nM |
10.6019/CHEMBL1201861 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
2.759 |
nM |
10.6019/CHEMBL1201861 |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
37.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
0.5694 |
nM |
10.6019/CHEMBL1201861 |
NPT2023 |
Cell Line |
NB7 |
Homo sapiens |
IC50 |
= |
16.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2376 |
Cell Line |
NBsusSR |
Homo sapiens |
IC50 |
= |
0.1936 |
nM |
10.6019/CHEMBL1201861 |
NPT2377 |
Cell Line |
NCI-H2087 |
Homo sapiens |
IC50 |
= |
5.074 |
nM |
10.6019/CHEMBL1201861 |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
0.04843 |
nM |
10.6019/CHEMBL1201861 |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
44.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
1009.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
296.49 |
nM |
10.6019/CHEMBL1201861 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
7.272 |
nM |
10.6019/CHEMBL1201861 |
NPT2379 |
Cell Line |
P12-Ichikawa |
Homo sapiens |
IC50 |
= |
0.1016 |
nM |
10.6019/CHEMBL1201861 |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
10.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2380 |
Cell Line |
SK-N-AS |
Homo sapiens |
IC50 |
= |
5.377 |
nM |
10.6019/CHEMBL1201861 |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
21.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2381 |
Cell Line |
SW900 |
Homo sapiens |
IC50 |
= |
31.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
260.2 |
nM |
10.6019/CHEMBL1201861 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
6.632 |
nM |
10.6019/CHEMBL1201861 |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
0.7956 |
nM |
10.6019/CHEMBL1201861 |
NPT2383 |
Cell Line |
ESS-1 |
Homo sapiens |
IC50 |
= |
7.079 |
nM |
10.6019/CHEMBL1201861 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
IC50 |
= |
0.6154 |
nM |
10.6019/CHEMBL1201861 |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
IC50 |
= |
0.3582 |
nM |
10.6019/CHEMBL1201861 |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
2.551 |
nM |
10.6019/CHEMBL1201861 |
NPT2384 |
Cell Line |
HPAF-II |
Homo sapiens |
IC50 |
= |
55.12 |
nM |
10.6019/CHEMBL1201861 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
11.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
IC50 |
= |
3.015 |
nM |
10.6019/CHEMBL1201861 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1077.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2386 |
Cell Line |
KYSE-270 |
Homo sapiens |
IC50 |
= |
5.223 |
nM |
10.6019/CHEMBL1201861 |
NPT2387 |
Cell Line |
KYSE-410 |
Homo sapiens |
IC50 |
= |
78.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
19.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
0.5865 |
nM |
10.6019/CHEMBL1201861 |
NPT2388 |
Cell Line |
LU-135 |
Homo sapiens |
IC50 |
= |
28.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
51.21 |
nM |
10.6019/CHEMBL1201861 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
27.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2389 |
Cell Line |
NCI-H1048 |
Homo sapiens |
IC50 |
= |
0.5292 |
nM |
10.6019/CHEMBL1201861 |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
43.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2390 |
Cell Line |
NCI-H2122 |
Homo sapiens |
IC50 |
= |
12.98 |
nM |
10.6019/CHEMBL1201861 |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
178.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2391 |
Cell Line |
NCI-H810 |
Homo sapiens |
IC50 |
= |
50.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
2.792 |
nM |
10.6019/CHEMBL1201861 |
NPT2392 |
Cell Line |
S-117 |
Homo sapiens |
IC50 |
= |
78.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
1.241 |
nM |
10.6019/CHEMBL1201861 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
106.62 |
nM |
10.6019/CHEMBL1201861 |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
1.227 |
nM |
10.6019/CHEMBL1201861 |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
20.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
20.51 |
nM |
10.6019/CHEMBL1201861 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
34.07 |
nM |
10.6019/CHEMBL1201861 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
1.869 |
nM |
10.6019/CHEMBL1201861 |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
34.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2047 |
Cell Line |
HC-1 |
Homo sapiens |
IC50 |
= |
3.344 |
nM |
10.6019/CHEMBL1201861 |
NPT2394 |
Cell Line |
HSC-4 |
Homo sapiens |
IC50 |
= |
0.1816 |
nM |
10.6019/CHEMBL1201861 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
29.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
3.201 |
nM |
10.6019/CHEMBL1201861 |
NPT2395 |
Cell Line |
KYSE-450 |
Homo sapiens |
IC50 |
= |
23.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2396 |
Cell Line |
KYSE-510 |
Homo sapiens |
IC50 |
= |
6.754 |
nM |
10.6019/CHEMBL1201861 |
NPT2397 |
Cell Line |
KYSE-520 cell line |
|
IC50 |
= |
82.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
16.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2398 |
Cell Line |
MKN-7 |
Homo sapiens |
IC50 |
= |
144.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
2.165 |
nM |
10.6019/CHEMBL1201861 |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
1.188 |
nM |
10.6019/CHEMBL1201861 |
NPT2399 |
Cell Line |
NCI-H2170 |
Homo sapiens |
IC50 |
= |
13.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
588.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
0.981 |
nM |
10.6019/CHEMBL1201861 |
NPT2401 |
Cell Line |
PANC-03-27 |
Homo sapiens |
IC50 |
= |
7.103 |
nM |
10.6019/CHEMBL1201861 |
NPT2402 |
Cell Line |
PANC-08-13 |
Homo sapiens |
IC50 |
= |
44.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
27.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2403 |
Cell Line |
SBC-5 |
Homo sapiens |
IC50 |
= |
32.15 |
nM |
10.6019/CHEMBL1201861 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
7210.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
1.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2404 |
Cell Line |
SW982 |
Homo sapiens |
IC50 |
= |
4.062 |
nM |
10.6019/CHEMBL1201861 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
17.77 |
nM |
10.6019/CHEMBL1201861 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
115.96 |
nM |
10.6019/CHEMBL1201861 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
31.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
1.777 |
nM |
10.6019/CHEMBL1201861 |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
314.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2406 |
Cell Line |
HCC1395 |
Homo sapiens |
IC50 |
= |
1367.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2407 |
Cell Line |
HCC1419 |
Homo sapiens |
IC50 |
= |
4155.69 |
nM |
10.6019/CHEMBL1201861 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
0.3944 |
nM |
10.6019/CHEMBL1201861 |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
1093.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
69.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
2892.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2408 |
Cell Line |
KYSE-70 cell line |
|
IC50 |
= |
92.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
1.869 |
nM |
10.6019/CHEMBL1201861 |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
276.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2409 |
Cell Line |
LU-99A |
Homo sapiens |
IC50 |
= |
3.854 |
nM |
10.6019/CHEMBL1201861 |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
8.145 |
nM |
10.6019/CHEMBL1201861 |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
38.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
9.425 |
nM |
10.6019/CHEMBL1201861 |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
59.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2411 |
Cell Line |
NCI-H2228 |
Homo sapiens |
IC50 |
= |
49 |
nM |
10.6019/CHEMBL1201861 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
8.743 |
nM |
10.6019/CHEMBL1201861 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
1.088 |
nM |
10.6019/CHEMBL1201861 |
NPT2412 |
Cell Line |
Panc1005 |
Homo sapiens |
IC50 |
= |
19.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
13.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
18.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2414 |
Cell Line |
SCC-25 |
Homo sapiens |
IC50 |
= |
56.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
3.067 |
nM |
10.6019/CHEMBL1201861 |
NPT2415 |
Cell Line |
SKG-IIIa |
Homo sapiens |
IC50 |
= |
4.582 |
nM |
10.6019/CHEMBL1201861 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
86.88 |
nM |
10.6019/CHEMBL1201861 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
1.614 |
nM |
10.6019/CHEMBL1201861 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
13.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2416 |
Cell Line |
UACC-893 |
Homo sapiens |
IC50 |
= |
383.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
3.093 |
nM |
10.6019/CHEMBL1201861 |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
2.659 |
nM |
10.6019/CHEMBL1201861 |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
3.267 |
nM |
10.6019/CHEMBL1201861 |
NPT2418 |
Cell Line |
HCC1569 |
Homo sapiens |
IC50 |
= |
267.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2419 |
Cell Line |
HT-1376 |
Homo sapiens |
IC50 |
= |
1780.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
17.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
134.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
148.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
7.054 |
nM |
10.6019/CHEMBL1201861 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
14.93 |
nM |
10.6019/CHEMBL1201861 |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
5.083 |
nM |
10.6019/CHEMBL1201861 |
NPT3466 |
Cell Line |
MOLT-13 |
Homo sapiens |
IC50 |
= |
1.787 |
nM |
10.6019/CHEMBL1201861 |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
66.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
110.1 |
nM |
10.6019/CHEMBL1201861 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
22.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2420 |
Cell Line |
NCI-H2291 |
Homo sapiens |
IC50 |
= |
975.25 |
nM |
10.6019/CHEMBL1201861 |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
42.71 |
nM |
10.6019/CHEMBL1201861 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
9.753 |
nM |
10.6019/CHEMBL1201861 |
NPT2421 |
Cell Line |
PFSK-1 |
Homo sapiens |
IC50 |
= |
26.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2422 |
Cell Line |
SCC-4 |
Homo sapiens |
IC50 |
= |
19.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2423 |
Cell Line |
SCC-9 |
Homo sapiens |
IC50 |
= |
33.19 |
nM |
10.6019/CHEMBL1201861 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
IC50 |
= |
4.503 |
nM |
10.6019/CHEMBL1201861 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
17.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
4602.33 |
nM |
10.6019/CHEMBL1201861 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
27.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2425 |
Cell Line |
UMC-11 |
Homo sapiens |
IC50 |
= |
2511.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
3.469 |
nM |
10.6019/CHEMBL1201861 |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
0.1214 |
nM |
10.6019/CHEMBL1201861 |
NPT2426 |
Cell Line |
HCC1806 |
Homo sapiens |
IC50 |
= |
3.143 |
nM |
10.6019/CHEMBL1201861 |
NPT1884 |
Cell Line |
HCC1937 |
Homo sapiens |
IC50 |
= |
349.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2427 |
Cell Line |
HCC1954 |
Homo sapiens |
IC50 |
= |
266.61 |
nM |
10.6019/CHEMBL1201861 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
85.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2428 |
Cell Line |
HT-3 |
Homo sapiens |
IC50 |
= |
0.2119 |
nM |
10.6019/CHEMBL1201861 |
NPT2429 |
Cell Line |
HT55 |
Homo sapiens |
IC50 |
= |
192.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2085 |
Cell Line |
Kasumi 1 |
|
IC50 |
= |
4.066 |
nM |
10.6019/CHEMBL1201861 |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
1.535 |
nM |
10.6019/CHEMBL1201861 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
7.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
124.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
4.095 |
nM |
10.6019/CHEMBL1201861 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
9.948 |
nM |
10.6019/CHEMBL1201861 |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
0.7318 |
nM |
10.6019/CHEMBL1201861 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
1.616 |
nM |
10.6019/CHEMBL1201861 |
NPT2431 |
Cell Line |
NCI-H1437 |
Homo sapiens |
IC50 |
= |
34.93 |
nM |
10.6019/CHEMBL1201861 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
40.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2432 |
Cell Line |
NCI-H2342 |
Homo sapiens |
IC50 |
= |
618.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
3.108 |
nM |
10.6019/CHEMBL1201861 |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
3.793 |
nM |
10.6019/CHEMBL1201861 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
3.069 |
nM |
10.6019/CHEMBL1201861 |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
628.09 |
nM |
10.6019/CHEMBL1201861 |
NPT890 |
Cell Line |
SNU-387 |
Homo sapiens |
IC50 |
= |
256.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2433 |
Cell Line |
SNU-423 |
Homo sapiens |
IC50 |
= |
128.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2434 |
Cell Line |
TCC-SUP |
Homo sapiens |
IC50 |
= |
39.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2435 |
Cell Line |
VM-CUB-1 |
Homo sapiens |
IC50 |
= |
2.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2436 |
Cell Line |
VMRC-RCZ |
Homo sapiens |
IC50 |
= |
47.35 |
nM |
10.6019/CHEMBL1201861 |
NPT1653 |
Cell Line |
WM-115 |
Homo sapiens |
IC50 |
= |
102.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
150.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2437 |
Cell Line |
EW-22 |
Homo sapiens |
IC50 |
= |
0.5566 |
nM |
10.6019/CHEMBL1201861 |
NPT2113 |
Cell Line |
EW-24 |
Homo sapiens |
IC50 |
= |
4.033 |
nM |
10.6019/CHEMBL1201861 |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
55.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2438 |
Cell Line |
HTC-C3 |
Homo sapiens |
IC50 |
= |
31.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
3.382 |
nM |
10.6019/CHEMBL1201861 |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
1.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
10.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
7.897 |
nM |
10.6019/CHEMBL1201861 |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
2.076 |
nM |
10.6019/CHEMBL1201861 |
NPT2439 |
Cell Line |
MC-IXC |
Homo sapiens |
IC50 |
= |
0.513 |
nM |
10.6019/CHEMBL1201861 |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
15.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
27.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2440 |
Cell Line |
NCI-H1563 |
Homo sapiens |
IC50 |
= |
150.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2441 |
Cell Line |
NCI-H2347 |
Homo sapiens |
IC50 |
= |
185.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2442 |
Cell Line |
NCI-H2405 |
Homo sapiens |
IC50 |
= |
58.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
0.441 |
nM |
10.6019/CHEMBL1201861 |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
19.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
0.7753 |
nM |
10.6019/CHEMBL1201861 |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
113.62 |
nM |
10.6019/CHEMBL1201861 |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
2.835 |
nM |
10.6019/CHEMBL1201861 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
3.379 |
nM |
10.6019/CHEMBL1201861 |
NPT2443 |
Cell Line |
SNU-449 |
Homo sapiens |
IC50 |
= |
194.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
35.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
147.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2444 |
Cell Line |
YAPC |
Homo sapiens |
IC50 |
= |
29.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2445 |
Cell Line |
YH-13 |
Homo sapiens |
IC50 |
= |
11.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
0.3192 |
nM |
10.6019/CHEMBL1201861 |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
0.2708 |
nM |
10.6019/CHEMBL1201861 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
150.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2446 |
Cell Line |
HCC38 |
Homo sapiens |
IC50 |
= |
12.86 |
nM |
10.6019/CHEMBL1201861 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
144.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2447 |
Cell Line |
HuCCT-1 |
Homo sapiens |
IC50 |
= |
73.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
332.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2448 |
Cell Line |
KLE |
Homo sapiens |
IC50 |
= |
411.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
87.25 |
nM |
10.6019/CHEMBL1201861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6.427 |
nM |
10.6019/CHEMBL1201861 |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
2.774 |
nM |
10.6019/CHEMBL1201861 |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
8.238 |
nM |
10.6019/CHEMBL1201861 |
NPT2449 |
Cell Line |
NCI-H1573 |
Homo sapiens |
IC50 |
= |
173.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
33.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2450 |
Cell Line |
NCI-H2452 |
Homo sapiens |
IC50 |
= |
90.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2451 |
Cell Line |
NCI-H28 |
Homo sapiens |
IC50 |
= |
38.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
2.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
1.557 |
nM |
10.6019/CHEMBL1201861 |
NPT2453 |
Cell Line |
RCM-1 |
Homo sapiens |
IC50 |
= |
28.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
15.74 |
nM |
10.6019/CHEMBL1201861 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
7.909 |
nM |
10.6019/CHEMBL1201861 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
9.009 |
nM |
10.6019/CHEMBL1201861 |
NPT2455 |
Cell Line |
SNU-C2B |
Homo sapiens |
IC50 |
= |
35.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2456 |
Cell Line |
TE-11 |
Homo sapiens |
IC50 |
= |
16.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
265.25 |
nM |
10.6019/CHEMBL1201861 |
NPT2457 |
Cell Line |
YKG-1 |
Homo sapiens |
IC50 |
= |
5.453 |
nM |
10.6019/CHEMBL1201861 |
NPT994 |
Cell Line |
ZR-75-30 |
Homo sapiens |
IC50 |
= |
261 |
nM |
10.6019/CHEMBL1201861 |
NPT1216 |
Cell Line |
FaDu |
Homo sapiens |
IC50 |
= |
0.5392 |
nM |
10.6019/CHEMBL1201861 |
NPT2458 |
Cell Line |
FTC-133 |
Homo sapiens |
IC50 |
= |
4.567 |
nM |
10.6019/CHEMBL1201861 |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
45.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2460 |
Cell Line |
HCE-4 |
Homo sapiens |
IC50 |
= |
1.814 |
nM |
10.6019/CHEMBL1201861 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
115.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2461 |
Cell Line |
HuO-3N1 |
Homo sapiens |
IC50 |
= |
12.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2462 |
Cell Line |
HuO9 |
Homo sapiens |
IC50 |
= |
2.881 |
nM |
10.6019/CHEMBL1201861 |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
55.67 |
nM |
10.6019/CHEMBL1201861 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
74.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
91.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
196.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
7.569 |
nM |
10.6019/CHEMBL1201861 |
NPT2464 |
Cell Line |
MDA-MB-175-VII |
Homo sapiens |
IC50 |
= |
83.02 |
nM |
10.6019/CHEMBL1201861 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
229.98 |
nM |
10.6019/CHEMBL1201861 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
0.7058 |
nM |
10.6019/CHEMBL1201861 |
NPT2465 |
Cell Line |
NCI-H1623 |
Homo sapiens |
IC50 |
= |
0.7479 |
nM |
10.6019/CHEMBL1201861 |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
38.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
105.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
91.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
0.2738 |
nM |
10.6019/CHEMBL1201861 |
NPT2467 |
Cell Line |
RERF-LC-MS |
Homo sapiens |
IC50 |
= |
22.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
3.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
59.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
1543.63 |
nM |
10.6019/CHEMBL1201861 |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
7.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
174.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
2544.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
IC50 |
= |
19.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2470 |
Cell Line |
G-402 |
Homo sapiens |
IC50 |
= |
24.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
5.469 |
nM |
10.6019/CHEMBL1201861 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5.051 |
nM |
10.6019/CHEMBL1201861 |
NPT2471 |
Cell Line |
HuP-T3 |
Homo sapiens |
IC50 |
= |
36.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2472 |
Cell Line |
HuP-T4 |
Homo sapiens |
IC50 |
= |
0.8814 |
nM |
10.6019/CHEMBL1201861 |
NPT2163 |
Cell Line |
KMOE-2 |
Homo sapiens |
IC50 |
= |
11.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
18.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
34.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2474 |
Cell Line |
MDA-MB-415 |
Homo sapiens |
IC50 |
= |
134.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
20.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
14.11 |
nM |
10.6019/CHEMBL1201861 |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
149.39 |
nM |
10.6019/CHEMBL1201861 |
NPT2475 |
Cell Line |
NCI-H1651 |
Homo sapiens |
IC50 |
= |
14.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2476 |
Cell Line |
NCI-H441 |
Homo sapiens |
IC50 |
= |
28.46 |
nM |
10.6019/CHEMBL1201861 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
56.63 |
nM |
10.6019/CHEMBL1201861 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
3.136 |
nM |
10.6019/CHEMBL1201861 |
NPT2478 |
Cell Line |
NY |
Homo sapiens |
IC50 |
= |
4356.62 |
nM |
10.6019/CHEMBL1201861 |
NPT2479 |
Cell Line |
OAW-28 |
Homo sapiens |
IC50 |
= |
7.263 |
nM |
10.6019/CHEMBL1201861 |
NPT2480 |
Cell Line |
RH-18 |
Homo sapiens |
IC50 |
= |
389.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
4.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2481 |
Cell Line |
SW1088 |
Homo sapiens |
IC50 |
= |
27.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2482 |
Cell Line |
SW 1116 |
Homo sapiens |
IC50 |
= |
190.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2483 |
Cell Line |
SW13 |
Homo sapiens |
IC50 |
= |
2.993 |
nM |
10.6019/CHEMBL1201861 |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
178.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
113.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2175 |
Cell Line |
GAK |
Homo sapiens |
IC50 |
= |
218.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2484 |
Cell Line |
GAMG |
Homo sapiens |
IC50 |
= |
1.527 |
nM |
10.6019/CHEMBL1201861 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
776.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
1.634 |
nM |
10.6019/CHEMBL1201861 |
NPT2485 |
Cell Line |
IA-LM |
Homo sapiens |
IC50 |
= |
12 |
nM |
10.6019/CHEMBL1201861 |
NPT2486 |
Cell Line |
IGR-1 |
Homo sapiens |
IC50 |
= |
151.26 |
nM |
10.6019/CHEMBL1201861 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
36.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
33.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2487 |
Cell Line |
KNS-62 |
Homo sapiens |
IC50 |
= |
7.701 |
nM |
10.6019/CHEMBL1201861 |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
2.806 |
nM |
10.6019/CHEMBL1201861 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
6.965 |
nM |
10.6019/CHEMBL1201861 |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
2.692 |
nM |
10.6019/CHEMBL1201861 |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
8.612 |
nM |
10.6019/CHEMBL1201861 |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
46.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2490 |
Cell Line |
NCI-H1666 |
Homo sapiens |
IC50 |
= |
18.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2491 |
Cell Line |
NCI-H1693 |
Homo sapiens |
IC50 |
= |
26.69 |
nM |
10.6019/CHEMBL1201861 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
24.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2184 |
Cell Line |
NCI-H510A |
Homo sapiens |
IC50 |
= |
1.699 |
nM |
10.6019/CHEMBL1201861 |
NPT2492 |
Cell Line |
OAW-42 |
Homo sapiens |
IC50 |
= |
8.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2493 |
Cell Line |
OC-314 |
Homo sapiens |
IC50 |
= |
2.506 |
nM |
10.6019/CHEMBL1201861 |
NPT2494 |
Cell Line |
RMG-I |
Homo sapiens |
IC50 |
= |
244.5 |
nM |
10.6019/CHEMBL1201861 |
NPT3467 |
Cell Line |
SJRH30 |
Homo sapiens |
IC50 |
= |
298.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
18 |
nM |
10.6019/CHEMBL1201861 |
NPT2495 |
Cell Line |
SW1417 |
Homo sapiens |
IC50 |
= |
52.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2496 |
Cell Line |
SW1463 |
Homo sapiens |
IC50 |
= |
51.69 |
nM |
10.6019/CHEMBL1201861 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
IC50 |
= |
2.348 |
nM |
10.6019/CHEMBL1201861 |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
4.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
23.65 |
nM |
10.6019/CHEMBL1201861 |
NPT1354 |
Cell Line |
TGBC11TKB |
Homo sapiens |
IC50 |
= |
12.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
4.677 |
nM |
10.6019/CHEMBL1201861 |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
486.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2497 |
Cell Line |
HEC-1 |
Homo sapiens |
IC50 |
= |
18.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
19.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2498 |
Cell Line |
KOSC-2 |
Homo sapiens |
IC50 |
= |
4.393 |
nM |
10.6019/CHEMBL1201861 |
NPT2499 |
Cell Line |
KP-4 |
Homo sapiens |
IC50 |
= |
3.162 |
nM |
10.6019/CHEMBL1201861 |
NPT2500 |
Cell Line |
LCLC-103H cell line |
|
IC50 |
= |
20.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
39.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2501 |
Cell Line |
MEL-HO |
Homo sapiens |
IC50 |
= |
7.628 |
nM |
10.6019/CHEMBL1201861 |
NPT2502 |
Cell Line |
MEL-JUSO |
Homo sapiens |
IC50 |
= |
35.62 |
nM |
10.6019/CHEMBL1201861 |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
111.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2503 |
Cell Line |
NCI-H1703 |
Homo sapiens |
IC50 |
= |
6.515 |
nM |
10.6019/CHEMBL1201861 |
NPT2504 |
Cell Line |
NCI-H1755 |
Homo sapiens |
IC50 |
= |
208.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
162.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
0.8868 |
nM |
10.6019/CHEMBL1201861 |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
38.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2506 |
Cell Line |
RO82-W-1 |
Homo sapiens |
IC50 |
= |
14.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2507 |
Cell Line |
RPMI-2650 |
Homo sapiens |
IC50 |
= |
2.217 |
nM |
10.6019/CHEMBL1201861 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
7.253 |
nM |
10.6019/CHEMBL1201861 |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
180.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2508 |
Cell Line |
SW1710 |
Homo sapiens |
IC50 |
= |
33.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2509 |
Cell Line |
SW1783 |
Homo sapiens |
IC50 |
= |
24.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
109.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
66.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2510 |
Cell Line |
GCT |
Homo sapiens |
IC50 |
= |
5.023 |
nM |
10.6019/CHEMBL1201861 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
6.311 |
nM |
10.6019/CHEMBL1201861 |
NPT2511 |
Cell Line |
HGC-27 |
Homo sapiens |
IC50 |
= |
4.073 |
nM |
10.6019/CHEMBL1201861 |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
3.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
10.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2207 |
Cell Line |
KP-N-YN |
Homo sapiens |
IC50 |
= |
102.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
736.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2512 |
Cell Line |
LCLC-97TM1 |
Homo sapiens |
IC50 |
= |
8.136 |
nM |
10.6019/CHEMBL1201861 |
NPT2513 |
Cell Line |
LK-2 |
Homo sapiens |
IC50 |
= |
35.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2514 |
Cell Line |
LN-405 |
Homo sapiens |
IC50 |
= |
517.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2515 |
Cell Line |
MFE-280 |
Homo sapiens |
IC50 |
= |
21.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
0.6143 |
nM |
10.6019/CHEMBL1201861 |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
44.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
157.32 |
nM |
10.6019/CHEMBL1201861 |
NPT1669 |
Cell Line |
NCI-H1792 |
Homo sapiens |
IC50 |
= |
40.12 |
nM |
10.6019/CHEMBL1201861 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4.76 |
% |
23501113 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4.94 |
% |
23501113 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
30.17 |
% |
23501113 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
60.44 |
% |
23501113 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
88 |
nM |
23578545 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
67 |
nM |
23578545 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
0.77 |
% |
23578545 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
30 |
nM |
23578545 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
280 |
nM |
23608763 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
70 |
nM |
23608763 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
37.2 |
% |
23608763 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
70.5 |
% |
23608763 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
32300 |
nM |
23562244 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio |
= |
0.64 |
|
23665106 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
52 |
% |
23602620 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
48.33 |
% |
23602620 |
NPT4475 |
Cell Line |
CEM/C2 |
Homo sapiens |
GI50 |
= |
1000 |
nM |
23750455 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
2 |
nM |
23750455 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
31620 |
nM |
23831811 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
160 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
790 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
50 |
nM |
23831811 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
23831811 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
13 |
nM |
24900725 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
162 |
nM |
24900725 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
99 |
nM |
24900725 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
78 |
nM |
24900725 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
31 |
nM |
24900725 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
26 |
nM |
24900725 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
24 |
nM |
24900725 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
0.04 |
nM |
24900725 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
23816880 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
16 |
nM |
24033077 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
GI50 |
= |
1800 |
nM |
23831507 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
2000 |
nM |
23831507 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
GI50 |
= |
250 |
nM |
23831507 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
600 |
nM |
23831507 |
NPT1723 |
Cell Line |
HBL-100 |
Homo sapiens |
GI50 |
= |
230 |
nM |
23831507 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
60 |
nM |
24041234 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24041234 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
190 |
nM |
24041234 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
50 |
nM |
24041234 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
24041234 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
Activity |
= |
0.67 |
% |
23974020 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
Activity |
= |
3.1 |
% |
23974020 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
Activity |
= |
4.08 |
% |
23974020 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
Activity |
= |
92.16 |
% |
23974020 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
230 |
nM |
23974020 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
37050 |
nM |
23974020 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4470 |
nM |
23974020 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
71.9 |
% |
24090914 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
30.6 |
% |
24090914 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
780 |
nM |
24013413 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
390 |
nM |
24013413 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
420 |
nM |
24013413 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
300 |
nM |
24013413 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
26.1 |
% |
24013413 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
21.6 |
% |
24056146 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
2.4 |
% |
24056146 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
74.8 |
% |
24056146 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
1.2 |
% |
24056146 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
50.5 |
% |
24056146 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
70 |
nM |
24069881 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
< |
1 |
nM |
24069881 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
650 |
nM |
24069881 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
LD50 |
= |
0.16 |
umol/ml |
24075143 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
74.81 |
% |
23571415 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
107.28 |
% |
23571415 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
< |
10 |
nM |
24180210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
24180210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
10 |
nM |
24180210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
24180210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
< |
10 |
nM |
24180210 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
< |
10 |
nM |
24180210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
24200393 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
20 |
nM |
24200393 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3.3 |
nM |
24200393 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
130 |
nM |
24200393 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
800 |
nM |
24303808 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
500 |
nM |
24303808 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
400 |
nM |
24303808 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24303808 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
60 |
nM |
24360564 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
24360564 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
40 |
nM |
24360564 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
> |
10000 |
nM |
24484281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
24484281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300 |
nM |
24484281 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80 |
nM |
24484281 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
35.48 |
nM |
24502276 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
17.38 |
nM |
24502276 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
1000 |
nM |
24502276 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
18.2 |
nM |
24502276 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
40.9 |
% |
24502276 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
13 |
nM |
24502276 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24502276 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
24502276 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
24502276 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24502276 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24502276 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
24502276 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24502276 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1584.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4466.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3548.1 |
nM |
PubChem BioAssay data set |
NPT105 |
Individual Protein |
Muscleblind-like protein 1 |
Homo sapiens |
Potency |
|
2511.9 |
nM |
PubChem BioAssay data set |
NPT105 |
Individual Protein |
Muscleblind-like protein 1 |
Homo sapiens |
Potency |
|
3162.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5011.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
580.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
28183.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2238.7 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
461.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3981.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1778.3 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
46.1 |
% |
10.1039/C3MD00055A |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
53.3 |
% |
10.1039/C3MD00055A |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
61.8 |
% |
10.1039/C3MD00055A |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
0 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
17 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
42 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
40 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
80.5 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
19.5 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
23.5 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
62 |
% |
10.1039/C3MD00399J |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
= |
53 |
% |
10.1039/C3MD00399J |
NPT2 |
Others |
Unspecified |
|
ED50 |
< |
2.8 |
10'-6umol/ml |
423214 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
8.6 |
10'-6umol/ml |
423214 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
2.8 |
10'-6umol/ml |
423214 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2780 |
nM |
24685545 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
24593048 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24800942 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
30 |
nM |
24800942 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
24800942 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
220 |
nM |
24800942 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
24800942 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24800942 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
24800942 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
270 |
nM |
24904965 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
280 |
nM |
24904965 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
4010 |
nM |
24904965 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10070 |
nM |
24904965 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
35.5 |
% |
24904965 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
74 |
% |
24904965 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
60.44 |
% |
24910974 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
30.17 |
% |
24910974 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4.94 |
% |
24910974 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4.76 |
% |
24910974 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
33.1 |
% |
10.1039/C2MD20098H |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
80 |
nM |
25481396 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
400 |
nM |
25481396 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
110 |
nM |
25481396 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
260 |
nM |
25481396 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
< |
0.024 |
ug/ml |
24940955 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
79.6 |
% |
25062005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11 |
% |
25062005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.9 |
% |
25062005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.2 |
% |
25062005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
30.8 |
% |
25062005 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
65.7 |
% |
25062006 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
280 |
nM |
25062006 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
950 |
nM |
25062006 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1980 |
nM |
25062006 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
750 |
nM |
25062006 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
24901491 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
65.1 |
nM |
24901491 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
474 |
nM |
24901491 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
510 |
nM |
24901491 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
786 |
nM |
24901491 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.64 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
15.22 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
36.98 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
51.12 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
81.62 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
83.26 |
% |
24980118 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
420 |
nM |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
56.16 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
41.38 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
13.7 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.4 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.1 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.18 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.76 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.32 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.04 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.12 |
% |
24980118 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
131 |
nM |
24980118 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
187 |
nM |
24980118 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
110 |
nM |
24980118 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
342 |
nM |
24980118 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
29 |
nM |
25003995 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
37 |
nM |
25003995 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
16 |
nM |
25003995 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
120 |
nM |
25003995 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
56.2 |
mg/kg |
25003995 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.5 |
nM |
25084144 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3 |
nM |
25084144 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
25084144 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3600 |
nM |
25237727 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6300 |
nM |
25237727 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
25237727 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1 |
nM |
25237727 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
900 |
nM |
25237727 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.15 |
nM |
25247770 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.6 |
nM |
25247770 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4 |
nM |
25247770 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500000 |
nM |
25221657 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
49 |
% |
25259515 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
96.1 |
% |
25259515 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
126 |
% |
25259515 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
29 |
% |
25881826 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
48.5 |
% |
25881826 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
30 |
% |
25881826 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
130 |
nM |
25590864 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
200 |
nM |
25590864 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
70 |
nM |
25599951 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
5370 |
nM |
25599951 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
11620 |
nM |
25599951 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
26450 |
nM |
25599951 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
2.05 |
ug/ml |
25867737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11.71 |
ug/ml |
25867737 |
NPT1893 |
Cell Line |
MEF |
Mus musculus |
IC50 |
= |
5.87 |
ug/ml |
25867737 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
11.3 |
ug |
25453788 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
45.31 |
% |
25453788 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
80.7 |
% |
25936262 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
40.8 |
% |
25936262 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25936262 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
2820 |
nM |
25936262 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1840 |
nM |
25936262 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
180 |
nM |
25936262 |
NPT1329 |
Cell Line |
Detroit 551 |
Homo sapiens |
IC50 |
= |
990 |
nM |
10.1039/C4MD00133H |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
3140 |
nM |
10.1039/C4MD00133H |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2110 |
nM |
10.1039/C4MD00133H |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
10.1039/C4MD00133H |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
23760 |
nM |
10.1039/C4MD00133H |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220 |
nM |
10.1039/C4MD00133H |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
6000 |
nM |
10.1039/C4MD00133H |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
180 |
nM |
10.1039/C4MD00133H |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
230 |
nM |
26063305 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
20.9 |
% |
26022080 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
58 |
% |
26022080 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
520 |
nM |
26022080 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
310 |
nM |
26022080 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
400 |
nM |
26022080 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
410 |
nM |
26022080 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
100 |
nM |
26226379 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
90 |
nM |
26226379 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
26226379 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
710 |
nM |
26226379 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
960 |
nM |
26226379 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2500 |
nM |
26226379 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
> |
200000 |
nM |
26226379 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
3 |
nM |
26226379 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
< |
3 |
nM |
26226379 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
140 |
nM |
26226379 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25000 |
nM |
26188908 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81 |
% |
26188908 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
15 |
nM |
26188908 |
NPT1917 |
Cell Line |
CA46 |
Homo sapiens |
IC50 |
= |
520 |
nM |
26188908 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
14000 |
nM |
26188908 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1600 |
nM |
26188908 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
44.7 |
% |
26361737 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
110 |
nM |
26361737 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
52.7 |
% |
26361737 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
300 |
nM |
26361737 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
80 |
nM |
26361737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
970 |
nM |
26361737 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
52.4 |
% |
26222449 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
10.1039/C4MD00306C |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
1000 |
nM |
10.1039/C4MD00306C |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25799376 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25799376 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
190 |
nM |
10.1039/C4MD00344F |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
10.1039/C4MD00344F |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
10.1039/C4MD00344F |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
26.9 |
% |
26334499 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
70.9 |
% |
26334499 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
6080 |
nM |
26334499 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1620 |
nM |
26334499 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1590 |
nM |
26334499 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
14760 |
nM |
26602827 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
5770 |
nM |
26602827 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6130 |
nM |
26602827 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4960 |
nM |
26602827 |
NPT2 |
Others |
Unspecified |
|
IC50 |
<= |
100 |
nM |
26810835 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
<= |
100 |
nM |
26810835 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
1000 |
nM |
26810835 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
26810835 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
26649907 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
26649907 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.5 |
|
26649907 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
19800 |
nM |
26649907 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.1 |
|
26649907 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
5500 |
nM |
26649907 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60.9 |
% |
10.1039/C5MD00289C |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
74.8 |
% |
10.1039/C5MD00289C |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
21.6 |
% |
10.1039/C5MD00289C |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
2.4 |
% |
10.1039/C5MD00289C |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
1.2 |
% |
10.1039/C5MD00289C |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
85 |
nM |
26890120 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
58.7 |
% |
26927425 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
27.6 |
% |
26927425 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1290 |
nM |
26927425 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
11170 |
nM |
26927425 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
590 |
nM |
26927425 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
34.7 |
% |
26945111 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
64.7 |
% |
26945111 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
26945111 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2820 |
nM |
26945111 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1840 |
nM |
26945111 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
180 |
nM |
26945111 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7000 |
nM |
26988802 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
73.6 |
% |
26988802 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
24.6 |
% |
26988802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7100 |
nM |
26988802 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
4100 |
nM |
26988802 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
37 |
nM |
26994847 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
16 |
nM |
26994847 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
120 |
nM |
26994847 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
70 |
nM |
27017547 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1 |
nM |
27017547 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.5 |
nM |
27017547 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
350 |
nM |
27156772 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
190 |
nM |
27156772 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
70 |
nM |
27156772 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
23.4 |
% |
27157005 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
8.9 |
% |
27157005 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
39.6 |
% |
27157005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
12.8 |
% |
27157005 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
11.4 |
% |
27157005 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
34.6 |
% |
27157005 |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
Activity |
= |
65 |
% |
27135370 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Activity |
= |
100 |
% |
27070999 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
27070999 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
30 |
nM |
27070999 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
220 |
nM |
27070999 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
20 |
nM |
27070999 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10 |
nM |
27070999 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3 |
nM |
27096049 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
13 |
nM |
27096049 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9 |
nM |
27096049 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
35 |
nM |
27096049 |