Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT1214 | Individual Protein | Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens | Inhibition | = | -7 | % | 10450977 |
NPT1214 | Individual Protein | Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens | Inhibition | = | 3 | % | 10450977 |
NPT3065 | Individual Protein | Acyl coenzyme A:cholesterol acyltransferase 1 | Rattus norvegicus | IC50 | = | 150000 | nM | 15261286 |
NPT1214 | Individual Protein | Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens | IC50 | = | 53000 | nM | 15261286 |
NPT1214 | Individual Protein | Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens | IC50 | = | 45000 | nM | 15261286 |
NPT698 | Individual Protein | Regulator of G-protein signaling 4 | Homo sapiens | Potency | 23778.1 | nM | PubChem BioAssay data set | |
NPT49 | Individual Protein | DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens | Potency | 8912.5 | nM | PubChem BioAssay data set |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC49494 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
1.0 | High Similarity | NPC188341 |
0.9792 | High Similarity | NPC261571 |
0.807 | Intermediate Similarity | NPC325550 |
0.807 | Intermediate Similarity | NPC326524 |
0.807 | Intermediate Similarity | NPC329003 |
0.7895 | Intermediate Similarity | NPC321030 |
0.7667 | Intermediate Similarity | NPC316674 |
0.7647 | Intermediate Similarity | NPC76976 |
0.75 | Intermediate Similarity | NPC28394 |
0.75 | Intermediate Similarity | NPC31557 |
0.7368 | Intermediate Similarity | NPC242930 |
0.7255 | Intermediate Similarity | NPC252978 |
0.7083 | Intermediate Similarity | NPC277333 |
0.7 | Intermediate Similarity | NPC325734 |
0.697 | Remote Similarity | NPC103712 |
0.697 | Remote Similarity | NPC291196 |
0.6769 | Remote Similarity | NPC113224 |
0.6667 | Remote Similarity | NPC261158 |
0.6667 | Remote Similarity | NPC24216 |
0.6667 | Remote Similarity | NPC306420 |
0.6667 | Remote Similarity | NPC4881 |
0.6667 | Remote Similarity | NPC104138 |
0.661 | Remote Similarity | NPC281972 |
0.661 | Remote Similarity | NPC88966 |
0.661 | Remote Similarity | NPC424 |
0.661 | Remote Similarity | NPC154245 |
0.661 | Remote Similarity | NPC87564 |
0.661 | Remote Similarity | NPC85813 |
0.661 | Remote Similarity | NPC6095 |
0.661 | Remote Similarity | NPC25417 |
0.661 | Remote Similarity | NPC32467 |
0.661 | Remote Similarity | NPC290563 |
0.661 | Remote Similarity | NPC261831 |
0.6571 | Remote Similarity | NPC288086 |
0.6552 | Remote Similarity | NPC92114 |
0.6538 | Remote Similarity | NPC241279 |
0.6508 | Remote Similarity | NPC130807 |
0.65 | Remote Similarity | NPC297020 |
0.65 | Remote Similarity | NPC273023 |
0.6491 | Remote Similarity | NPC59051 |
0.6481 | Remote Similarity | NPC108195 |
0.6479 | Remote Similarity | NPC264417 |
0.6479 | Remote Similarity | NPC217095 |
0.6452 | Remote Similarity | NPC210999 |
0.6441 | Remote Similarity | NPC294548 |
0.6441 | Remote Similarity | NPC36061 |
0.6441 | Remote Similarity | NPC321062 |
0.6441 | Remote Similarity | NPC70387 |
0.6441 | Remote Similarity | NPC26102 |
0.6441 | Remote Similarity | NPC187361 |
0.6441 | Remote Similarity | NPC477724 |
0.6441 | Remote Similarity | NPC139029 |
0.6441 | Remote Similarity | NPC1813 |
0.6406 | Remote Similarity | NPC47333 |
0.6393 | Remote Similarity | NPC477201 |
0.6393 | Remote Similarity | NPC18951 |
0.6379 | Remote Similarity | NPC129263 |
0.6349 | Remote Similarity | NPC312826 |
0.6333 | Remote Similarity | NPC49059 |
0.6333 | Remote Similarity | NPC256209 |
0.6316 | Remote Similarity | NPC98284 |
0.6308 | Remote Similarity | NPC55068 |
0.629 | Remote Similarity | NPC302569 |
0.629 | Remote Similarity | NPC168308 |
0.6275 | Remote Similarity | NPC40434 |
0.6275 | Remote Similarity | NPC34873 |
0.6271 | Remote Similarity | NPC281245 |
0.623 | Remote Similarity | NPC477726 |
0.623 | Remote Similarity | NPC477725 |
0.6207 | Remote Similarity | NPC329773 |
0.6167 | Remote Similarity | NPC474496 |
0.6167 | Remote Similarity | NPC303672 |
0.6167 | Remote Similarity | NPC34577 |
0.6154 | Remote Similarity | NPC29468 |
0.614 | Remote Similarity | NPC91495 |
0.614 | Remote Similarity | NPC91044 |
0.6129 | Remote Similarity | NPC187777 |
0.6129 | Remote Similarity | NPC470967 |
0.6129 | Remote Similarity | NPC470969 |
0.6129 | Remote Similarity | NPC471960 |
0.6129 | Remote Similarity | NPC161838 |
0.6129 | Remote Similarity | NPC470966 |
0.6129 | Remote Similarity | NPC475384 |
0.6129 | Remote Similarity | NPC473847 |
0.6129 | Remote Similarity | NPC179764 |
0.6129 | Remote Similarity | NPC477661 |
0.6129 | Remote Similarity | NPC470968 |
0.6102 | Remote Similarity | NPC262968 |
0.6102 | Remote Similarity | NPC474495 |
0.6102 | Remote Similarity | NPC473672 |
0.6094 | Remote Similarity | NPC106851 |
0.6094 | Remote Similarity | NPC274927 |
0.6071 | Remote Similarity | NPC276825 |
0.6061 | Remote Similarity | NPC477106 |
0.6042 | Remote Similarity | NPC151719 |
0.6042 | Remote Similarity | NPC95174 |
0.6034 | Remote Similarity | NPC207815 |
0.6034 | Remote Similarity | NPC5413 |
0.6034 | Remote Similarity | NPC149821 |
0.6032 | Remote Similarity | NPC225929 |
0.6032 | Remote Similarity | NPC470970 |
0.6027 | Remote Similarity | NPC3094 |
0.6 | Remote Similarity | NPC323153 |
0.6 | Remote Similarity | NPC243532 |
0.6 | Remote Similarity | NPC195986 |
0.5974 | Remote Similarity | NPC82799 |
0.5968 | Remote Similarity | NPC475353 |
0.5968 | Remote Similarity | NPC473721 |
0.5968 | Remote Similarity | NPC473896 |
0.5968 | Remote Similarity | NPC52264 |
0.5968 | Remote Similarity | NPC473735 |
0.5968 | Remote Similarity | NPC54766 |
0.5968 | Remote Similarity | NPC473863 |
0.5968 | Remote Similarity | NPC473910 |
0.5968 | Remote Similarity | NPC471992 |
0.5968 | Remote Similarity | NPC274290 |
0.5968 | Remote Similarity | NPC473725 |
0.5965 | Remote Similarity | NPC319709 |
0.5965 | Remote Similarity | NPC289484 |
0.5932 | Remote Similarity | NPC224227 |
0.5932 | Remote Similarity | NPC131623 |
0.5921 | Remote Similarity | NPC477485 |
0.5909 | Remote Similarity | NPC328776 |
0.5909 | Remote Similarity | NPC201939 |
0.5909 | Remote Similarity | NPC320305 |
0.5909 | Remote Similarity | NPC321838 |
0.5902 | Remote Similarity | NPC39633 |
0.5902 | Remote Similarity | NPC139545 |
0.5902 | Remote Similarity | NPC309606 |
0.5897 | Remote Similarity | NPC477487 |
0.5897 | Remote Similarity | NPC474312 |
0.5882 | Remote Similarity | NPC477525 |
0.5873 | Remote Similarity | NPC274396 |
0.5862 | Remote Similarity | NPC207292 |
0.5857 | Remote Similarity | NPC249713 |
0.5857 | Remote Similarity | NPC474812 |
0.5846 | Remote Similarity | NPC5698 |
0.5846 | Remote Similarity | NPC122239 |
0.5833 | Remote Similarity | NPC243539 |
0.5833 | Remote Similarity | NPC151782 |
0.5833 | Remote Similarity | NPC304223 |
0.5833 | Remote Similarity | NPC267340 |
0.5833 | Remote Similarity | NPC54542 |
0.5833 | Remote Similarity | NPC145032 |
0.5821 | Remote Similarity | NPC477707 |
0.5818 | Remote Similarity | NPC249801 |
0.5818 | Remote Similarity | NPC46248 |
0.5818 | Remote Similarity | NPC149668 |
0.5811 | Remote Similarity | NPC212008 |
0.5811 | Remote Similarity | NPC51055 |
0.5811 | Remote Similarity | NPC62293 |
0.5811 | Remote Similarity | NPC140327 |
0.5806 | Remote Similarity | NPC110732 |
0.5806 | Remote Similarity | NPC13011 |
0.5806 | Remote Similarity | NPC124382 |
0.5806 | Remote Similarity | NPC137538 |
0.5806 | Remote Similarity | NPC473532 |
0.5789 | Remote Similarity | NPC475363 |
0.5789 | Remote Similarity | NPC140501 |
0.5789 | Remote Similarity | NPC269074 |
0.5789 | Remote Similarity | NPC210560 |
0.5789 | Remote Similarity | NPC117572 |
0.5789 | Remote Similarity | NPC473972 |
0.5789 | Remote Similarity | NPC24824 |
0.5789 | Remote Similarity | NPC473971 |
0.5789 | Remote Similarity | NPC165651 |
0.5789 | Remote Similarity | NPC474833 |
0.5781 | Remote Similarity | NPC281230 |
0.5781 | Remote Similarity | NPC52012 |
0.5781 | Remote Similarity | NPC192843 |
0.5763 | Remote Similarity | NPC302310 |
0.5758 | Remote Similarity | NPC309877 |
0.5758 | Remote Similarity | NPC174447 |
0.5758 | Remote Similarity | NPC122521 |
0.5758 | Remote Similarity | NPC252809 |
0.5758 | Remote Similarity | NPC251042 |
0.5758 | Remote Similarity | NPC235242 |
0.575 | Remote Similarity | NPC477199 |
0.5738 | Remote Similarity | NPC35519 |
0.5738 | Remote Similarity | NPC179169 |
0.5738 | Remote Similarity | NPC306195 |
0.5738 | Remote Similarity | NPC157781 |
0.5738 | Remote Similarity | NPC181255 |
0.5735 | Remote Similarity | NPC328089 |
0.5735 | Remote Similarity | NPC68343 |
0.5714 | Remote Similarity | NPC270796 |
0.5714 | Remote Similarity | NPC281590 |
0.5714 | Remote Similarity | NPC326521 |
0.5714 | Remote Similarity | NPC28779 |
0.5714 | Remote Similarity | NPC128061 |
0.5714 | Remote Similarity | NPC223677 |
0.5714 | Remote Similarity | NPC10316 |
0.5714 | Remote Similarity | NPC228473 |
0.5714 | Remote Similarity | NPC15162 |
0.5714 | Remote Similarity | NPC200845 |
0.5714 | Remote Similarity | NPC471991 |
0.5694 | Remote Similarity | NPC324638 |
0.5692 | Remote Similarity | NPC469373 |
0.5692 | Remote Similarity | NPC226848 |
0.5692 | Remote Similarity | NPC10017 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC49494 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
0.661 | Remote Similarity | NPD3195 | Phase 2 |
0.661 | Remote Similarity | NPD4266 | Approved |
0.661 | Remote Similarity | NPD3196 | Approved |
0.661 | Remote Similarity | NPD3194 | Approved |
0.6441 | Remote Similarity | NPD3172 | Approved |
0.6308 | Remote Similarity | NPD3210 | Clinical (unspecified phase) |
0.6164 | Remote Similarity | NPD819 | Approved |
0.6164 | Remote Similarity | NPD818 | Approved |
0.6154 | Remote Similarity | NPD6949 | Clinical (unspecified phase) |
0.6102 | Remote Similarity | NPD29 | Approved |
0.6102 | Remote Similarity | NPD28 | Approved |
0.6071 | Remote Similarity | NPD39 | Approved |
0.6066 | Remote Similarity | NPD9652 | Approved |
0.6034 | Remote Similarity | NPD3173 | Approved |
0.6 | Remote Similarity | NPD15 | Approved |
0.6 | Remote Similarity | NPD791 | Approved |
0.6 | Remote Similarity | NPD1082 | Approved |
0.5965 | Remote Similarity | NPD3211 | Approved |
0.5789 | Remote Similarity | NPD4265 | Approved |
0.5789 | Remote Similarity | NPD4222 | Approved |
0.5789 | Remote Similarity | NPD3732 | Approved |
0.5735 | Remote Similarity | NPD3197 | Phase 1 |
0.5714 | Remote Similarity | NPD5326 | Phase 3 |
0.5694 | Remote Similarity | NPD3212 | Clinical (unspecified phase) |
0.5672 | Remote Similarity | NPD835 | Approved |
0.5672 | Remote Similarity | NPD834 | Approved |
PubChem CID   | 6435901 |
ChEMBL   | CHEMBL64122 |
ZINC   |
Molecular Weight:   | 279.26 |
ALogP:   | -0.7903 |
MLogP:   | 3.22 |
XLogP:   | 8.271 |
# Rotatable Bonds:   | 16 |
Polar Surface Area:   | 44.08 |
# H-Bond Aceptor:   | 2 |
# H-Bond Donor:   | 2 |
# Rings:   | 0 |
# Heavy Atoms:   | 20 |