Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
2500 |
nM |
10.1016/S0960-894X(01)81034-9 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
< |
0.3 |
ug/ml |
1992152 |
NPT561 |
Organism |
Tetrahymena pyriformis |
Tetrahymena pyriformis |
MIC |
> |
20 |
ug/ml |
1992152 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
2500 |
nM |
7381854 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Ki |
= |
5750 |
nM |
7381854 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
IC50 |
= |
1900 |
nM |
10.1016/S0960-894X(01)81233-6 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED |
= |
0.05 |
ug/ml |
2362275 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
IC50 |
= |
1500 |
nM |
10.1016/S0960-894X(00)80225-5 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.62 |
nM |
10.1016/S0960-894X(00)80225-5 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
71 |
nM |
10.1016/S0960-894X(00)80225-5 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
IC50 |
= |
4168.69 |
nM |
10649972 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.4 |
nM |
1433180 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Inhibition |
= |
100 |
% |
9836614 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
1900 |
nM |
9836614 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25 |
nM |
12431060 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
12431060 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ID50 |
= |
2.2 |
ug/ml |
6502608 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ID50 |
= |
6 |
nM ml-1 |
6502608 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
IC50 |
= |
800 |
nM |
8164254 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12852768 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
12852768 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
30 |
nM |
12852768 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50 |
nM |
12852768 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
50 |
nM |
12852768 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
70 |
nM |
12852768 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
20 |
nM |
12852768 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
10000 |
nM |
12852768 |
NPT2688 |
Organism |
Sus scrofa |
Sus scrofa |
IC50 |
= |
1400 |
nM |
12852768 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1260 |
nM |
12852768 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
1.6 |
mg/kg |
4032423 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
IC50 |
= |
800 |
nM |
11689079 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1500 |
nM |
9083485 |
NPT1917 |
Cell Line |
CA46 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
9083485 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
10000 |
nM |
9873473 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
1.6 |
mg/kg |
7241524 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
1.4 |
mg/kg |
7241524 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
Inhibition |
= |
4 |
% |
10571149 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
Inhibition |
= |
3 |
% |
10571149 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
Inhibition |
= |
0 |
% |
10571149 |
NPT309 |
Cell Line |
1A9 |
Homo sapiens |
IC50 |
> |
2500 |
nM |
10571149 |
NPT310 |
Cell Line |
1A9/ptx-10 |
Homo sapiens |
IC50 |
> |
2500 |
nM |
10571149 |
NPT5191 |
Cell Line |
1A9/ptx-22 |
Homo sapiens |
IC50 |
> |
2500 |
nM |
10571149 |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
IC50 |
= |
93.1 |
nM |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
228.3 |
nM |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
51.5 |
nM |
10.1016/0960-894X(95)00300-I |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
4.4 |
|
10.1016/0960-894X(95)00300-I |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.4 |
nM |
2795608 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
50 |
nM |
9871709 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
< |
50 |
nM |
9871709 |
NPT2505 |
Cell Line |
NCI-H520 |
|
GI50 |
< |
50 |
nM |
9871709 |
NPT875 |
Organism |
Bos taurus |
Bos taurus |
IC50 |
= |
11800 |
nM |
9871709 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
140 |
nM |
11814821 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
46 |
nM |
11814821 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
Ki |
= |
780 |
nM |
11814821 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
29300 |
nM |
12372531 |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
GI50 |
= |
0.0315 |
ug/ml |
12372531 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
0.0084 |
ug/ml |
12372531 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
11200 |
nM |
10091693 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
8700 |
nM |
10091693 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
< |
50 |
nM |
10091693 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
50 |
nM |
10091693 |
NPT2505 |
Cell Line |
NCI-H520 |
|
GI50 |
< |
50 |
nM |
10091693 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
800000 |
nM |
11354375 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7500 |
nM |
10.1016/S0960-894X(01)81108-2 |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
Ki |
= |
2500 |
nM |
10.1016/S0960-894X(01)81108-2 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
IC50 |
= |
11200000 |
nM |
9371249 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Activity |
= |
1 |
|
9371249 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1900 |
nM |
8387598 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1.8 |
nM |
10602712 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
10602712 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
IC50 |
= |
5100 |
nM |
8459402 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
37.2 |
% |
8459402 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
89.7 |
% |
8459402 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Potency |
= |
0.4 |
uM/kg |
6620299 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.4 |
nM |
1479582 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
11200 |
nM |
10.1016/S0960-894X(97)00327-2 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Potency |
= |
0.4 |
uM/kg |
7265112 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Inhibition |
= |
100 |
% |
9357519 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
2100 |
nM |
9357519 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
1700 |
nM |
9357519 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
30 |
nM |
9357519 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
= |
2.4 |
mg/kg |
6218302 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
= |
13.2 |
mg/kg |
6218302 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
3.5 |
mg/kg |
6218302 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
13.5 |
mg/kg |
6218302 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
10743950 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
IC50 |
= |
3500 |
nM |
10.1016/S0960-894X(01)81230-0 |
NPT1597 |
Cell Line |
J774.2 |
|
ED50 |
= |
0.06 |
nM |
1956052 |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
ED50 |
= |
0.2 |
nM |
1956052 |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
ED50 |
= |
0.017 |
nM |
1956052 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.012 |
nM |
1956052 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.47 |
nM |
1956052 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
800 |
nM |
11087572 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
IC50 |
= |
800 |
nM |
9216846 |
NPT3804 |
Cell Line |
Human Tumor Cell lines |
|
GI50 |
= |
57.54 |
nM |
9216846 |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
IC50 |
= |
2400 |
nM |
2299625 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
40 |
nM |
2299625 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11.9 |
nM |
12270161 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
> |
100 |
nM |
12270161 |
NPT309 |
Cell Line |
1A9 |
Homo sapiens |
IC50 |
= |
11.9 |
nM |
12270161 |
NPT1298 |
Cell Line |
A9 |
Mus musculus |
IC50 |
= |
13.8 |
nM |
12270161 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
9544215 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
9544215 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
ED50 |
= |
0.016 |
ug/ml |
9544215 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
ED50 |
|
0.4 |
ug/ml |
9544215 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
> |
0.4 |
ug/ml |
9544215 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.008 |
ug/ml |
9544215 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
800 |
nM |
9544215 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
23 |
nM |
11741473 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
11741473 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1400 |
nM |
9632366 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
800 |
nM |
9301667 |
NPT3804 |
Cell Line |
Human Tumor Cell lines |
|
GI50 |
= |
57.54 |
nM |
9301667 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
800 |
nM |
7932568 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
63.1 |
nM |
8496915 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
GI50 |
< |
112.2 |
nM |
8496915 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
< |
63.1 |
nM |
8496915 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
< |
63.1 |
nM |
8496915 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
< |
63.1 |
nM |
8496915 |
NPT5198 |
Cell Line |
OVCAR |
Homo sapiens |
GI50 |
< |
63.1 |
nM |
8496915 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
4200 |
nM |
8496915 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
2 |
nM |
8496935 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
18 |
nM |
8496935 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
ED50 |
= |
175 |
nM |
8496935 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
100 |
nM |
8496935 |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
ED50 |
= |
1 |
nM |
8496935 |
NPT672 |
Cell Line |
TE-671 |
Homo sapiens |
ED50 |
= |
1 |
nM |
8496935 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
4200 |
nM |
8496935 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Inhibition |
= |
26 |
% |
8496935 |
NPT5292 |
Cell Line |
Burkitts lymphoma cells |
|
IC50 |
= |
50 |
nM |
8496935 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
14 |
nM |
12773051 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
EC50 |
= |
6 |
nM |
12773051 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
EC50 |
= |
190 |
nM |
12773051 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
IC50 |
> |
50000 |
nM |
12699389 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
0.1 |
nM/mg*min |
12699389 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Inhibition |
= |
8 |
% |
12699389 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
> |
50000 |
nM |
12699389 |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
IC50 |
> |
50000 |
nM |
12699389 |
NPT1456 |
Individual Protein |
P-glycoprotein 1 |
Mus musculus |
IC50 |
> |
50000 |
nM |
12699389 |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
Ratio |
= |
0.8 |
|
12699389 |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
Ratio |
= |
1.8 |
|
12699389 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1500 |
nM |
9599244 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
0.002 |
ug/ml |
9599244 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
0.022 |
ug/ml |
9599244 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
> |
0.4 |
ug/ml |
9599244 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
EC50 |
= |
0.4 |
ug/ml |
9599244 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
EC50 |
= |
0.008 |
ug/ml |
9599244 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15.3 |
nM |
7990108 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
5 |
nM |
7990108 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
6.9 |
nM |
7990108 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
14 |
nM |
7990108 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
6 |
nM |
7990108 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
5.6 |
nM |
7990108 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
14.1 |
nM |
7990108 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
5.2 |
nM |
7990108 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
9.5 |
nM |
7990108 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
14.7 |
nM |
7990108 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
20.5 |
nM |
7990108 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
18 |
nM |
7990108 |
NPT3360 |
Individual Protein |
Tubulin alpha-1 chain |
Rattus norvegicus |
Inhibition |
= |
93 |
% |
6094813 |
NPT517 |
Cell Line |
Panel NCI-60 (60 carcinoma cell lines) |
Homo sapiens |
GI50 |
= |
1.7 |
nM |
15743190 |
NPT2688 |
Organism |
Sus scrofa |
Sus scrofa |
Inhibition |
= |
78 |
% |
15603947 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Inhibition |
= |
80 |
% |
16198562 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
Inhibition |
= |
80 |
% |
16198562 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
EC50 |
= |
2.8 |
nM |
16198562 |
NPT517 |
Cell Line |
Panel NCI-60 (60 carcinoma cell lines) |
Homo sapiens |
GI50 |
= |
5.8 |
|
16539384 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
19.6 |
|
16539384 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
2700 |
nM |
16570932 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1700 |
nM |
16504507 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
11 |
nM |
16504507 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Inhibition |
= |
78 |
% |
16870433 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
16 |
nM |
16970401 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
5000 |
nM |
16970401 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
500 |
nM |
16970401 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
17034147 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
15 |
nM |
17154496 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
13.3 |
nM |
17154496 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
117 |
nM |
17154496 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3300 |
nM |
17154496 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17181164 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
17181164 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
17181164 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17181164 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17181164 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
70 |
nM |
17181164 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
10000 |
nM |
17181164 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
20 |
nM |
17181164 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
1.06 |
nM |
17181164 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
14 |
nM |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
26.6 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.4 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.1 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
35.7 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11.9 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.1 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.2 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.1 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.6 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.1 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
87.6 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.7 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.5 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
63.3 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.7 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.3 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.2 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.5 |
% |
17181164 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.3 |
% |
17181164 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2.75 |
nM |
17249649 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
522 |
nM |
17249649 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1.84 |
nM |
17249649 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.3 |
nM |
17286393 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
63 |
nM |
17286393 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17286393 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
39.8 |
nM |
17286393 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
15566282 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13 |
nM |
15566282 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
14 |
nM |
15566300 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
34 |
nM |
15566300 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
EC50 |
= |
190 |
nM |
15566300 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3 |
% |
16279766 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
14 |
% |
16279766 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
83 |
% |
16279766 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
18 |
nM |
17275318 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
17497841 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13 |
nM |
17497841 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Ki |
= |
1600 |
10^5/M |
17497841 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
4 |
nM |
17498960 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
15 |
nM |
17498960 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
9 |
nM |
17498960 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
84.1 |
% |
17567121 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
4 |
% |
17567121 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
11.9 |
% |
17567121 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
59 |
% |
17602466 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
71.2 |
% |
17602466 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
17602466 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12 |
nM |
17685504 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
120 |
nM |
17685504 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
19 |
nM |
17685504 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
13 |
nM |
17685504 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
2900 |
nM |
17685504 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
57.9 |
% |
17512729 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
23.1 |
% |
17512729 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
19 |
% |
17512729 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17889547 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1 |
% |
17889547 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17973361 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
17973361 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1050 |
nM |
17973361 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
17973361 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17973361 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
70 |
nM |
17973361 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
20 |
nM |
17973361 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
14000 |
nM |
17973361 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17973361 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
14 |
nM |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
26.6 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.4 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.1 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
35.7 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11.9 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.1 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.2 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.1 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
63.3 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.7 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.6 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.1 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
87.6 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.7 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.5 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.3 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.2 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.5 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.3 |
% |
17973361 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
371.54 |
nM |
17890094 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
22.91 |
nM |
17890094 |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
IC50 |
= |
210 |
nM |
17637068 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
9 |
nM |
18197614 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
15 |
nM |
18197614 |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
EC50 |
= |
4 |
nM |
18197614 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7 |
nM |
18197614 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3800 |
nM |
18083556 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
18083520 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1995.26 |
nM |
18083520 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
44900 |
nM |
18321710 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
50 |
% |
18366178 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
4 |
nM |
18502639 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
15 |
nM |
18502639 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
9 |
nM |
18502639 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
19 |
% |
18502639 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
62 |
% |
18502639 |
NPT2 |
Others |
Unspecified |
|
ID50 |
= |
0.006 |
nM |
3598594 |
NPT24 |
Organism |
Human immunodeficiency virus 1 |
Human immunodeficiency virus 1 |
IC50 |
= |
18 |
nM |
1919593 |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
EC50 |
= |
10 |
nM |
1919593 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
21 |
ug/ml |
11473441 |
NPT1881 |
Uncleic Acid |
Calf thymus DNA |
Bos taurus |
Activity |
< |
30 |
% |
1812211 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Activity |
< |
30 |
% |
1812211 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
12.59 |
nM |
18386884 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
125.89 |
nM |
18386884 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
25.12 |
nM |
18386884 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
25.12 |
nM |
18386884 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
15.85 |
nM |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
316.23 |
nM |
18386884 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
10 |
nM |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
23.3 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
10.2 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
55.2 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
11.3 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
60 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
6.9 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
21.6 |
% |
18386884 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
11.5 |
% |
18386884 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Activity |
= |
72 |
% |
18678497 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7 |
nM |
19282188 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
19282188 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
8.8 |
% |
18440099 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
16.6 |
% |
18440099 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
74.6 |
% |
18440099 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
14.59 |
% |
18440099 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2400 |
nM |
2095370 |
NPT26 |
Individual Protein |
Reverse transcriptase |
Human immunodeficiency virus 1 |
IC50 |
> |
200 |
ug/ml |
1710653 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
32 |
nM |
19530698 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
29 |
nM |
19530698 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
19530698 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
26 |
nM |
19530698 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2100 |
nM |
19530698 |
NPT3638 |
Organism |
BK polyomavirus |
BK polyomavirus |
EC50 |
= |
22 |
nM |
17893158 |
NPT2 |
Others |
Unspecified |
|
Ratio CC50/EC50 |
= |
3.63 |
|
17893158 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
100 |
nM |
8988604 |
NPT76 |
Cell Line |
C6 |
Rattus norvegicus |
LC50 |
= |
200 |
nM |
8988604 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
650 |
nM |
14987069 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
15043436 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
90 |
% |
3879267 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
3 |
umol/kg |
3879267 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.6 |
ug/ml |
15165134 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
15165134 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
15165134 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
15165134 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
20 |
nM |
18503262 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2200 |
nM |
18503262 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
29 |
nM |
18503262 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
45 |
nM |
18503262 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
40 |
nM |
18503262 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
70 |
nM |
18503262 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
40 |
nM |
18503262 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
18503262 |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
Activity |
= |
101 |
% |
18457386 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
990 |
nM |
18778046 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2200 |
nM |
18778046 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.7 |
nM |
18783207 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
Inhibition |
= |
31.9 |
% |
18788725 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
19117761 |
NPT2433 |
Cell Line |
SNU-423 |
Homo sapiens |
IC50 |
= |
25 |
nM |
19117761 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19117761 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
25 |
nM |
19117761 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19220018 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
19220018 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
19220018 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19220018 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19220018 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19220018 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
10 |
nM |
19220018 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
3000 |
nM |
19220018 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
14 |
nM |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
26.6 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.1 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
63.3 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.4 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.7 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.1 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10.6 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
64.3 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
35.7 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.1 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.2 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11.9 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
87.6 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.5 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.1 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.7 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.3 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.2 |
% |
19220018 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94.5 |
% |
19220018 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1060 |
nM |
19220018 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1400 |
nM |
7623025 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
8277312 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
70 |
% |
8277312 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
8277312 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
8133298 |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
8133298 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.007 |
ug/ml |
8133298 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.005 |
ug/ml |
8133298 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
8133298 |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
7528785 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
7528785 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.6 |
ug/ml |
7528785 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
3.5 |
ug/ml |
7528785 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
7528785 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
7528785 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
18 |
nM |
2778449 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
> |
40 |
mm |
2778449 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
40 |
mm |
2778449 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
25 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
24 |
nM |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
> |
40 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
40 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
17.5 |
mm |
2778449 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
8133298 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
70 |
% |
8133298 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
8133298 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
7.4 |
ug/ml |
8133298 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
8133298 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.008 |
ug/ml |
8133298 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
8133298 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
ED50 |
= |
0.004 |
ug/ml |
8133298 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
8133298 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
3.5 |
ug/ml |
8133298 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
15620246 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.2 |
ug/ml |
15620246 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
0.3 |
ug/ml |
15620246 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
15620246 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.7 |
ug/ml |
15620246 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.6 |
ug/ml |
15620246 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.23 |
ug/ml |
7130986 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.01078 |
ug/ml |
19138858 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
= |
16 |
nM |
15730238 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
EC50 |
= |
30 |
nM |
15730238 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
EC50 |
= |
25 |
nM |
15730238 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
3.7 |
ug/ml |
15730238 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
2.8 |
ug/ml |
15730238 |
NPT729 |
Organism |
Micrococcus luteus |
Micrococcus luteus |
MIC |
> |
500 |
ug/ml |
15730238 |
NPT602 |
Organism |
Mycobacterium smegmatis |
Mycobacterium smegmatis |
MIC |
> |
500 |
ug/ml |
15730238 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
MIC |
> |
500 |
ug/ml |
15730238 |
NPT21 |
Organism |
Aspergillus niger |
Aspergillus niger |
MIC |
> |
500 |
ug/ml |
15730238 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
10395506 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
9 |
nM |
18617414 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
15 |
nM |
18617414 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
4 |
nM |
18617414 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
19 |
% |
18617414 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
62 |
% |
18617414 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
9 |
nM |
18651728 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
15 |
nM |
18651728 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
18651728 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11.4 |
nM |
18588280 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
20.2 |
nM |
18588280 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
11 |
nM |
18588280 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
125 |
nM |
18588280 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3000 |
nM |
18588280 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
4 |
nM |
18579387 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
15 |
nM |
18579387 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
9 |
nM |
18579387 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
19 |
% |
18579387 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
62 |
% |
18579387 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1 |
|
18583138 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
31 |
nM |
18583138 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.003 |
nM |
18583138 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
39 |
nM |
18684625 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
31 |
nM |
18684625 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
EC50 |
= |
14 |
nM |
18684625 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
EC50 |
= |
530 |
nM |
18684625 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
EC50 |
= |
390 |
nM |
18684625 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
EC50 |
= |
270 |
nM |
18684625 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11 |
nM |
19053773 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
116 |
nM |
19053773 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
18 |
nM |
19053773 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19053773 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
13 |
nM |
19053773 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
19053773 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29 |
nM |
19243174 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19243174 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19243174 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
11 |
nM |
19243174 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
16 |
nM |
19243174 |
NPT5294 |
Cell Line |
PPC-1 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19243174 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
19394823 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
9 |
nM |
19464890 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
50 |
nM |
19464890 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
19464890 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.043 |
nM |
19394222 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11 |
nM |
19586033 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
18 |
nM |
19586033 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19586033 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
42.83 |
% |
19586033 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
76.95 |
% |
19586033 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
977 |
nM |
19586033 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
19586033 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
19369076 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
14 |
nM |
19500976 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
EC50 |
= |
180 |
nM |
19500976 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
50 |
nM |
19500976 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
140 |
nM |
19500976 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
63 |
nM |
19500976 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
19502058 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
548 |
nM |
19502058 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7.3 |
nM |
19502058 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2600 |
nM |
19837594 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
8.9 |
% |
20034800 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
20170097 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
290 |
nM |
20170097 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12 |
nM |
20148562 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
12.4 |
nM |
20148562 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
13.2 |
nM |
20148562 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
20.1 |
nM |
20148562 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
128 |
nM |
20148562 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4200 |
nM |
20148562 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13.4 |
nM |
20334421 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
8 |
nM |
20334421 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
13 |
nM |
20363142 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10900 |
nM |
20363142 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
59 |
% |
20411988 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
4 |
% |
20411988 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
53 |
nM |
20411988 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
20411988 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Ratio IC50 |
> |
1000 |
|
20411988 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20529690 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12 |
nM |
20529690 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17 |
nM |
20493717 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
20493717 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
24.31 |
% |
20493717 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.96 |
% |
20493717 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
32.28 |
% |
20493717 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
800 |
nM |
20187635 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1500 |
nM |
20187635 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20537765 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
20537765 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
20537765 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50 |
nM |
20537765 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
50 |
nM |
20537765 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
70 |
nM |
20537765 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
20 |
nM |
20537765 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
10000 |
nM |
20537765 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
14 |
nM |
20537765 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20546980 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
1400 |
nM |
20546980 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
LD50 |
= |
0.02 |
nM |
20674369 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
= |
85 |
% |
20674369 |
NPT1893 |
Cell Line |
MEF |
Mus musculus |
Activity |
= |
57 |
% |
20674369 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
ED50 |
= |
0.054 |
ug/ml |
20542428 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.0199 |
ug/ml |
20542428 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
ED50 |
= |
0.0027 |
ug/ml |
20542428 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
ED50 |
= |
0.0027 |
ug/ml |
20542428 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.0038 |
ug/ml |
20542428 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.1578 |
ug/ml |
20542428 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
12589.25 |
nM |
19734910 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2400000 |
nM |
18070965 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2500000 |
nM |
18070965 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2500 |
nM |
18070965 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20919720 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29 |
nM |
20919720 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
16 |
nM |
20919720 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
11 |
nM |
20919720 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
20919720 |
NPT5294 |
Cell Line |
PPC-1 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20919720 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
20919720 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
658 |
nM |
20919720 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
65.8 |
nM |
20919720 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
20919720 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
= |
0 |
mm |
20739103 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
53.8 |
% |
20833451 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
20833451 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
20833451 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
< |
1000 |
nM |
20833451 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17 |
nM |
21036623 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
21036623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
14.58 |
% |
21036623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
8.58 |
% |
21036623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
8.16 |
% |
21036623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
43.11 |
% |
21036623 |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
63.1 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
50.1 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
8.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
125.9 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
31.6 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
158.5 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
100 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
39.8 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
125.9 |
nM |
PubChem BioAssay data set |
NPT537 |
Individual Protein |
Ras-related protein Rab-9A |
Homo sapiens |
Potency |
= |
580478.9 |
nM |
PubChem BioAssay data set |
NPT537 |
Individual Protein |
Ras-related protein Rab-9A |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
79.4 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
12.6 |
nM |
PubChem BioAssay data set |
NPT442 |
Individual Protein |
Ferritin light chain |
Equus caballus |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
10 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
20 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
20 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
11220.2 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
25.1 |
nM |
PubChem BioAssay data set |
NPT794 |
Individual Protein |
Endonuclease 4 |
Escherichia coli K-12 |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
70.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
62.79 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
14125.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
631 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
501.2 |
nM |
PubChem BioAssay data set |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
100 |
nM |
PubChem BioAssay data set |
NPT56 |
Individual Protein |
Beta-lactamase AmpC |
Escherichia coli K-12 |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
50.1 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
100000 |
nM |
PubChem BioAssay data set |
NPT1834 |
Individual Protein |
CREB-binding protein |
Homo sapiens |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Potency |
= |
891.3 |
nM |
PubChem BioAssay data set |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
501.2 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
1584.9 |
nM |
PubChem BioAssay data set |
NPT277 |
Individual Protein |
Caspase-1 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
50.1 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
199.5 |
nM |
PubChem BioAssay data set |
NPT1416 |
Individual Protein |
Neuropeptide S receptor |
Homo sapiens |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Potency |
= |
794.3 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
= |
39.8 |
nM |
PubChem BioAssay data set |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3548.1 |
nM |
PubChem BioAssay data set |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Kd |
= |
3700 |
nM |
21106379 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
16.6 |
nM |
21106379 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
17 |
nM |
21126027 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21126027 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
IC50 |
= |
14 |
nM |
21126027 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
14 |
nM |
21126027 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
13 |
nM |
21126027 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
16 |
nM |
21126027 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
33 |
nM |
21126027 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
2000 |
nM |
21126027 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
79 |
% |
21126027 |
NPT61 |
Individual Protein |
Beta-glucocerebrosidase |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
460.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
30 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
73.1 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
58 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
843.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
160 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
10000 |
nM |
PubChem BioAssay data set |
NPT62 |
Individual Protein |
6-phospho-1-fructokinase |
Trypanosoma brucei |
Potency |
|
37.9 |
nM |
PubChem BioAssay data set |
NPT135 |
Individual Protein |
Chromobox protein homolog 1 |
Homo sapiens |
Potency |
|
3.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
80000 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
33.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2310.9 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
23099.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
58 |
nM |
PubChem BioAssay data set |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
AC50 |
= |
3162.28 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
AC50 |
= |
12589.25 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
AC50 |
= |
2511.89 |
nM |
PubChem BioAssay data set |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
25118.86 |
nM |
PubChem BioAssay data set |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
AC50 |
= |
794.33 |
nM |
PubChem BioAssay data set |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
21440448 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
21440448 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
0.5 |
ug/ml |
21440448 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.3 |
ug/ml |
21440448 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
90.46 |
% |
21440448 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
2.65 |
% |
21440448 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
2.29 |
% |
21440448 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
40 |
nM |
21480626 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
53.2 |
nM |
21480626 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
71.2 |
nM |
21480626 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
21.9 |
nM |
21480626 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
50.6 |
nM |
21480626 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
37 |
nM |
21480626 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
10 |
nM |
21480626 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
2680 |
nM |
21480626 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
7.3 |
nM |
21536450 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
101 |
nM |
21536450 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
17.2 |
nM |
21536450 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
63.6 |
% |
21530013 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21530013 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
50 |
% |
21530013 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21563750 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
27 |
nM |
21563750 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
29 |
nM |
21563750 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
23 |
nM |
21563750 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17 |
nM |
21563750 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21563750 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
21 |
nM |
21563750 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
89 |
nM |
21563750 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
21563750 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
220 |
nM |
21604746 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
21604746 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.9 |
nM |
21604746 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28 |
nM |
21604746 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13 |
nM |
21604746 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21604746 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
1.1 |
nM |
21604746 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
21604746 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2.1 |
nM |
21604746 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
7.9 |
nM |
21604746 |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
IC50 |
= |
140 |
nM |
21604746 |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
Ratio IC50 |
= |
0.64 |
|
21604746 |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
IC50 |
= |
620 |
nM |
21604746 |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
Ratio IC50 |
= |
2.8 |
|
21604746 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
21604746 |
NPT2828 |
Cell Line |
CEM-VLB |
Homo sapiens |
Ratio IC50 |
= |
46 |
|
21604746 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21705223 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
21705223 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50 |
nM |
21705223 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
50 |
nM |
21705223 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
70 |
nM |
21705223 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
21705223 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
21705223 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
14 |
nM |
21705223 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1400 |
nM |
21705223 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1060 |
nM |
21705223 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
21576023 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
21576023 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
21724404 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21775150 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
21775150 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
20 |
nM |
21775150 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21775150 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21775150 |
NPT5294 |
Cell Line |
PPC-1 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21775150 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
0.5 |
ug/ml |
21783370 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.3 |
ug/ml |
21783370 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
1.58 |
% |
21783370 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
1.3 |
% |
21783370 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
61.11 |
% |
21783370 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
10 |
nM |
21641700 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
121 |
nM |
21641700 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21641700 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
15 |
nM |
21641700 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
12 |
nM |
21641700 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4100 |
nM |
21641700 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
27 |
nM |
21873068 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
17 |
nM |
21557538 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
1113 |
nM |
21557538 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
65 |
|
21557538 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1960 |
nM |
21851083 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
58 |
% |
21851083 |
NPT546 |
Individual Protein |
Retinoid X receptor alpha |
Homo sapiens |
Potency |
|
31.6 |
nM |
PubChem BioAssay data set |
NPT546 |
Individual Protein |
Retinoid X receptor alpha |
Homo sapiens |
Potency |
|
25.1 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
9285 |
nM |
PubChem BioAssay data set |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
|
1.3 |
nM |
PubChem BioAssay data set |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
|
44.7 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
9528.3 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
31.6 |
nM |
PubChem BioAssay data set |
NPT249 |
Individual Protein |
Glucocorticoid receptor |
Homo sapiens |
Potency |
|
4466.8 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
29934.9 |
nM |
PubChem BioAssay data set |
NPT803 |
Individual Protein |
Flap endonuclease 1 |
Homo sapiens |
Potency |
|
6701.6 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
11.2 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
35.5 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
112.2 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
17.8 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
25.1 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
70.8 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
10 |
nM |
PubChem BioAssay data set |
NPT108 |
Individual Protein |
Estrogen receptor alpha |
Homo sapiens |
Potency |
|
4466.8 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
7943.3 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
31.6 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
18526 |
nM |
PubChem BioAssay data set |
NPT154 |
Individual Protein |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
Potency |
|
1122 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
73 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1412.5 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
79.4 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
25.1 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
50.1 |
nM |
PubChem BioAssay data set |
NPT249 |
Individual Protein |
Glucocorticoid receptor |
Homo sapiens |
Potency |
|
707.9 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
9466.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
163.5 |
nM |
PubChem BioAssay data set |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT546 |
Individual Protein |
Retinoid X receptor alpha |
Homo sapiens |
Potency |
|
39.8 |
nM |
PubChem BioAssay data set |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
220 |
nM |
21920638 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
21920638 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.9 |
nM |
21920638 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28 |
nM |
21920638 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13 |
nM |
21920638 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21920638 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
1.1 |
nM |
21920638 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
21920638 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2.1 |
nM |
21920638 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
7.9 |
nM |
21920638 |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
IC50 |
= |
140 |
nM |
21920638 |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
Ratio IC50 |
= |
0.64 |
|
21920638 |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
IC50 |
= |
620 |
nM |
21920638 |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
Ratio IC50 |
= |
2.8 |
|
21920638 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
21920638 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
46 |
|
21920638 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
2 |
% |
22189271 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
3 |
% |
22189271 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
85 |
% |
22189271 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
3.42 |
% |
22192936 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
2.43 |
% |
22192936 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
Activity |
= |
75.24 |
% |
22192936 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.53 |
ug/ml |
22261027 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.75 |
ug/ml |
22261027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.72 |
ug/ml |
22261027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
2 |
% |
22261027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3 |
% |
22261027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
79 |
% |
22261027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5 |
nM |
22044164 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
22044164 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
10.3 |
nM |
22060033 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
16.2 |
nM |
22060033 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
19.2 |
nM |
22060033 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
54 |
nM |
24900316 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8 |
nM |
24900316 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
11 |
nM |
24900316 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
32.8 |
% |
24900316 |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
41.3 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
199.07 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
16.41 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
559.76 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
659.17 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
11.38 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
14.59 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
13.46 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
19.19 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
30.69 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
23.71 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
845.28 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
25.82 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
24.15 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
21.13 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
28.18 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
7177.94 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
89.1 |
nM |
PubChem BioAssay data set |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
GI50 |
|
14.29 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
345.14 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
23659.2 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
22.13 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
11.94 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
14.26 |
nM |
PubChem BioAssay data set |
NPT573 |
Cell Line |
M19-MEL |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
14.55 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
17.26 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
24.66 |
nM |
PubChem BioAssay data set |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
GI50 |
|
18.54 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
101.8 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
12882.5 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
17.46 |
nM |
PubChem BioAssay data set |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
20.61 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
11.67 |
nM |
PubChem BioAssay data set |
NPT575 |
Cell Line |
KM-20L2 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
17.54 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
59.43 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
25.88 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
121.9 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
16.83 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
64.27 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
48977.88 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
23.17 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT731 |
Cell Line |
LXFL 529 |
Homo sapiens |
GI50 |
|
11.22 |
nM |
PubChem BioAssay data set |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
GI50 |
|
44.77 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
75.68 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
78342.96 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
20.56 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
100.93 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
24.6 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
14.39 |
nM |
PubChem BioAssay data set |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
GI50 |
|
1361.44 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
10 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
24.77 |
nM |
PubChem BioAssay data set |
NPT577 |
Cell Line |
RXF 631 |
Homo sapiens |
GI50 |
|
36.31 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
32.43 |
nM |
PubChem BioAssay data set |
NPT578 |
Cell Line |
SNB-78 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
341.19 |
nM |
PubChem BioAssay data set |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
13.24 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
18.97 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
99.08 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
56.62 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
11.91 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
25.47 |
nM |
PubChem BioAssay data set |
NPT732 |
Cell Line |
HOP-18 |
Homo sapiens |
GI50 |
|
68865.23 |
nM |
PubChem BioAssay data set |
NPT738 |
Cell Line |
SN12K1 |
Homo sapiens |
GI50 |
|
62.52 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.51 |
ug/ml |
22503741 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.74 |
ug/ml |
22503741 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.7 |
ug/ml |
22503741 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
1.96 |
% |
22503741 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
1.34 |
% |
22503741 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
78.1 |
% |
22503741 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
530 |
nM |
22512906 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
230 |
nM |
22512906 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
750 |
nM |
22512906 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1720 |
nM |
22512906 |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
3300 |
nM |
22185476 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
16 |
nM |
22185476 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4120 |
nM |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
47.5 |
% |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
31.5 |
% |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
21 |
% |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
1.3 |
% |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
8.9 |
% |
22185476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
89.9 |
% |
22185476 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
16 |
nM |
22611477 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
22611477 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10 |
nM |
22542017 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8 |
nM |
22542017 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.4 |
ug/ml |
22578453 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
0.8 |
ug/ml |
22578453 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
22578453 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.3 |
ug/ml |
22578453 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
30 |
nM |
22564383 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
20 |
nM |
22608389 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
22608389 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
22608389 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
22608389 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
20 |
nM |
22608389 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
9.3 |
nM |
22727370 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
20.2 |
nM |
22727370 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
50.6 |
nM |
22727370 |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
3300 |
nM |
22727370 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4120 |
nM |
22727370 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
16 |
nM |
22727370 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
6.4 |
nM |
22850214 |
NPT1018 |
Organism |
Trypanosoma brucei |
Trypanosoma brucei |
IC50 |
= |
14000 |
nM |
22850214 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Ratio IC50 |
< |
2 |
|
22931300 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
8 |
% |
12699389 |
NPT1546 |
Individual Protein |
Solute carrier family 22 member 3 |
Homo sapiens |
Ki |
= |
120 |
nM |
10196521 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
206 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
42.2 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
75 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
153.6 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
188.3 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
53.1 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
4.6 |
nM |
PubChem BioAssay data set |
NPT158 |
Individual Protein |
Nuclear receptor subfamily 1 group I member 2 |
Rattus norvegicus |
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT158 |
Individual Protein |
Nuclear receptor subfamily 1 group I member 2 |
Rattus norvegicus |
Potency |
|
1584.9 |
nM |
PubChem BioAssay data set |
NPT102 |
Individual Protein |
Interleukin-8 |
Homo sapiens |
Potency |
|
53.1 |
nM |
PubChem BioAssay data set |
NPT102 |
Individual Protein |
Interleukin-8 |
Homo sapiens |
Potency |
|
47.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
206 |
nM |
PubChem BioAssay data set |
NPT103 |
Individual Protein |
Nuclear receptor ROR-gamma |
Homo sapiens |
Potency |
|
334.9 |
nM |
PubChem BioAssay data set |
NPT103 |
Individual Protein |
Nuclear receptor ROR-gamma |
Homo sapiens |
Potency |
|
118.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23350 |
nM |
23022053 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
550 |
nM |
23022053 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
100 |
nM |
23022053 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
50 |
nM |
23022053 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23022053 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
11.2 |
nM |
22783954 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
11.5 |
nM |
22783954 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
16.3 |
nM |
22783954 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29 |
nM |
22783954 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
20.6 |
nM |
22783954 |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Inhibition |
= |
24.4 |
% |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
-3.9 |
% |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
45.2 |
% |
22541068 |
NPT140 |
Organism |
Artemia |
Artemia |
LD50 |
= |
71.1 |
nM |
23148724 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
23017885 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
0.14 |
% |
23062825 |
NPT67 |
Individual Protein |
Cholinesterase |
Equus caballus |
Inhibition |
= |
0.1 |
% |
23062825 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Ratio IC50 |
= |
1.2 |
|
23176628 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9.7 |
nM |
23176628 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8.2 |
nM |
23176628 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
Ratio IC50 |
= |
2.5 |
|
23176628 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16.8 |
nM |
23176628 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
6.7 |
nM |
23176628 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
37 |
nM |
23176628 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
69.25 |
nM |
23176628 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
15.6 |
nM |
23176628 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
7850 |
nM |
23176628 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Ki |
= |
1.614 |
nM |
23176628 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
12 |
nM |
23063401 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1700 |
nM |
23063401 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Ratio IC50 |
= |
1.2 |
|
23103097 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9700 |
nM |
23103097 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8200 |
nM |
23103097 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
2.5 |
|
23103097 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16800 |
nM |
23103097 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
6700 |
nM |
23103097 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
45.5 |
nM |
23103097 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
20 |
nM |
11378362 |
NPT5296 |
Individual Protein |
Tubulin polymerization-promoting protein |
Bos taurus |
EC50 |
= |
750 |
nM |
11378362 |
NPT3478 |
Organism |
Nicotiana tabacum |
Nicotiana tabacum |
EC50 |
= |
356000 |
nM |
11378362 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
7070 |
nM |
10.1007/s00044-012-0428-9 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
21.81 |
% |
10.1007/s00044-012-0428-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13 |
nM |
23220647 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
329 |
nM |
23214452 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11 |
nM |
23214452 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
86 |
nM |
23214452 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23214452 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23214452 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
18 |
nM |
23214452 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
28 |
nM |
23214452 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5 |
nM |
23214452 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
23214452 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1700 |
nM |
23313639 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
58.5 |
|
23547728 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
643 |
nM |
23547728 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
11 |
nM |
23547728 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1780 |
nM |
23419737 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
780 |
nM |
23419737 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
3500 |
nM |
23419737 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
660 |
nM |
23419737 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
7.6 |
nM |
23360369 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
Activity |
= |
56 |
% |
23360369 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
Ratio IC50 |
= |
0.85 |
|
23360369 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
8.91 |
nM |
23360369 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46.74 |
nM |
23360369 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
15.38 |
nM |
23360369 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
37.38 |
nM |
23360369 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23360369 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1450 |
nM |
23419737 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
60 |
nM |
23419737 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
50 |
nM |
23419737 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
70 |
nM |
23419737 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
23425970 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
11800 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3120 |
nM |
23425970 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
300 |
nM |
23425970 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
40 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
90 |
nM |
23425970 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
120 |
nM |
23425970 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
290 |
nM |
23425970 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
170 |
nM |
23425970 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
1310 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27000 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
80000 |
nM |
23425970 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23425970 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23425970 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
80 |
nM |
23425970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1720 |
nM |
23425970 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
23.58 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
24.14 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
21.75 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
18.02 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
17.78 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
16.86 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
23.71 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
24.03 |
% |
23353745 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
21.12 |
% |
23353745 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
17.8 |
nM |
23445405 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
47.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8.2 |
nM |
PubChem BioAssay data set |
NPT35 |
Others |
n.a. |
|
IC50 |
> |
67568 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
188.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
266.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
66.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16.4 |
nM |
PubChem BioAssay data set |
NPT585 |
Individual Protein |
Nuclear receptor subfamily 0 group B member 1 |
Homo sapiens |
IC50 |
> |
67568 |
nM |
PubChem BioAssay data set |
NPT861 |
Individual Protein |
Isocitrate dehydrogenase [NADP] cytoplasmic |
Homo sapiens |
Potency |
|
7.3 |
nM |
PubChem BioAssay data set |
NPT1283 |
Individual Protein |
Paired box protein Pax-8 |
Homo sapiens |
AC50 |
< |
260 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
475 |
nM |
23524161 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
> |
100000 |
nM |
23524161 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
74 |
% |
23524161 |
NPT2142 |
Cell Line |
REH |
Homo sapiens |
IC50 |
= |
9.5 |
nM |
23524161 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
32.5 |
nM |
23524161 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
15.9 |
% |
23524161 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
23524161 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
23 |
nM |
23524161 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
7.7 |
nM |
23524161 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
2.6 |
nM |
23524161 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
74 |
nM |
23602523 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17 |
nM |
23602523 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
37 |
nM |
23602523 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
23 |
nM |
23602523 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
19 |
nM |
23602523 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.97 |
|
23747810 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.85 |
|
23747810 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
> |
10000 |
nM |
23747810 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
710 |
nM |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23747810 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17 |
nM |
23747810 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
70 |
nM |
23747810 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
40.5 |
% |
23747810 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
60.1 |
% |
23747810 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
72.3 |
% |
23747810 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
41.8 |
% |
23747810 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
58.7 |
% |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
14.3 |
% |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
63.6 |
% |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
63.3 |
% |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
5.6 |
% |
23747810 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
16.8 |
% |
23747810 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3200 |
nM |
23810282 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1800 |
nM |
23735826 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
30.2 |
nM |
23961916 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
30 |
nM |
23961916 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
9 |
nM |
23932339 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
19 |
nM |
23932339 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22 |
nM |
23932339 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18 |
nM |
23932339 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Ki |
= |
2400 |
nM |
24106982 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
72 |
% |
24106982 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
32 |
% |
24106982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4200 |
nM |
24106982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
51.8 |
nM |
24106982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
35.4 |
nM |
24106982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
122 |
nM |
24106982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19.8 |
nM |
24106982 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
11.5 |
nM |
24106982 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
15.2 |
nM |
24106982 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
10.3 |
nM |
24106982 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
75.12 |
% |
23571415 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
101.04 |
% |
23571415 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
9.1 |
% |
24210503 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
7.7 |
% |
24210503 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Inhibition |
= |
11.1 |
% |
24210503 |
NPT628 |
Individual Protein |
Cytochrome P450 2C8 |
Homo sapiens |
Inhibition |
= |
20.4 |
% |
24210503 |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
Inhibition |
= |
12.4 |
% |
24210503 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
13.2 |
nM |
24210503 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
2.1 |
nM |
24210503 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
5.4 |
nM |
24210503 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
3.8 |
nM |
24210503 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
77 |
% |
24360827 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
76 |
% |
24360827 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
30.2 |
nM |
23457660 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
30 |
nM |
23457660 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16 |
nM |
23457660 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
8120 |
nM |
10.1039/C3MD00287J |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
10.6 |
nM |
10.1039/C3MD00287J |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8.2 |
nM |
10.1039/C3MD00287J |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
54.4 |
nM |
10.1039/C3MD00287J |
NPT2 |
Others |
Unspecified |
|
Potency |
|
501.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43.6 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
6.2 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
8.6 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
17.2 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
30.3 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
60.1 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
188.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
60.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
760.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3757.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
136.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
118.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
19.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
150.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
89.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
39.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
562.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1188.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1368.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
891.3 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
42.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3349.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
67753.4 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
19.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1516.8 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
23.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
172.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
494.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
13685.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
86.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
135.2 |
nM |
PubChem BioAssay data set |
NPT105 |
Individual Protein |
Muscleblind-like protein 1 |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT105 |
Individual Protein |
Muscleblind-like protein 1 |
Homo sapiens |
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
96.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
67.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
530.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
42.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
237.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7.7 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
10.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
334.9 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
67.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
379 |
nM |
PubChem BioAssay data set |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
5.6 |
nM |
PubChem BioAssay data set |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
70794.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
12 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
87.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
95.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
75.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
68.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
354.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3981.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
375.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
266 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
13.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21425.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3162.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
84.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43277.1 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
1083.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10.7 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
375.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8634.9 |
nM |
PubChem BioAssay data set |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
10.3 |
nM |
10.1039/C0MD00052C |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19.8 |
nM |
10.1039/C0MD00052C |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
15.2 |
nM |
10.1039/C0MD00052C |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11.5 |
nM |
10.1039/C0MD00052C |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
121.2 |
nM |
10.1039/C0MD00052C |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
4100 |
nM |
10.1039/C0MD00052C |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8 |
nM |
10.1039/C3MD00077J |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8 |
nM |
10.1039/C3MD00077J |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
14 |
% |
10.1039/C2MD20250F |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
92.6 |
% |
10.1039/C2MD20250F |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
54.4 |
nM |
10.1039/C2MD20250F |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
8.2 |
nM |
10.1039/C2MD20250F |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
10.6 |
nM |
10.1039/C2MD20250F |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
15 |
% |
430477 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Activity |
= |
3 |
% |
430477 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12.4 |
nM |
24657567 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14.9 |
nM |
24657567 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
12.8 |
nM |
24657567 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
4900 |
nM |
24657567 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
32.2 |
% |
24657567 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
72 |
% |
24657567 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.8 |
nM |
24773591 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
31 |
nM |
24773591 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.9 |
nM |
24773591 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
10 |
nM |
24773591 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
13 |
nM |
24773591 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8.7 |
nM |
24773591 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
EC50 |
= |
30 |
nM |
24842619 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
EC25 |
= |
0.02 |
nM |
24842619 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
30 |
nM |
24842619 |
NPT2 |
Others |
Unspecified |
|
EC25 |
= |
0.02 |
nM |
24842619 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Ratio EC50 |
= |
10 |
|
24842619 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
10 |
|
24842619 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.39 |
ug/ml |
24916028 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.58 |
ug/ml |
24916028 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.48 |
ug/ml |
24916028 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
1340 |
nM |
24916028 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
4.6 |
% |
24916028 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
11.78 |
% |
24916028 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
83.62 |
% |
24916028 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11 |
nM |
25025991 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
329 |
nM |
25025991 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
5400 |
nM |
25059503 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
34.5 |
% |
25059503 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
64.4 |
% |
25059503 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
21 |
nM |
25091926 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
3 |
nM |
25091926 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1 |
nM |
25091926 |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
IC50 |
= |
8 |
nM |
25091926 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1710 |
nM |
25091926 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
704 |
nM |
25091926 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7 |
nM |
25091926 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
25025991 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5 |
nM |
25025991 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
25025991 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
420 |
nM |
25025991 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
4 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
344 |
nM |
25208345 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
16 |
nM |
25208345 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
12 |
nM |
25208345 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
42 |
nM |
25208345 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
58 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4 |
nM |
25208345 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
9 |
nM |
25208345 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25208345 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.8 |
nM |
25282265 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
31 |
nM |
25282265 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.9 |
nM |
25282265 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
14 |
nM |
25282265 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
31 |
nM |
25282265 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
28 |
nM |
25282265 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
6 |
% |
25282265 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
5 |
% |
25282265 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
10 |
% |
25282265 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
80 |
% |
25282265 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
50 |
nM |
25426924 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12 |
nM |
25426924 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
5 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
> |
0.015 |
nM |
25426924 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.4 |
|
25426924 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.1 |
|
25426924 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
15 |
nM |
25426924 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
306 |
nM |
25426924 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
20 |
|
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
3.3 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
3.9 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
4.3 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
6.6 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
12.9 |
nM |
25426924 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Activity |
= |
13.7 |
nM |
25426924 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
50 |
nM |
25061803 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
34 |
nM |
25061803 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
33 |
nM |
25061803 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
160 |
nM |
25061803 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
35 |
nM |
25061803 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
57 |
nM |
25061803 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
590 |
nM |
25061803 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
59 |
nM |
25061803 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1100 |
nM |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
81 |
nM |
25061803 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
25061803 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
10 |
|
25061803 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
19 |
|
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Ratio IC50 |
= |
2.3 |
|
25061803 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
169 |
|
25061803 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
2600 |
nM |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
36.19 |
% |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
37.72 |
% |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
6.93 |
% |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
19.16 |
% |
25061803 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40 |
% |
25496412 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25499929 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
690 |
nM |
25499929 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
25499929 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
25499929 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
Inhibition |
= |
87 |
% |
25499929 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
1700 |
nM |
25499929 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1800 |
nM |
25778766 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
40 |
nM |
25827522 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
< |
10 |
nM |
25827522 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
25827522 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
30 |
nM |
25827522 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
390 |
nM |
25703297 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
580 |
nM |
25703297 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
480 |
nM |
25703297 |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
1340 |
nM |
25703297 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6.94 |
% |
25703297 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
12.44 |
% |
25703297 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
80.62 |
% |
25703297 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
360 |
nM |
25659770 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
97.2 |
% |
25874341 |
NPT684 |
Individual Protein |
Histone deacetylase 1 |
Homo sapiens |
IC50 |
> |
20 |
ug/ml |
25805446 |
NPT685 |
Individual Protein |
Histone deacetylase 2 |
Homo sapiens |
IC50 |
> |
20 |
ug/ml |
25805446 |
NPT686 |
Individual Protein |
Histone deacetylase 3 |
Homo sapiens |
IC50 |
> |
20 |
ug/ml |
25805446 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
105 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
25805446 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
5 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14 |
nM |
25805446 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
27 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
110 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
34 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
21 |
nM |
25805446 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
8 |
nM |
25805446 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
132 |
nM |
25768706 |
NPT2588 |
Organism |
Paracentrotus lividus |
Paracentrotus lividus |
EC |
= |
0.05 |
nM |
25768706 |
NPT2588 |
Organism |
Paracentrotus lividus |
Paracentrotus lividus |
EC |
= |
0.1 |
nM |
25768706 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
120 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
0.8 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
4.3 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
3 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
-5 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
8 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
16 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
1 |
|
21051535 |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
FC |
= |
-0.4 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
4.2 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
6.4 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
85 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
67 |
|
21051535 |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
320 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
18.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
38.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
316.2 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
309 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
42.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
171.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
977 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
354.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
1.71 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
52.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
100 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
172.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
10000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
1.88 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
685.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
860.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
26.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
538.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
549.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
305.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
11.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
216.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
1.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
96.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
37.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
1.73 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LD50 |
= |
19.4 |
nM |
25730346 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LD50 |
= |
8.1 |
nM |
26039736 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
Activity |
= |
2.4 |
% |
26069928 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
Activity |
= |
27.9 |
% |
26069928 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
Activity |
= |
11.8 |
% |
26069928 |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
Activity |
= |
57.9 |
% |
26069928 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
13500 |
nM |
26070164 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
10500 |
nM |
26070164 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
4400 |
nM |
26070164 |
NPT5180 |
Protein Complex |
Tubulin |
Bos taurus |
IC50 |
= |
2620 |
nM |
26070164 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14.9 |
nM |
26160020 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12.4 |
nM |
26160020 |
NPT5180 |
Protein Complex |
Tubulin |
Bos taurus |
IC50 |
= |
1900 |
nM |
26160020 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
86.2 |
% |
26160020 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
Inhibition |
= |
82.8 |
% |
26160020 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5 |
nM |
26132075 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
30 |
nM |
26132075 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
420 |
nM |
26132075 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11 |
nM |
26132075 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
329 |
nM |
26132075 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
96 |
nM |
25811651 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.36 |
nM |
25811651 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5023 |
nM |
25937236 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
3200 |
nM |
26132075 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
2210 |
nM |
26241032 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
40 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
4 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
20 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
6 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
5 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
48 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
30 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
43 |
% |
26094121 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
19 |
% |
26094121 |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
7800 |
nM |
26226379 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
63.6 |
% |
26344588 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
20 |
nM |
26344588 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17 |
nM |
26344588 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.85 |
|
26344588 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
Activity |
= |
8.9 |
% |
26454648 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
Activity |
= |
21.5 |
% |
26454648 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
Activity |
= |
12.6 |
% |
26454648 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
Activity |
= |
57.5 |
% |
26454648 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
2100 |
nM |
26580420 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
15 |
nM |
26602281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
26602281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
26778612 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
4.2 |
nM |
26778612 |
NPT5129 |
Cell Line |
BJAB |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1039/C5MD00320B |
NPT5129 |
Cell Line |
BJAB |
Homo sapiens |
AC50 |
= |
30 |
nM |
10.1039/C5MD00320B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
375 |
nM |
10.1039/C5MD00320B |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
37 |
nM |
26927488 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
3790 |
nM |
26927488 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
10 |
nM |
27094151 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Inhibition |
= |
52 |
% |
27094151 |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
6.7 |
nM |
26985296 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18.6 |
nM |
26985296 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
23.9 |
nM |
26985296 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
21.8 |
nM |
26985296 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
13.5 |
nM |
26985296 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20.4 |
nM |
26985296 |