Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6 |
ug |
8709115 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.001 |
nM |
7131481 |
NPT3845 |
Cell Line |
LFCl2A |
|
IC50 |
= |
28500 |
nM |
10.1016/S0960-894X(01)81055-6 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
12877593 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
AC50 |
= |
6500 |
nM |
12877593 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
300 |
nM |
2967375 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3 |
ug/ml |
10.1016/S0960-894X(97)00365-X |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.32 |
ug/ml |
3373480 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
40 |
ug/ml |
3373480 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
3.8 |
ug/ml |
3373480 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
38 |
ug/ml |
3373480 |
NPT3846 |
Cell Line |
PC10 |
Homo sapiens |
IC50 |
> |
100 |
ug/ml |
3373480 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
3.3 |
ug/ml |
3373480 |
NPT3847 |
Cell Line |
TE-2 |
Homo sapiens |
IC50 |
= |
3.9 |
ug/ml |
3373480 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
6.1 |
ug/ml |
3373480 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6810 |
nM |
10072683 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
90500 |
nM |
10072683 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
37900 |
nM |
10072683 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
10072683 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
10072683 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
13100 |
nM |
10072683 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
41000 |
nM |
10072683 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
> |
100000 |
nM |
10072683 |
NPT3848 |
Cell Line |
9L |
Rattus norvegicus |
IC50 |
= |
1000 |
nM |
10072683 |
NPT793 |
Cell Line |
MOLT-3 |
Homo sapiens |
IC50 |
= |
1.2 |
ug/ml |
8648611 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
0.5 |
ug/ml |
8648611 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
4.3 |
ug/ml |
8648611 |
NPT2193 |
Cell Line |
IM-9 |
Homo sapiens |
IC50 |
= |
0.34 |
ug/ml |
8648611 |
NPT3849 |
Cell Line |
PHA-Ly |
Homo sapiens |
IC50 |
= |
1.4 |
ug/ml |
8648611 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.26 |
ug/ml |
11814824 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
11814824 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
11814824 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.63 |
ug/ml |
11814824 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
2500 |
nM |
11728193 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
1010 |
nM |
11728193 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
360 |
nM |
11728193 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
200 |
nM |
11728193 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
85000 |
nM |
10.1016/0960-894X(96)00418-0 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8000 |
nM |
10.1016/0960-894X(96)00418-0 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
0.09 |
|
10.1016/0960-894X(96)00418-0 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
11229742 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3500 |
nM |
11229742 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1600 |
nM |
11229742 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
68000 |
nM |
11229742 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
2500 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT3850 |
Cell Line |
KKLS |
|
IC50 |
= |
6200 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT3851 |
Cell Line |
AZ-521 cell line |
|
IC50 |
= |
3900 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
4400 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT3852 |
Cell Line |
COLO 320DM |
Homo sapiens |
IC50 |
= |
1100 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT3853 |
Cell Line |
SNU- |
|
IC50 |
= |
2700 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
IC50 |
> |
78000 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
22000 |
nM |
10.1016/0960-894X(96)00339-3 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Activity |
= |
44 |
|
6387121 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Activity |
= |
40 |
|
6387121 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Activity |
= |
30 |
|
6387121 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Activity |
= |
22 |
|
6387121 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
MIC |
= |
1 |
ug/ml |
6387121 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
MIC |
= |
4 |
ug/ml |
6387121 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
620 |
nM |
10229634 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2300 |
nM |
10229634 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
2200 |
nM |
11063625 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
630 |
nM |
11063625 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
220 |
nM |
11063625 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
125 |
nM |
11063625 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
79.8 |
% |
3918171 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
81.2 |
% |
3918171 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
90.3 |
% |
3918171 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
5000 |
nM |
7853342 |
NPT3857 |
Cell Line |
CHO-FU |
Cricetulus griseus |
IC50 |
= |
100000 |
nM |
7853342 |
NPT3845 |
Cell Line |
LFCl2A |
|
IC50 |
= |
28500 |
nM |
10.1016/S0960-894X(00)80263-2 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.208 |
ug/ml |
3007759 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.286 |
ug/ml |
3007759 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
ID50 |
= |
1.35 |
ug/ml |
3007759 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
ID50 |
= |
3.37 |
ug/ml |
3007759 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2000 |
nM |
10.1016/0960-894X(96)00451-9 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.32 |
ug/ml |
1992123 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
40 |
ug/ml |
1992123 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
3.8 |
ug/ml |
1992123 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
3.8 |
ug/ml |
1992123 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
3.5 |
ug/ml |
1992123 |
NPT3846 |
Cell Line |
PC10 |
Homo sapiens |
IC50 |
> |
100 |
ug/ml |
1992123 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
10 |
ug/ml |
1992123 |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
3.7 |
ug/ml |
1992123 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
3.3 |
ug/ml |
1992123 |
NPT3847 |
Cell Line |
TE-2 |
Homo sapiens |
IC50 |
= |
3.9 |
ug/ml |
1992123 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
6.1 |
ug/ml |
1992123 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
2.6 |
ug/ml |
1995905 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
40 |
ug/ml |
1995905 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
3.8 |
ug/ml |
1995905 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.3 |
ug/ml |
1995905 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
3.5 |
ug/ml |
1995905 |
NPT3846 |
Cell Line |
PC10 |
Homo sapiens |
IC50 |
> |
100 |
ug/ml |
1995905 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
10 |
ug/ml |
1995905 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
10.7 |
ug/ml |
1995905 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12.1 |
ug/ml |
1995905 |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
3.7 |
ug/ml |
1995905 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
3.3 |
ug/ml |
1995905 |
NPT3847 |
Cell Line |
TE-2 |
Homo sapiens |
IC50 |
= |
3.9 |
ug/ml |
1995905 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
6.1 |
ug/ml |
1995905 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2.1 |
ug/ml |
1995901 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.33 |
ug/ml |
1995901 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2.2 |
ug/ml |
1995901 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
1995901 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
0.07 |
ug/ml |
1995901 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
0.18 |
ug/ml |
1995901 |
NPT1307 |
Cell Line |
Calu-1 |
Homo sapiens |
IC50 |
> |
3.3 |
ug/ml |
1995901 |
NPT3860 |
Cell Line |
QG-90 |
Homo sapiens |
IC50 |
= |
0.22 |
ug/ml |
1995901 |
NPT3556 |
Cell Line |
PC-8 |
|
IC50 |
= |
0.42 |
ug/ml |
1995901 |
NPT3861 |
Cell Line |
KU-2 cell line |
|
IC50 |
= |
0.28 |
ug/ml |
1995901 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
1995901 |
NPT3862 |
Cell Line |
HT-137 |
|
IC50 |
= |
0.58 |
ug/ml |
1995901 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
IC50 |
= |
0.22 |
ug/ml |
1995901 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
0.79 |
ug/ml |
1995901 |
NPT3863 |
Cell Line |
G-292 |
Homo sapiens |
IC50 |
> |
3.3 |
ug/ml |
1995901 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
0.78 |
ug/ml |
1995901 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ID50 |
= |
6.1 |
nM |
3625714 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ID50 |
= |
0.8 |
nM |
3625714 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ID50 |
= |
13.8 |
nM |
3625714 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ID50 |
= |
0.002 |
nM |
3625714 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ID50 |
= |
0.3 |
nM |
3625714 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
= |
0.1 |
nM |
3625714 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.4 |
nM |
3625714 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ID50 |
= |
0.3 |
nM |
6827533 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
ID50 |
= |
0.0023 |
uM/ml |
7086837 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.00018 |
uM/ml |
7086837 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
500 |
nM |
7120290 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
5000 |
nM |
7120290 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
ID50 |
= |
0.0046 |
uM/ml |
7086837 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.001 |
uM/ml |
7086837 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.00023 |
uM/ml |
7086837 |
NPT3864 |
Cell Line |
MDAY-D2 |
Mus musculus |
ID50 |
= |
0.0002 |
uM/ml |
7086837 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
1.00E-06 |
nM |
7328578 |
NPT3865 |
Cell Line |
L1210/C |
Mus musculus |
IC50 |
= |
0.2 |
ug/ml |
10.1016/S0960-894X(01)80742-3 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
4 |
ug/ml |
10.1016/S0960-894X(01)80742-3 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
6 |
ug/ml |
10.1016/S0960-894X(01)80742-3 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
11 |
ug/ml |
10.1016/S0960-894X(01)80742-3 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
6 |
ug/ml |
10.1016/S0960-894X(01)80742-3 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
490 |
nM |
11052798 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
280 |
nM |
11052798 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
23000 |
nM |
11052798 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
8900 |
nM |
11052798 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
150 |
nM |
2547068 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
310 |
nM |
2547068 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2000 |
nM |
2362278 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
300 |
nM |
2362278 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
17 |
|
6447210 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
22 |
|
6447210 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
90 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
77 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
63.5 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
34.3 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
70 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
55 |
% |
2666666 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
19 |
% |
2666666 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
2200 |
nM |
7629806 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
630 |
nM |
7629806 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
220 |
nM |
7629806 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
120 |
nM |
7629806 |
NPT3869 |
Cell Line |
C170 |
|
IC50 |
= |
0.3 |
ug/ml |
8496926 |
NPT3869 |
Cell Line |
C170 |
|
IC50 |
= |
2000 |
nM |
8496926 |
NPT3870 |
Cell Line |
791T cell line |
|
IC50 |
= |
0.7 |
ug/ml |
8496926 |
NPT3870 |
Cell Line |
791T cell line |
|
IC50 |
= |
5500 |
nM |
8496926 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
0.5 |
ug/ml |
8496926 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
4100 |
nM |
8496926 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
0 |
% |
7365742 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Survival |
= |
9.66 |
day |
7365742 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.36 |
ug/ml |
10.1016/S0960-894X(01)81041-6 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.95 |
ug/ml |
10.1016/S0960-894X(01)81041-6 |
NPT3846 |
Cell Line |
PC10 |
Homo sapiens |
IC50 |
= |
42 |
ug/ml |
10.1016/S0960-894X(01)81041-6 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12.1 |
ug/ml |
10.1016/S0960-894X(01)81041-6 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.04 |
ug/ml |
11123990 |
NPT1759 |
Cell Line |
FM3A |
Mus musculus |
IC50 |
= |
0.02 |
ug/ml |
11123990 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
2.9 |
ug/ml |
11123990 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
1.2 |
ug/ml |
11123990 |
NPT1868 |
Cell Line |
L1210 (1565) |
|
ID50 |
< |
0.1 |
ug/ml |
8258836 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
ID50 |
< |
0.1 |
ug/ml |
8258836 |
NPT3871 |
Cell Line |
N592 |
|
IC50 |
= |
5400 |
nM |
8258835 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8400 |
nM |
8258835 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
28 |
% |
8277499 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
17 |
% |
8277499 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
9 |
% |
8277499 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
6 |
% |
8277499 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
1 |
% |
8277499 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4800 |
nM |
15658875 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9600 |
nM |
15658875 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
11900 |
nM |
15341952 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
15341952 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
4900 |
nM |
15341952 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6400 |
nM |
15341952 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3600 |
nM |
15341952 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
11900 |
nM |
15454213 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
15454213 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
4900 |
nM |
15454213 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6400 |
nM |
15454213 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3600 |
nM |
15454213 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
65300 |
nM |
15380199 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
50500 |
nM |
15380199 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
11900 |
nM |
16005217 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
16005217 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
4900 |
nM |
16005217 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6400 |
nM |
16005217 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3600 |
nM |
16005217 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
11900 |
nM |
15801848 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
15801848 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
4900 |
nM |
15801848 |
NPT3873 |
Cell Line |
Prostatic carcinoma cells |
Homo sapiens |
IC50 |
= |
6400 |
nM |
15801848 |
NPT3874 |
Cell Line |
TSU |
Homo sapiens |
IC50 |
= |
3600 |
nM |
15801848 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
40 |
% |
16275069 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
67 |
% |
16275069 |
NPT76 |
Cell Line |
C6 |
Rattus norvegicus |
IC50 |
= |
6100 |
nM |
16970409 |
NPT3875 |
Cell Line |
Astrocytes |
|
IC50 |
> |
100000 |
nM |
16970409 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37000 |
nM |
17253861 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
65 |
% |
16990003 |
NPT3876 |
Cell Line |
BEL-7404 tumor cell line |
|
Activity |
= |
29 |
% |
16997554 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
29 |
% |
16997554 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
25.2 |
ug |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
119.49 |
% |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
3.96 |
U/mg |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
20.4 |
U/mg |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
16.2 |
U/mg |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.97 |
U/mg |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.99 |
nmol |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.85 |
nmol |
17000104 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
3.65 |
nmol |
17000104 |
NPT820 |
Organism |
Clavispora lusitaniae |
Clavispora lusitaniae |
MIC |
<= |
0.5 |
ug/ml |
17060521 |
NPT820 |
Organism |
Clavispora lusitaniae |
Clavispora lusitaniae |
MIC |
>= |
512 |
ug/ml |
17060521 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
0.008 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
0.25 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
4 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
0.5 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
16 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
8 |
ug/ml |
17043122 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
= |
256 |
ug/ml |
17043122 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
160 |
nM |
17291040 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300000 |
nM |
17411027 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
300000 |
nM |
17411027 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
300000 |
nM |
17411027 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
3390 |
nM |
16996657 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2040 |
nM |
16996657 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
6610 |
nM |
16996657 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
7940 |
nM |
16996657 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
18600 |
nM |
16996657 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
5750 |
nM |
16996657 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
126000 |
nM |
16996657 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
IC50 |
= |
60300 |
nM |
16996657 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
13400 |
nM |
17000031 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
CC50 |
= |
3843800 |
nM |
17337193 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
CC50 |
= |
384400 |
nM |
17337193 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
46100 |
nM |
17337193 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
768800 |
nM |
17337193 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
17337193 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
31622.78 |
nM |
17446077 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
19952.62 |
nM |
17446077 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
17446077 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
17446077 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
3981.07 |
nM |
17446077 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
1995.26 |
nM |
17446077 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
316227.77 |
nM |
17446077 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
17446077 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
17446077 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
251188.64 |
nM |
17446077 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
1000 |
nM |
17446077 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
17446077 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
17446077 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
17446077 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
17446077 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
17446077 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
17446077 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17446077 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
17446077 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
17446077 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
17446077 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
1258.93 |
nM |
17446077 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
125892.54 |
nM |
17446077 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
199526.23 |
nM |
17446077 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
17446077 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
17446077 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
17446077 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
17446077 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
17446077 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
17446077 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
63095.73 |
nM |
17446077 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
17446077 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
17446077 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
17446077 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
17446077 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17446077 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17446077 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
3981.07 |
nM |
17446077 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
17446077 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
17446077 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
125892.54 |
nM |
17446077 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
17446077 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
17446077 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17446077 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
17446077 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
17446077 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
501187.23 |
nM |
17446077 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
251188.64 |
nM |
17446077 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
17446077 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
17446077 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9200 |
nM |
17604394 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
51000 |
nM |
17604394 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
370000 |
nM |
17604394 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
540000 |
nM |
17604394 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
200 |
nM |
17234303 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
100 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
73.68 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
65.79 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
42.11 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
37360 |
nM |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
60.71 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
32.14 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
17.86 |
% |
17239491 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
90550 |
nM |
17239491 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
17320246 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
17320246 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
600 |
nM |
17320246 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
17320246 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7300 |
nM |
17110105 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
2.30E-05 |
ug |
17174089 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
80.4 |
% |
17174089 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18600 |
nM |
17524655 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
128700 |
nM |
17524655 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14500 |
nM |
17524655 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
8100 |
nM |
17524655 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
17548198 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
300 |
nM |
17548198 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
17548198 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
3500 |
nM |
17548198 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
17553685 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
CC50 |
= |
3843800 |
nM |
17555969 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
CC50 |
= |
384400 |
nM |
17555969 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
230600 |
nM |
17555969 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
10 |
|
17555969 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
16.67 |
|
17555969 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
17555969 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
52500 |
nM |
17562365 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5750 |
nM |
17562365 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
20 |
% |
17950603 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
31 |
% |
17950603 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Inhibition |
= |
36 |
% |
17950603 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
25 |
% |
17950603 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Inhibition |
= |
41 |
% |
17950603 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
72.4 |
% |
17275295 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Activity |
= |
0.56 |
ug |
17275295 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
9600 |
nM |
17336074 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4800 |
nM |
17336074 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
42.8 |
% |
17428583 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
15.6 |
% |
17428583 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
5.87 |
/10^6mm3 |
17428583 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
83.6 |
10^6/100microL |
17428583 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
14.7 |
/10^3mm3 |
17428583 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
280 |
nM |
17931862 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23000 |
nM |
17931862 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
9000 |
nM |
17931862 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
CD100 |
> |
0.1 |
nM |
17950610 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4320 |
nM |
18194866 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
18205316 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.54 |
ug/ml |
18205316 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.7 |
ug/ml |
18205316 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.54 |
ug/ml |
18205316 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
0.65 |
ug/ml |
18205316 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
2.47 |
ug/ml |
1800632 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
5.64 |
ug/ml |
1800632 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
1.28 |
ug/ml |
1800632 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
3.72 |
ug/ml |
3443857 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.94 |
ug/ml |
3443857 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.5 |
nM |
11277741 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
0.008 |
nM |
11277741 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
ED50 |
= |
0.044 |
nM |
12027771 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.53 |
nM |
11325233 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
0.008 |
nM |
11325233 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
> |
10 |
ug/ml |
11374943 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
> |
10 |
ug/ml |
11374943 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
6.3 |
ug/ml |
11374943 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.015 |
ug/ml |
11374950 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
0.48 |
ug/ml |
11374950 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
EC50 |
= |
0.29 |
ug/ml |
12444707 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
0.07 |
ug/ml |
12444707 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.53 |
nM |
11430002 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
0.008 |
nM |
11430002 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.075 |
ug/ml |
12502333 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.08 |
ug/ml |
1812210 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
11575942 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
11575942 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
11575942 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26800 |
nM |
18271558 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
47 |
% |
18271558 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
18700 |
nM |
18302336 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
CC50 |
= |
3843800 |
nM |
17548129 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
CC50 |
= |
384400 |
nM |
17548129 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
768800 |
nM |
17548129 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
46100 |
nM |
17548129 |
NPT2891 |
Cell Line |
H4 |
Homo sapiens |
Ratio |
= |
10 |
|
17548129 |
NPT2891 |
Cell Line |
H4 |
Homo sapiens |
Ratio |
= |
83.4 |
|
17548129 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
5 |
|
17548129 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
17548129 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
CC50 |
= |
3843800 |
nM |
18037195 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
CC50 |
= |
384400 |
nM |
18037195 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
46100 |
nM |
18037195 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
768800 |
nM |
18037195 |
NPT2891 |
Cell Line |
H4 |
Homo sapiens |
CC50 |
= |
10000 |
nM |
18037195 |
NPT2891 |
Cell Line |
H4 |
Homo sapiens |
CC50 |
= |
83400 |
nM |
18037195 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
CC50 |
= |
5000 |
nM |
18037195 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
18037195 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
40 |
% |
19201604 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
25 |
% |
19201604 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
44 |
% |
19201604 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
GI |
= |
56 |
% |
19201604 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
4300 |
nM |
19233650 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
19233650 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
LC50 |
= |
0.2 |
ug/ml |
8594149 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.41 |
ug/ml |
1800632 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
2.14 |
ug/ml |
1800632 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
1.25 |
ug/ml |
1800632 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
ED50 |
= |
3.09 |
ug/ml |
1800632 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Activity |
= |
32.9 |
% |
12662110 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
7.15 |
ug/ml |
11908984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
ED50 |
= |
3.3 |
ug/ml |
11908984 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
ED50 |
= |
0.48 |
ug/ml |
11908984 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
7.4 |
ug/ml |
11908984 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.4 |
ug/ml |
16309328 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.6 |
ug/ml |
16309328 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
16309328 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
16309328 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
18424155 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
6500 |
nM |
18424155 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
8700 |
nM |
18424155 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
9200 |
nM |
18424155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
460 |
nM |
18440233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5780 |
nM |
18440233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2590 |
nM |
18440233 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9190 |
nM |
18440233 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
770 |
nM |
18440233 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
9450 |
nM |
18440233 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16000 |
nM |
18424155 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
9230 |
nM |
18424155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20000 |
nM |
18424155 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
690 |
nM |
18424155 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
57 |
% |
18707881 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI |
= |
37 |
% |
18707881 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
30 |
% |
18707881 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
27 |
% |
18707881 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI |
= |
29 |
% |
18707881 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI |
= |
46 |
% |
18707881 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
29 |
% |
18707881 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
77 |
% |
18707881 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
11 |
% |
18707881 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
Inhibition |
= |
0.9 |
% |
18788725 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
16700 |
nM |
18798609 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
14600 |
nM |
18798609 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
8900 |
nM |
18798609 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
22400 |
nM |
18798609 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6500 |
nM |
18798609 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
15400 |
nM |
18798609 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
4100 |
nM |
18798609 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
GI50 |
< |
1540 |
nM |
18798609 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
23.8 |
% |
18951805 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
> |
100000 |
nM |
19324555 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
65300 |
nM |
19324555 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
50500 |
nM |
19324555 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
19324555 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
7380 |
nM |
15387639 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4930 |
nM |
15387639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5400 |
nM |
15387656 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
3700 |
nM |
14640513 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5400 |
nM |
15568771 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
690 |
nM |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
609 |
nM |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
> |
40 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
15 |
mm |
2778449 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
0 |
Zone units |
2809606 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
Activity |
= |
800 |
Zone units |
2809606 |
NPT693 |
Organism |
Xenopus laevis |
Xenopus laevis |
GI |
= |
47 |
% |
12762796 |
NPT826 |
Organism |
Magnaporthe oryzae |
Magnaporthe oryzae |
Activity |
<= |
5 |
ug/ml |
12932123 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
3800 |
nM |
18491866 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
TGI |
= |
95 |
% |
18508273 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
Activity |
= |
-7 |
% |
18508273 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
63.8 |
% |
18539036 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4320 |
nM |
18069093 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4000 |
nM |
18640746 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
18640746 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
18640746 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
18640746 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
18640746 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
400 |
nM |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
10 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
12 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
26 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
60 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
59 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
57 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
39 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
41 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
43 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
1 |
% |
18640746 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
0 |
% |
18640746 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
1230 |
nM |
12027739 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
EC50 |
= |
1380 |
nM |
12027739 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
3610 |
nM |
12027739 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
230 |
nM |
12027739 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
310 |
nM |
12027739 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.93 |
ug/ml |
10425135 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
0.073 |
ug/ml |
17067147 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.44 |
ug/ml |
10425135 |
NPT2914 |
Organism |
Xanthomonas oryzae |
Xanthomonas oryzae |
Activity |
= |
4 |
ug/ml |
17067169 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.02 |
ug/ml |
10579858 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
10579858 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
10579858 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.1 |
ug/ml |
10579858 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.0012 |
ug/ml |
16038565 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.072 |
ug/ml |
16038565 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC60 |
= |
7.4 |
ug/ml |
16038565 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
0.008 |
nM |
11141109 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
16499317 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
16499317 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
16499317 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
4200 |
nM |
16499317 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
4200 |
nM |
16499317 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1.3 |
ug/ml |
16499328 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI50 |
= |
0.073 |
ug/ml |
16562827 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
18606546 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
18606546 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
18606546 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
600 |
nM |
18606546 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16350 |
nM |
18644718 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
13160 |
nM |
18644718 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
21380 |
nM |
18644718 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
14410 |
nM |
18644718 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10850 |
nM |
18644718 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
8730 |
nM |
18644718 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
73.5 |
% |
18644718 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
53200 |
nM |
19463000 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
5710 |
nM |
19463000 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
4.46 |
nM |
19345581 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
17700 |
nM |
19398334 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
18950904 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
TGI |
> |
100000 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15090 |
nM |
18950904 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
GI50 |
> |
100000 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8370 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72070 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
18950904 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
18950904 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
19338315 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.2 |
ug/ml |
19338315 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
19338315 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
19338315 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
19338315 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
GI50 |
> |
10000 |
nM |
19406645 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
> |
10000 |
nM |
19406645 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19743863 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1100 |
nM |
19743863 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
600 |
nM |
19743863 |
NPT2064 |
Cell Line |
UACC-812 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
19743863 |
NPT2186 |
Cell Line |
RL |
Homo sapiens |
IC50 |
= |
3200 |
nM |
19743863 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
125000 |
nM |
19743863 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2600 |
nM |
19743863 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
4400 |
nM |
19743863 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
19743863 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20800 |
nM |
19422203 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
CD100 |
> |
0.1 |
nM |
19572611 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
10000 |
nM |
19572613 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
15000 |
nM |
19572613 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
16 |
nM |
19423198 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
18 |
nM |
19423198 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2 |
ug/ml |
19700322 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
9772.37 |
nM |
19740574 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
2290.87 |
nM |
19740574 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
19740574 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
354.81 |
nM |
19740574 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
44.67 |
nM |
19740574 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
23.99 |
nM |
19740574 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
190.55 |
nM |
19740574 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
61659.5 |
nM |
19740574 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
19740574 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
77624.71 |
nM |
19740574 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
54954.09 |
nM |
19740574 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
19740574 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
56.23 |
nM |
19740574 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
7244.36 |
nM |
19740574 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
331.13 |
nM |
19740574 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
158.49 |
nM |
19740574 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
52.48 |
nM |
19740574 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
19740574 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
109.65 |
nM |
19740574 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
19740574 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
213.8 |
nM |
19740574 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
933.25 |
nM |
19740574 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
19740574 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
19740574 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
63.1 |
nM |
19740574 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
3801.89 |
nM |
19740574 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
19740574 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
912.01 |
nM |
19740574 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
245.47 |
nM |
19740574 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
51.29 |
nM |
19740574 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
977.24 |
nM |
19740574 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
56234.13 |
nM |
19740574 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
1023.29 |
nM |
19740574 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
467.74 |
nM |
19740574 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
19740574 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
524.81 |
nM |
19740574 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
1230.27 |
nM |
19740574 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
15.85 |
nM |
19740574 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
4466.84 |
nM |
19740574 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
10964.78 |
nM |
19740574 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
1737.8 |
nM |
19740574 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
21877.62 |
nM |
19740574 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
724.44 |
nM |
19740574 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
19740574 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
295.12 |
nM |
19740574 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
72.44 |
nM |
19740574 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
2630.27 |
nM |
19740574 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
501.19 |
nM |
19740574 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
1122.02 |
nM |
19740574 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
1412.54 |
nM |
19740574 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
2344.23 |
nM |
19740574 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
363.08 |
nM |
19740574 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
79.43 |
nM |
19740574 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
316.23 |
nM |
19740574 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
6606.93 |
nM |
19740574 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
9772.37 |
nM |
19740574 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
72.44 |
nM |
19740574 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
10715.19 |
nM |
19740574 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
8128.31 |
nM |
19740574 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.67 |
ug/ml |
19932530 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1.01 |
ug/ml |
19932530 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
12 |
% |
19939522 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
20 |
% |
19939522 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
21000 |
nM |
19939522 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI |
= |
26 |
% |
19939522 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
0 |
% |
19926172 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
29 |
% |
19926172 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
25 |
% |
19926172 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
40 |
% |
19926172 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
29 |
% |
19926172 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
0 |
% |
19926172 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
58 |
% |
19926172 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12500 |
nM |
19846302 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
58 |
uL |
19527933 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
10 |
g/dl |
19527933 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
42.3 |
% |
19527933 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
13.8 |
|
19527933 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4300 |
nM |
19560842 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
19560842 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
GI50 |
= |
50000 |
nM |
19664930 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
29000 |
nM |
19664930 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
19000 |
nM |
19664930 |
NPT1723 |
Cell Line |
HBL-100 |
Homo sapiens |
GI50 |
= |
5500 |
nM |
19664930 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
4400 |
nM |
19664930 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
GI50 |
= |
4100 |
nM |
19664930 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
49 |
% |
19913412 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
54 |
% |
19913412 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
64200 |
nM |
20171096 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
67200 |
nM |
20171096 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
78000 |
nM |
20151671 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
5200 |
nM |
19919052 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10000 |
nM |
19919065 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
19919065 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
Inhibition |
= |
64.2 |
% |
19879023 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
45.4 |
% |
19879023 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Inhibition |
= |
73.7 |
% |
19879023 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
Inhibition |
= |
71.3 |
% |
19879023 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
65.1 |
% |
19879023 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
Inhibition |
= |
70.5 |
% |
19879023 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
19795843 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10000 |
nM |
19795843 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10000 |
nM |
19618920 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
19618920 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
8580 |
nM |
19689125 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5910 |
nM |
19689125 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
440 |
nM |
19689125 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
410 |
nM |
19689125 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7390 |
nM |
19689125 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
/ml |
19447526 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
23 |
% |
19447526 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.4 |
/10'3mm'-3 |
19447526 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
40.86 |
% |
19447526 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
10.73 |
% |
19447526 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
GI50 |
< |
3000 |
nM |
20356752 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
2300 |
nM |
20356752 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
5300 |
nM |
20356752 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
4500 |
nM |
20356752 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
32400 |
nM |
20356752 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
14900 |
nM |
20356752 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
89900 |
nM |
20356752 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
20350811 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
20350811 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
30 |
nM |
20211564 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
20211564 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
20211564 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
20211564 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
20211564 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
27.5 |
ug |
20353152 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
80.7 |
% |
20353152 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3030 |
nM |
20163895 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
54000 |
nM |
20438092 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
6200 |
nM |
20438092 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
8300 |
nM |
20438092 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10000 |
nM |
20405881 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
47000 |
nM |
20438092 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
GI50 |
= |
3000 |
nM |
20438092 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
20403701 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
20403701 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15200 |
nM |
20403701 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3500 |
nM |
20403701 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
CC50 |
= |
70 |
nM |
20227144 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
4460 |
nM |
20356655 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
52430 |
nM |
20409617 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
100000 |
nM |
20409617 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
43730 |
nM |
20409617 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
79790 |
nM |
20409617 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
48500 |
nM |
20398972 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
7.38 |
ug/ml |
20538457 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1930 |
nM |
20494492 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
2950 |
nM |
20494492 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2190 |
nM |
20494492 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45400 |
nM |
20494492 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9700 |
nM |
20494492 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
87960 |
nM |
18469809 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
18469809 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
> |
100000 |
nM |
18469809 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
26260 |
nM |
18469809 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
11630 |
nM |
18469809 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28910 |
nM |
18469809 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
87730 |
nM |
18469809 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38670 |
nM |
18469809 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
96370 |
nM |
18469809 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
26670 |
nM |
18469809 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6360 |
nM |
18469809 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
18240 |
nM |
18469809 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
50090 |
nM |
18469809 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
13180 |
nM |
18469809 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7210 |
nM |
18469809 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
13770 |
nM |
18469809 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
IC50 |
= |
14670 |
nM |
18469809 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT2 |
Others |
Unspecified |
|
Activity |
< |
3 |
% |
18469809 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
10 |
% |
18469809 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
Activity |
< |
3 |
% |
18469809 |
NPT742 |
Organism |
Influenza A virus |
Influenza A virus |
EC50 |
= |
26 |
ug/ml |
20674371 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
23 |
ug/ml |
20674371 |
NPT616 |
Cell Line |
MDCK |
Canis lupus familiaris |
IC50 |
> |
100 |
ug/ml |
20674371 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
57.6 |
% |
20729093 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
41.7 |
% |
20729093 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
46.1 |
% |
20729093 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3981.07 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
15848.93 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
7943.28 |
nM |
19734910 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
7.38 |
ug/ml |
20800480 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2.48 |
ug/ml |
20800480 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
2.17 |
ug/ml |
20800480 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
16000 |
nM |
20873740 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
43000 |
nM |
20873740 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
30000 |
nM |
20873740 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
IC50 |
= |
30000 |
nM |
20873740 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
64000 |
nM |
20873740 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
87000 |
nM |
20873740 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
48000 |
nM |
20873740 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
20873740 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
20873740 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
20873740 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
90000 |
nM |
20873740 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
57000 |
nM |
20873740 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
> |
100000 |
nM |
20873740 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50000 |
nM |
20873740 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
20873740 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
20873740 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
7.36 |
ug/ml |
20947362 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
3.3 |
% |
20943401 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
41.6 |
% |
20943401 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
9772.37 |
nM |
20850204 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
2290.87 |
nM |
20850204 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
20850204 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
354.81 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
44.67 |
nM |
20850204 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
23.99 |
nM |
20850204 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
190.55 |
nM |
20850204 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
61659.5 |
nM |
20850204 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
20850204 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
77624.71 |
nM |
20850204 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
54954.09 |
nM |
20850204 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
20850204 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
56.23 |
nM |
20850204 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
7244.36 |
nM |
20850204 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
331.13 |
nM |
20850204 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
158.49 |
nM |
20850204 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
52.48 |
nM |
20850204 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
20850204 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
109.65 |
nM |
20850204 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
20850204 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
213.8 |
nM |
20850204 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
933.25 |
nM |
20850204 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
20850204 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
20850204 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
63.1 |
nM |
20850204 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
3801.89 |
nM |
20850204 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
20850204 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
912.01 |
nM |
20850204 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
245.47 |
nM |
20850204 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
51.29 |
nM |
20850204 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
977.24 |
nM |
20850204 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
56234.13 |
nM |
20850204 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
1023.29 |
nM |
20850204 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
467.74 |
nM |
20850204 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
20850204 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
524.81 |
nM |
20850204 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
1230.27 |
nM |
20850204 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
15.85 |
nM |
20850204 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
4466.84 |
nM |
20850204 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
10964.78 |
nM |
20850204 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
1737.8 |
nM |
20850204 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
21877.62 |
nM |
20850204 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
724.44 |
nM |
20850204 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
20850204 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
295.12 |
nM |
20850204 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
72.44 |
nM |
20850204 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
2630.27 |
nM |
20850204 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
501.19 |
nM |
20850204 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
1122.02 |
nM |
20850204 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
1412.54 |
nM |
20850204 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
2344.23 |
nM |
20850204 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
363.08 |
nM |
20850204 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
79.43 |
nM |
20850204 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
316.23 |
nM |
20850204 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
6606.93 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
9772.37 |
nM |
20850204 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
72.44 |
nM |
20850204 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
10715.19 |
nM |
20850204 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
8128.31 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
562.34 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1995.26 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
186.21 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1348.96 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
933.25 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1819.7 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
575.44 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
912.01 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1380.38 |
nM |
20850204 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4600 |
nM |
21074444 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
3600 |
nM |
21074444 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
21074444 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
18000 |
nM |
21074444 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
21074444 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
4800 |
nM |
21074444 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
21074444 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
125.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
14125.4 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
1258.9 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
11.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
4466.8 |
nM |
PubChem BioAssay data set |
NPT1197 |
Individual Protein |
Huntingtin |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
1258.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3981.1 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
1584.9 |
nM |
PubChem BioAssay data set |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Potency |
= |
2909.3 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
631 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
794.3 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
7943.3 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
5623.4 |
nM |
PubChem BioAssay data set |
NPT794 |
Individual Protein |
Endonuclease 4 |
Escherichia coli K-12 |
Potency |
= |
8912.5 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20470 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
37650.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4170 |
nM |
PubChem BioAssay data set |
NPT796 |
Individual Protein |
Peripheral myelin protein 22 |
Homo sapiens |
Potency |
= |
4775.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
4250 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
158.5 |
nM |
PubChem BioAssay data set |
NPT54 |
Individual Protein |
Nonstructural protein 1 |
Influenza A virus |
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT54 |
Individual Protein |
Nonstructural protein 1 |
Influenza A virus |
Potency |
= |
1000 |
nM |
PubChem BioAssay data set |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Potency |
= |
23280.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
7079.5 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9780 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2530 |
nM |
PubChem BioAssay data set |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
Potency |
= |
1258.9 |
nM |
PubChem BioAssay data set |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
12.6 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2990 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
6240 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
378 |
nM |
PubChem BioAssay data set |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
51.2 |
% |
20970893 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
7.2 |
ug/ml |
20961091 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
34 |
ug/ml |
20961091 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14.1 |
ug/ml |
21109433 |
NPT2580 |
Organism |
Candida dubliniensis |
Candida dubliniensis |
MIC |
= |
32 |
ug/ml |
19704126 |
NPT2580 |
Organism |
Candida dubliniensis |
Candida dubliniensis |
MIC |
= |
16 |
ug/ml |
19704126 |
NPT2580 |
Organism |
Candida dubliniensis |
Candida dubliniensis |
MIC |
= |
8 |
ug/ml |
19704126 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
8.6 |
ug/ml |
21130542 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6.5 |
ug/ml |
21130542 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.3 |
ug/ml |
21130542 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
99.5 |
% |
21130542 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
38000 |
nM |
21131104 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2160 |
nM |
21131104 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2780 |
nM |
21131104 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11900 |
nM |
21144621 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13100 |
nM |
21144621 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
12600 |
nM |
21144621 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15200 |
nM |
21144621 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
25 |
ug/ml |
21115211 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
35.39 |
% |
21126804 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
25.63 |
% |
21126804 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
38.98 |
% |
21126804 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6.06 |
% |
21126804 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
8.06 |
% |
21126804 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
87.4 |
% |
21126804 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4320 |
nM |
21126804 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
15900 |
nM |
21273072 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
560 |
nM |
21232828 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
570 |
nM |
21232828 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
14000 |
nM |
21232828 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9600 |
nM |
21295381 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
21295381 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
120000 |
nM |
21226488 |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
3262.9 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
2592.9 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
11582.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
12995.3 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
28183.8 |
nM |
PubChem BioAssay data set |
NPT62 |
Individual Protein |
6-phospho-1-fructokinase |
Trypanosoma brucei |
Potency |
|
8492.1 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
22.4 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
9285 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
10417.9 |
nM |
PubChem BioAssay data set |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
560 |
nM |
21330014 |
NPT1759 |
Cell Line |
FM3A |
Mus musculus |
IC50 |
= |
180 |
nM |
21330014 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
14000 |
nM |
21330014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
450 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
21000 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
1300 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
620 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
470 |
nM |
21330014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
21330014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
180 |
nM |
21330014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1100 |
nM |
21330014 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
> |
500000 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
970 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
51000 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
370 |
nM |
21330014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
4900 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
= |
7000 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
= |
220 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
= |
20 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
>= |
10000 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
= |
600 |
nM |
21330014 |
NPT3791 |
Individual Protein |
Thymidylate synthase |
Mus musculus |
IC50 |
= |
60 |
nM |
21330014 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
9500 |
nM |
21250700 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
11300 |
nM |
21250700 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21250700 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21250700 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21250700 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
21250700 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
IC50 |
= |
54100 |
nM |
21250700 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20300 |
nM |
21486694 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
41460 |
nM |
21486694 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
29300 |
nM |
21486694 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26920 |
nM |
21486694 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7540 |
nM |
21486694 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
31460 |
nM |
21486698 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
18850 |
nM |
21486698 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
15690 |
nM |
21486698 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.5 |
ug/ml |
21353349 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
31 |
% |
21482109 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
9100 |
nM |
21381696 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
21381696 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
20000 |
nM |
21381696 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
21381696 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
4170 |
nM |
21449610 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
21449610 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8510 |
nM |
21449610 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
9710 |
nM |
21449610 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10200 |
nM |
21449610 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
8320 |
nM |
21449610 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21449610 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
33100 |
nM |
21449610 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21449610 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
21449610 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
2300 |
nM |
21489802 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2800 |
nM |
21489802 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
5200 |
nM |
21489802 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
3100 |
nM |
21489802 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
6100 |
nM |
21489802 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
2800 |
nM |
21489802 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
2400 |
nM |
21489802 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
4100 |
nM |
21489802 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
12000 |
nM |
21489802 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
6300 |
nM |
21489802 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
3500 |
nM |
21489802 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16100 |
nM |
21515044 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5600 |
nM |
21515044 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14100 |
nM |
21515044 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
15000 |
nM |
21439690 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
8000 |
nM |
21439690 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
40000 |
nM |
21439690 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
30000 |
nM |
21439690 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
0 |
% |
21531049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
7 |
% |
21531049 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
21612935 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4000 |
nM |
21612935 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
21612935 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.0017 |
nM |
21640594 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.0027 |
nM |
21640594 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.0011 |
nM |
21640594 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.0077 |
nM |
21640594 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
21458113 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
7400 |
nM |
21458113 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
21458113 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8700 |
nM |
21458113 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
13000 |
nM |
21495659 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
13700 |
nM |
21495659 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
21800 |
nM |
21495659 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
34.7 |
% |
21620530 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Activity |
= |
1.11 |
ug |
21620530 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
46.5 |
% |
21620530 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
832.28 |
ug |
21620534 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
51.28 |
% |
21620534 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
18500 |
nM |
21524829 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
11450 |
nM |
21524829 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
3380 |
nM |
21524829 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
38250 |
nM |
21524829 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21524829 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
42010 |
nM |
21524829 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10310 |
nM |
21524829 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11000 |
nM |
21530016 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
21530016 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
21530016 |
NPT769 |
Organism |
Mucor mucedo |
Mucor mucedo |
Inhibition |
= |
75 |
% |
21885289 |
NPT769 |
Organism |
Mucor mucedo |
Mucor mucedo |
Inhibition |
= |
61 |
% |
21885289 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
42.86 |
% |
21705114 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
15.6 |
% |
21705114 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
5.87 |
% |
21705114 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
14.7 |
% |
21705114 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.9 |
% |
21705114 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3300 |
nM |
21774474 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
109000 |
nM |
21774474 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
31000 |
nM |
21774474 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
8500 |
nM |
21774474 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
59000 |
nM |
21774474 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
121000 |
nM |
21774474 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
52000 |
nM |
21774474 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4320 |
nM |
21684047 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
IC50 |
= |
730 |
nM |
21684047 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1080 |
nM |
21684047 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
660 |
nM |
21684047 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
0.17 |
|
21684047 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Ratio IC50 |
= |
0.61 |
|
21684047 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21689869 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
> |
100000 |
nM |
21689869 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
23.31 |
ug/ml |
21889345 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
31.02 |
ug/ml |
21889345 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
28.52 |
ug/ml |
21889345 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
EC50 |
= |
17.37 |
ug/ml |
21889345 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12500 |
nM |
21843939 |
NPT478 |
Individual Protein |
Ataxin-2 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT108 |
Individual Protein |
Estrogen receptor alpha |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
4653.5 |
nM |
PubChem BioAssay data set |
NPT135 |
Individual Protein |
Chromobox protein homolog 1 |
Homo sapiens |
Potency |
|
100000 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
4256.2 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT249 |
Individual Protein |
Glucocorticoid receptor |
Homo sapiens |
Potency |
|
22.4 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
446.7 |
nM |
PubChem BioAssay data set |
NPT803 |
Individual Protein |
Flap endonuclease 1 |
Homo sapiens |
Potency |
|
150 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14.1 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
6573.3 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
6745.6 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
1299.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14125.4 |
nM |
PubChem BioAssay data set |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
490 |
nM |
21917363 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
21917363 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
21917363 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
420 |
nM |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
22000925 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6150 |
nM |
22000925 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
72900 |
nM |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
38.68 |
% |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
35.12 |
% |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
21.51 |
% |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
20.6 |
% |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
39.81 |
% |
22000925 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
44.28 |
% |
22000925 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Activity |
= |
50 |
% |
21644529 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
110010 |
nM |
21962523 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
110160 |
nM |
21962523 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
95170 |
nM |
21962523 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
100020 |
nM |
21962523 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
85500 |
nM |
22093761 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
76000 |
nM |
22093761 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
76700 |
nM |
22093761 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
22056277 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
42900 |
nM |
22093761 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
22119151 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
GI50 |
> |
100000 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
22119151 |
NPT3880 |
Cell Line |
Melanoma cells |
Homo sapiens |
GI50 |
= |
70600 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
22056277 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
GI50 |
> |
100000 |
nM |
22056277 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22056277 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
TGI |
> |
100000 |
nM |
22056277 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
22119151 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
TGI |
> |
100000 |
nM |
22119151 |
NPT3880 |
Cell Line |
Melanoma cells |
Homo sapiens |
TGI |
> |
100000 |
nM |
22119151 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
22119151 |
NPT3877 |
Cell Line |
NSCLC |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22119151 |
NPT3880 |
Cell Line |
Melanoma cells |
Homo sapiens |
LC50 |
> |
100000 |
nM |
22119151 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
70 |
% |
22071256 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
GI |
= |
68 |
% |
22071256 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI |
= |
22 |
% |
22047801 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
21 |
% |
22047801 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
44 |
% |
22047801 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
76 |
% |
22047801 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI |
= |
44 |
% |
22047801 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
GI |
= |
7 |
% |
22047801 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
71 |
% |
22047801 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
9850 |
nM |
22079378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17200 |
nM |
22079378 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
16600 |
nM |
22079378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15500 |
nM |
22079378 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
> |
50000 |
nM |
22079378 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9670 |
nM |
22079378 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
9000 |
nM |
22200404 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13500 |
nM |
22200404 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
8.6 |
ug/ml |
22204901 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
3.2 |
ug/ml |
22204901 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6.5 |
ug/ml |
22204901 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.3 |
ug/ml |
22204901 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.32 |
ug/ml |
22011319 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
22011319 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.22 |
ug/ml |
22011319 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.0082 |
ug/ml |
22011319 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
0.023 |
ug/ml |
22011319 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
0.36 |
ug/ml |
22011319 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
41 |
% |
22123322 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
44 |
% |
22123322 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
29 |
% |
22123322 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
29 |
% |
22123322 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
35 |
% |
22123322 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
16 |
% |
22123322 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.67 |
ug/ml |
22154835 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6 |
ug/ml |
22154835 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5640 |
nM |
22182926 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14300 |
nM |
22182926 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16320 |
nM |
22182926 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
15710 |
nM |
22182926 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
76 |
% |
22245048 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
75 |
% |
22245048 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI |
= |
75 |
% |
22245048 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
79 |
% |
22245048 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI |
= |
71 |
% |
22245048 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
85 |
% |
22245048 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
23.8 |
nM |
22305543 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
7280 |
nM |
22305543 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
68300 |
nM |
22244588 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
54800 |
nM |
22244588 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
82200 |
nM |
22244588 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
218000 |
nM |
22244588 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
75 |
% |
22245048 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
63 |
% |
22245048 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
22130132 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
22130132 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
22130132 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7900 |
nM |
22381354 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
266000 |
nM |
22424614 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
22424614 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
22424614 |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
8072.35 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
24945.95 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
9616.12 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
12161.86 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
5636.38 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
20892.96 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
161808 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
9289.66 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
1333.52 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
11587.77 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
22490.55 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
21183.61 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
10185.91 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
13963.68 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
27289.78 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
21827.3 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
41304.75 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
20183.66 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
44258.84 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
172186.86 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
5619.2 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
115611.22 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
488652.36 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
4355.12 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
136144.47 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
27669.42 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
9506.05 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
36982.82 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
46451.53 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
14381.8 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
22542.39 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
4909.08 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
69662.65 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
6025.6 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
109900.58 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
372391.71 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
1595.88 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
2113.49 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
181134.01 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
4083.19 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
5688.53 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
298538.26 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
51404.37 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
50582.47 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
1753.88 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
170608.24 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
1051.96 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
75509.22 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
13931.57 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
4446.31 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
10592.54 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
14321.88 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
51880 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
11912.42 |
nM |
PubChem BioAssay data set |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
|
224905.46 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
95719.41 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
35156.04 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
6714.29 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
250034.54 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
50234.26 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
6839.12 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
54075.43 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
LC50 |
= |
25000 |
nM |
22381050 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
33000 |
nM |
22304344 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
34000 |
nM |
22304344 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
45000 |
nM |
22304344 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
43000 |
nM |
22304344 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
29000 |
nM |
22304344 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
35000 |
nM |
22304344 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
490 |
nM |
22405290 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
22405290 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
22405290 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
22405290 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
22405290 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
22405290 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
300 |
nM |
22405290 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
7110 |
nM |
22405648 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3420 |
nM |
22405648 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
5330 |
nM |
22405648 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
4170 |
nM |
22409967 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
22409967 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8510 |
nM |
22409967 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
9710 |
nM |
22409967 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10200 |
nM |
22409967 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
8320 |
nM |
22409967 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
380000 |
nM |
22409967 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
> |
2512000 |
nM |
22409967 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
22409967 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
108000 |
nM |
22283451 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
108000 |
nM |
22283451 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
31000 |
nM |
22283451 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
62000 |
nM |
22283451 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
22283451 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
22283451 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
123000 |
nM |
22283451 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
65 |
% |
22472045 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
74 |
% |
22472045 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
35050 |
nM |
22483608 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
31720 |
nM |
22483608 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46310 |
nM |
22483608 |
NPT3377 |
Cell Line |
PC-9 |
|
IC50 |
= |
23470 |
nM |
22483608 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
46550 |
nM |
22483608 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
9900 |
nM |
22512908 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
21000 |
nM |
22512908 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
9370 |
nM |
22512908 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
21000 |
nM |
22512908 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
9900 |
nM |
22512908 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
9100 |
nM |
22512908 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
20000 |
nM |
22512908 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
76000 |
nM |
22512908 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
82000 |
nM |
22512908 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
6500 |
nM |
22512908 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
22512908 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
22512908 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100000 |
nM |
22512908 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
100000 |
nM |
22512908 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
100000 |
nM |
22512908 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
22450132 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
9600 |
nM |
22450132 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7300 |
nM |
22450132 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
22512908 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
GI50 |
= |
30000 |
nM |
22512908 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
GI50 |
= |
8200 |
nM |
22512908 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
GI50 |
= |
6300 |
nM |
22512908 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
9720 |
nM |
22512908 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
LC50 |
= |
100000 |
nM |
22512908 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
TGI |
= |
100000 |
nM |
22512908 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8920 |
nM |
22512908 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
86060 |
nM |
22512908 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
Inhibition |
= |
3.25 |
% |
22512908 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
Activity |
= |
700 |
% |
22512908 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
22537362 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
22537362 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
6800 |
nM |
22537362 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
33400 |
nM |
22537362 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
22537362 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
22537362 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
46570 |
nM |
22579780 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5640 |
nM |
22579780 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16320 |
nM |
22579780 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14300 |
nM |
22579780 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
15710 |
nM |
22579780 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
6040 |
nM |
22579780 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
13650 |
nM |
22579780 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
24660 |
nM |
22555152 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
11670 |
nM |
22555152 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
6680 |
nM |
22555152 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
56200 |
nM |
22555152 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
66910 |
nM |
22555152 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
14930 |
nM |
22555152 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
81.3 |
% |
22727445 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
GI |
= |
80.8 |
% |
22727445 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
GI |
= |
85.7 |
% |
22727445 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
89.7 |
% |
22727445 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
80.4 |
% |
22727445 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4800 |
nM |
22727445 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
6300 |
nM |
22727445 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
22727445 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46830 |
nM |
22809558 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
35410 |
nM |
22809558 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22630 |
nM |
22809558 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
41730 |
nM |
22809558 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
22727445 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12500 |
nM |
22727445 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
30700 |
nM |
22409771 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
22409771 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
22409771 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3500 |
nM |
22409771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
22409771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7600 |
nM |
22409771 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
8280 |
nM |
22749192 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15100 |
nM |
22749192 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
18500 |
nM |
22749192 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14200 |
nM |
22749192 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17400 |
nM |
22749192 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
280 |
ug/ml |
22796042 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
ug/ml |
22796042 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
690 |
ug/ml |
22796042 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
40 |
ug/ml |
22796042 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
115 |
mg/kg |
22796042 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
12320 |
nM |
22687745 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
14490 |
nM |
22687745 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8830 |
nM |
22687745 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
1090 |
nM |
22687745 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
32220 |
nM |
22687745 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
15990 |
nM |
22687745 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
1380 |
nM |
22687745 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
100000 |
nM |
22687745 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
15920 |
nM |
22209486 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
22765897 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
9600 |
nM |
22765897 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7300 |
nM |
22765897 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
Activity |
= |
1645 |
mm3 |
22339362 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
Ratio |
= |
9.13 |
|
22339362 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
GI |
= |
20 |
% |
22339362 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10360 |
nM |
22801644 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
15650 |
nM |
22801644 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
24580 |
nM |
22801644 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
31570 |
nM |
22801644 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
35750 |
nM |
22801644 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
10450 |
nM |
22801644 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
31520 |
nM |
22801644 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9920 |
nM |
22801644 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
3060 |
nM |
22801644 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
24580 |
nM |
22801644 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
70 |
% |
22818042 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
GI |
= |
68 |
% |
22818042 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16200 |
nM |
22840493 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
12800 |
nM |
22840493 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
3300 |
nM |
22840493 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25600 |
nM |
22840493 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
42.5 |
% |
22840493 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
79 |
% |
22982123 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
78 |
% |
22982123 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
22867707 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
30700 |
nM |
22867707 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9970 |
nM |
22867707 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7690 |
nM |
22867707 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
18700 |
nM |
22867707 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
8910 |
nM |
22867707 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3500 |
nM |
22867707 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
47300 |
nM |
22867707 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
1280 |
nM |
22867707 |
NPT3882 |
Cell Line |
MFE-296 |
Homo sapiens |
IC50 |
= |
30680 |
nM |
22867707 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
97.3 |
ug |
23022735 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
9.1 |
ug/ml |
23022735 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
4 |
ug/ml |
23022735 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6.4 |
ug/ml |
23022735 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.5 |
ug/ml |
23022735 |
NPT2 |
Others |
Unspecified |
|
ED100 |
= |
68 |
ug |
23022735 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
38.6 |
ug |
23022735 |
NPT2 |
Others |
Unspecified |
|
ED25 |
= |
32.26 |
ug |
23022735 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
22959205 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
9600 |
nM |
22959205 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7300 |
nM |
22959205 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
25929 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
|
3981.1 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
10590.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
1258.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
3505 |
nM |
PubChem BioAssay data set |
NPT101 |
Individual Protein |
Glucagon-like peptide 1 receptor |
Homo sapiens |
Potency |
|
11220.2 |
nM |
PubChem BioAssay data set |
NPT158 |
Individual Protein |
Nuclear receptor subfamily 1 group I member 2 |
Rattus norvegicus |
Potency |
|
56234.1 |
nM |
PubChem BioAssay data set |
NPT102 |
Individual Protein |
Interleukin-8 |
Homo sapiens |
Potency |
|
66824.2 |
nM |
PubChem BioAssay data set |
NPT159 |
Individual Protein |
Aberrant vpr protein |
Human immunodeficiency virus 1 |
Potency |
|
10000 |
nM |
PubChem BioAssay data set |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
280 |
nM |
22959518 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
60 |
nM |
22959518 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
1070 |
nM |
22959518 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Activity |
= |
98 |
% |
22959518 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Activity |
= |
94 |
% |
22959518 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Activity |
= |
87 |
% |
22959518 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Activity |
= |
76 |
% |
22959518 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12500 |
nM |
22955095 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
Inhibition |
= |
20 |
% |
22607122 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
22995621 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
22995621 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9500 |
nM |
23002924 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12000 |
nM |
23002924 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3250 |
nM |
23018096 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2410 |
nM |
23018096 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
1520 |
nM |
23018096 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
23018096 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4210 |
nM |
23044370 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
Inhibition |
= |
20 |
% |
22715973 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
4500 |
nM |
23075414 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12300 |
nM |
23075414 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5100 |
nM |
23075414 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8500 |
nM |
23075414 |
NPT1719 |
Cell Line |
2008 |
Homo sapiens |
IC50 |
= |
4200 |
nM |
23075414 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
230 |
nM |
21892829 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
21892829 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
12000 |
nM |
21892829 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18000 |
nM |
21892829 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
320 |
nM |
21892829 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
15200 |
nM |
23067549 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
36400 |
nM |
23067549 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
51500 |
nM |
23067549 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
88900 |
nM |
23067549 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
78600 |
nM |
23067549 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
63400 |
nM |
23067549 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
66.8 |
% |
22647218 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
GI |
= |
66.8 |
% |
22647218 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
GI |
= |
66.8 |
% |
22647218 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
66.8 |
% |
22647218 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
7.2 |
ug/ml |
22647218 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
8.2 |
ug/ml |
22647218 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
8.7 |
ug/ml |
22647218 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
9.3 |
ug/ml |
22647218 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
GI50 |
= |
62.02 |
nM |
23094992 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1 |
nM |
23094992 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
3.6 |
nM |
23094992 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
GI50 |
= |
7.6 |
nM |
23094992 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
GI50 |
= |
2.9 |
nM |
23094992 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
GI50 |
= |
30.6 |
nM |
23094992 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23094992 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
69.6 |
nM |
23094992 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
26.4 |
nM |
23094992 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
8.12 |
nM |
23094992 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
14.5 |
nM |
23094992 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
10.45 |
nM |
23094992 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
20 |
nM |
23094992 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
21.1 |
nM |
23094992 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
8.8 |
nM |
23094992 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
1 |
nM |
23094992 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
TGI |
= |
8.4 |
nM |
23094992 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
100 |
nM |
23094992 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
TGI |
= |
36.66 |
% |
23094992 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
TGI |
= |
23.66 |
% |
23094992 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
1 |
nM |
23094992 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
= |
100 |
nM |
23094992 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
33 |
% |
10.1007/s00044-011-9899-3 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
21 |
% |
10.1007/s00044-011-9899-3 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
22 |
% |
10.1007/s00044-011-9899-3 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
GI |
= |
27 |
% |
10.1007/s00044-011-9899-3 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
51 |
% |
10.1007/s00044-011-9899-3 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
4700 |
nM |
10.1007/s00044-011-9778-y |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
266000 |
nM |
10.1007/s00044-011-9778-y |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
85113803.82 |
nM |
10.1007/s00044-011-9906-8 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
45708818.96 |
nM |
10.1007/s00044-011-9906-8 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
9332543.01 |
nM |
10.1007/s00044-011-9906-8 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
21877616.24 |
nM |
10.1007/s00044-011-9906-8 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
8128.31 |
nM |
10.1007/s00044-011-9789-8 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
10715.19 |
nM |
10.1007/s00044-011-9789-8 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
= |
9772.37 |
nM |
10.1007/s00044-011-9789-8 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
6606.93 |
nM |
10.1007/s00044-011-9789-8 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
79.43 |
nM |
10.1007/s00044-011-9789-8 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
363.08 |
nM |
10.1007/s00044-011-9789-8 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
2344.23 |
nM |
10.1007/s00044-011-9789-8 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
1412.54 |
nM |
10.1007/s00044-011-9789-8 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
1122.02 |
nM |
10.1007/s00044-011-9789-8 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
501.19 |
nM |
10.1007/s00044-011-9789-8 |
NPT3121 |
Cell Line |
RXF-393 |
Homo sapiens |
GI50 |
= |
2630.27 |
nM |
10.1007/s00044-011-9789-8 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
72.44 |
nM |
10.1007/s00044-011-9789-8 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
295.12 |
nM |
10.1007/s00044-011-9789-8 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
10.1007/s00044-011-9789-8 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
724.44 |
nM |
10.1007/s00044-011-9789-8 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
21877.62 |
nM |
10.1007/s00044-011-9789-8 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
1737.8 |
nM |
10.1007/s00044-011-9789-8 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
10964.78 |
nM |
10.1007/s00044-011-9789-8 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
4466.84 |
nM |
10.1007/s00044-011-9789-8 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
15.85 |
nM |
10.1007/s00044-011-9789-8 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
1230.27 |
nM |
10.1007/s00044-011-9789-8 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
524.81 |
nM |
10.1007/s00044-011-9789-8 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
10.1007/s00044-011-9789-8 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
467.74 |
nM |
10.1007/s00044-011-9789-8 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
1023.29 |
nM |
10.1007/s00044-011-9789-8 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
56234.13 |
nM |
10.1007/s00044-011-9789-8 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
977.24 |
nM |
10.1007/s00044-011-9789-8 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
51.29 |
nM |
10.1007/s00044-011-9789-8 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
245.47 |
nM |
10.1007/s00044-011-9789-8 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
GI50 |
= |
912.01 |
nM |
10.1007/s00044-011-9789-8 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
10.1007/s00044-011-9789-8 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
3801.89 |
nM |
10.1007/s00044-011-9789-8 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
63.1 |
nM |
10.1007/s00044-011-9789-8 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
10.1007/s00044-011-9789-8 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
10.1007/s00044-011-9789-8 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
933.25 |
nM |
10.1007/s00044-011-9789-8 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
213.8 |
nM |
10.1007/s00044-011-9789-8 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
10.1007/s00044-011-9789-8 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
109.65 |
nM |
10.1007/s00044-011-9789-8 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
229.09 |
nM |
10.1007/s00044-011-9789-8 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
52.48 |
nM |
10.1007/s00044-011-9789-8 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
158.49 |
nM |
10.1007/s00044-011-9789-8 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
7244.36 |
nM |
10.1007/s00044-011-9789-8 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
56.23 |
nM |
10.1007/s00044-011-9789-8 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
177.83 |
nM |
10.1007/s00044-011-9789-8 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
331.13 |
nM |
10.1007/s00044-011-9789-8 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
54954.09 |
nM |
10.1007/s00044-011-9789-8 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
77624.71 |
nM |
10.1007/s00044-011-9789-8 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
398.11 |
nM |
10.1007/s00044-011-9789-8 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
61659.5 |
nM |
10.1007/s00044-011-9789-8 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
190.55 |
nM |
10.1007/s00044-011-9789-8 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
23.99 |
nM |
10.1007/s00044-011-9789-8 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
44.67 |
nM |
10.1007/s00044-011-9789-8 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
354.81 |
nM |
10.1007/s00044-011-9789-8 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
3548.13 |
nM |
10.1007/s00044-011-9789-8 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
2290.87 |
nM |
10.1007/s00044-011-9789-8 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
9772.37 |
nM |
10.1007/s00044-011-9789-8 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
69 |
% |
10.1007/s00044-011-9887-7 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
74 |
% |
10.1007/s00044-011-9887-7 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
18 |
% |
10.1007/s00044-011-9850-7 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
8 |
% |
10.1007/s00044-011-9850-7 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
5 |
% |
10.1007/s00044-011-9850-7 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
GI |
= |
10 |
% |
10.1007/s00044-011-9850-7 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
24 |
% |
10.1007/s00044-011-9850-7 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
29190 |
nM |
10.1007/s00044-011-9549-9 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
9720 |
nM |
10.1007/s00044-011-9549-9 |
NPT3884 |
Individual Protein |
Uracil phosphoribosyltransferase |
Escherichia coli (strain K12) |
Ki |
= |
13000 |
nM |
10.1007/s00044-011-9627-z |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
10.1007/s00044-010-9500-5 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
10.1007/s00044-010-9500-5 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
10.1007/s00044-010-9500-5 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
2190 |
nM |
10.1007/s00044-010-9395-1 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
45400 |
nM |
10.1007/s00044-010-9395-1 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2950 |
nM |
10.1007/s00044-010-9395-1 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9700 |
nM |
10.1007/s00044-010-9395-1 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1930 |
nM |
10.1007/s00044-010-9395-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
37 |
% |
10.1007/s00044-011-9610-8 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
58 |
% |
10.1007/s00044-011-9610-8 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
93 |
% |
10.1007/s00044-011-9610-8 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
90.76 |
% |
10.1007/s00044-010-9455-6 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
92.7 |
% |
10.1007/s00044-010-9455-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
85.17 |
% |
10.1007/s00044-010-9455-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
14.83 |
% |
10.1007/s00044-010-9455-6 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
25.4 |
ug/ml |
10.1007/s00044-009-9193-9 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
10.26 |
ug/ml |
10.1007/s00044-009-9193-9 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
0.58 |
ug/ml |
10.1007/s00044-009-9193-9 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
g/dl |
10.1007/s00044-009-9199-3 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
42.3 |
% |
10.1007/s00044-009-9199-3 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
123 |
10'6/ml |
10.1007/s00044-009-9199-3 |
NPT2 |
Others |
Unspecified |
|
ED25 |
= |
0 |
nM |
10.1007/s00044-009-9199-3 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
96.3 |
nM |
10.1007/s00044-009-9199-3 |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
Inhibition |
= |
30.7 |
% |
16190646 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
41.1 |
% |
16190646 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
69 |
% |
10.1007/s00044-012-0106-y |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
29 |
% |
10.1007/s00044-012-0106-y |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
30 |
% |
10.1007/s00044-012-0106-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI |
= |
36 |
% |
10.1007/s00044-012-0106-y |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI |
= |
38 |
% |
10.1007/s00044-012-0106-y |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
42 |
% |
10.1007/s00044-012-0106-y |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
47 |
% |
10.1007/s00044-012-0106-y |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2720 |
nM |
10.1007/s00044-012-0209-5 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
3240 |
nM |
10.1007/s00044-012-0209-5 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0 |
% |
10.1007/s00044-012-0116-9 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Activity |
= |
0 |
% |
10.1007/s00044-012-0116-9 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
Activity |
= |
0 |
% |
10.1007/s00044-012-0116-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
0 |
% |
10.1007/s00044-012-0116-9 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
79 |
% |
10.1007/s00044-012-0032-z |
NPT3885 |
Cell Line |
CV-1 |
Chlorocebus aethiops |
GI |
= |
43 |
% |
10.1007/s00044-012-0032-z |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
87 |
% |
10.1007/s00044-012-0032-z |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
79 |
% |
10.1007/s00044-012-0032-z |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.2 |
% |
10.1007/s00044-013-0478-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
27.8 |
% |
10.1007/s00044-013-0478-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
71 |
% |
10.1007/s00044-013-0478-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
15.6 |
mm3 |
10.1007/s00044-013-0478-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
13.99 |
g% |
10.1007/s00044-013-0478-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
4.67 |
million/mm3 |
10.1007/s00044-013-0478-7 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
57.29 |
% |
10.1007/s00044-013-0478-7 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
70.68 |
% |
10.1007/s00044-013-0478-7 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
21000 |
nM |
10.1007/s00044-012-0424-0 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
18 |
% |
10.1007/s00044-012-0438-7 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
GI |
= |
22 |
% |
10.1007/s00044-012-0438-7 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
19 |
% |
10.1007/s00044-012-0438-7 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
24 |
% |
10.1007/s00044-012-0438-7 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
15 |
% |
10.1007/s00044-012-0438-7 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
28 |
% |
10.1007/s00044-012-0439-6 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
GI |
= |
18 |
% |
10.1007/s00044-012-0439-6 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
15 |
% |
10.1007/s00044-012-0439-6 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
18 |
% |
10.1007/s00044-012-0439-6 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
10 |
% |
10.1007/s00044-012-0439-6 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
19200 |
nM |
10.1007/s00044-012-0461-8 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
21900 |
nM |
10.1007/s00044-012-0181-0 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
46200 |
nM |
10.1007/s00044-012-0181-0 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5200 |
nM |
10.1007/s00044-012-0181-0 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
= |
251188.64 |
nM |
10.1007/s00044-012-0192-x |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
79432.82 |
nM |
10.1007/s00044-012-0192-x |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
10.1007/s00044-012-0192-x |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
501187.23 |
nM |
10.1007/s00044-012-0192-x |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
10.1007/s00044-012-0192-x |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
10.1007/s00044-012-0192-x |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
10.1007/s00044-012-0192-x |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
125892.54 |
nM |
10.1007/s00044-012-0192-x |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.1007/s00044-012-0192-x |
NPT3121 |
Cell Line |
RXF-393 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
3981.07 |
nM |
10.1007/s00044-012-0192-x |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
10000 |
nM |
10.1007/s00044-012-0192-x |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
10.1007/s00044-012-0192-x |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
10.1007/s00044-012-0192-x |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
10.1007/s00044-012-0192-x |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
63095.73 |
nM |
10.1007/s00044-012-0192-x |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.1007/s00044-012-0192-x |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
100000 |
nM |
10.1007/s00044-012-0192-x |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
398107.17 |
nM |
10.1007/s00044-012-0192-x |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
10.1007/s00044-012-0192-x |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
10.1007/s00044-012-0192-x |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
199526.23 |
nM |
10.1007/s00044-012-0192-x |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
125892.54 |
nM |
10.1007/s00044-012-0192-x |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
1258.93 |
nM |
10.1007/s00044-012-0192-x |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
50118.72 |
nM |
10.1007/s00044-012-0192-x |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
25118.86 |
nM |
10.1007/s00044-012-0192-x |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
10.1007/s00044-012-0192-x |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
10.1007/s00044-012-0192-x |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
10.1007/s00044-012-0192-x |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
3981.07 |
nM |
10.1007/s00044-012-0192-x |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
1584.89 |
nM |
10.1007/s00044-012-0192-x |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
6309.57 |
nM |
10.1007/s00044-012-0192-x |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
39810.72 |
nM |
10.1007/s00044-012-0192-x |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
1000 |
nM |
10.1007/s00044-012-0192-x |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
251188.64 |
nM |
10.1007/s00044-012-0192-x |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
158489.32 |
nM |
10.1007/s00044-012-0192-x |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
= |
316227.77 |
nM |
10.1007/s00044-012-0192-x |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
1995.26 |
nM |
10.1007/s00044-012-0192-x |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
5011.87 |
nM |
10.1007/s00044-012-0192-x |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
12589.25 |
nM |
10.1007/s00044-012-0192-x |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
19952.62 |
nM |
10.1007/s00044-012-0192-x |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
31622.78 |
nM |
10.1007/s00044-012-0192-x |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
72.53 |
% |
10.1007/s00044-012-0201-0 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
13.8 |
10'3cm |
10.1007/s00044-012-0201-0 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
42.3 |
% |
10.1007/s00044-012-0201-0 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
10 |
g/dl |
10.1007/s00044-012-0201-0 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
123 |
10'6/ml |
10.1007/s00044-012-0201-0 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
70000 |
nM |
10.1007/s00044-012-0201-0 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
20000 |
nM |
10.1007/s00044-012-0201-0 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
2150 |
nM |
10.1007/s00044-012-0260-2 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1250 |
nM |
10.1007/s00044-012-0260-2 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
10.1007/s00044-012-0260-2 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
50000 |
nM |
10.1007/s00044-012-0201-0 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
20000 |
nM |
10.1007/s00044-012-0201-0 |
NPT2 |
Others |
Unspecified |
|
ED25 |
= |
40 |
microg/cm3 |
10.1007/s00044-012-0336-z |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
63 |
microg/cm3 |
10.1007/s00044-012-0336-z |
NPT2 |
Others |
Unspecified |
|
ED100 |
= |
97 |
microg/cm3 |
10.1007/s00044-012-0336-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
19200 |
nM |
10.1007/s00044-012-0283-8 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2950 |
nM |
10.1007/s00044-012-0283-8 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1930 |
nM |
10.1007/s00044-012-0283-8 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
10.1007/s00044-012-0283-8 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
10.1007/s00044-012-0240-6 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
19200 |
nM |
10.1007/s00044-012-0240-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
13.8 |
10'3/mm3 |
10.1007/s00044-012-0396-0 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
42.3 |
g% |
10.1007/s00044-012-0396-0 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
g% |
10.1007/s00044-012-0396-0 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
16.7 |
% |
10.1007/s00044-012-0396-0 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.3 |
ml |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.7 |
ug |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94 |
% |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
162.3 |
U/L |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
42.45 |
U/L |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
56.3 |
U/L |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
156.42 |
mg/dl |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
112.52 |
mg/dl |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.65 |
10'5/mm3 |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17.45 |
% |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11.5 |
g/dl |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.1 |
million/mm3 |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11.3 |
ml |
10.1007/s00044-012-0407-1 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7120 |
nM |
23164710 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3850 |
nM |
23164710 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
23164710 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1540 |
nM |
23164710 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
3840 |
nM |
23164710 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
5380 |
nM |
23164710 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
114500 |
nM |
23356786 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
126200 |
nM |
23356786 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
158200 |
nM |
23356786 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
142600 |
nM |
23356786 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
56000 |
nM |
23356786 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17200 |
nM |
23279864 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
28500 |
nM |
23279864 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
21900 |
nM |
23279864 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
23313635 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
23313635 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
14780 |
nM |
23313635 |
NPT3886 |
Cell Line |
COS-1 |
Chlorocebus aethiops |
IC50 |
= |
110000 |
nM |
23202484 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
29870 |
nM |
23202484 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
39500 |
nM |
23202484 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
45010 |
nM |
23202484 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
IC50 |
= |
56760 |
nM |
23202484 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
51800 |
nM |
23202484 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
19 |
% |
23202484 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
32 |
% |
23202484 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
GI |
= |
22 |
% |
23202484 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
13 |
% |
23202484 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
15 |
% |
23202484 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
7 |
|
23305919 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
FC |
= |
2.6 |
|
23305919 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
25000 |
nM |
23305919 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3560 |
nM |
23305919 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
IC50 |
= |
50000 |
nM |
23360104 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1.28 |
ug/ml |
23352638 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
0.87 |
ug/ml |
23352638 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
4.03 |
ug/ml |
23352638 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
0.54 |
ug/ml |
23352638 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
84 |
% |
23419739 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
72 |
% |
23419739 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5640 |
nM |
23353737 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16320 |
nM |
23353737 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
15850 |
nM |
23353737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14300 |
nM |
23353737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
46570 |
nM |
23353737 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
46350 |
nM |
23312949 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
21410 |
nM |
23312949 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
70.31 |
% |
23167526 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
55 |
% |
23387901 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
Activity |
= |
84 |
% |
23387901 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
22 |
% |
23387901 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3340 |
nM |
23353743 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
27070 |
nM |
23353743 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7540 |
nM |
23353743 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
7010 |
nM |
23353743 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
LC50 |
= |
25000 |
nM |
23321564 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16700 |
nM |
23490159 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
28900 |
nM |
23490159 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
22800 |
nM |
23490159 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
18356.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8199.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16360.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14963.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33498.3 |
nM |
PubChem BioAssay data set |
NPT861 |
Individual Protein |
Isocitrate dehydrogenase [NADP] cytoplasmic |
Homo sapiens |
Potency |
|
2310.9 |
nM |
PubChem BioAssay data set |
NPT1357 |
Cell Line |
H22 |
Mus musculus |
Activity |
= |
81 |
% |
23597099 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LC90 |
= |
736.49 |
ug/ml |
23474904 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LC50 |
= |
409.16 |
ug/ml |
23474904 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
9.874 |
ug/ml |
23548704 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
4.562 |
ug/ml |
23548704 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
23550 |
nM |
23558238 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
23930 |
nM |
23558238 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
10050 |
nM |
23558238 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
35620 |
nM |
23558238 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6670 |
nM |
23558238 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
44050 |
nM |
23558238 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
27760 |
nM |
23558238 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
40340 |
nM |
23558238 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11500 |
nM |
23558238 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7340 |
nM |
23558238 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4900 |
nM |
23501113 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
23501113 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
23501113 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
23501113 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
32000 |
nM |
23535322 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
28000 |
nM |
23535322 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
23474899 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
23474899 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
70800 |
nM |
23647462 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
56.7 |
% |
23611732 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
89 |
% |
23584541 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
83 |
% |
23584541 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
75 |
% |
23584541 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
73 |
% |
23584541 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
72 |
% |
23584541 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
72 |
% |
23584541 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
64 |
% |
23584541 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI |
= |
37.8 |
% |
23611732 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
78.1 |
% |
23611732 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
11.5 |
% |
23611732 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
35.5 |
% |
23611732 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
58.2 |
% |
23611732 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI |
= |
41.3 |
% |
23611732 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI |
= |
66.9 |
% |
23611732 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI |
= |
54 |
% |
23611732 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI |
= |
34.3 |
% |
23611732 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI |
= |
39.4 |
% |
23611732 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI |
= |
39.3 |
% |
23611732 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI |
= |
48.7 |
% |
23611732 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI |
= |
77.5 |
% |
23611732 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI |
= |
47.6 |
% |
23611732 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI |
= |
44.3 |
% |
23611732 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI |
= |
59.4 |
% |
23611732 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI |
= |
47.4 |
% |
23611732 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI |
= |
51.2 |
% |
23611732 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI |
= |
39.7 |
% |
23611732 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI |
= |
19.5 |
% |
23611732 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI |
= |
33.7 |
% |
23611732 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI |
= |
95.5 |
% |
23611732 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI |
= |
36.6 |
% |
23611732 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI |
= |
58.2 |
% |
23611732 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI |
= |
30.4 |
% |
23611732 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI |
= |
50.3 |
% |
23611732 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI |
= |
65.9 |
% |
23611732 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI |
= |
65.9 |
% |
23611732 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
69.1 |
% |
23611732 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI |
= |
59 |
% |
23611732 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
50.1 |
% |
23611732 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI |
= |
40.7 |
% |
23611732 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
27.1 |
% |
23611732 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
26.5 |
% |
23611732 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
17.8 |
% |
23611732 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
40.2 |
% |
23611732 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
58 |
% |
23611732 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
13 |
% |
23611732 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI |
= |
59.5 |
% |
23611732 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI |
= |
39 |
% |
23611732 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI |
= |
69.5 |
% |
23611732 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI |
= |
50.6 |
% |
23611732 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI |
= |
47.8 |
% |
23611732 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
58.4 |
% |
23611732 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
34.2 |
% |
23611732 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI |
= |
24.8 |
% |
23611732 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI |
= |
41.4 |
% |
23611732 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI |
= |
43.1 |
% |
23611732 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
42.3 |
% |
23611732 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
47.9 |
% |
23611732 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI |
= |
57.1 |
% |
23611732 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
6.81 |
% |
23665106 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
47.75 |
% |
23665106 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
45.44 |
% |
23665106 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5530 |
nM |
23665106 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
24500 |
nM |
23665106 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
43710 |
nM |
23665106 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
32180 |
nM |
23665106 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3520 |
nM |
23665106 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
320 |
nM |
23644193 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
26710 |
nM |
23644193 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7330 |
nM |
23644193 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
7140 |
nM |
23644193 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6350 |
nM |
23644215 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4520 |
nM |
23644215 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
23644215 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
23644215 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
9710 |
nM |
23685571 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
970 |
nM |
23685571 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3240 |
nM |
23685571 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10140 |
nM |
23685571 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8710 |
nM |
23685571 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
24960 |
nM |
23685571 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
23683592 |
NPT1357 |
Cell Line |
H22 |
Mus musculus |
Inhibition |
= |
57.55 |
% |
23617697 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
23683592 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
23683592 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
56.7 |
% |
23642480 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI |
= |
37.8 |
% |
23642480 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
78.1 |
% |
23642480 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
11.5 |
% |
23642480 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
35.5 |
% |
23642480 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
58.2 |
% |
23642480 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI |
= |
41.3 |
% |
23642480 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI |
= |
54 |
% |
23642480 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI |
= |
39.4 |
% |
23642480 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI |
= |
39.3 |
% |
23642480 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI |
= |
77.5 |
% |
23642480 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
47.6 |
% |
23642480 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI |
= |
44.3 |
% |
23642480 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI |
= |
59.4 |
% |
23642480 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI |
= |
47.4 |
% |
23642480 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI |
= |
51.2 |
% |
23642480 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI |
= |
39.7 |
% |
23642480 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI |
= |
33.7 |
% |
23642480 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI |
= |
19.5 |
% |
23642480 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI |
= |
95.5 |
% |
23642480 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI |
= |
58.2 |
% |
23642480 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI |
= |
30.4 |
% |
23642480 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI |
= |
50.3 |
% |
23642480 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI |
= |
65.9 |
% |
23642480 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
69 |
% |
23642480 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI |
= |
59 |
% |
23642480 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
< |
20 |
% |
23642480 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI |
= |
40.7 |
% |
23642480 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
26.5 |
% |
23642480 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
17.8 |
% |
23642480 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
58 |
% |
23642480 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI |
= |
59.5 |
% |
23642480 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI |
= |
39 |
% |
23642480 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI |
= |
69.5 |
% |
23642480 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI |
= |
50.6 |
% |
23642480 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI |
= |
47.8 |
% |
23642480 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
34.2 |
% |
23642480 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI |
= |
24.8 |
% |
23642480 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI |
= |
41.4 |
% |
23642480 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI |
= |
43.1 |
% |
23642480 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
42.3 |
% |
23642480 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
47.9 |
% |
23642480 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI |
= |
57.1 |
% |
23642480 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
27070 |
nM |
23735281 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
31440 |
nM |
23735281 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
23800391 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
8000 |
nM |
23800391 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
23800391 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
23800391 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
9780 |
nM |
23792764 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
24760 |
nM |
23792764 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7540 |
nM |
23792764 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
6920 |
nM |
23792764 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10610 |
nM |
23792764 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
96 |
% |
23811086 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
76 |
% |
23811086 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
86 |
% |
23811086 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
15710 |
nM |
23920246 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
13650 |
nM |
23920246 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
3600 |
nM |
23964677 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
6040 |
nM |
23920246 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14300 |
nM |
23920246 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16520 |
nM |
23920246 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5620 |
nM |
23920246 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
8120 |
nM |
23887055 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
10600 |
nM |
23887055 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
9770 |
nM |
23887055 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
6600 |
nM |
23887055 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
70 |
nM |
23887055 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
360 |
nM |
23887055 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
2360 |
nM |
23887055 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
1420 |
nM |
23887055 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
1120 |
nM |
23887055 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
490 |
nM |
23887055 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
2610 |
nM |
23887055 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
70 |
nM |
23887055 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
290 |
nM |
23887055 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
350 |
nM |
23887055 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
720 |
nM |
23887055 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
21800 |
nM |
23887055 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
310 |
nM |
23887055 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
1740 |
nM |
23887055 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
10900 |
nM |
23887055 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
4430 |
nM |
23887055 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
10 |
nM |
23887055 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
1220 |
nM |
23887055 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
520 |
nM |
23887055 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
3550 |
nM |
23887055 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
460 |
nM |
23887055 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
1030 |
nM |
23887055 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
56700 |
nM |
23887055 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
70 |
nM |
23887055 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
980 |
nM |
23887055 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
50 |
nM |
23887055 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
240 |
nM |
23887055 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
900 |
nM |
23887055 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
78700 |
nM |
23887055 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
3810 |
nM |
23887055 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
60 |
nM |
23887055 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
220 |
nM |
23887055 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
1620 |
nM |
23887055 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
920 |
nM |
23887055 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
210 |
nM |
23887055 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
170 |
nM |
23887055 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
110 |
nM |
23887055 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
220 |
nM |
23887055 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
50 |
nM |
23887055 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
150 |
nM |
23887055 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
7270 |
nM |
23887055 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
50 |
nM |
23887055 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
330 |
nM |
23887055 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
54700 |
nM |
23887055 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
77900 |
nM |
23887055 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
390 |
nM |
23887055 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61800 |
nM |
23887055 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
180 |
nM |
23887055 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
20 |
nM |
23887055 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
40 |
nM |
23887055 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
350 |
nM |
23887055 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
9790 |
nM |
23887055 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
3580 |
nM |
23887055 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
2300 |
nM |
23887055 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26700 |
nM |
23867385 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
22300 |
nM |
23867385 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3600 |
nM |
23792763 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
128700 |
nM |
23792763 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
8100 |
nM |
23792763 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14500 |
nM |
23792763 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3400 |
nM |
23792763 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18600 |
nM |
23792763 |
NPT2 |
Others |
Unspecified |
|
IC25 |
= |
0.19 |
nM |
10.1007/s00044-013-0859-y |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
380 |
nM |
10.1007/s00044-013-0859-y |
NPT2 |
Others |
Unspecified |
|
IC100 |
= |
0.77 |
nM |
10.1007/s00044-013-0859-y |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6530 |
nM |
23867603 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
4840 |
nM |
23867603 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6230 |
nM |
23867603 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
ED50 |
= |
50.2 |
nM |
24020806 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
ED50 |
= |
15.07 |
nM |
24020806 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
ED50 |
= |
16.22 |
nM |
24020806 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1510 |
nM |
23994328 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
56.7 |
% |
23994328 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI |
= |
37.8 |
% |
23994328 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
78.1 |
% |
23994328 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
11.5 |
% |
23994328 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
35.5 |
% |
23994328 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
58.2 |
% |
23994328 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI |
= |
41.3 |
% |
23994328 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI |
= |
66.9 |
% |
23994328 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI |
= |
54 |
% |
23994328 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI |
= |
34.3 |
% |
23994328 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI |
= |
39.4 |
% |
23994328 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI |
= |
39.3 |
% |
23994328 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI |
= |
48.7 |
% |
23994328 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI |
= |
77.5 |
% |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
47.6 |
% |
23994328 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI |
= |
44.3 |
% |
23994328 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI |
= |
59.4 |
% |
23994328 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI |
= |
47.4 |
% |
23994328 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI |
= |
51.2 |
% |
23994328 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI |
= |
39.7 |
% |
23994328 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI |
= |
19.5 |
% |
23994328 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI |
= |
33.7 |
% |
23994328 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI |
= |
95.5 |
% |
23994328 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI |
= |
36.6 |
% |
23994328 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI |
= |
58.2 |
% |
23994328 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI |
= |
30.4 |
% |
23994328 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI |
= |
50.3 |
% |
23994328 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI |
= |
65.9 |
% |
23994328 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI |
= |
65.9 |
% |
23994328 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
69.1 |
% |
23994328 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI |
= |
59 |
% |
23994328 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
50.1 |
% |
23994328 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI |
= |
40.7 |
% |
23994328 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
27.1 |
% |
23994328 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
26.5 |
% |
23994328 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
17.8 |
% |
23994328 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
40.2 |
% |
23994328 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI |
= |
58 |
% |
23994328 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
13 |
% |
23994328 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI |
= |
59.5 |
% |
23994328 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI |
= |
39 |
% |
23994328 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI |
= |
69.5 |
% |
23994328 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI |
= |
50.6 |
% |
23994328 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI |
= |
47.8 |
% |
23994328 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
58.4 |
% |
23994328 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
34.2 |
% |
23994328 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI |
= |
24.8 |
% |
23994328 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI |
= |
41.4 |
% |
23994328 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI |
= |
43.1 |
% |
23994328 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI |
= |
42.3 |
% |
23994328 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
47.9 |
% |
23994328 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI |
= |
57.1 |
% |
23994328 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.8 |
ug/ml |
23994872 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
23550 |
nM |
23999046 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
23930 |
nM |
23999046 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
10050 |
nM |
23999046 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
35620 |
nM |
23999046 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6670 |
nM |
23999046 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
44050 |
nM |
23999046 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
27760 |
nM |
23999046 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
40340 |
nM |
23999046 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11500 |
nM |
23999046 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7340 |
nM |
23999046 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
5950 |
nM |
10.1007/s00044-013-0798-7 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
49210 |
nM |
10.1007/s00044-013-0798-7 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
8400 |
nM |
10.1007/s00044-013-0798-7 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
9510 |
nM |
10.1007/s00044-013-0798-7 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
> |
100000 |
nM |
10.1007/s00044-013-0798-7 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
> |
100000 |
nM |
10.1007/s00044-013-0798-7 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
> |
100000 |
nM |
10.1007/s00044-013-0798-7 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
> |
100000 |
nM |
10.1007/s00044-013-0798-7 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
7.7 |
nM |
24128077 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
ED50 |
= |
0.021 |
nM |
24128077 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
ED50 |
= |
7.7 |
nM |
24128077 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ED50 |
= |
6.2 |
nM |
24128077 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
28.07 |
% |
23988357 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
0 |
% |
23988357 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
71.93 |
% |
23988357 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
16.8 |
% |
23988357 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
6.5 |
% |
23988357 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
24430 |
nM |
23988357 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
29980 |
nM |
23988357 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
34330 |
nM |
23988357 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
44040 |
nM |
23988357 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
24430 |
nM |
24095745 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
29980 |
nM |
24095745 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
34330 |
nM |
24095745 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
44040 |
nM |
24095745 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
24013415 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
14550 |
nM |
24013415 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
12480 |
nM |
24013415 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15660 |
nM |
24013415 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
24056146 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
24056146 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.887 |
ug/ml |
24021891 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
2.48 |
ug/ml |
24021891 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1100 |
nM |
24060486 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
24060486 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24060486 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
24060486 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7540 |
nM |
24077182 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
24760 |
nM |
24077182 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
9780 |
nM |
24077182 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
6920 |
nM |
24077182 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10610 |
nM |
24077182 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
6920 |
nM |
24095094 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
8300 |
nM |
24095094 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8920 |
nM |
24095094 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
91.17 |
% |
23571415 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
86.84 |
% |
23571415 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
1000000 |
nM |
24177365 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
264000 |
nM |
24177365 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
8500 |
nM |
24195466 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3400 |
nM |
24195466 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
28.07 |
% |
24211021 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
0 |
% |
24211021 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
71.93 |
% |
24211021 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
6.5 |
% |
24211021 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
16.8 |
% |
24211021 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
15320 |
nM |
24211021 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
19450 |
nM |
24211021 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8320 |
nM |
24211021 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20130 |
nM |
24211021 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
23320 |
nM |
24211021 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4900 |
nM |
24332497 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
4200 |
nM |
24332497 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3500 |
nM |
24332497 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI |
= |
62 |
% |
24332623 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7480 |
nM |
24286761 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5260 |
nM |
24286761 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9790 |
nM |
24286761 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7430 |
nM |
24286761 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
28 |
% |
24378217 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
65.6 |
% |
24378217 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
56000 |
nM |
24378217 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5780 |
nM |
24378217 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
35340 |
nM |
24378217 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
42200 |
nM |
24378217 |
NPT3887 |
Cell Line |
CNE |
Homo sapiens |
IC50 |
= |
40210 |
nM |
24378217 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
29980 |
nM |
24378217 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
8100 |
nM |
24359303 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
24359303 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5500 |
nM |
24359303 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
23792352 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
24.87 |
ug/ml |
24342667 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
20.03 |
ug/ml |
24342667 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
25.6 |
ug/ml |
24342667 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7600 |
nM |
24547794 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2300 |
nM |
24547794 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
76400 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
22700 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
45600 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
61400 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
70600 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
72100 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
8400 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
100000 |
nM |
24469112 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
15100 |
nM |
24469112 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4350 |
nM |
24119869 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
5580 |
nM |
24119869 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3680 |
nM |
24119869 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7370 |
nM |
24119869 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
24430 |
nM |
24565905 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
80480 |
nM |
24565905 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26800 |
nM |
24565905 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
24430 |
nM |
24565905 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
26980 |
nM |
24565905 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
36040 |
nM |
24565905 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15800 |
nM |
24534537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15700 |
nM |
24534537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14300 |
nM |
24534537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16300 |
nM |
24534537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16400 |
nM |
24534537 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6678 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5623.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6309.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9905.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4216.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
22373.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1569.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3567.4 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
28336.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9439.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
570.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27918.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
20060.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11220.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5955.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35673.7 |
nM |
PubChem BioAssay data set |
NPT104 |
Individual Protein |
Cerebroside-sulfatase |
Homo sapiens |
Potency |
|
26854.5 |
nM |
PubChem BioAssay data set |
NPT105 |
Individual Protein |
Muscleblind-like protein 1 |
Homo sapiens |
Potency |
|
158489.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4730.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2488.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
57044.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1787.9 |
nM |
PubChem BioAssay data set |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Potency |
|
18356.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
793.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10583.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33491.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
50390.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
22710 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
44641.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35992.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21131.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9432.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
62500.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7497.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7868.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10054.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7986.4 |
nM |
PubChem BioAssay data set |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
0.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17615.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1059.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
40026.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
990.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
356.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10590.9 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
19940.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6682.4 |
nM |
PubChem BioAssay data set |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
21000 |
nM |
10.1039/C3MD00055A |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
TGI |
= |
25.93 |
% |
24629450 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
330 |
nM |
24631358 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1800 |
nM |
24641975 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1800 |
nM |
24641975 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
24641975 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
24641975 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
86870 |
nM |
24684840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
67650 |
nM |
24684840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
500000 |
nM |
24684840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
95360 |
nM |
24684840 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
24631358 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
24631358 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
980 |
nM |
24727462 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
31.7 |
% |
385879 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
35.8 |
% |
385879 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
45.7 |
% |
385879 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
MIC |
= |
1.25 |
ug/ml |
385880 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
MIC |
= |
2.5 |
ug/ml |
385880 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
MIC |
> |
20 |
ug/ml |
385880 |
NPT187 |
Organism |
Issatchenkia orientalis |
Pichia kudriavzevii |
MIC |
= |
2.5 |
ug/ml |
385880 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
47 |
mg/kg |
490545 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
70 |
mg/kg |
490545 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Survival |
= |
18 |
day |
316462 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2860 |
nM |
24704691 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
18120 |
nM |
24704691 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
10560 |
nM |
24704691 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
280 |
nM |
24704691 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8060 |
nM |
24704691 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2580 |
nM |
24704691 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
4390 |
nM |
24704691 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
3690 |
nM |
24704691 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9260 |
nM |
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.82 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.44 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.76 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
28.79 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.76 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.6 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.11 |
|
24704691 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.51 |
|
24704691 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11500 |
nM |
24767839 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
44050 |
nM |
24767839 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7340 |
nM |
24767839 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
17200 |
nM |
24767839 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7080 |
nM |
24819956 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
10540 |
nM |
24819956 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11120 |
nM |
24819956 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3520 |
nM |
24835817 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9450 |
nM |
24835817 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
11340 |
nM |
24835817 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Survival |
= |
11 |
day |
592323 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
72.3 |
nM |
338900 |
NPT729 |
Organism |
Micrococcus luteus |
Micrococcus luteus |
MIC |
= |
72.3 |
nM |
338900 |
NPT3888 |
Organism |
Micrococcus flavus |
Micrococcus flavus |
MIC |
= |
4.25 |
nM |
338900 |
NPT79 |
Organism |
Bacillus subtilis |
Bacillus subtilis |
MIC |
= |
4620 |
nM |
338900 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
18600 |
nM |
338900 |
NPT173 |
Organism |
Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
= |
601000 |
nM |
338900 |
NPT766 |
Organism |
Proteus vulgaris |
Proteus vulgaris |
MIC |
= |
18500 |
nM |
338900 |
NPT3889 |
Organism |
Brevundimonas diminuta |
Brevundimonas diminuta |
MIC |
> |
1000000 |
nM |
338900 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
200 |
mg/kg |
357721 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
145 |
mg/kg |
357721 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
115 |
mg/kg |
357721 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
42 |
% |
357721 |
NPT2870 |
Cell Line |
Sarcoma-180 |
Mus musculus |
TGI |
= |
48 |
% |
357721 |
NPT3890 |
Cell Line |
YOSHIDA |
Rattus norvegicus |
TGI |
= |
41 |
% |
357721 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
33 |
% |
357721 |
NPT1842 |
Cell Line |
W256 |
Rattus norvegicus |
TGI |
= |
24 |
% |
357721 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
42.1 |
ug |
357721 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
151.21 |
U/ml |
25010935 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
32.75 |
U/ml |
25010935 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4210 |
nM |
24956552 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
24956552 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
4550 |
nM |
24797798 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
24910974 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4500 |
nM |
24910974 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4900 |
nM |
24910974 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
8130 |
nM |
24798098 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7760 |
nM |
24798098 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24140 |
nM |
24798098 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
4680 |
nM |
24798098 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2450 |
nM |
24941129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3520 |
nM |
24941129 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2780 |
nM |
24941129 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
24835633 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1300 |
nM |
24835633 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
24835633 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
24835633 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1650 |
nM |
24996138 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
10050 |
nM |
24953029 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
46930 |
nM |
24953029 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
45140 |
nM |
24953029 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
34340 |
nM |
24953029 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1230 |
nM |
24953029 |
NPT3887 |
Cell Line |
CNE |
Homo sapiens |
IC50 |
= |
45100 |
nM |
24953029 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
23330 |
nM |
24953029 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
38340 |
nM |
24953029 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
24120 |
nM |
24953029 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
7640 |
nM |
25506718 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9670 |
nM |
25506718 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
13450 |
nM |
25506718 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
26900 |
nM |
25462264 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
31600 |
nM |
25462264 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30900 |
nM |
25462264 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.357 |
ug |
25462264 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
15.7 |
ug |
25462264 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
49.6 |
ug |
25462264 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
319.2 |
ug |
25462264 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
7900 |
nM |
25462277 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6000 |
nM |
25462277 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30700 |
nM |
25462277 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
35600 |
nM |
25453794 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
18100 |
nM |
25453794 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16300 |
nM |
25453794 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38200 |
nM |
25453794 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
36200 |
nM |
25453794 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
12700 |
nM |
25453794 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9340 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11780 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10450 |
nM |
25529742 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
30450 |
nM |
25462253 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9090 |
nM |
25529742 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
10520 |
nM |
25529742 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
70.3 |
% |
25529742 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
36040 |
nM |
25462253 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
36530 |
nM |
25462253 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
12000 |
nM |
25086915 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4700 |
nM |
25086915 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
25086915 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4600 |
nM |
25086915 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
46 |
% |
25043312 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
LC50 |
= |
25000 |
nM |
25078313 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Activity |
= |
13 |
% |
25066282 |
NPT2 |
Others |
Unspecified |
|
Activity |
< |
10 |
% |
25066282 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
FC |
= |
1.9 |
|
25066282 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
FC |
= |
1.1 |
|
25066282 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
25066282 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
25066282 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46830 |
nM |
25016234 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
35410 |
nM |
25016234 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
24600 |
nM |
25016234 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
39880 |
nM |
25016234 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
7760 |
nM |
25113877 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19840 |
nM |
25113877 |
NPT3887 |
Cell Line |
CNE |
Homo sapiens |
IC50 |
= |
15070 |
nM |
25113877 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7620 |
nM |
25113877 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3450 |
nM |
25001482 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7120 |
nM |
25001482 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8070 |
nM |
25001482 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15080 |
nM |
25001482 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
24906510 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
330 |
nM |
24906510 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
24906510 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4.1 |
ug/ml |
25017036 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12.1 |
ug/ml |
25017036 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4.8 |
ug/ml |
25017036 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5.7 |
ug/ml |
25017036 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2.9 |
ug/ml |
25017036 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11640 |
nM |
24583355 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29140 |
nM |
24583355 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
24870 |
nM |
24583355 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29500 |
nM |
24657568 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
3390 |
nM |
24657568 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
5750 |
nM |
24657568 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6610 |
nM |
24657568 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
7940 |
nM |
24657568 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
18600 |
nM |
24657568 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
85100 |
nM |
24657568 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
126000 |
nM |
24657568 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3550 |
nM |
24657568 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
IC50 |
= |
60300 |
nM |
24657568 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
30210 |
nM |
24934992 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
28760 |
nM |
24934992 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50000 |
nM |
25124114 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5620 |
nM |
25442303 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14260 |
nM |
25442303 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8130 |
nM |
25442303 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
EC50 |
> |
50000 |
nM |
25198997 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
16300 |
nM |
25198997 |
NPT2 |
Others |
Unspecified |
|
EC50 |
> |
50000 |
nM |
25198997 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
38060 |
nM |
25198997 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
48700 |
nM |
25198997 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50/EC50 |
= |
0.97 |
|
25198997 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50/EC50 |
= |
2.98 |
|
25198997 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50/EC50 |
= |
1.2 |
|
25198997 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16300 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14600 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1300 |
nM |
25176329 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
25176329 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
70.3 |
% |
25247772 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
26.2 |
ug |
25247772 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15400 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15300 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15600 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16800 |
nM |
25261825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10810 |
nM |
25180925 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8930 |
nM |
25180925 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
7690 |
nM |
25180925 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
870 |
nM |
25180925 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2600 |
nM |
25435471 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
25435471 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
330 |
nM |
25435471 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
67700 |
nM |
25164762 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
59900 |
nM |
25164762 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
17850 |
nM |
25164762 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
51640 |
nM |
25164762 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
53520 |
nM |
25164762 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27010 |
nM |
25164762 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
78.43 |
% |
25203783 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
6690 |
nM |
25203783 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
72.25 |
% |
25203783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3540 |
nM |
25203783 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
80.36 |
% |
25203783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2230 |
nM |
25203783 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
56.06 |
% |
25203783 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4610 |
nM |
25203783 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
40 |
nM |
25259515 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10 |
nM |
25259515 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
46930 |
nM |
25151580 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
44040 |
nM |
25151580 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
29980 |
nM |
25151580 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
35340 |
nM |
25151580 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40210 |
nM |
25151580 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
56000 |
nM |
25151580 |
NPT2 |
Others |
Unspecified |
|
TC50 |
= |
21.68 |
nM |
25461891 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6560 |
nM |
25554922 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3710 |
nM |
25554922 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
5180 |
nM |
25554922 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11610 |
nM |
25655718 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9120 |
nM |
25655718 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
8430 |
nM |
25655718 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1430 |
nM |
25655718 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
5820 |
nM |
25870131 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7510 |
nM |
25870131 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
6370 |
nM |
25870131 |
NPT2 |
Others |
Unspecified |
|
TC50 |
= |
6.12 |
ug/ml |
25600408 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12240 |
nM |
25707012 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
10720 |
nM |
25707012 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15670 |
nM |
25707012 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
20400 |
nM |
25707012 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22540 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
21150 |
nM |
25644674 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
4690 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6000 |
nM |
25644674 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
25080 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38920 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20460 |
nM |
25644674 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
3230 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.94 |
|
25644674 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.28 |
|
25644674 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
1920 |
nM |
25644674 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
3850 |
nM |
25644674 |
NPT17 |
Organism |
Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
= |
3850 |
nM |
25644674 |
NPT17 |
Organism |
Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
= |
1920 |
nM |
25644674 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
7690 |
nM |
25644674 |
NPT17 |
Organism |
Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
= |
960 |
nM |
25644674 |
NPT17 |
Organism |
Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
= |
480 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5500 |
nM |
25752525 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
GI50 |
= |
4300 |
nM |
25752525 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
15000 |
nM |
25752525 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
47000 |
nM |
25752525 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
GI50 |
= |
49000 |
nM |
25752525 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3580 |
nM |
25812966 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4870 |
nM |
25812966 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6120 |
nM |
25812966 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5860 |
nM |
25812966 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
36638 |
nM |
25675144 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
910 |
nM |
25675144 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
47390 |
nM |
25841196 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
38230 |
nM |
25841196 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
31980 |
nM |
25841196 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40570 |
nM |
25841196 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
44100 |
nM |
25841196 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
46150 |
nM |
25841196 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27340 |
nM |
25841196 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
56370 |
nM |
25841196 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
40940 |
nM |
25841199 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29580 |
nM |
25841199 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37560 |
nM |
25841199 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
30790 |
nM |
25841199 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
36340 |
nM |
25841199 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
58740 |
nM |
25841199 |
NPT3891 |
Cell Line |
S180 |
Mus musculus |
TGI |
= |
52.54 |
% |
25825934 |
NPT3891 |
Cell Line |
S180 |
Mus musculus |
TGI |
= |
96.92 |
% |
25825934 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
25969171 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
70.3 |
% |
25984840 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
26.2 |
ug |
25984840 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
69.1 |
% |
25958244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
27.43 |
ug |
25958244 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22360 |
nM |
25959813 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
40380 |
nM |
25959813 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19910 |
nM |
25959813 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8930 |
nM |
25959813 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9560 |
nM |
25959813 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2050 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2080 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2930 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2970 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3940 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3950 |
nM |
20930123 |
NPT3123 |
Cell Line |
DAN-G |
Homo sapiens |
IC50 |
= |
4380 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2.4 |
|
20930123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
33200 |
nM |
20930123 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2.5 |
|
20930123 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
4.3 |
|
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
26.4 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
45.4 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
54.6 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
53 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
16.4 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
31.2 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
39.1 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
44.9 |
% |
20930123 |
NPT1027 |
Individual Protein |
Multidrug resistance-associated protein 5 |
Homo sapiens |
Activity |
= |
59.2 |
% |
20930123 |
NPT1027 |
Individual Protein |
Multidrug resistance-associated protein 5 |
Homo sapiens |
FC |
= |
2.1 |
|
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
36 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
80 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
94 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
10 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
27 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
63 |
% |
20930123 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
66 |
% |
20930123 |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
16077.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
707.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
45312.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
1000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
10000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
20000 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
3161.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10682.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
|
1962.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4491.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1899.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14329 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
63437.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
28166.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6343.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
2238.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
14125.4 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
77280 |
nM |
25466196 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38880 |
nM |
25466196 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
34480 |
nM |
25466196 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
5200 |
nM |
25919052 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
4400 |
nM |
25919052 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3700 |
nM |
25919052 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5800 |
nM |
25919052 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
25919052 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8400 |
nM |
25919052 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
540 |
nM |
26001344 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
18000 |
nM |
26001344 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
330 |
nM |
26001344 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4900 |
nM |
10.1039/C4MD00209A |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4710 |
nM |
10.1039/C4MD00209A |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
860 |
nM |
10.1039/C4MD00209A |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TGI |
= |
37.3 |
% |
25937236 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10070 |
nM |
26227777 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
16420 |
nM |
26227777 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6300 |
nM |
26227777 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14150 |
nM |
26227777 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
44050 |
nM |
26259802 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
40340 |
nM |
26259802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1500 |
nM |
26259802 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
5580 |
nM |
26259802 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11500 |
nM |
26259802 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
26222449 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4900 |
nM |
26222449 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
26222449 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2130 |
nM |
26231080 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2360 |
nM |
26231080 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4600 |
nM |
26231080 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
15260 |
nM |
26231080 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
6072 |
nM |
26301558 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8317 |
nM |
26301558 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7244 |
nM |
26301558 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5012 |
nM |
26301558 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30700 |
nM |
10.1039/C4MD00306C |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
10.1039/C4MD00306C |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Inhibition |
= |
68.2 |
% |
26312434 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
68.2 |
% |
26312434 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
> |
150000 |
nM |
26320625 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
26320625 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
150000 |
nM |
26320625 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
700000 |
nM |
26320625 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
78.66 |
% |
26364944 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
64.47 |
% |
26364944 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
66500 |
nM |
26291038 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
790 |
nM |
26291038 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11670 |
nM |
26291038 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
55200 |
nM |
26291038 |
NPT2788 |
Cell Line |
3T3 |
Mus musculus |
IC50 |
= |
28300 |
nM |
26291038 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
15830 |
nM |
26413725 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
22630 |
nM |
26363869 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46830 |
nM |
26363869 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22280 |
nM |
26363869 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
19390 |
nM |
26363869 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.3 |
ug/ml |
26383125 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.4 |
ug/ml |
26383125 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
1 |
ug/ml |
26383125 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.3 |
ug/ml |
26383125 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
0.7 |
ug/ml |
26383125 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.4 |
ug/ml |
26383125 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
0.9 |
ug/ml |
26383125 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19820 |
nM |
26413726 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
45430 |
nM |
26413726 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68280 |
nM |
26413726 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
39170 |
nM |
26413726 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7590 |
nM |
26413726 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10.41 |
ug/ml |
26546214 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17.41 |
ug/ml |
26546214 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
35.99 |
ug/ml |
26546214 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
GI50 |
= |
1500 |
nM |
26539626 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
2200 |
nM |
26539626 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
2.60E-05 |
ug |
26638042 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
68.2 |
% |
26638042 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
42500 |
nM |
26595184 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11900 |
nM |
26595184 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
6760 |
nM |
26595184 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15190 |
nM |
26595184 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25900 |
nM |
26595184 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.83 |
|
26595184 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
32720 |
nM |
10.1039/C5MD00163C |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
10.1039/C5MD00163C |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
40180 |
nM |
10.1039/C5MD00163C |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
520 |
nM |
26725029 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
64 |
nM |
26725029 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
83 |
% |
26725029 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
60 |
% |
26725029 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
10.1039/C5MD00240K |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14200 |
nM |
10.1039/C5MD00240K |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15900 |
nM |
10.1039/C5MD00240K |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9200 |
nM |
10.1039/C5MD00240K |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5620 |
nM |
26786698 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
17210 |
nM |
26786698 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8130 |
nM |
26786698 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
2980 |
nM |
26786698 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
90 |
nM |
26617970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
790 |
nM |
26617970 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
> |
100000 |
nM |
26617970 |
NPT2788 |
Cell Line |
3T3 |
Mus musculus |
IC50 |
= |
28300 |
nM |
26617970 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
26629861 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
113.6 |
|
26629861 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
26629861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3520 |
nM |
26703795 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
90.9 |
|
26629861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
26629861 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
124 |
|
26629861 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
26629861 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
75.7 |
|
26629861 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
136400 |
nM |
26629861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
32180 |
nM |
26703795 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
43710 |
nM |
26703795 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
24500 |
nM |
26703795 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5530 |
nM |
26703795 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
5.42 |
% |
26703795 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
91.11 |
% |
26703795 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
3.48 |
% |
26703795 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24580 |
nM |
26706349 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
31330 |
nM |
26706349 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30230 |
nM |
26706349 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22430 |
nM |
26706349 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
35520 |
nM |
26706349 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
10.1039/C5MD00289C |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
500 |
nM |
10.1039/C5MD00289C |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14800 |
nM |
26727215 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
14800 |
nM |
26727215 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
14800 |
nM |
26727215 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
1862000 |
nM |
26727215 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
> |
1862000 |
nM |
26727215 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
TGI |
> |
1862000 |
nM |
26727215 |
NPT2 |
Others |
Unspecified |
|
CC50 |
> |
2512000 |
nM |
26727215 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
CC50 |
> |
2512000 |
nM |
26727215 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
CC50 |
> |
2512000 |
nM |
26727215 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3610 |
nM |
26735909 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3470 |
nM |
26735909 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1440 |
nM |
26735909 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
26606140 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6400 |
nM |
26606140 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
400 |
nM |
26606140 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
8700 |
nM |
26606140 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
26606140 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
33000 |
nM |
10.1039/C5MD00382B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
46000 |
nM |
10.1039/C5MD00382B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37000 |
nM |
10.1039/C5MD00382B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38000 |
nM |
10.1039/C5MD00382B |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
20000 |
nM |
10.1039/C5MD00382B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29000 |
nM |
10.1039/C5MD00382B |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
26140 |
nM |
26922223 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
26180 |
nM |
26922223 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27430 |
nM |
26922223 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38300 |
nM |
26922223 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
> |
50000 |
nM |
26922223 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
49020 |
nM |
26922223 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
82270 |
nM |
26873416 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
54820 |
nM |
26873416 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
32310 |
nM |
26873416 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
41620 |
nM |
26873416 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38910 |
nM |
26873416 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
7030 |
nM |
26883149 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
2210 |
nM |
26883149 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
3350 |
nM |
26883149 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
50000 |
nM |
26922233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27800 |
nM |
26922233 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
> |
50000 |
nM |
26922233 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
25000 |
nM |
26922233 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6300 |
nM |
26922233 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
> |
50000 |
nM |
26922233 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
41100 |
nM |
26922233 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
6800 |
nM |
26922233 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
26731300 |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
6200 |
nM |
26731300 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4900 |
nM |
26731300 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
900 |
nM |
26731300 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
79 |
% |
26854375 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
82 |
% |
26854375 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
92 |
% |
26854375 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
89 |
% |
26854375 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
26854375 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
26854375 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
26854375 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1700 |
nM |
26854375 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
56960 |
nM |
27017265 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
222600 |
nM |
27017265 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
174500 |
nM |
27017265 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6530 |
nM |
27073055 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
4840 |
nM |
27073055 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6230 |
nM |
27073055 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
6600 |
nM |
27073055 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7020 |
nM |
27073055 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.13 |
|
27073055 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.45 |
|
27073055 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.08 |
|
27073055 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.06 |
|
27073055 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.54 |
|
27073055 |
NPT3792 |
Cell Line |
143B |
Homo sapiens |
IC50 |
= |
13010 |
nM |
27073055 |
NPT3792 |
Cell Line |
143B |
Homo sapiens |
IC50 |
= |
16310 |
nM |
27073055 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
89200 |
nM |
26714048 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68300 |
nM |
26714048 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
126400 |
nM |
26714048 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
26714048 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
34270 |
nM |
26883148 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
49720 |
nM |
26883148 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10530 |
nM |
26883148 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
47090 |
nM |
26883148 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
42780 |
nM |
26883148 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17530 |
nM |
27133593 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
25170 |
nM |
27133593 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
15470 |
nM |
27133593 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
IC50 |
= |
24690 |
nM |
27133593 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
27133593 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
21580 |
nM |
27133593 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
30 |
nM |
27156770 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
27156770 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18250 |
nM |
27081742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
219600 |
nM |
27081742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
49298000 |
nM |
27081742 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
27092413 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2760 |
nM |
27092413 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3980 |
nM |
27092413 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3650 |
nM |
27092413 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
16150 |
nM |
27092413 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7610 |
nM |
27105028 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5610 |
nM |
27105028 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
3260 |
nM |
27105028 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1250 |
nM |
27105028 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3170 |
nM |
27105028 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
44050 |
nM |
27189676 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22990 |
nM |
27189676 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
40340 |
nM |
27189676 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
5180 |
nM |
27189676 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11500 |
nM |
27189676 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11100 |
nM |
27234893 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8510 |
nM |
27210438 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15480 |
nM |
27210438 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
47180 |
nM |
27210438 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
32270 |
nM |
27210438 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10.89 |
ug/ml |
27262600 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10.5 |
ug/ml |
27262600 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14.53 |
ug/ml |
27262600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10.8 |
ug/ml |
27262600 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10.72 |
ug/ml |
27262600 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
9.23 |
ug/ml |
27262600 |
NPT2 |
Others |
Unspecified |
|
TC50 |
= |
21.68 |
nM |
10.1039/C6MD00008H |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
55740 |
nM |
10.1039/C6MD00061D |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22620 |
nM |
10.1039/C6MD00061D |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8820 |
nM |
10.1039/C6MD00061D |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
21470 |
nM |
10.1039/C6MD00061D |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12230 |
nM |
10.1039/C6MD00061D |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
24600 |
nM |
27128180 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
35410 |
nM |
27128180 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46830 |
nM |
27128180 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
30410 |
nM |
27128180 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
27311895 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5800 |
nM |
27311895 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
5200 |
nM |
27311895 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
57170 |
nM |
27287368 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
57040 |
nM |
27287368 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68710 |
nM |
27287368 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
46830 |
nM |
27287368 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
39860 |
nM |
27448774 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
72070 |
nM |
27448774 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
35910 |
nM |
27448774 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
98000 |
nM |
27448774 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15380 |
nM |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
74.3 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
15.3 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
11.7 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
93.2 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
5.2 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
1 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
0.6 |
% |
27448774 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
FC |
= |
4.2 |
|
27448774 |