Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
3900.0 |
ug.mL-1 |
PMID[501791] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
1.7 |
nM |
PMID[501793] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
8.2 |
nM |
PMID[501793] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ILS |
~ |
50.0 |
% |
PMID[501793] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ILS |
~ |
100.0 |
% |
PMID[501793] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED |
= |
0.0015 |
ug ml-1 |
PMID[501794] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
T/C |
= |
140.0 |
% |
PMID[501794] |
NPT319 |
Cell Line |
B16 |
Mus musculus |
T/C |
= |
180.0 |
% |
PMID[501794] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Log CR |
= |
1.28 |
n.a. |
PMID[501798] |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Log CR |
= |
1.46 |
n.a. |
PMID[501798] |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
IC50 |
= |
2.1 |
nM |
PMID[501799] |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
15.9 |
nM |
PMID[501799] |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
0.8 |
nM |
PMID[501799] |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
90.9 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
163.3 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
43.0 |
nM |
PMID[501800] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
3.4 |
nM |
PMID[501800] |
NPT3597 |
Individual Protein |
Tubulin beta chain |
Bos taurus |
Ki |
> |
100000.0 |
nM |
PMID[501800] |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
Relative IC50 |
= |
1.0 |
nM |
PMID[501801] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Relative IC50 |
= |
2000.0 |
nM |
PMID[501801] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Relative IC50 |
= |
1.3 |
nM |
PMID[501801] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Relative IC50 |
= |
1.0 |
nM |
PMID[501801] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Relative IC50 |
= |
17500.0 |
nM |
PMID[501801] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Relative IC50 |
= |
0.5 |
nM |
PMID[501801] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Relative IC50 |
= |
1.0 |
nM |
PMID[501801] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Relative IC50 |
= |
19.0 |
nM |
PMID[501801] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Relative IC50 |
= |
0.2 |
nM |
PMID[501801] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Reduction |
~ |
88.0 |
% |
PMID[501802] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Reduction |
~ |
94.0 |
% |
PMID[501802] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Reduction |
~ |
95.0 |
% |
PMID[501802] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Reduction |
= |
0.0 |
% |
PMID[501802] |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
GI50 |
= |
0.0102 |
ug.mL-1 |
PMID[501803] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
0.001 |
ug.mL-1 |
PMID[501803] |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Survival |
< |
0.01 |
n.a. |
PMID[501804] |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Reduction |
> |
99.0 |
% |
PMID[501804] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2.3 |
nM |
PMID[501805] |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
350.0 |
nM |
PMID[501805] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI50 |
= |
4.1 |
nM |
PMID[501805] |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
GI50 |
= |
470.0 |
nM |
PMID[501805] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
0.02 |
nM |
PMID[501807] |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
< |
0.25 |
nM |
PMID[501807] |
NPT708 |
Cell Line |
HuT78 |
Homo sapiens |
GI50 |
< |
0.25 |
nM |
PMID[501807] |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
0.003 |
nM |
PMID[501807] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
< |
0.25 |
nM |
PMID[501807] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
0.036 |
nM |
PMID[501807] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
TGI |
= |
1.91 |
nM |
PMID[501807] |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
TGI |
< |
0.25 |
nM |
PMID[501807] |
NPT708 |
Cell Line |
HuT78 |
Homo sapiens |
TGI |
< |
0.25 |
nM |
PMID[501807] |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
TGI |
= |
0.8 |
nM |
PMID[501807] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
< |
0.25 |
nM |
PMID[501807] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
TGI |
= |
0.25 |
nM |
PMID[501807] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
LC50 |
= |
5.73 |
nM |
PMID[501807] |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
LC50 |
< |
0.25 |
nM |
PMID[501807] |
NPT708 |
Cell Line |
HuT78 |
Homo sapiens |
LC50 |
= |
0.25 |
nM |
PMID[501807] |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
LC50 |
= |
3.28 |
nM |
PMID[501807] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
< |
0.25 |
nM |
PMID[501807] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
LC50 |
= |
1.51 |
nM |
PMID[501807] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
11.0 |
nM |
PMID[501808] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.1 |
ug.mL-1 |
PMID[501809] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Permeability |
= |
1.54 |
*10e6 |
PMID[501810] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Permeability |
= |
12.5 |
*10e6 |
PMID[501810] |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
EC50 |
< |
3700.0 |
nM |
PMID[501811] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
IC50 |
= |
26000.0 |
nM |
PMID[501813] |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
IC50 |
> |
50000.0 |
nM |
PMID[501813] |
NPT1456 |
Individual Protein |
P-glycoprotein 1 |
Mus musculus |
IC50 |
= |
8000.0 |
nM |
PMID[501813] |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
Ratio |
= |
3.0 |
n.a. |
PMID[501813] |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
Ratio |
= |
5.2 |
n.a. |
PMID[501813] |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
Ratio |
= |
4.3 |
n.a. |
PMID[501813] |
NPT3871 |
Cell Line |
N592 |
|
IC50 |
= |
4.0 |
nM |
PMID[501814] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
3.15 |
nM |
PMID[501815] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
T/C |
= |
157.0 |
% |
PMID[501815] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
LTS |
= |
2.0 |
n.a. |
PMID[501815] |
NPT2698 |
Individual Protein |
Beta tubulin |
Leishmania donovani |
IC50 |
= |
1000.0 |
nM |
PMID[501817] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
1.2 |
nM |
PMID[501818] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9.9 |
nM |
PMID[501818] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8.7 |
nM |
PMID[501818] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[501819] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
3000.0 |
nM |
PMID[501820] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
33.0 |
% |
PMID[501820] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
30.0 |
% |
PMID[501820] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
37.0 |
% |
PMID[501820] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Log 1/Km |
= |
-0.834 |
n.a. |
PMID[501821] |
NPT1527 |
Cell Line |
WRL68 |
Homo sapiens |
IC50 |
= |
1.45 |
ug.mL-1 |
PMID[501822] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.22 |
ug.mL-1 |
PMID[501822] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.02 |
ug.mL-1 |
PMID[501822] |
NPT1527 |
Cell Line |
WRL68 |
Homo sapiens |
IC50 |
= |
2.6 |
ug.mL-1 |
PMID[501822] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.046 |
ug.mL-1 |
PMID[501822] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.46 |
ug.mL-1 |
PMID[501822] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
0.025 |
ug.mL-1 |
PMID[501822] |
NPT3852 |
Cell Line |
COLO 320DM |
Homo sapiens |
IC50 |
= |
0.52 |
ug.mL-1 |
PMID[501822] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
1.15 |
ug.mL-1 |
PMID[501822] |
NPT3852 |
Cell Line |
COLO 320DM |
Homo sapiens |
IC50 |
= |
1.6 |
ug.mL-1 |
PMID[501822] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.4 |
nM |
PMID[501823] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
28.7 |
nM |
PMID[501823] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
206.6 |
nM |
PMID[501823] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1.1 |
nM |
PMID[501823] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[501823] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.0 |
nM |
PMID[501823] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
EC50 |
= |
2.0 |
nM |
PMID[501824] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
= |
3.0 |
nM |
PMID[501824] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
EC50 |
= |
1.0 |
nM |
PMID[501824] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
81.0 |
% |
PMID[501826] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
72.0 |
% |
PMID[501826] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
42.0 |
% |
PMID[501826] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
4.4 |
nM |
PMID[501827] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Ratio IC50 |
= |
22.0 |
n.a. |
PMID[501827] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.34 |
nM |
PMID[501827] |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
95.0 |
nM |
PMID[501827] |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
4.3 |
nM |
PMID[501827] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Ratio IC50 |
= |
15.0 |
n.a. |
PMID[501827] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Ratio IC50 |
= |
10.0 |
n.a. |
PMID[501827] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.29 |
nM |
PMID[501827] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.42 |
nM |
PMID[501827] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
4.1 |
nM |
PMID[501827] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
79.4 |
nM |
PMID[501828] |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
25.0 |
nM |
PMID[501828] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
1.6 |
nM |
PMID[501828] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[501829] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
89.0 |
n.a. |
PMID[501829] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
2.0 |
n.a. |
PMID[501829] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
25.0 |
nM |
PMID[501830] |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
EC50 |
= |
73.0 |
nM |
PMID[501830] |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
EC50 |
= |
129.0 |
nM |
PMID[501830] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
0.9 |
nM |
PMID[501831] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
0.5 |
nM |
PMID[501831] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
2.0 |
nM |
PMID[501832] |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
10.0 |
nM |
PMID[501832] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2.0 |
nM |
PMID[501832] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.8 |
nM |
PMID[501833] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
83.3 |
% |
PMID[501833] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
6.6 |
% |
PMID[501833] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
10.1 |
% |
PMID[501833] |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
6880.0 |
nM |
PMID[501834] |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
61.66 |
nM |
PMID[501836] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
43.0 |
nM |
PMID[501837] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
44.0 |
nM |
PMID[501837] |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
EC50 |
= |
38.0 |
nM |
PMID[501837] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7.0 |
nM |
PMID[501837] |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
28.0 |
nM |
PMID[501838] |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
IC50 |
= |
9271000.0 |
nM |
PMID[501840] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.07 |
nM |
PMID[501840] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
440.0 |
nM |
PMID[501840] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.88 |
nM |
PMID[501840] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5946000.0 |
nM |
PMID[501840] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
170.0 |
nM |
PMID[501840] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
193000.0 |
nM |
PMID[501840] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.27 |
nM |
PMID[501841] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.53 |
nM |
PMID[501841] |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
0.49 |
nM |
PMID[501841] |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
3.6 |
ug.mL-1 |
PMID[501847] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1.0 |
nM |
PMID[501849] |
NPT6402 |
Individual Protein |
Tubulin beta-5 chain |
Homo sapiens |
Activity |
= |
25.0 |
% |
PMID[501849] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Papp |
= |
5.1 |
nm/s |
PMID[501850] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7.0 |
nM |
PMID[501851] |
NPT459 |
Individual Protein |
Human immunodeficiency virus type 1 reverse transcriptase |
Human immunodeficiency virus 1 |
IC50 |
> |
200.0 |
ug.mL-1 |
PMID[501852] |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
ED50 |
= |
0.05 |
ug ml-1 |
PMID[501853] |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
ED50 |
= |
0.01 |
ug ml-1 |
PMID[501853] |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
ED50 |
= |
0.02 |
ug ml-1 |
PMID[501853] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.002 |
ug ml-1 |
PMID[501853] |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
0.1 |
ug ml-1 |
PMID[501853] |
NPT1034 |
Cell Line |
Lu1 |
Homo sapiens |
ED50 |
= |
0.02 |
ug ml-1 |
PMID[501853] |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.01 |
ug ml-1 |
PMID[501853] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.02 |
ug ml-1 |
PMID[501853] |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
ED50 |
= |
0.3 |
ug ml-1 |
PMID[501853] |
NPT76 |
Cell Line |
C6 |
Rattus norvegicus |
LC50 |
= |
66.0 |
nM |
PMID[501854] |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501856] |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
TGI |
= |
2440.0 |
nM |
PMID[501856] |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
LC50 |
= |
2480.0 |
nM |
PMID[501856] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501856] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
= |
1640.0 |
nM |
PMID[501856] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
= |
2480.0 |
nM |
PMID[501856] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501856] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
1600.0 |
nM |
PMID[501856] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
2500.0 |
nM |
PMID[501856] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501856] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
350.0 |
nM |
PMID[501856] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
2100.0 |
nM |
PMID[501856] |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501856] |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
< |
10.0 |
nM |
PMID[501856] |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
LC50 |
= |
920.0 |
nM |
PMID[501856] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
1.7 |
ug ml-1 |
PMID[501857] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.0 |
nM |
PMID[501858] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
135.0 |
nM |
PMID[501858] |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[501858] |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[501858] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio IC50 |
= |
45.0 |
n.a. |
PMID[501858] |
NPT319 |
Cell Line |
B16 |
Mus musculus |
T/C |
= |
309.0 |
% |
PMID[501859] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501860] |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
Activity |
= |
78.0 |
% |
PMID[501861] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.73 |
nM |
PMID[501860] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
78.0 |
nM |
PMID[501860] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
496.0 |
nM |
PMID[501860] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
PMID[501860] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.8 |
nM |
PMID[501860] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501860] |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
Inhibition |
= |
1.9 |
% |
PMID[501862] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[501865] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
40.0 |
mm |
PMID[501865] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
25.0 |
mm |
PMID[501865] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
10.0 |
mm |
PMID[501865] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.7 |
nM |
PMID[501865] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
> |
40.0 |
mm |
PMID[501865] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
32.5 |
mm |
PMID[501865] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
12.5 |
mm |
PMID[501865] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.1 |
10'-4 ug/ml |
PMID[501867] |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
ED50 |
> |
1.0 |
10'-1 ug/ml |
PMID[501867] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.03 |
ug.mL-1 |
PMID[501869] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.002 |
ug ml-1 |
PMID[501870] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED50 |
> |
20.0 |
ug ml-1 |
PMID[501871] |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
ED50 |
> |
20.0 |
ug ml-1 |
PMID[501871] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
> |
20.0 |
ug ml-1 |
PMID[501871] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.26 |
nM |
PMID[501872] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.73 |
nM |
PMID[501873] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.1 |
nM |
PMID[501873] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.2 |
nM |
PMID[501873] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
78.0 |
nM |
PMID[501873] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
496.0 |
nM |
PMID[501873] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501873] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501873] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
permeability |
= |
0.1 |
10'-6 cm/s |
PMID[501874] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
permeability |
= |
41.9 |
10'-6 cm/s |
PMID[501874] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.05 |
ug ml-1 |
PMID[501876] |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
ED50 |
= |
0.001 |
ug ml-1 |
PMID[501876] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.1 |
10'-4 ug/ml |
PMID[501878] |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
ED50 |
> |
1.0 |
ug ml-1 |
PMID[501878] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
27.0 |
nM |
PMID[501879] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.6 |
nM |
PMID[501879] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
2.0 |
nM |
PMID[501880] |
NPT2815 |
Cell Line |
M21 |
Homo sapiens |
GI50 |
= |
10.0 |
nM |
PMID[501880] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2.0 |
nM |
PMID[501880] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.4 |
nM |
PMID[501882] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
0.9 |
nM |
PMID[501882] |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
GI50 |
= |
5.0 |
nM |
PMID[501886] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7.0 |
nM |
PMID[501886] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
10.0 |
nM |
PMID[501886] |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
EC50 |
= |
26.0 |
nM |
PMID[501886] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
32.0 |
nM |
PMID[501886] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
36.0 |
nM |
PMID[501886] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
32.0 |
nM |
PMID[501890] |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
EC50 |
= |
160.0 |
nM |
PMID[501890] |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
EC50 |
= |
82.0 |
nM |
PMID[501890] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.1 |
nM |
PMID[501891] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.2 |
nM |
PMID[501891] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
685.0 |
n.a. |
PMID[501891] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
107.0 |
n.a. |
PMID[501891] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[501891] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
78.0 |
nM |
PMID[501891] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.73 |
nM |
PMID[501891] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[501893] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.0 |
nM |
PMID[501893] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.3 |
nM |
PMID[501893] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.6 |
nM |
PMID[501893] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
10.0 |
nM |
PMID[501893] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
60.0 |
nM |
PMID[501896] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
10000.0 |
nM |
PMID[501896] |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501896] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
300.0 |
nM |
PMID[501896] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
32.0 |
nM |
PMID[501897] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
36.0 |
nM |
PMID[501897] |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
EC50 |
= |
26.0 |
nM |
PMID[501897] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
7.0 |
nM |
PMID[501897] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
10.0 |
nM |
PMID[501897] |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
GI50 |
= |
5.0 |
nM |
PMID[501897] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.8 |
nM |
PMID[501898] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
PMID[501898] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501898] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501898] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
496.0 |
nM |
PMID[501898] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
78.0 |
nM |
PMID[501898] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.73 |
nM |
PMID[501898] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501899] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501899] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
= |
1640.0 |
nM |
PMID[501899] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
= |
2480.0 |
nM |
PMID[501899] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
10.0 |
nM |
PMID[501899] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
1600.0 |
nM |
PMID[501899] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
2500.0 |
nM |
PMID[501899] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
350.0 |
nM |
PMID[501899] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
2100.0 |
nM |
PMID[501899] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.6 |
nM |
PMID[501900] |
NPT984 |
Cell Line |
Hepatocyte |
|
TC50 |
= |
5.45 |
10'4nM |
PMID[501906] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
11.0 |
nM |
PMID[501908] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
27.5 |
nM |
PMID[501908] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.0 |
nM |
PMID[501909] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
PMID[501909] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[501909] |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
11220.2 |
nM |
PMID[501911] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[501914] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80.0 |
nM |
PMID[501914] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[501914] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501914] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501914] |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
PMID[501914] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.8 |
nM |
PMID[501914] |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
49.0 |
nM |
PMID[501915] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.0 |
nM |
PMID[501916] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
27.0 |
nM |
PMID[501916] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.79 |
nM |
PMID[501916] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
17.0 |
nM |
PMID[501916] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[501917] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80.0 |
nM |
PMID[501917] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[501917] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501917] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501917] |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
Activity |
= |
51.5 |
% |
PMID[501918] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.11 |
nM |
PMID[501919] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[501919] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.42 |
nM |
PMID[501919] |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2.7 |
nM |
PMID[501919] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
5.5 |
nM |
PMID[501919] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
28.5 |
nM |
PMID[501921] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
28.5 |
nM |
PMID[501922] |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
n.a. |
3162.3 |
nM |
PMID[501911] |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
0.018 |
ug.mL-1 |
PMID[501928] |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
Activity |
= |
60.06 |
% |
PMID[501929] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[501930] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80.0 |
nM |
PMID[501930] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[501930] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.2 |
n.a. |
PMID[501930] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
679.5 |
n.a. |
PMID[501930] |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
17.0 |
nM |
PMID[501931] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.36 |
nM |
PMID[501931] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.16 |
nM |
PMID[501931] |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
0.063 |
nM |
PMID[501931] |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
0.099 |
nM |
PMID[501931] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.12 |
nM |
PMID[501931] |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.039 |
nM |
PMID[501931] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.38 |
nM |
PMID[501931] |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
IC50 |
= |
6.9 |
nM |
PMID[501931] |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
Ratio IC50 |
= |
0.41 |
n.a. |
PMID[501931] |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
IC50 |
= |
66.0 |
nM |
PMID[501931] |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
Ratio IC50 |
= |
3.9 |
n.a. |
PMID[501931] |
NPT2828 |
Cell Line |
CEM-VLB |
Homo sapiens |
Ratio IC50 |
= |
1579.0 |
n.a. |
PMID[501931] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
4.1 |
nM |
PMID[501932] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
56.1 |
n.a. |
PMID[501932] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
1.1 |
n.a. |
PMID[501933] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
> |
134.0 |
n.a. |
PMID[501933] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.8 |
nM |
PMID[501933] |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
4.5 |
nM |
PMID[501934] |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
0.31 |
nM |
PMID[501934] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
3.9 |
nM |
PMID[501935] |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
582.0 |
nM |
PMID[501935] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
Ratio IC50 |
= |
149.0 |
n.a. |
PMID[501935] |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
n.a. |
44668.4 |
nM |
PMID[501911] |
NPT154 |
Individual Protein |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
Potency |
n.a. |
11220.2 |
nM |
PMID[501936] |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
n.a. |
56234.1 |
nM |
PMID[501911] |
NPT257 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Oryctolagus cuniculus |
IC50 |
= |
5037.0 |
nM |
PMID[501938] |
NPT300 |
Individual Protein |
Thromboxane-A synthase |
Homo sapiens |
IC50 |
= |
1870.0 |
nM |
PMID[501938] |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
17.0 |
nM |
PMID[501940] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.36 |
nM |
PMID[501940] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.16 |
nM |
PMID[501940] |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
0.063 |
nM |
PMID[501940] |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
0.099 |
nM |
PMID[501940] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.12 |
nM |
PMID[501940] |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.039 |
nM |
PMID[501940] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.38 |
nM |
PMID[501940] |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
IC50 |
= |
6.9 |
nM |
PMID[501940] |
NPT5195 |
Cell Line |
CHO-TAX 5-6 |
Cricetulus griseus |
Ratio IC50 |
= |
0.41 |
n.a. |
PMID[501940] |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
IC50 |
= |
66.0 |
nM |
PMID[501940] |
NPT5196 |
Cell Line |
CHO-VV 3-2 |
Cricetulus griseus |
Ratio IC50 |
= |
3.9 |
n.a. |
PMID[501940] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
1579.0 |
n.a. |
PMID[501940] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[501941] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
56.1 |
n.a. |
PMID[501941] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
80.0 |
% |
PMID[501942] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
15.0 |
nM |
PMID[501942] |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
n.a. |
223.7 |
nM |
PMID[501911] |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
n.a. |
720.8 |
nM |
PMID[501911] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[501943] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80.0 |
nM |
PMID[501943] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[501943] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
106.0 |
n.a. |
PMID[501943] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
680.0 |
n.a. |
PMID[501943] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
9.4 |
nM |
PMID[501944] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
31.0 |
nM |
PMID[501944] |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
8.1 |
nM |
PMID[501944] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8.7 |
nM |
PMID[501944] |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
24.0 |
nM |
PMID[501944] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[501945] |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
0.91 |
nM |
PMID[501947] |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
Km |
= |
137300.0 |
nM |
PMID[501949] |
NPT304 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Rattus norvegicus |
Activity |
= |
29.0 |
% |
PMID[501970] |
NPT2613 |
Individual Protein |
Bile salt export pump |
Mus musculus |
Km |
= |
38300.0 |
nM |
PMID[501976] |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
IC50 |
= |
21000.0 |
nM |
PMID[501979] |
NPT1594 |
Individual Protein |
Multidrug resistance-associated protein 1 |
Homo sapiens |
IC50 |
= |
30000.0 |
nM |
PMID[501980] |
NPT1456 |
Individual Protein |
P-glycoprotein 1 |
Mus musculus |
IC50 |
= |
8000.0 |
nM |
PMID[501972] |
NPT1455 |
Individual Protein |
P-glycoprotein 3 |
Mus musculus |
IC50 |
> |
50000.0 |
nM |
PMID[501972] |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
n.a. |
5.3 |
nM |
PMID[501911] |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
n.a. |
749.9 |
nM |
PMID[501911] |
NPT1853 |
Individual Protein |
Putative uncharacterized protein |
Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
Potency |
n.a. |
31622.8 |
nM |
PMID[501911] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Activity |
= |
49.0 |
% |
PMID[501986] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.08 |
ug.mL-1 |
PMID[501987] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.37 |
ug.mL-1 |
PMID[501987] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.047 |
ug.mL-1 |
PMID[501987] |
NPT4599 |
Cell Line |
S9 |
Homo sapiens |
Activity |
= |
6.06 |
% |
PMID[501988] |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Inhibition |
= |
-9.3 |
% |
PMID[501989] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.42 |
nM |
PMID[501991] |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[501991] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.11 |
nM |
PMID[501991] |
NPT4465 |
Cell Line |
HCT-116/VM46 |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[501992] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
PMID[501992] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.0 |
nM |
PMID[501992] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
256.2 |
n.a. |
PMID[501994] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[501994] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
76.24 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
72.13 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
60.35 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
55.0 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
48.75 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
45.13 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
29.6 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
24.25 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
16.13 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.18 |
% |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
14.38 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
7.82 |
% |
PMID[501995] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6.1 |
ug.mL-1 |
PMID[501995] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4.6 |
ug.mL-1 |
PMID[501995] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
2.8 |
ug.mL-1 |
PMID[501996] |
NPT1527 |
Cell Line |
WRL68 |
Homo sapiens |
IC50 |
= |
2.6 |
ug.mL-1 |
PMID[501996] |
NPT2641 |
Cell Line |
COLO 320 |
Homo sapiens |
IC50 |
= |
1.6 |
ug.mL-1 |
PMID[501996] |
NPT1527 |
Cell Line |
WRL68 |
Homo sapiens |
IC50 |
= |
1.45 |
ug.mL-1 |
PMID[501996] |
NPT2641 |
Cell Line |
COLO 320 |
Homo sapiens |
IC50 |
= |
0.52 |
ug.mL-1 |
PMID[501996] |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
0.46 |
ug.mL-1 |
PMID[501996] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.22 |
ug.mL-1 |
PMID[501996] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
0.15 |
ug.mL-1 |
PMID[501996] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
0.03 |
ug.mL-1 |
PMID[501996] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.02 |
ug.mL-1 |
PMID[501996] |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
27060.0 |
nM |
PMID[501997] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1900.0 |
nM |
PMID[501997] |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI |
= |
84.0 |
% |
PMID[501998] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
14.38 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6.1 |
ug.mL-1 |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
76.24 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
60.35 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
48.75 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
29.6 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.18 |
% |
PMID[501999] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
7.82 |
% |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4.6 |
ug.mL-1 |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
72.13 |
% |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
55.0 |
% |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
45.13 |
% |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
24.25 |
% |
PMID[501999] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
16.13 |
% |
PMID[501999] |
NPT4465 |
Cell Line |
HCT-116/VM46 |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[502000] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
PMID[502000] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.0 |
nM |
PMID[502000] |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
200.0 |
nM |
PMID[502001] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
15.0 |
nM |
PMID[502001] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
24.0 |
nM |
PMID[502001] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.0 |
nM |
PMID[502001] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[502001] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
30.0 |
nM |
PMID[502001] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10.0 |
nM |
PMID[502001] |
NPT4465 |
Cell Line |
HCT-116/VM46 |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[502002] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
PMID[502002] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.4 |
nM |
PMID[502003] |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
Ratio IC50 |
> |
250.0 |
n.a. |
PMID[502004] |
NPT4490 |
Cell Line |
IMR-90 |
Homo sapiens |
IC50 |
> |
1000.0 |
nM |
PMID[502004] |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[502004] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
2.3 |
nM |
PMID[502005] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
105.0 |
n.a. |
PMID[502006] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2.0 |
nM |
PMID[502006] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[502007] |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[502007] |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
n.a. |
141.3 |
nM |
PMID[501936] |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
n.a. |
70.8 |
nM |
PMID[501936] |
NPT2268 |
Cell Line |
DOK |
Homo sapiens |
IC50 |
= |
4.196 |
nM |
PMID[502008] |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
23.21 |
nM |
PMID[502008] |
NPT1184 |
Cell Line |
Daoy |
Homo sapiens |
IC50 |
= |
3.102 |
nM |
PMID[502008] |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
98.66 |
nM |
PMID[502008] |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
383.01 |
nM |
PMID[502008] |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
278.22 |
nM |
PMID[502008] |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
5.316 |
nM |
PMID[502008] |
NPT2269 |
Cell Line |
EPLC-272H |
Homo sapiens |
IC50 |
= |
10.78 |
nM |
PMID[502008] |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
13.83 |
nM |
PMID[502008] |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
3.882 |
nM |
PMID[502008] |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
4.714 |
nM |
PMID[502008] |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
2.766 |
nM |
PMID[502008] |
NPT2270 |
Cell Line |
Detroit562 |
Homo sapiens |
IC50 |
= |
5.531 |
nM |
PMID[502008] |
NPT2271 |
Cell Line |
DoTc2-4510 |
Homo sapiens |
IC50 |
= |
16.52 |
nM |
PMID[502008] |
NPT1908 |
Cell Line |
EC-GI-10 |
Homo sapiens |
IC50 |
= |
3.531 |
nM |
PMID[502008] |
NPT3465 |
Cell Line |
ECC10 |
Homo sapiens |
IC50 |
= |
21.16 |
nM |
PMID[502008] |
NPT2272 |
Cell Line |
EFM-19 |
Homo sapiens |
IC50 |
= |
5.242 |
nM |
PMID[502008] |
NPT2273 |
Cell Line |
EFO-21 |
Homo sapiens |
IC50 |
= |
44.03 |
nM |
PMID[502008] |
NPT2274 |
Cell Line |
EFO-27 |
Homo sapiens |
IC50 |
= |
7.449 |
nM |
PMID[502008] |
NPT2275 |
Cell Line |
EGI-1 |
Homo sapiens |
IC50 |
= |
10.81 |
nM |
PMID[502008] |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
5.938 |
nM |
PMID[502008] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4.954 |
nM |
PMID[502008] |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
6.875 |
nM |
PMID[502008] |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
8.01 |
nM |
PMID[502008] |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
12.66 |
nM |
PMID[502008] |
NPT2278 |
Cell Line |
COLO-741 |
Homo sapiens |
IC50 |
= |
2.139 |
nM |
PMID[502008] |
NPT2279 |
Cell Line |
COLO-792 |
Homo sapiens |
IC50 |
= |
25.63 |
nM |
PMID[502008] |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
2816.86 |
nM |
PMID[502008] |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
119.71 |
nM |
PMID[502008] |
NPT2281 |
Cell Line |
ABC-1 |
Homo sapiens |
IC50 |
= |
15.49 |
nM |
PMID[502008] |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
16.88 |
nM |
PMID[502008] |
NPT2282 |
Cell Line |
C32 |
Homo sapiens |
IC50 |
= |
866.85 |
nM |
PMID[502008] |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
3.342 |
nM |
PMID[502008] |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
136.2 |
nM |
PMID[502008] |
NPT2283 |
Cell Line |
DK-MG |
Homo sapiens |
IC50 |
= |
6.646 |
nM |
PMID[502008] |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
20.94 |
nM |
PMID[502008] |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
59.04 |
nM |
PMID[502008] |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
40.29 |
nM |
PMID[502008] |
NPT2284 |
Cell Line |
C3A |
Homo sapiens |
IC50 |
= |
332.14 |
nM |
PMID[502008] |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
27.01 |
nM |
PMID[502008] |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
19.17 |
nM |
PMID[502008] |
NPT2285 |
Cell Line |
COR-L105 |
Homo sapiens |
IC50 |
= |
65.75 |
nM |
PMID[502008] |
NPT1918 |
Cell Line |
DMS-79 |
Homo sapiens |
IC50 |
= |
534.65 |
nM |
PMID[502008] |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
1.809 |
nM |
PMID[502008] |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
12.3 |
nM |
PMID[502008] |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
5.215 |
nM |
PMID[502008] |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
IC50 |
= |
24.61 |
nM |
PMID[502008] |
NPT2286 |
Cell Line |
CAL-120 |
Homo sapiens |
IC50 |
= |
87.26 |
nM |
PMID[502008] |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
3.623 |
nM |
PMID[502008] |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
24.32 |
nM |
PMID[502008] |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
IC50 |
= |
3.396 |
nM |
PMID[502008] |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
36.92 |
nM |
PMID[502008] |
NPT2288 |
Cell Line |
AN3-CA |
Homo sapiens |
IC50 |
= |
9.765 |
nM |
PMID[502008] |
NPT2289 |
Cell Line |
CAL-12T |
Homo sapiens |
IC50 |
= |
55.97 |
nM |
PMID[502008] |
NPT2290 |
Cell Line |
CAL-27 |
Homo sapiens |
IC50 |
= |
2.086 |
nM |
PMID[502008] |
NPT2291 |
Cell Line |
CP50-MEL-B |
Homo sapiens |
IC50 |
= |
13.12 |
nM |
PMID[502008] |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
48.58 |
nM |
PMID[502008] |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
9.815 |
nM |
PMID[502008] |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
1.034 |
nM |
PMID[502008] |
NPT2292 |
Cell Line |
CAL-33 |
Homo sapiens |
IC50 |
= |
6.184 |
nM |
PMID[502008] |
NPT2293 |
Cell Line |
CAL-39 |
Homo sapiens |
IC50 |
= |
5.114 |
nM |
PMID[502008] |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
1.636 |
nM |
PMID[502008] |
NPT2294 |
Cell Line |
23132-87 |
Homo sapiens |
IC50 |
= |
20.64 |
nM |
PMID[502008] |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
0.951 |
nM |
PMID[502008] |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
3.448 |
nM |
PMID[502008] |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
13.21 |
nM |
PMID[502008] |
NPT2298 |
Cell Line |
BALL-1 |
Homo sapiens |
IC50 |
= |
313.17 |
nM |
PMID[502008] |
NPT2299 |
Cell Line |
CAL-51 |
Homo sapiens |
IC50 |
= |
16.39 |
nM |
PMID[502008] |
NPT2300 |
Cell Line |
CAL-54 |
Homo sapiens |
IC50 |
= |
60.59 |
nM |
PMID[502008] |
NPT2301 |
Cell Line |
CAL-62 |
Homo sapiens |
IC50 |
= |
10.1 |
nM |
PMID[502008] |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
1.405 |
nM |
PMID[502008] |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
101.38 |
nM |
PMID[502008] |
NPT2302 |
Cell Line |
639-V |
Homo sapiens |
IC50 |
= |
5.605 |
nM |
PMID[502008] |
NPT2303 |
Cell Line |
647-V |
Homo sapiens |
IC50 |
= |
23.03 |
nM |
PMID[502008] |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
8.315 |
nM |
PMID[502008] |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
12.56 |
nM |
PMID[502008] |
NPT2304 |
Cell Line |
CAL-72 |
Homo sapiens |
IC50 |
= |
647.18 |
nM |
PMID[502008] |
NPT2305 |
Cell Line |
CAL-85-1 |
Homo sapiens |
IC50 |
= |
6079.95 |
nM |
PMID[502008] |
NPT2306 |
Cell Line |
Ca-Ski |
Homo sapiens |
IC50 |
= |
4.694 |
nM |
PMID[502008] |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
6.391 |
nM |
PMID[502008] |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
6.225 |
nM |
PMID[502008] |
NPT2307 |
Cell Line |
769-P |
Homo sapiens |
IC50 |
= |
25.55 |
nM |
PMID[502008] |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
15.58 |
nM |
PMID[502008] |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
20.7 |
nM |
PMID[502008] |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
32.01 |
nM |
PMID[502008] |
NPT2309 |
Cell Line |
CAPAN-1 |
Homo sapiens |
IC50 |
= |
52.3 |
nM |
PMID[502008] |
NPT2310 |
Cell Line |
CaR-1 |
Homo sapiens |
IC50 |
= |
45.73 |
nM |
PMID[502008] |
NPT2311 |
Cell Line |
Calu-3 |
Homo sapiens |
IC50 |
= |
551.0 |
nM |
PMID[502008] |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
6.335 |
nM |
PMID[502008] |
NPT2312 |
Cell Line |
8305C |
Homo sapiens |
IC50 |
= |
3.67 |
nM |
PMID[502008] |
NPT2313 |
Cell Line |
BCPAP |
Homo sapiens |
IC50 |
= |
2.33 |
nM |
PMID[502008] |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
93.12 |
nM |
PMID[502008] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
10.05 |
nM |
PMID[502008] |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
149.1 |
nM |
PMID[502008] |
NPT1313 |
Cell Line |
Capan-2 |
Homo sapiens |
IC50 |
= |
114.18 |
nM |
PMID[502008] |
NPT1215 |
Cell Line |
8505C |
Homo sapiens |
IC50 |
= |
3.109 |
nM |
PMID[502008] |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
31.39 |
nM |
PMID[502008] |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
1.416 |
nM |
PMID[502008] |
NPT2314 |
Cell Line |
BEN |
Homo sapiens |
IC50 |
= |
81.23 |
nM |
PMID[502008] |
NPT2315 |
Cell Line |
BFTC-905 |
Homo sapiens |
IC50 |
= |
3.773 |
nM |
PMID[502008] |
NPT2316 |
Cell Line |
CFPAC-1 |
Homo sapiens |
IC50 |
= |
93.2 |
nM |
PMID[502008] |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
5.556 |
nM |
PMID[502008] |
NPT2317 |
Cell Line |
ChaGo-K-1 |
Homo sapiens |
IC50 |
= |
1.013 |
nM |
PMID[502008] |
NPT1944 |
Cell Line |
D-247MG |
Homo sapiens |
IC50 |
= |
6.979 |
nM |
PMID[502008] |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
9.616 |
nM |
PMID[502008] |
NPT2319 |
Cell Line |
A204 |
Homo sapiens |
IC50 |
= |
8.765 |
nM |
PMID[502008] |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
1.218 |
nM |
PMID[502008] |
NPT2320 |
Cell Line |
BFTC-909 |
Homo sapiens |
IC50 |
= |
7.532 |
nM |
PMID[502008] |
NPT2321 |
Cell Line |
BHT-101 |
Homo sapiens |
IC50 |
= |
31.36 |
nM |
PMID[502008] |
NPT2322 |
Cell Line |
CHL-1 |
Homo sapiens |
IC50 |
= |
12.0 |
nM |
PMID[502008] |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
9.278 |
nM |
PMID[502008] |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
4.608 |
nM |
PMID[502008] |
NPT2323 |
Cell Line |
BHY |
Homo sapiens |
IC50 |
= |
15.33 |
nM |
PMID[502008] |
NPT2324 |
Cell Line |
CHP-212 |
Homo sapiens |
IC50 |
= |
3.547 |
nM |
PMID[502008] |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
39.1 |
nM |
PMID[502008] |
NPT1953 |
Cell Line |
D-336MG |
Homo sapiens |
IC50 |
= |
7.255 |
nM |
PMID[502008] |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
18.86 |
nM |
PMID[502008] |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
4.32 |
nM |
PMID[502008] |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
23.53 |
nM |
PMID[502008] |
NPT2325 |
Cell Line |
BPH-1 |
Homo sapiens |
IC50 |
= |
3.263 |
nM |
PMID[502008] |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
37.68 |
nM |
PMID[502008] |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
203.92 |
nM |
PMID[502008] |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
562.6 |
nM |
PMID[502008] |
NPT2327 |
Cell Line |
D-423MG |
Homo sapiens |
IC50 |
= |
8.639 |
nM |
PMID[502008] |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
23.49 |
nM |
PMID[502008] |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
6.915 |
nM |
PMID[502008] |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
1.867 |
nM |
PMID[502008] |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
94.15 |
nM |
PMID[502008] |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
7.977 |
nM |
PMID[502008] |
NPT2328 |
Cell Line |
COLO-678 |
Homo sapiens |
IC50 |
= |
2480.78 |
nM |
PMID[502008] |
NPT2329 |
Cell Line |
COLO-679 |
Homo sapiens |
IC50 |
= |
5415.81 |
nM |
PMID[502008] |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
3876.68 |
nM |
PMID[502008] |
NPT2330 |
Cell Line |
D-566MG |
Homo sapiens |
IC50 |
= |
2.043 |
nM |
PMID[502008] |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
12.55 |
nM |
PMID[502008] |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
4975.15 |
nM |
PMID[502008] |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
42.27 |
nM |
PMID[502008] |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
1.126 |
nM |
PMID[502008] |
NPT2332 |
Cell Line |
COLO-680N |
Homo sapiens |
IC50 |
= |
74.71 |
nM |
PMID[502008] |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
7.666 |
nM |
PMID[502008] |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
1.687 |
nM |
PMID[502008] |
NPT2333 |
Cell Line |
DBTRG-05MG |
Homo sapiens |
IC50 |
= |
225.99 |
nM |
PMID[502008] |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
2.16 |
nM |
PMID[502008] |
NPT2334 |
Cell Line |
NCI-H1793 |
Homo sapiens |
IC50 |
= |
29.6 |
nM |
PMID[502008] |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
191.13 |
nM |
PMID[502008] |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
5.136 |
nM |
PMID[502008] |
NPT2335 |
Cell Line |
NCI-H596 |
|
IC50 |
= |
156.07 |
nM |
PMID[502008] |
NPT2336 |
Cell Line |
OE19 |
Homo sapiens |
IC50 |
= |
412.2 |
nM |
PMID[502008] |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
28.59 |
nM |
PMID[502008] |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
IC50 |
= |
1.658 |
nM |
PMID[502008] |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
2.852 |
nM |
PMID[502008] |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
18.71 |
nM |
PMID[502008] |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
67.32 |
nM |
PMID[502008] |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
61.39 |
nM |
PMID[502008] |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
6.943 |
nM |
PMID[502008] |
NPT2339 |
Cell Line |
TGBC24TKB |
Homo sapiens |
IC50 |
= |
32.52 |
nM |
PMID[502008] |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
4.362 |
nM |
PMID[502008] |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
6.367 |
nM |
PMID[502008] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
4.371 |
nM |
PMID[502008] |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
1.187 |
nM |
PMID[502008] |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
7.987 |
nM |
PMID[502008] |
NPT2340 |
Cell Line |
KU-19-19 |
Homo sapiens |
IC50 |
= |
43.72 |
nM |
PMID[502008] |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
8.279 |
nM |
PMID[502008] |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
588.37 |
nM |
PMID[502008] |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
135.5 |
nM |
PMID[502008] |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
3.274 |
nM |
PMID[502008] |
NPT2341 |
Cell Line |
NCI-H1975 |
Homo sapiens |
IC50 |
= |
24.23 |
nM |
PMID[502008] |
NPT2342 |
Cell Line |
NCI-H630 |
Homo sapiens |
IC50 |
= |
241.69 |
nM |
PMID[502008] |
NPT2343 |
Cell Line |
NCI-H650 |
Homo sapiens |
IC50 |
= |
27.08 |
nM |
PMID[502008] |
NPT1968 |
Cell Line |
OMC-1 |
Homo sapiens |
IC50 |
= |
144.1 |
nM |
PMID[502008] |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
3.742 |
nM |
PMID[502008] |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
1.966 |
nM |
PMID[502008] |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
53.3 |
nM |
PMID[502008] |
NPT2344 |
Cell Line |
SK-MEL-24 |
Homo sapiens |
IC50 |
= |
31.55 |
nM |
PMID[502008] |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
8.836 |
nM |
PMID[502008] |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
23.21 |
nM |
PMID[502008] |
NPT2346 |
Cell Line |
TI-73 |
Homo sapiens |
IC50 |
= |
3.212 |
nM |
PMID[502008] |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
42.4 |
nM |
PMID[502008] |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
6.076 |
nM |
PMID[502008] |
NPT2347 |
Cell Line |
GMS-10 |
Homo sapiens |
IC50 |
= |
11.28 |
nM |
PMID[502008] |
NPT2348 |
Cell Line |
HLE |
Homo sapiens |
IC50 |
= |
4.235 |
nM |
PMID[502008] |
NPT2349 |
Cell Line |
HMV-2 cell line |
|
IC50 |
= |
3.905 |
nM |
PMID[502008] |
NPT2350 |
Cell Line |
HN |
Homo sapiens |
IC50 |
= |
4.15 |
nM |
PMID[502008] |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
0.7882 |
nM |
PMID[502008] |
NPT1505 |
Cell Line |
J82 |
Homo sapiens |
IC50 |
= |
68.47 |
nM |
PMID[502008] |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
16.79 |
nM |
PMID[502008] |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
6.977 |
nM |
PMID[502008] |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
14.16 |
nM |
PMID[502008] |
NPT2352 |
Cell Line |
MHH-ES-1 |
Homo sapiens |
IC50 |
= |
5.129 |
nM |
PMID[502008] |
NPT1980 |
Cell Line |
NB14 |
Homo sapiens |
IC50 |
= |
4.953 |
nM |
PMID[502008] |
NPT1995 |
Cell Line |
NB17 |
Homo sapiens |
IC50 |
= |
21.77 |
nM |
PMID[502008] |
NPT2353 |
Cell Line |
NCI-H1993 |
Homo sapiens |
IC50 |
= |
3395.38 |
nM |
PMID[502008] |
NPT2354 |
Cell Line |
NCI-H2009 |
Homo sapiens |
IC50 |
= |
53.45 |
nM |
PMID[502008] |
NPT2355 |
Cell Line |
NCI-H2029 |
Homo sapiens |
IC50 |
= |
203.7 |
nM |
PMID[502008] |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
8.047 |
nM |
PMID[502008] |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
525.78 |
nM |
PMID[502008] |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
69.84 |
nM |
PMID[502008] |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
4.508 |
nM |
PMID[502008] |
NPT2357 |
Cell Line |
RT-112 |
Homo sapiens |
IC50 |
= |
2.708 |
nM |
PMID[502008] |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
17.04 |
nM |
PMID[502008] |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
IC50 |
= |
717.01 |
nM |
PMID[502008] |
NPT2359 |
Cell Line |
SK-MEL-30 |
Homo sapiens |
IC50 |
= |
415.46 |
nM |
PMID[502008] |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
101.3 |
nM |
PMID[502008] |
NPT2360 |
Cell Line |
SW756 |
Homo sapiens |
IC50 |
= |
14.7 |
nM |
PMID[502008] |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
2.329 |
nM |
PMID[502008] |
NPT2362 |
Cell Line |
TYK-nu |
Homo sapiens |
IC50 |
= |
11.9 |
nM |
PMID[502008] |
NPT2363 |
Cell Line |
U-118-MG |
Homo sapiens |
IC50 |
= |
45.16 |
nM |
PMID[502008] |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
8.207 |
nM |
PMID[502008] |
NPT2364 |
Cell Line |
GP5d |
Homo sapiens |
IC50 |
= |
4.674 |
nM |
PMID[502008] |
NPT2365 |
Cell Line |
HO-1-N-1 |
Homo sapiens |
IC50 |
= |
1.756 |
nM |
PMID[502008] |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
1406.87 |
nM |
PMID[502008] |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
0.608 |
nM |
PMID[502008] |
NPT2366 |
Cell Line |
JEG-3 |
Homo sapiens |
IC50 |
= |
12.48 |
nM |
PMID[502008] |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
233.07 |
nM |
PMID[502008] |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
3.69 |
nM |
PMID[502008] |
NPT2367 |
Cell Line |
KYSE-140 |
Homo sapiens |
IC50 |
= |
44.94 |
nM |
PMID[502008] |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
2844.0 |
nM |
PMID[502008] |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
53.33 |
nM |
PMID[502008] |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
38.85 |
nM |
PMID[502008] |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
15.7 |
nM |
PMID[502008] |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
80.02 |
nM |
PMID[502008] |
NPT2368 |
Cell Line |
NCI-H2030 |
Homo sapiens |
IC50 |
= |
27.72 |
nM |
PMID[502008] |
NPT2369 |
Cell Line |
NCI-H2052 |
Homo sapiens |
IC50 |
= |
24.65 |
nM |
PMID[502008] |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
46.86 |
nM |
PMID[502008] |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
27.94 |
nM |
PMID[502008] |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
IC50 |
= |
13.6 |
nM |
PMID[502008] |
NPT2370 |
Cell Line |
RVH-421 |
Homo sapiens |
IC50 |
= |
7.249 |
nM |
PMID[502008] |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
1.439 |
nM |
PMID[502008] |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
8.645 |
nM |
PMID[502008] |
NPT2371 |
Cell Line |
SW837 |
Homo sapiens |
IC50 |
= |
120.44 |
nM |
PMID[502008] |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
255.22 |
nM |
PMID[502008] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
25.72 |
nM |
PMID[502008] |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
10.8 |
nM |
PMID[502008] |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
115.12 |
nM |
PMID[502008] |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
5.753 |
nM |
PMID[502008] |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
7.631 |
nM |
PMID[502008] |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
1.92 |
nM |
PMID[502008] |
NPT2372 |
Cell Line |
H-EMC-SS |
Homo sapiens |
IC50 |
= |
255.94 |
nM |
PMID[502008] |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
IC50 |
= |
25.92 |
nM |
PMID[502008] |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
6.25 |
nM |
PMID[502008] |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
5585.18 |
nM |
PMID[502008] |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
1.705 |
nM |
PMID[502008] |
NPT2373 |
Cell Line |
KYSE-150 cell line |
|
IC50 |
= |
46.53 |
nM |
PMID[502008] |
NPT2374 |
Cell Line |
KYSE-180 |
Homo sapiens |
IC50 |
= |
6.385 |
nM |
PMID[502008] |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
66.35 |
nM |
PMID[502008] |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
1.493 |
nM |
PMID[502008] |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
3.388 |
nM |
PMID[502008] |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
10.1 |
nM |
PMID[502008] |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
5.73 |
nM |
PMID[502008] |
NPT2023 |
Cell Line |
NB7 |
Homo sapiens |
IC50 |
= |
195.12 |
nM |
PMID[502008] |
NPT2376 |
Cell Line |
NBsusSR |
Homo sapiens |
IC50 |
= |
3.232 |
nM |
PMID[502008] |
NPT2377 |
Cell Line |
NCI-H2087 |
Homo sapiens |
IC50 |
= |
30.53 |
nM |
PMID[502008] |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
13.15 |
nM |
PMID[502008] |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
6.88 |
nM |
PMID[502008] |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
175.7 |
nM |
PMID[502008] |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
81.18 |
nM |
PMID[502008] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
6.554 |
nM |
PMID[502008] |
NPT2379 |
Cell Line |
P12-Ichikawa |
Homo sapiens |
IC50 |
= |
1.704 |
nM |
PMID[502008] |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
1.546 |
nM |
PMID[502008] |
NPT2380 |
Cell Line |
SK-N-AS |
Homo sapiens |
IC50 |
= |
8.669 |
nM |
PMID[502008] |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
37.37 |
nM |
PMID[502008] |
NPT2381 |
Cell Line |
SW900 |
Homo sapiens |
IC50 |
= |
25.41 |
nM |
PMID[502008] |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
75.99 |
nM |
PMID[502008] |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
29.98 |
nM |
PMID[502008] |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
3.24 |
nM |
PMID[502008] |
NPT2383 |
Cell Line |
ESS-1 |
Homo sapiens |
IC50 |
= |
4.876 |
nM |
PMID[502008] |
NPT2891 |
Cell Line |
H4 |
Homo sapiens |
IC50 |
= |
5.837 |
nM |
PMID[502008] |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
IC50 |
= |
2.248 |
nM |
PMID[502008] |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
233.41 |
nM |
PMID[502008] |
NPT2384 |
Cell Line |
HPAF-II |
Homo sapiens |
IC50 |
= |
40.05 |
nM |
PMID[502008] |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
20.2 |
nM |
PMID[502008] |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
IC50 |
= |
4.389 |
nM |
PMID[502008] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1082.28 |
nM |
PMID[502008] |
NPT2386 |
Cell Line |
KYSE-270 |
Homo sapiens |
IC50 |
= |
9.632 |
nM |
PMID[502008] |
NPT2387 |
Cell Line |
KYSE-410 |
Homo sapiens |
IC50 |
= |
9.297 |
nM |
PMID[502008] |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
56.27 |
nM |
PMID[502008] |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
8.582 |
nM |
PMID[502008] |
NPT2388 |
Cell Line |
LU-135 |
Homo sapiens |
IC50 |
= |
35.58 |
nM |
PMID[502008] |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
2.698 |
nM |
PMID[502008] |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
48.42 |
nM |
PMID[502008] |
NPT2389 |
Cell Line |
NCI-H1048 |
Homo sapiens |
IC50 |
= |
10.06 |
nM |
PMID[502008] |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
223.56 |
nM |
PMID[502008] |
NPT2390 |
Cell Line |
NCI-H2122 |
Homo sapiens |
IC50 |
= |
3.436 |
nM |
PMID[502008] |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
25.9 |
nM |
PMID[502008] |
NPT2391 |
Cell Line |
NCI-H810 |
Homo sapiens |
IC50 |
= |
68.69 |
nM |
PMID[502008] |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
11.07 |
nM |
PMID[502008] |
NPT2392 |
Cell Line |
S-117 |
Homo sapiens |
IC50 |
= |
5.576 |
nM |
PMID[502008] |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
28.13 |
nM |
PMID[502008] |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
642.78 |
nM |
PMID[502008] |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
1.505 |
nM |
PMID[502008] |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
9.662 |
nM |
PMID[502008] |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
19.39 |
nM |
PMID[502008] |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
13.94 |
nM |
PMID[502008] |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
5.018 |
nM |
PMID[502008] |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
5.788 |
nM |
PMID[502008] |
NPT2047 |
Cell Line |
HC-1 |
Homo sapiens |
IC50 |
= |
4.211 |
nM |
PMID[502008] |
NPT2394 |
Cell Line |
HSC-4 |
Homo sapiens |
IC50 |
= |
2.355 |
nM |
PMID[502008] |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
15.64 |
nM |
PMID[502008] |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
4.682 |
nM |
PMID[502008] |
NPT2395 |
Cell Line |
KYSE-450 |
Homo sapiens |
IC50 |
= |
9.649 |
nM |
PMID[502008] |
NPT2396 |
Cell Line |
KYSE-510 |
Homo sapiens |
IC50 |
= |
5.875 |
nM |
PMID[502008] |
NPT2397 |
Cell Line |
KYSE-520 cell line |
|
IC50 |
= |
47.62 |
nM |
PMID[502008] |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
14.08 |
nM |
PMID[502008] |
NPT2398 |
Cell Line |
MKN-7 |
Homo sapiens |
IC50 |
= |
76.69 |
nM |
PMID[502008] |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
8.652 |
nM |
PMID[502008] |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
43.74 |
nM |
PMID[502008] |
NPT2399 |
Cell Line |
NCI-H2170 |
Homo sapiens |
IC50 |
= |
33.41 |
nM |
PMID[502008] |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
1642.17 |
nM |
PMID[502008] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
8.092 |
nM |
PMID[502008] |
NPT2401 |
Cell Line |
PANC-03-27 |
Homo sapiens |
IC50 |
= |
5.472 |
nM |
PMID[502008] |
NPT2402 |
Cell Line |
PANC-08-13 |
Homo sapiens |
IC50 |
= |
61.47 |
nM |
PMID[502008] |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
8.104 |
nM |
PMID[502008] |
NPT2403 |
Cell Line |
SBC-5 |
Homo sapiens |
IC50 |
= |
7.471 |
nM |
PMID[502008] |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
8155.03 |
nM |
PMID[502008] |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
6.138 |
nM |
PMID[502008] |
NPT2404 |
Cell Line |
SW982 |
Homo sapiens |
IC50 |
= |
8.919 |
nM |
PMID[502008] |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
32.31 |
nM |
PMID[502008] |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
90.53 |
nM |
PMID[502008] |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
8.062 |
nM |
PMID[502008] |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
3.148 |
nM |
PMID[502008] |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
2.754 |
nM |
PMID[502008] |
NPT2406 |
Cell Line |
HCC1395 |
Homo sapiens |
IC50 |
= |
29.25 |
nM |
PMID[502008] |
NPT2407 |
Cell Line |
HCC1419 |
Homo sapiens |
IC50 |
= |
57.16 |
nM |
PMID[502008] |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
4.228 |
nM |
PMID[502008] |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
99.76 |
nM |
PMID[502008] |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
7.787 |
nM |
PMID[502008] |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
1657.4 |
nM |
PMID[502008] |
NPT2408 |
Cell Line |
KYSE-70 cell line |
|
IC50 |
= |
48.35 |
nM |
PMID[502008] |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
5.997 |
nM |
PMID[502008] |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
115.72 |
nM |
PMID[502008] |
NPT2409 |
Cell Line |
LU-99A |
Homo sapiens |
IC50 |
= |
20.83 |
nM |
PMID[502008] |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
4.652 |
nM |
PMID[502008] |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
15.09 |
nM |
PMID[502008] |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
16.42 |
nM |
PMID[502008] |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
133.77 |
nM |
PMID[502008] |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
5.671 |
nM |
PMID[502008] |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
1.622 |
nM |
PMID[502008] |
NPT2412 |
Cell Line |
Panc1005 |
Homo sapiens |
IC50 |
= |
42.8 |
nM |
PMID[502008] |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
3.534 |
nM |
PMID[502008] |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
23.15 |
nM |
PMID[502008] |
NPT2414 |
Cell Line |
SCC-25 |
Homo sapiens |
IC50 |
= |
15.68 |
nM |
PMID[502008] |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
11.75 |
nM |
PMID[502008] |
NPT2415 |
Cell Line |
SKG-IIIa |
Homo sapiens |
IC50 |
= |
17.24 |
nM |
PMID[502008] |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
109.77 |
nM |
PMID[502008] |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
5.104 |
nM |
PMID[502008] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
7.711 |
nM |
PMID[502008] |
NPT2416 |
Cell Line |
UACC-893 |
Homo sapiens |
IC50 |
= |
98.3 |
nM |
PMID[502008] |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
5.107 |
nM |
PMID[502008] |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
7.151 |
nM |
PMID[502008] |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
36.52 |
nM |
PMID[502008] |
NPT2418 |
Cell Line |
HCC1569 |
Homo sapiens |
IC50 |
= |
92.26 |
nM |
PMID[502008] |
NPT2419 |
Cell Line |
HT-1376 |
Homo sapiens |
IC50 |
= |
60.4 |
nM |
PMID[502008] |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
3.319 |
nM |
PMID[502008] |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
1.793 |
nM |
PMID[502008] |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
309.15 |
nM |
PMID[502008] |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
10.29 |
nM |
PMID[502008] |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
6.025 |
nM |
PMID[502008] |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
29.44 |
nM |
PMID[502008] |
NPT3466 |
Cell Line |
MOLT-13 |
Homo sapiens |
IC50 |
= |
5.603 |
nM |
PMID[502008] |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
19.54 |
nM |
PMID[502008] |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
4.277 |
nM |
PMID[502008] |
NPT2411 |
Cell Line |
NCI-H2228 |
Homo sapiens |
IC50 |
= |
41.09 |
nM |
PMID[502008] |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
13.81 |
nM |
PMID[502008] |
NPT2420 |
Cell Line |
NCI-H2291 |
Homo sapiens |
IC50 |
= |
232.1 |
nM |
PMID[502008] |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
132.84 |
nM |
PMID[502008] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
33.37 |
nM |
PMID[502008] |
NPT2421 |
Cell Line |
PFSK-1 |
Homo sapiens |
IC50 |
= |
4.972 |
nM |
PMID[502008] |
NPT2422 |
Cell Line |
SCC-4 |
Homo sapiens |
IC50 |
= |
2.395 |
nM |
PMID[502008] |
NPT2423 |
Cell Line |
SCC-9 |
Homo sapiens |
IC50 |
= |
10.66 |
nM |
PMID[502008] |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
IC50 |
= |
16.06 |
nM |
PMID[502008] |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
11.25 |
nM |
PMID[502008] |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
8147.21 |
nM |
PMID[502008] |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
11.4 |
nM |
PMID[502008] |
NPT2425 |
Cell Line |
UMC-11 |
Homo sapiens |
IC50 |
= |
76.22 |
nM |
PMID[502008] |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
3.273 |
nM |
PMID[502008] |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
7.832 |
nM |
PMID[502008] |
NPT2426 |
Cell Line |
HCC1806 |
Homo sapiens |
IC50 |
= |
0.6303 |
nM |
PMID[502008] |
NPT1884 |
Cell Line |
HCC1937 |
Homo sapiens |
IC50 |
= |
2049.18 |
nM |
PMID[502008] |
NPT2427 |
Cell Line |
HCC1954 |
Homo sapiens |
IC50 |
= |
121.72 |
nM |
PMID[502008] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
45.85 |
nM |
PMID[502008] |
NPT2428 |
Cell Line |
HT-3 |
Homo sapiens |
IC50 |
= |
37.07 |
nM |
PMID[502008] |
NPT2429 |
Cell Line |
HT55 |
Homo sapiens |
IC50 |
= |
391.6 |
nM |
PMID[502008] |
NPT2085 |
Cell Line |
Kasumi 1 |
|
IC50 |
= |
8.059 |
nM |
PMID[502008] |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
3.993 |
nM |
PMID[502008] |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
7.015 |
nM |
PMID[502008] |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
47.7 |
nM |
PMID[502008] |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
15.06 |
nM |
PMID[502008] |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
3.191 |
nM |
PMID[502008] |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
2.429 |
nM |
PMID[502008] |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
3.847 |
nM |
PMID[502008] |
NPT2431 |
Cell Line |
NCI-H1437 |
Homo sapiens |
IC50 |
= |
7.76 |
nM |
PMID[502008] |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
5.706 |
nM |
PMID[502008] |
NPT2432 |
Cell Line |
NCI-H2342 |
Homo sapiens |
IC50 |
= |
950.45 |
nM |
PMID[502008] |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
5.122 |
nM |
PMID[502008] |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
26.35 |
nM |
PMID[502008] |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
1.248 |
nM |
PMID[502008] |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
29.72 |
nM |
PMID[502008] |
NPT890 |
Cell Line |
SNU-387 |
Homo sapiens |
IC50 |
= |
11.42 |
nM |
PMID[502008] |
NPT2433 |
Cell Line |
SNU-423 |
Homo sapiens |
IC50 |
= |
19.47 |
nM |
PMID[502008] |
NPT2434 |
Cell Line |
TCC-SUP |
Homo sapiens |
IC50 |
= |
23.63 |
nM |
PMID[502008] |
NPT2435 |
Cell Line |
VM-CUB-1 |
Homo sapiens |
IC50 |
= |
4.281 |
nM |
PMID[502008] |
NPT2436 |
Cell Line |
VMRC-RCZ |
Homo sapiens |
IC50 |
= |
19.27 |
nM |
PMID[502008] |
NPT1653 |
Cell Line |
WM-115 |
Homo sapiens |
IC50 |
= |
10.16 |
nM |
PMID[502008] |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
510.36 |
nM |
PMID[502008] |
NPT2437 |
Cell Line |
EW-22 |
Homo sapiens |
IC50 |
= |
29.35 |
nM |
PMID[502008] |
NPT2113 |
Cell Line |
EW-24 |
Homo sapiens |
IC50 |
= |
18.01 |
nM |
PMID[502008] |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
79.26 |
nM |
PMID[502008] |
NPT2438 |
Cell Line |
HTC-C3 |
Homo sapiens |
IC50 |
= |
10.38 |
nM |
PMID[502008] |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
12.28 |
nM |
PMID[502008] |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
18.38 |
nM |
PMID[502008] |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
33.33 |
nM |
PMID[502008] |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
40.27 |
nM |
PMID[502008] |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
10.12 |
nM |
PMID[502008] |
NPT2439 |
Cell Line |
MC-IXC |
Homo sapiens |
IC50 |
= |
2.985 |
nM |
PMID[502008] |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
7.953 |
nM |
PMID[502008] |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
30.28 |
nM |
PMID[502008] |
NPT2440 |
Cell Line |
NCI-H1563 |
Homo sapiens |
IC50 |
= |
21.46 |
nM |
PMID[502008] |
NPT2441 |
Cell Line |
NCI-H2347 |
Homo sapiens |
IC50 |
= |
135.12 |
nM |
PMID[502008] |
NPT2442 |
Cell Line |
NCI-H2405 |
Homo sapiens |
IC50 |
= |
826.38 |
nM |
PMID[502008] |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
1.273 |
nM |
PMID[502008] |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
8.484 |
nM |
PMID[502008] |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
8.95 |
nM |
PMID[502008] |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
510.4 |
nM |
PMID[502008] |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
21.9 |
nM |
PMID[502008] |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
16.19 |
nM |
PMID[502008] |
NPT2443 |
Cell Line |
SNU-449 |
Homo sapiens |
IC50 |
= |
127.72 |
nM |
PMID[502008] |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
10.85 |
nM |
PMID[502008] |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
21.47 |
nM |
PMID[502008] |
NPT2444 |
Cell Line |
YAPC |
Homo sapiens |
IC50 |
= |
86.99 |
nM |
PMID[502008] |
NPT2445 |
Cell Line |
YH-13 |
Homo sapiens |
IC50 |
= |
3.702 |
nM |
PMID[502008] |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
37.21 |
nM |
PMID[502008] |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
19.83 |
nM |
PMID[502008] |
NPT2446 |
Cell Line |
HCC38 |
Homo sapiens |
IC50 |
= |
58.38 |
nM |
PMID[502008] |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
17.31 |
nM |
PMID[502008] |
NPT2447 |
Cell Line |
HuCCT-1 |
Homo sapiens |
IC50 |
= |
17.29 |
nM |
PMID[502008] |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
9.324 |
nM |
PMID[502008] |
NPT2448 |
Cell Line |
KLE |
Homo sapiens |
IC50 |
= |
309.24 |
nM |
PMID[502008] |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
145.03 |
nM |
PMID[502008] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
31.6 |
nM |
PMID[502008] |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
30.83 |
nM |
PMID[502008] |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
12.22 |
nM |
PMID[502008] |
NPT2449 |
Cell Line |
NCI-H1573 |
Homo sapiens |
IC50 |
= |
30.74 |
nM |
PMID[502008] |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
4.236 |
nM |
PMID[502008] |
NPT2450 |
Cell Line |
NCI-H2452 |
Homo sapiens |
IC50 |
= |
9.587 |
nM |
PMID[502008] |
NPT2451 |
Cell Line |
NCI-H28 |
Homo sapiens |
IC50 |
= |
34.26 |
nM |
PMID[502008] |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
3.03 |
nM |
PMID[502008] |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
7.859 |
nM |
PMID[502008] |
NPT2453 |
Cell Line |
RCM-1 |
Homo sapiens |
IC50 |
= |
1369.69 |
nM |
PMID[502008] |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
4.172 |
nM |
PMID[502008] |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
36.31 |
nM |
PMID[502008] |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
1.211 |
nM |
PMID[502008] |
NPT2455 |
Cell Line |
SNU-C2B |
Homo sapiens |
IC50 |
= |
24.67 |
nM |
PMID[502008] |
NPT2456 |
Cell Line |
TE-11 |
Homo sapiens |
IC50 |
= |
5.128 |
nM |
PMID[502008] |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
700.72 |
nM |
PMID[502008] |
NPT2457 |
Cell Line |
YKG-1 |
Homo sapiens |
IC50 |
= |
5.534 |
nM |
PMID[502008] |
NPT994 |
Cell Line |
ZR-75-30 |
Homo sapiens |
IC50 |
= |
402.55 |
nM |
PMID[502008] |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
1.261 |
nM |
PMID[502008] |
NPT1216 |
Cell Line |
FaDu |
Homo sapiens |
IC50 |
= |
20.02 |
nM |
PMID[502008] |
NPT2458 |
Cell Line |
FTC-133 |
Homo sapiens |
IC50 |
= |
8.444 |
nM |
PMID[502008] |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
20.8 |
nM |
PMID[502008] |
NPT2460 |
Cell Line |
HCE-4 |
Homo sapiens |
IC50 |
= |
18.09 |
nM |
PMID[502008] |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
87.74 |
nM |
PMID[502008] |
NPT2461 |
Cell Line |
HuO-3N1 |
Homo sapiens |
IC50 |
= |
4.827 |
nM |
PMID[502008] |
NPT2462 |
Cell Line |
HuO9 |
Homo sapiens |
IC50 |
= |
12.64 |
nM |
PMID[502008] |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
5.339 |
nM |
PMID[502008] |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
14.42 |
nM |
PMID[502008] |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
64.11 |
nM |
PMID[502008] |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
9.064 |
nM |
PMID[502008] |
NPT2464 |
Cell Line |
MDA-MB-175-VII |
Homo sapiens |
IC50 |
= |
267.63 |
nM |
PMID[502008] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
44.59 |
nM |
PMID[502008] |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
2.805 |
nM |
PMID[502008] |
NPT2465 |
Cell Line |
NCI-H1623 |
Homo sapiens |
IC50 |
= |
503.24 |
nM |
PMID[502008] |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
5.519 |
nM |
PMID[502008] |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
37.01 |
nM |
PMID[502008] |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
40.88 |
nM |
PMID[502008] |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
5.893 |
nM |
PMID[502008] |
NPT2467 |
Cell Line |
RERF-LC-MS |
Homo sapiens |
IC50 |
= |
15.15 |
nM |
PMID[502008] |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
3.4 |
nM |
PMID[502008] |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
43.54 |
nM |
PMID[502008] |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
148.18 |
nM |
PMID[502008] |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
6.135 |
nM |
PMID[502008] |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
270.54 |
nM |
PMID[502008] |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
4123.67 |
nM |
PMID[502008] |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
IC50 |
= |
8.671 |
nM |
PMID[502008] |
NPT2470 |
Cell Line |
G-402 |
Homo sapiens |
IC50 |
= |
17.58 |
nM |
PMID[502008] |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
20.01 |
nM |
PMID[502008] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.626 |
nM |
PMID[502008] |
NPT2471 |
Cell Line |
HuP-T3 |
Homo sapiens |
IC50 |
= |
17.96 |
nM |
PMID[502008] |
NPT2472 |
Cell Line |
HuP-T4 |
Homo sapiens |
IC50 |
= |
43.18 |
nM |
PMID[502008] |
NPT2163 |
Cell Line |
KMOE-2 |
Homo sapiens |
IC50 |
= |
20.76 |
nM |
PMID[502008] |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
8.574 |
nM |
PMID[502008] |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
21.23 |
nM |
PMID[502008] |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
1.662 |
nM |
PMID[502008] |
NPT2474 |
Cell Line |
MDA-MB-415 |
Homo sapiens |
IC50 |
= |
18.55 |
nM |
PMID[502008] |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
24.19 |
nM |
PMID[502008] |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
60.31 |
nM |
PMID[502008] |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
126.77 |
nM |
PMID[502008] |
NPT2475 |
Cell Line |
NCI-H1651 |
Homo sapiens |
IC50 |
= |
23.0 |
nM |
PMID[502008] |
NPT2476 |
Cell Line |
NCI-H441 |
Homo sapiens |
IC50 |
= |
473.3 |
nM |
PMID[502008] |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
2.122 |
nM |
PMID[502008] |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
3.455 |
nM |
PMID[502008] |
NPT2478 |
Cell Line |
NY |
Homo sapiens |
IC50 |
= |
5315.23 |
nM |
PMID[502008] |
NPT2479 |
Cell Line |
OAW-28 |
Homo sapiens |
IC50 |
= |
40.72 |
nM |
PMID[502008] |
NPT2480 |
Cell Line |
RH-18 |
Homo sapiens |
IC50 |
= |
1128.93 |
nM |
PMID[502008] |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
8.239 |
nM |
PMID[502008] |
NPT2481 |
Cell Line |
SW1088 |
Homo sapiens |
IC50 |
= |
16.97 |
nM |
PMID[502008] |
NPT2482 |
Cell Line |
SW 1116 |
Homo sapiens |
IC50 |
= |
1163.6 |
nM |
PMID[502008] |
NPT2483 |
Cell Line |
SW13 |
Homo sapiens |
IC50 |
= |
5.49 |
nM |
PMID[502008] |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
56.47 |
nM |
PMID[502008] |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
38.83 |
nM |
PMID[502008] |
NPT2175 |
Cell Line |
GAK |
Homo sapiens |
IC50 |
= |
219.86 |
nM |
PMID[502008] |
NPT2484 |
Cell Line |
GAMG |
Homo sapiens |
IC50 |
= |
19.38 |
nM |
PMID[502008] |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
78.58 |
nM |
PMID[502008] |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
3.33 |
nM |
PMID[502008] |
NPT2485 |
Cell Line |
IA-LM |
Homo sapiens |
IC50 |
= |
68.58 |
nM |
PMID[502008] |
NPT2486 |
Cell Line |
IGR-1 |
Homo sapiens |
IC50 |
= |
2.076 |
nM |
PMID[502008] |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
215.27 |
nM |
PMID[502008] |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
18.69 |
nM |
PMID[502008] |
NPT2487 |
Cell Line |
KNS-62 |
Homo sapiens |
IC50 |
= |
5.802 |
nM |
PMID[502008] |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
7.896 |
nM |
PMID[502008] |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
3.285 |
nM |
PMID[502008] |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
4.473 |
nM |
PMID[502008] |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
11.08 |
nM |
PMID[502008] |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
9.134 |
nM |
PMID[502008] |
NPT2490 |
Cell Line |
NCI-H1666 |
Homo sapiens |
IC50 |
= |
20.12 |
nM |
PMID[502008] |
NPT2491 |
Cell Line |
NCI-H1693 |
Homo sapiens |
IC50 |
= |
78.21 |
nM |
PMID[502008] |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
46.39 |
nM |
PMID[502008] |
NPT2184 |
Cell Line |
NCI-H510A |
Homo sapiens |
IC50 |
= |
2.753 |
nM |
PMID[502008] |
NPT2492 |
Cell Line |
OAW-42 |
Homo sapiens |
IC50 |
= |
233.12 |
nM |
PMID[502008] |
NPT2493 |
Cell Line |
OC-314 |
Homo sapiens |
IC50 |
= |
2.225 |
nM |
PMID[502008] |
NPT2494 |
Cell Line |
RMG-I |
Homo sapiens |
IC50 |
= |
116.58 |
nM |
PMID[502008] |
NPT3467 |
Cell Line |
SJRH30 |
Homo sapiens |
IC50 |
= |
59.36 |
nM |
PMID[502008] |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
12.06 |
nM |
PMID[502008] |
NPT2495 |
Cell Line |
SW1417 |
Homo sapiens |
IC50 |
= |
423.54 |
nM |
PMID[502008] |
NPT2496 |
Cell Line |
SW1463 |
Homo sapiens |
IC50 |
= |
69.69 |
nM |
PMID[502008] |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
IC50 |
= |
33.25 |
nM |
PMID[502008] |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
6.156 |
nM |
PMID[502008] |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
4.27 |
nM |
PMID[502008] |
NPT1354 |
Cell Line |
TGBC11TKB |
Homo sapiens |
IC50 |
= |
15.83 |
nM |
PMID[502008] |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
39.85 |
nM |
PMID[502008] |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
642.79 |
nM |
PMID[502008] |
NPT2497 |
Cell Line |
HEC-1 |
Homo sapiens |
IC50 |
= |
11.35 |
nM |
PMID[502008] |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
20.16 |
nM |
PMID[502008] |
NPT2498 |
Cell Line |
KOSC-2 |
Homo sapiens |
IC50 |
= |
0.6975 |
nM |
PMID[502008] |
NPT2499 |
Cell Line |
KP-4 |
Homo sapiens |
IC50 |
= |
2.369 |
nM |
PMID[502008] |
NPT2500 |
Cell Line |
LCLC-103H cell line |
|
IC50 |
= |
1.502 |
nM |
PMID[502008] |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
14.74 |
nM |
PMID[502008] |
NPT2501 |
Cell Line |
MEL-HO |
Homo sapiens |
IC50 |
= |
53.86 |
nM |
PMID[502008] |
NPT2502 |
Cell Line |
MEL-JUSO |
Homo sapiens |
IC50 |
= |
17.51 |
nM |
PMID[502008] |
NPT2503 |
Cell Line |
NCI-H1703 |
Homo sapiens |
IC50 |
= |
1.431 |
nM |
PMID[502008] |
NPT2504 |
Cell Line |
NCI-H1755 |
Homo sapiens |
IC50 |
= |
19.36 |
nM |
PMID[502008] |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
30.13 |
nM |
PMID[502008] |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
138.49 |
nM |
PMID[502008] |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
7.561 |
nM |
PMID[502008] |
NPT2506 |
Cell Line |
RO82-W-1 |
Homo sapiens |
IC50 |
= |
5.57 |
nM |
PMID[502008] |
NPT2507 |
Cell Line |
RPMI-2650 |
Homo sapiens |
IC50 |
= |
26.61 |
nM |
PMID[502008] |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
12.05 |
nM |
PMID[502008] |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
58.6 |
nM |
PMID[502008] |
NPT2508 |
Cell Line |
SW1710 |
Homo sapiens |
IC50 |
= |
5.607 |
nM |
PMID[502008] |
NPT2509 |
Cell Line |
SW1783 |
Homo sapiens |
IC50 |
= |
85.55 |
nM |
PMID[502008] |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
31.21 |
nM |
PMID[502008] |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
49.73 |
nM |
PMID[502008] |
NPT2510 |
Cell Line |
GCT |
Homo sapiens |
IC50 |
= |
4.728 |
nM |
PMID[502008] |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
32.84 |
nM |
PMID[502008] |
NPT2511 |
Cell Line |
HGC-27 |
Homo sapiens |
IC50 |
= |
1.012 |
nM |
PMID[502008] |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
4.526 |
nM |
PMID[502008] |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
67.68 |
nM |
PMID[502008] |
NPT2207 |
Cell Line |
KP-N-YN |
Homo sapiens |
IC50 |
= |
46.36 |
nM |
PMID[502008] |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
22.91 |
nM |
PMID[502008] |
NPT2512 |
Cell Line |
LCLC-97TM1 |
Homo sapiens |
IC50 |
= |
5.491 |
nM |
PMID[502008] |
NPT2513 |
Cell Line |
LK-2 |
Homo sapiens |
IC50 |
= |
7.503 |
nM |
PMID[502008] |
NPT2514 |
Cell Line |
LN-405 |
Homo sapiens |
IC50 |
= |
12.4 |
nM |
PMID[502008] |
NPT2515 |
Cell Line |
MFE-280 |
Homo sapiens |
IC50 |
= |
36.08 |
nM |
PMID[502008] |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
7.317 |
nM |
PMID[502008] |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
61.41 |
nM |
PMID[502008] |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
28.46 |
nM |
PMID[502008] |
NPT1669 |
Cell Line |
NCI-H1792 |
Homo sapiens |
IC50 |
= |
4.391 |
nM |
PMID[502008] |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
3.7 |
nM |
PMID[502009] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.5 |
nM |
PMID[502010] |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
0.8 |
nM |
PMID[502010] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
7.0 |
nM |
PMID[502010] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10.9 |
nM |
PMID[502013] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio IC50 |
= |
90.0 |
n.a. |
PMID[502016] |
NPT4465 |
Cell Line |
HCT-116/VM46 |
Homo sapiens |
IC50 |
> |
110.0 |
nM |
PMID[502016] |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
4.6 |
nM |
PMID[502016] |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
8.0 |
nM |
PMID[502016] |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[502016] |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
4.6 |
nM |
PMID[502016] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
110.0 |
nM |
PMID[502016] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6.8 |
nM |
PMID[502016] |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
3.5 |
nM |
PMID[502016] |
NPT4609 |
Cell Line |
HCC1143 |
Homo sapiens |
IC50 |
= |
3.8 |
nM |
PMID[502016] |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
4.5 |
nM |
PMID[502016] |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
4.0 |
nM |
PMID[502016] |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
6.0 |
nM |
PMID[502016] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
5.2 |
nM |
PMID[502019] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
RatioGI50 |
= |
500.0 |
n.a. |
PMID[502019] |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
GI50 |
= |
1.5 |
nM |
PMID[502019] |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
GI50 |
= |
86.8 |
nM |
PMID[502019] |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
RatioGI50 |
= |
58.0 |
n.a. |
PMID[502019] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.5 |
nM |
PMID[502020] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2.7 |
nM |
PMID[502020] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
PMID[502020] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2.9 |
nM |
PMID[502021] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
870.0 |
nM |
PMID[502021] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
300.0 |
n.a. |
PMID[502021] |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
2.0 |
nM |
PMID[502022] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
105.0 |
n.a. |
PMID[502022] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.02 |
ug.mL-1 |
PMID[502023] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.22 |
ug.mL-1 |
PMID[502023] |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.047 |
ug.mL-1 |
PMID[502023] |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
52.5 |
nM |
PMID[502024] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
80.7 |
nM |
PMID[502024] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Activity |
= |
21.0 |
% |
PMID[502025] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
44.0 |
% |
PMID[502025] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
1.3 |
nM |
PMID[502026] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
670.0 |
nM |
PMID[502026] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
248.86 |
n.a. |
PMID[502026] |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
1.0 |
nM |
PMID[502027] |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
193.0 |
n.a. |
PMID[502027] |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
200.0 |
nM |
PMID[502024] |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
GI50 |
= |
4.0 |
nM |
PMID[502028] |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
GI50 |
= |
210.0 |
nM |
PMID[502028] |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
Ratio |
= |
525.0 |
n.a. |
PMID[502028] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10.0 |
nM |
PMID[502029] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
0.25 |
nM |
PMID[502032] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
TGI |
= |
0.25 |
nM |
PMID[502032] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
LC50 |
= |
1.0 |
nM |
PMID[502032] |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
1.0 |
nM |
PMID[502032] |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
TGI |
= |
50.0 |
nM |
PMID[502032] |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
LC50 |
= |
2510.0 |
nM |
PMID[502032] |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
0.6 |
nM |
PMID[502032] |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
TGI |
= |
2.5 |
nM |
PMID[502032] |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
LC50 |
= |
790.0 |
nM |
PMID[502032] |
NPT616 |
Cell Line |
MDCK |
Canis lupus familiaris |
Ratio |
= |
1.8 |
n.a. |
PMID[502034] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.49 |
nM |
PMID[502035] |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8.78 |
nM |
PMID[502035] |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
1.82 |
nM |
PMID[502035] |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
4.5 |
nM |
PMID[502037] |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.5 |
nM |
PMID[502037] |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
15.0 |
nM |
PMID[502038] |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
> |
80.0 |
% |
PMID[502038] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
766.0 |
nM |
PMID[502038] |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
53.0 |
nM |
PMID[502038] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
81.0 |
nM |
PMID[502038] |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
30.0 |
% |
PMID[502039] |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
880.24 |
nM |
PMID[21401115] |
NPT27 |
Others |
Unspecified |
|
Activity |
= |
1.0 |
n.a. |
PMID[501791] |
NPT27 |
Others |
Unspecified |
|
Bullatacin index |
= |
18.8 |
n.a. |
PMID[501791] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Log kill |
= |
2.8 |
n.a. |
PMID[501792] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Log kill |
= |
1.9 |
n.a. |
PMID[501792] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Log kill |
< |
0.7 |
n.a. |
PMID[501792] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival days |
= |
11.0 |
n.a. |
PMID[501795] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival days |
= |
15.5 |
n.a. |
PMID[501795] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
14.6 |
% |
PMID[501795] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
89.0 |
% |
PMID[501795] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
18.0 |
nM |
PMID[501796] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
246.0 |
nM |
PMID[501796] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.1 |
ug.mL-1 |
PMID[501797] |
NPT2 |
Others |
Unspecified |
|
Log CR |
= |
2.38 |
n.a. |
PMID[501798] |
NPT35 |
Others |
n.a. |
|
LogD |
= |
3.69 |
n.a. |
PMID[501798] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
19.9 |
n.a. |
PMID[501799] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
31.3 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
69.7 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
84.8 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
140.3 |
pM of drug (10e6*cells)-1 |
PMID[501799] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1000.0 |
nM |
PMID[501800] |
NPT2 |
Others |
Unspecified |
|
Fold_increase |
= |
8.0 |
n.a. |
PMID[501802] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
600.0 |
nM |
PMID[501803] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
30.8 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
42.3 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
47.1 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
48.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
59.3 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
72.9 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
49.5 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
81.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
40.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survivors |
= |
0.0 |
n.a. |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survivors |
= |
1.0 |
n.a. |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survivors |
= |
4.0 |
n.a. |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
112.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survivors |
= |
5.0 |
n.a. |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survivors |
= |
2.0 |
n.a. |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
52.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
58.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
35.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
30.3 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
31.9 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
37.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
24.7 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
57.6 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
21.6 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
54.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
63.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
0.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
61.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ILS |
= |
74.0 |
% |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
26.0 |
mg.kg-1 |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
28.0 |
mg.kg-1 |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
27.4 |
mg.kg-1 |
PMID[501806] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
10.0 |
mg.kg-1 |
PMID[501806] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LD50 |
= |
2.9 |
mg.kg-1 |
PMID[501806] |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
700.0 |
nM |
PMID[501808] |
NPT781 |
Individual Protein |
Tubulin alpha chain |
Sus scrofa |
Inhibition |
= |
64.0 |
% |
PMID[501808] |
NPT27 |
Others |
Unspecified |
|
EC50 |
= |
1.2 |
nM |
PMID[501811] |
NPT679 |
Individual Protein |
Monoamine oxidase B |
Bos taurus |
Ki |
= |
77000.0 |
nM |
PMID[501812] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
5.2 |
n.a. |
PMID[501813] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
33.0 |
nM/mg*min |
PMID[501813] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Inhibition |
= |
75.0 |
% |
PMID[501813] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[501813] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
> |
50000.0 |
nM |
PMID[501813] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5.0 |
nM |
PMID[501814] |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
70.0 |
nM |
PMID[501815] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
100.0 |
nM |
PMID[501816] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Binding site fraction |
= |
0.4 |
n.a. |
PMID[501816] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
34000.0 |
nM |
PMID[501816] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
1300.0 |
nM |
PMID[501816] |
NPT35 |
Others |
n.a. |
|
pKa |
= |
7.59 |
n.a. |
PMID[501816] |
NPT35 |
Others |
n.a. |
|
pKa |
= |
5.96 |
n.a. |
PMID[501816] |
NPT35 |
Others |
n.a. |
|
pKa |
= |
7.4 |
n.a. |
PMID[501816] |
NPT35 |
Others |
n.a. |
|
pKa |
= |
5.4 |
n.a. |
PMID[501816] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
540.0 |
nM |
PMID[501818] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
20.0 |
nM |
PMID[501818] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.6 |
nM |
PMID[501828] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
8.9 |
nM |
PMID[501828] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
356.0 |
nM |
PMID[501829] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
8.0 |
nM |
PMID[501829] |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
300.0 |
nM |
PMID[501830] |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
EC50 |
= |
200.0 |
nM |
PMID[501831] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
375.0 |
nM |
PMID[501833] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.0 |
nM |
PMID[501833] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2818.38 |
nM |
PMID[501836] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
10000.0 |
nM |
PMID[501836] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
10471.29 |
nM |
PMID[501836] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
114815362149.69 |
nM |
PMID[501836] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1000.0 |
nM |
PMID[501838] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
950.0 |
nM |
PMID[501839] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1660.0 |
nM |
PMID[501839] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.11 |
nM |
PMID[501840] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1040.0 |
nM |
PMID[501840] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.38 |
nM |
PMID[501841] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
210.0 |
n.a. |
PMID[501843] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.7 |
uM |
PMID[501844] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40.0 |
uM |
PMID[501844] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
4.5 |
uM |
PMID[501844] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
42.0 |
uM |
PMID[501844] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
1.2 |
uM |
PMID[501844] |
NPT1881 |
Uncleic Acid |
Calf thymus DNA |
Bos taurus |
Activity |
> |
70.0 |
% |
PMID[501846] |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Activity |
= |
100.0 |
% |
PMID[501846] |
NPT679 |
Individual Protein |
Monoamine oxidase B |
Bos taurus |
Ki |
= |
77000.0 |
nM |
PMID[501848] |
NPT27 |
Others |
Unspecified |
|
Drug uptake |
= |
18.7 |
% |
PMID[501848] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.0 |
n.a. |
PMID[501849] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2100.0 |
nM |
PMID[501849] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500.0 |
nM |
PMID[501851] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
0.06 |
ug ml-1 |
PMID[501853] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
0.5 |
ug ml-1 |
PMID[501853] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
2.6 |
ug ml-1 |
PMID[501853] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
1.1 |
ug ml-1 |
PMID[501853] |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
8200.0 |
nM |
PMID[501854] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
90.0 |
nM |
PMID[501855] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
2.4 |
ug ml-1 |
PMID[501857] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4000.0 |
nM |
PMID[501863] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
100.0 |
% |
PMID[501864] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
0.0 |
% |
PMID[501864] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4000.0 |
nM |
PMID[501866] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
ED50 |
= |
2.6 |
ug ml-1 |
PMID[501870] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
260.0 |
nM |
PMID[501872] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
210.0 |
n.a. |
PMID[501875] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
210.0 |
n.a. |
PMID[501877] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
35.0 |
% |
PMID[501883] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
31.0 |
% |
PMID[501883] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000.0 |
nM |
PMID[501884] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500.0 |
nM |
PMID[501885] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1150.0 |
nM |
PMID[501887] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CL |
= |
3.1 |
mL.min-1.kg-1 |
PMID[501888] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CL_renal |
= |
2.64 |
mL.min-1.kg-1 |
PMID[501888] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500.0 |
nM |
PMID[501889] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Fg |
= |
1.02 |
n.a. |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CL_renal |
= |
2.6 |
mL.min-1.kg-1 |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CL |
= |
3.1 |
mL.min-1.kg-1 |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Vdss |
= |
28.0 |
L.kg-1 |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
F_fraction |
= |
0.05 |
n.a. |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Fa |
= |
0.05 |
n.a. |
PMID[501894] |
NPT614 |
Tissue |
Plasma |
Rattus norvegicus |
Fu |
= |
0.14 |
n.a. |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CL |
= |
0.5 |
mL.min-1.kg-1 |
PMID[501894] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Fh |
= |
0.98 |
n.a. |
PMID[501894] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
< |
100.0 |
nM |
PMID[501896] |
NPT35 |
Others |
n.a. |
|
LogP |
= |
3.9 |
n.a. |
PMID[501901] |
NPT2 |
Others |
Unspecified |
|
RBA |
= |
0.98 |
n.a. |
PMID[501903] |
NPT2 |
Others |
Unspecified |
|
RBA |
= |
1.37 |
n.a. |
PMID[501903] |
NPT2 |
Others |
Unspecified |
|
RBA |
= |
1.21 |
n.a. |
PMID[501903] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
12.6 |
nM |
PMID[501904] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
2037.0 |
nM |
PMID[501904] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
162.0 |
nM |
PMID[501904] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
8.5 |
nM |
PMID[501904] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
13.0 |
nM |
PMID[501904] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
EC50 |
= |
28.0 |
nM |
PMID[501905] |
NPT1188 |
Organism |
Plasmodium yoelii yoelii |
Plasmodium yoelii yoelii |
IC50 |
= |
7950.0 |
nM |
PMID[501906] |
NPT2 |
Others |
Unspecified |
|
Selectivity Index |
= |
6.85 |
n.a. |
PMID[501906] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
680.0 |
nM |
PMID[501907] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17.0 |
nM |
PMID[501907] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.4 |
nM |
PMID[501908] |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
= |
6.0 |
mm |
PMID[501910] |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
= |
0.0 |
mm |
PMID[501910] |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PMID[501911] |
NPT27 |
Others |
Unspecified |
|
T1/2 |
= |
67.0 |
hr |
PMID[501912] |
NPT27 |
Others |
Unspecified |
|
MRT |
= |
150.0 |
hr |
PMID[501912] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Fu |
= |
0.14 |
n.a. |
PMID[501912] |
NPT27 |
Others |
Unspecified |
|
Vdss |
= |
1.5 |
L.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
Vdss |
= |
2.3 |
L.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
3.1 |
mL.min-1.kg-1 |
PMID[501912] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
7.0 |
mL.min-1.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
Vdss |
= |
12.0 |
mL/min/kg |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
12.0 |
mL.min-1.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
22.0 |
mL.min-1.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
Vdss |
= |
24.0 |
L.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
CL |
= |
25.0 |
mL.min-1.kg-1 |
PMID[501913] |
NPT27 |
Others |
Unspecified |
|
Vdss |
= |
28.0 |
L.kg-1 |
PMID[501912] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1600.0 |
nM |
PMID[501916] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
100.0 |
nM |
PMID[501919] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.63 |
nM |
PMID[501919] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.24 |
nM |
PMID[501919] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2.0 |
nM |
PMID[501920] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.28 |
nM |
PMID[501921] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
439.73 |
nM |
PMID[501921] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Ratio IC50 |
= |
224.18 |
n.a. |
PMID[501921] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.28 |
nM |
PMID[501922] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
224.18 |
n.a. |
PMID[501922] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
439.73 |
nM |
PMID[501922] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.0086 |
ug.mL-1 |
PMID[501928] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.8 |
nM |
PMID[501931] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.099 |
nM |
PMID[501931] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
600.0 |
nM |
PMID[501931] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
230.0 |
nM |
PMID[501932] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.0 |
nM |
PMID[501933] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
375000.0 |
nM |
PMID[501933] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
n.a. |
849.2 |
nM |
PMID[501911] |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
n.a. |
11220.2 |
nM |
PMID[501936] |
NPT8 |
Individual Protein |
DNA polymerase iota |
Homo sapiens |
Potency |
n.a. |
44668.4 |
nM |
PMID[501936] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
n.a. |
477.5 |
nM |
PMID[501911] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Papp |
< |
10.0 |
nm/s |
PMID[501937] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Papp |
= |
232.0 |
nm/s |
PMID[501937] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ratio_Papp |
> |
23.0 |
n.a. |
PMID[501937] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ratio_ATPase activity |
= |
4.31 |
n.a. |
PMID[501937] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
% maximum response |
= |
24.4 |
% |
PMID[501937] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25191.0 |
nM |
PMID[501938] |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
22585.0 |
nM |
PMID[501938] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_bilirubinemia |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_cholecystitis |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_cholelithiasis |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_cirrhosis |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_elevated liver function tests |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_hepatic failure |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_hepatic necrosis |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_hepatitis |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_hepatomegaly |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_jaundice |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_liver disease |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_liver fatty |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_liver function tests abnormal |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20596 |
PHENOTYPE |
Hepatotoxicity |
n.a. |
HepSE_Combined Scores |
= |
0.0 |
n.a. |
PMID[501939] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.8 |
nM |
PMID[501940] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
0.099 |
nM |
PMID[501940] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
600.0 |
nM |
PMID[501940] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
230.0 |
nM |
PMID[501941] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
200.0 |
nM |
PMID[501942] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
2.3 |
nM |
PMID[501911] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
11.0 |
nM |
PMID[501944] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.5 |
nM |
PMID[501944] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
15.0 |
nM |
PMID[501944] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
4.2 |
nM |
PMID[501944] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
205.0 |
nM |
PMID[501945] |
NPT1018 |
Organism |
Trypanosoma brucei |
Trypanosoma brucei |
IC50 |
= |
410.0 |
nM |
PMID[501947] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Km |
= |
800.0 |
nM |
PMID[501948] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
44.0 |
% |
PMID[501971] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Activity |
= |
75.0 |
% |
PMID[501972] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Km |
= |
18990.0 |
nM |
PMID[501973] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Km |
= |
252800.0 |
nM |
PMID[501974] |
NPT713 |
Individual Protein |
Bile salt export pump |
Homo sapiens |
IC50 |
= |
114700.0 |
nM |
PMID[501975] |
NPT713 |
Individual Protein |
Bile salt export pump |
Homo sapiens |
IC50 |
= |
62000.0 |
nM |
PMID[501975] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Km |
= |
5710.0 |
nM |
PMID[501966] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
EC50 |
= |
14600.0 |
nM |
PMID[501977] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
EC50 |
= |
34000.0 |
nM |
PMID[501977] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Km |
= |
99400.0 |
nM |
PMID[501976] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
17700.0 |
nM |
PMID[501978] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
19900.0 |
nM |
PMID[501978] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
29500.0 |
nM |
PMID[501978] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
29000.0 |
nM |
PMID[501979] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
> |
50000.0 |
nM |
PMID[501972] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Kd |
= |
3000.0 |
nM |
PMID[501950] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
140000.0 |
nM |
PMID[501974] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
15000.0 |
nM |
PMID[501981] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
2100.0 |
nM |
PMID[501982] |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
36500.0 |
nM |
PMID[501983] |
NPT1188 |
Organism |
Plasmodium yoelii yoelii |
Plasmodium yoelii yoelii |
IC50 |
= |
7950.0 |
nM |
PMID[501985] |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
54.3 |
% |
PMID[501989] |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
57.6 |
% |
PMID[501989] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
100.0 |
nM |
PMID[501991] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
32.4 |
10'-7 cm/s |
PMID[501993] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
2.2 |
10'-7 cm/s |
PMID[501993] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
15.0 |
n.a. |
PMID[501993] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
205.0 |
nM |
PMID[501994] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
53.42 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
47.54 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
38.06 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
28.2 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
21.68 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
16.27 |
% |
PMID[501995] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.6 |
ug.mL-1 |
PMID[501995] |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
6.0 |
n.a. |
PMID[501996] |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
2.0 |
n.a. |
PMID[501996] |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
0.6 |
cm |
PMID[501996] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.6 |
ug.mL-1 |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
53.42 |
% |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
47.54 |
% |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
38.06 |
% |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
28.2 |
% |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
21.68 |
% |
PMID[501999] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Activity |
= |
16.27 |
% |
PMID[501999] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Inhibition |
= |
50.0 |
% |
PMID[502000] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
144.0 |
nM |
PMID[502001] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.0 |
nM |
PMID[502001] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Inhibition |
= |
50.0 |
% |
PMID[502002] |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
27.5 |
n.a. |
PMID[502003] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
11.0 |
nM |
PMID[502003] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.0 |
nM |
PMID[502004] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
9.0 |
nM |
PMID[502004] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1500.0 |
nM |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
50.0 |
% |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
0.5 |
n.a. |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
37.0 |
% |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
16.0 |
% |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
53.0 |
% |
PMID[502005] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
45.0 |
% |
PMID[502005] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
211.0 |
nM |
PMID[502006] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
9.0 |
nM |
PMID[502007] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.0 |
nM |
PMID[502007] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5.2 |
nM |
PMID[502009] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.0 |
nM |
PMID[502010] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2100.0 |
nM |
PMID[502010] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
5000.0 |
nM |
PMID[502011] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
6.0 |
nM |
PMID[502011] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
1.6 |
nM |
PMID[502014] |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
IC50 |
= |
94.0 |
nM |
PMID[502015] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
7.9 |
nM |
PMID[502016] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
19.6 |
nM |
PMID[502016] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5.1 |
nM |
PMID[502016] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.9 |
nM |
PMID[502016] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Activity |
= |
50.0 |
% |
PMID[502016] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
52.89 |
% |
PMID[502017] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (moderate) |
= |
5.0 |
n.a. |
PMID[502018] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (moderate) |
= |
22.6 |
% |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (acute) |
= |
1.0 |
n.a. |
PMID[502018] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (acute) |
= |
0.0 |
% |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (cytolytic) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (choleostasis) |
= |
1.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (severe hepatitis) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (chronic liver disease) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (cirrhosis) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (granulomatous hepatitis) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (association with vascular disease) |
= |
1.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (steatosis) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Hepatotoxicity (malignant tumour) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Hepatotoxicity (benign tumour) |
= |
0.0 |
n.a. |
PMID[502018] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
1412.5 |
nM |
PMID[501936] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
251.2 |
nM |
PMID[501936] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
2.8 |
nM |
PMID[502019] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
1402.0 |
nM |
PMID[502019] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2100.0 |
nM |
PMID[502020] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.0 |
nM |
PMID[502020] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
21.0 |
nM |
PMID[502022] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.0 |
nM |
PMID[502024] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
144.0 |
nM |
PMID[502024] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
193.0 |
nM |
PMID[502027] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
15.0 |
nM |
PMID[502024] |
NPT518 |
Protein Complex |
Tubulin |
Homo sapiens |
IC50 |
= |
2100.0 |
nM |
PMID[502029] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
2.0 |
nM |
PMID[502029] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1.0 |
nM |
PMID[502029] |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Ki |
= |
18600.0 |
nM |
PMID[502030] |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Ki |
= |
10200.0 |
nM |
PMID[502030] |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
64.1 |
% |
PMID[502030] |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
IC50 |
= |
46800.0 |
nM |
PMID[502030] |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
IC50 |
= |
43500.0 |
nM |
PMID[502030] |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
81.5 |
% |
PMID[502030] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
6.0 |
nM |
PMID[502031] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
5000.0 |
nM |
PMID[502031] |
NPT782 |
Protein Family |
Tubulin |
Bos taurus |
IC50 |
= |
600.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
1.37 |
nM |
PMID[502032] |
NPT2588 |
Organism |
Paracentrotus lividus |
Paracentrotus lividus |
EC |
= |
2.0 |
uM |
PMID[502032] |
NPT2588 |
Organism |
Paracentrotus lividus |
Paracentrotus lividus |
EC |
= |
0.2 |
uM |
PMID[502032] |
NPT2588 |
Organism |
Paracentrotus lividus |
Paracentrotus lividus |
EC |
= |
0.1 |
uM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
0.3 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
TGI |
= |
1.6 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
LC50 |
= |
500.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
1.6 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
TGI |
= |
320.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
LC50 |
= |
2000.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
100.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
TGI |
= |
790.0 |
nM |
PMID[502032] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
LC50 |
= |
1580.0 |
nM |
PMID[502032] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
340.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
2.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
6.5 |
ucm/s |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
3.2 |
ucm/s |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
13.5 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
-4.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
7.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
-11.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
11.9 |
ucm/s |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
1.0 |
ucm/s |
PMID[502034] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Fabs |
= |
5.0 |
% |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
14.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
12.3 |
ucm/s |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Papp |
= |
0.9 |
ucm/s |
PMID[502034] |
NPT23140 |
TISSUE |
Intestine |
Mus musculus |
Ratio AUC |
= |
0.7 |
n.a. |
PMID[502034] |
NPT624 |
Tissue |
Plasma |
Mus musculus |
Ratio AUC |
= |
1.5 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
88.0 |
n.a. |
PMID[502034] |
NPT27 |
Others |
Unspecified |
|
Ratio |
= |
46.0 |
n.a. |
PMID[502034] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
200.0 |
nM |
PMID[502038] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3.0 |
nM |
PMID[502038] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
144.0 |
nM |
PMID[502038] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
IC50 |
= |
1100.0 |
nM |
PMID[502040] |
NPT3014 |
Protein Family |
Tubulin |
Sus scrofa |
Inhibition |
= |
73.93 |
% |
PMID[502041] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
6.0 |
nM |
PMID[502042] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
GI50 |
= |
5000.0 |
nM |
PMID[502042] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
55.5 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
42200.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
406.83 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
101.5 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
135.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
30330000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
102.17 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
636.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
732.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
2.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1570.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
442.5 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
10.83 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
126.8 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.67 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
144.0 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
1.5 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
60200.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
15.5 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BASO |
= |
0.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
21.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
10193.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
165.83 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
702.17 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BASOLE |
= |
0.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
0.17 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5390000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
34.62 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
138000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
11080.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
91.83 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
25.68 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
399000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
64.37 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
1.5 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
6.5 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
= |
0.0 |
/100WBC |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1202830.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
51.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
41200.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
392.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
81.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
161.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
30670000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
100.5 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
648.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
242.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1868.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
188.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
116.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.51 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
142.55 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
2.2 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
60800.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
18.5 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
17.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
11849.17 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
69.83 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
730.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5930000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
37.42 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
144000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
12670.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
93.17 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
24.32 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
385000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
63.08 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
0.5 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
6.17 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1170500.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
47.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
41000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
395.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
99.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
140.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
32330000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
103.33 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
673.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
526.33 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
1.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1350.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
170.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
10.33 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
119.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
6.35 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
144.8 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
1.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
56000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
11.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
42.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
6254.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
40.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
297.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
0.67 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
4480000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
28.87 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
116300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
6630.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
94.33 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
26.0 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
403300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
64.43 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
0.67 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
4.33 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
825330.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
44.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
39300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
340.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
88.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
166.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
28000000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
101.33 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
696.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
599.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
2120.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
334.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LIPASE |
= |
10.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
133.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.71 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
141.27 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
2.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PROT |
= |
58300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
17.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
0.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
7180.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
26.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
293.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
0.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5150000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
32.43 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
130000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
7500.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
95.67 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
25.27 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
400700.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
63.1 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONOLE |
= |
0.33 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
4.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
1437000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
129.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
40300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
429.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
337.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
150.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
31000000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
102.0 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
1040.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
645.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
1.6 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1673.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
246.33 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
116.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.31 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
144.2 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
4.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
10.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
5650.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
34.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
381.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
4960000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
31.5 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
126700.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
6070.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
93.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
25.5 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
402300.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
63.4 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
6.33 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
588330.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALT |
= |
423.33 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALB |
= |
36000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ALP |
= |
438.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
AST |
= |
923.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BUN |
= |
146.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CO2 |
= |
33000000.0 |
nM |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
= |
96.0 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CHOL |
= |
1923.3 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CK |
= |
622.67 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
CREAT |
= |
1.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
GLUC |
= |
1210.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LDH |
= |
415.0 |
U.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PHOS |
= |
106.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
= |
5.16 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
SODIUM |
= |
141.4 |
mEq.L-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
BILI |
= |
56.7 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
URATE |
= |
7.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOS |
= |
11.33 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYM |
= |
4520.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MONO |
= |
22.67 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
= |
46.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
EOSLE |
= |
0.33 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBC |
= |
5700000.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HCT |
= |
34.73 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
HGB |
= |
135000.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
WBC |
= |
4600.0 |
cells.uL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
LYMLE |
= |
98.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCH |
= |
23.7 |
pg |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCHC |
= |
388700.0 |
ug.mL-1 |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
MCV |
= |
61.03 |
fL |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
= |
1.0 |
% |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
= |
0.33 |
/100WBC |
PMID[502043] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PLAT |
= |
95670.0 |
cells.uL-1 |
PMID[502043] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Hit score |
= |
0.2235 |
n.a. |
PMID[502044] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
11.78 |
% |
PMID[502045] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
2.15 |
% |
PMID[502046] |