Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
900 |
nM |
10841789 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
2400 |
nM |
10841789 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
300 |
nM |
15177438 |
NPT1851 |
Cell Line |
Col2 |
Homo sapiens |
IC50 |
= |
520 |
nM |
15177438 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
690 |
nM |
15177438 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
25 |
nM |
12182872 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.029 |
nM |
1875350 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.031 |
nM |
1875350 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.055 |
nM |
1875350 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
ED50 |
= |
0.032 |
nM |
1875350 |
NPT3958 |
Cell Line |
MLM |
|
ED50 |
= |
0.13 |
nM |
1875350 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
620 |
nM |
11720862 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
750 |
nM |
11720862 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.005 |
ug |
8709115 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
69 |
nM |
3806589 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
5.6 |
|
3806589 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
TD50 |
= |
0.02 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TD50 |
= |
0.17 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
TD50 |
= |
0.02 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT4464 |
Cell Line |
L1210/Adr |
Mus musculus |
TD50 |
= |
0.3 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TD50 |
= |
0.2 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
TD50 |
= |
0.05 |
ug/ml |
10.1016/0960-894X(96)00395-2 |
NPT1868 |
Cell Line |
L1210 (1565) |
|
IC50 |
= |
22 |
nM |
10.1016/0960-894X(95)00067-4 |
NPT1868 |
Cell Line |
L1210 (1565) |
|
IC50 |
= |
315 |
nM |
10.1016/0960-894X(95)00067-4 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
14.1 |
|
10.1016/0960-894X(95)00067-4 |
NPT5499 |
Cell Line |
H2981 cell line |
|
IC50 |
= |
700 |
nM |
8464046 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
26 |
nM |
10411474 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
1000 |
nM |
10411474 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
91000 |
nM |
10411474 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
10411474 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
17 |
nM |
10411474 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
IC50 |
= |
6.3 |
nM |
10411474 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
10411474 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
78 |
nM |
10411474 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
5370 |
ug/ml |
9207950 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.5 |
nM |
7086816 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
7086816 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.03 |
nM |
3806576 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
14971899 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
10000 |
nM |
14971899 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
300 |
nM |
14971899 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
150 |
nM |
14971899 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.257 |
ug/ml |
8027979 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.000104 |
ug/ml |
8027979 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.0176 |
ug/ml |
8027979 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.000153 |
ug/ml |
8027979 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
60 |
nM |
1354750 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
6000 |
nM |
1354750 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
200 |
nM |
1995877 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
1220 |
nM |
1995877 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
40 |
nM |
1995877 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
4200 |
nM |
1995877 |
NPT5500 |
Cell Line |
KBM-3 cell line |
|
IC50 |
= |
26 |
nM |
1995877 |
NPT5501 |
Cell Line |
KBM-3/DOX cell line |
|
IC50 |
= |
490 |
nM |
1995877 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1990 |
nM |
9873387 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1770 |
nM |
9873387 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
4150 |
nM |
9873387 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
0.17 |
ug/ml |
15013011 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
0.31 |
ug/ml |
15013011 |
NPT4705 |
Cell Line |
MG-22A |
Mus musculus |
IC50 |
< |
0.001 |
ug/ml |
15013011 |
NPT4705 |
Cell Line |
MG-22A |
Mus musculus |
IC50 |
= |
0.73 |
ug/ml |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.001 |
ug/ml |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
< |
0.001 |
ug/ml |
15013011 |
NPT3908 |
Cell Line |
N2a |
Mus musculus |
IC50 |
= |
0.004 |
ug/ml |
15013011 |
NPT3908 |
Cell Line |
N2a |
Mus musculus |
IC50 |
< |
0.001 |
ug/ml |
15013011 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
7 |
% |
15013011 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
28 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
11 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
16 |
% |
15013011 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
35 |
% |
15013011 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Inhibition |
= |
37 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
65 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
75 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
25 |
% |
15013011 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
70 |
% |
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
83 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
40 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
90 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
114 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
60 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
39 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
81 |
|
15013011 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
130 |
|
15013011 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
26 |
nM |
11123989 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
11123989 |
NPT571 |
Cell Line |
A2780cisR |
Homo sapiens |
IC50 |
= |
17 |
nM |
11123989 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
IC50 |
= |
6.3 |
nM |
11123989 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
IC50 |
= |
450 |
nM |
11123989 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
78 |
nM |
11123989 |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
640 |
nM |
10698436 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
10698436 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
640 |
nM |
10698436 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
220 |
nM |
10698436 |
NPT5502 |
Cell Line |
Human melanoma cell line |
|
IC50 |
= |
280 |
nM |
10698436 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10698436 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
20 |
nM |
10698436 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
> |
900 |
nM |
10698436 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
50 |
nM |
10698436 |
NPT1386 |
Protein Family |
Adrenergic receptor beta |
Homo sapiens |
Activity |
= |
-4.61 |
|
10.1016/S0960-894X(97)00046-2 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
390 |
nM |
9876111 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
9876111 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
135000 |
nM |
9876111 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.066 |
nM |
7086818 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
100 |
nM |
10476861 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10476861 |
NPT1307 |
Cell Line |
Calu-1 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
10476861 |
NPT5503 |
Cell Line |
MEL-AC cell line |
|
IC50 |
= |
1200 |
nM |
10476861 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
10476861 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
39400 |
nM |
10476861 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
70 |
nM |
10.1016/0960-894X(96)00167-9 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10.1016/0960-894X(96)00167-9 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
150 |
nM |
10.1016/0960-894X(96)00167-9 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
60 |
nM |
10.1016/0960-894X(96)00167-9 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
14980672 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
25 |
nM |
14980672 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
7 |
nM |
14980672 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
7 |
nM |
14980672 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.08 |
ug/ml |
10.1016/0960-894X(94)80019-7 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.000153 |
ug/ml |
10.1016/0960-894X(94)80019-7 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.0138 |
ug/ml |
10.1016/0960-894X(94)80019-7 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.000558 |
ug/ml |
10.1016/0960-894X(94)80019-7 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
7.2 |
nM |
10.1016/S0960-894X(96)00486-6 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
35 |
nM |
10.1016/S0960-894X(96)00486-6 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
60 |
nM |
9526570 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
6000 |
nM |
9526570 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
IC50 |
= |
65 |
nM |
9526570 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
14 |
nM |
9526570 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.016 |
ug/ml |
11055343 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.01 |
ug/ml |
11055343 |
NPT2831 |
Cell Line |
P388/S |
Mus musculus |
IC50 |
= |
19 |
nM |
8544183 |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
360 |
nM |
8544183 |
NPT5504 |
Cell Line |
UACC-375 |
|
IC50 |
= |
112 |
nM |
8960558 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
35 |
nM |
8960558 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
35 |
nM |
8960558 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
3884 |
nM |
8960558 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
28 |
nM |
8960558 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
8960558 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
53 |
nM |
8960558 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
130 |
nM |
8960558 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22 |
nM |
8960558 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
10 |
nM |
11454467 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
27.3 |
nM |
11806724 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
3874 |
nM |
11806724 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
20.1 |
nM |
11806724 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
319.3 |
nM |
11806724 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
0.58 |
ug/ml |
9876113 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
53 |
ug/ml |
9876113 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
7.2 |
nM |
10.1016/S0960-894X(97)00071-1 |
NPT4452 |
Cell Line |
CCD 19Lu |
Homo sapiens |
IC50 |
= |
2 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.003 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT4453 |
Cell Line |
Lu-99 cell line |
|
IC50 |
= |
0.002 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
10.1016/S0960-894X(97)00071-1 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
33 |
nM |
10.1016/0960-894X(96)00457-X |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
IC50 |
= |
21 |
nM |
10.1016/0960-894X(96)00457-X |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
7010 |
nM |
10.1016/0960-894X(96)00457-X |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.04 |
ug/ml |
8496904 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.02 |
ug/ml |
8496904 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.9 |
ug/ml |
8496904 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.06 |
ug/ml |
8496904 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
8496904 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
8496904 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
8496904 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
52 |
nM |
12431060 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
620 |
nM |
12431060 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
20 |
nM |
14971893 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
GI50 |
= |
20 |
nM |
14971893 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
4400 |
nM |
14971893 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
2400 |
nM |
14971893 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
GI50 |
= |
1100 |
nM |
14971893 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
3100 |
nM |
14971893 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
70 |
nM |
14971893 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
GI50 |
= |
3500 |
nM |
14971893 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
3100 |
nM |
14971893 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
10 |
nM |
14971893 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
2400 |
nM |
14971893 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
10 |
nM |
14971893 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
30 |
nM |
14971893 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
830 |
nM |
10.1016/0960-894X(96)00230-2 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
331 |
nM |
7853331 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
42 |
nM |
7853331 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
72 |
nM |
7853331 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
36 |
nM |
7853331 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
= |
5650 |
nM |
7853331 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.00399 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.42 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0243 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.00226 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.0349 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
0.00136 |
ug/ml |
10.1016/0960-894X(95)00182-S |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
26 |
nM |
11563932 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.09 |
ug/ml |
9873721 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
2.15 |
ug/ml |
9873721 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
970 |
nM |
14643344 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1170 |
nM |
14643344 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
4780 |
nM |
14643344 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
14643344 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10 |
nM |
12852768 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
1720 |
nM |
12852768 |
NPT5505 |
Cell Line |
Human lung LXF 629L tumor cell line |
|
IC50 |
= |
70 |
nM |
12852768 |
NPT731 |
Cell Line |
LXFL 529 |
Homo sapiens |
IC50 |
= |
30 |
nM |
12852768 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
50 |
nM |
12852768 |
NPT5506 |
Cell Line |
MAXF401 cell line |
|
IC50 |
= |
10 |
nM |
12852768 |
NPT5184 |
Cell Line |
RXF 944 |
Homo sapiens |
IC50 |
= |
60 |
nM |
12852768 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
26 |
nM |
8057291 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
IC50 |
= |
10 |
nM |
8057291 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
43 |
nM |
7853345 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
6000 |
nM |
7853345 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.004 |
ug/ml |
15056007 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
8.65 |
|
12570378 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431048 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431048 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
10 |
nM |
12431048 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
12431048 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
40 |
nM |
12431048 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431048 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431048 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431048 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431048 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
60 |
nM |
12431048 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
90 |
nM |
12431048 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
50 |
nM |
12431048 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431048 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
120 |
nM |
12431048 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
40 |
nM |
12431048 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431048 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
150 |
nM |
12431048 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431048 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
10 |
nM |
12431048 |
NPT5507 |
Cell Line |
CRL-7065 cell line |
|
IC50 |
= |
500 |
nM |
12431048 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
90 |
nM |
12431048 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
40 |
nM |
12431048 |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
CC50 |
= |
20 |
nM |
12431048 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
< |
0.5 |
ug/ml |
10.1016/0960-894X(95)00338-T |
NPT789 |
Cell Line |
SNU-354 |
Homo sapiens |
IC50 |
< |
0.5 |
ug/ml |
10.1016/0960-894X(95)00338-T |
NPT5508 |
Cell Line |
SNU-C4 |
Homo sapiens |
IC50 |
< |
0.5 |
ug/ml |
10.1016/0960-894X(95)00338-T |
NPT4266 |
Individual Protein |
NADH-ubiquinone oxidoreductase chain 4 |
Homo sapiens |
Activity |
= |
0.15 |
units ml-1 |
8421288 |
NPT5504 |
Cell Line |
UACC-375 |
|
IC50 |
= |
112 |
nM |
10956214 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
35 |
nM |
10956214 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
35 |
nM |
10956214 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
3884 |
nM |
10956214 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
28 |
nM |
10956214 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
10956214 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
53 |
nM |
10956214 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
130 |
nM |
10956214 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22 |
nM |
10956214 |
NPT568 |
Individual Protein |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
1322986 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
20 |
nM |
1322986 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.39 |
ug/ml |
12620075 |
NPT4590 |
Cell Line |
EL4 |
Mus musculus |
IC50 |
= |
0.67 |
ug/ml |
12620075 |
NPT2609 |
Cell Line |
BeWo |
Homo sapiens |
IC50 |
= |
6.24 |
ug/ml |
12620075 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
12620075 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
12620075 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5 |
nM |
8831755 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
357 |
nM |
8831755 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
63 |
nM |
8831755 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
56 |
nM |
8831755 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
43 |
nM |
8182705 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
> |
10000 |
nM |
8182705 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
180 |
nM |
8182705 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
IC50 |
> |
75000 |
nM |
8176712 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
4 |
nM |
9873661 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
9873661 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
100 |
nM |
9873661 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
35 |
nM |
9873661 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
ID50 |
= |
0.1 |
nM |
1548681 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ID50 |
= |
0.02 |
nM |
1548681 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
ID50 |
= |
0.01 |
nM |
1548681 |
NPT2 |
Others |
Unspecified |
|
ID50 |
= |
0.01 |
nM |
1548681 |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
ID50 |
= |
0.01 |
nM |
1548681 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
510 |
nM |
14971909 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
1700 |
nM |
14971909 |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
IC50 |
= |
79.4 |
nM |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
2752.5 |
nM |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
IC50 |
= |
368.4 |
nM |
10.1016/0960-894X(95)00300-I |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
7.5 |
|
10.1016/0960-894X(95)00300-I |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
Activity |
= |
66.8 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT1886 |
Cell Line |
J774 |
Mus musculus |
Activity |
= |
153.4 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
52.8 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
87 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
69.6 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT1597 |
Cell Line |
J774.2 |
|
Activity |
= |
130.5 |
pM of drug (10e6*cells)-1 |
10.1016/0960-894X(95)00300-I |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
230 |
nM |
10411476 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
IC50 |
= |
20 |
nM |
10411476 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
10 |
nM |
10411476 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
100 |
nM |
10411476 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
30 |
nM |
10411476 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10411476 |
NPT913 |
Cell Line |
CHO-K1 |
Cricetulus griseus |
IC50 |
= |
400 |
nM |
10411476 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
50 |
nM |
10411476 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
200 |
nM |
10411476 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
400 |
nM |
10411476 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10411476 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
10 |
nM |
10411476 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
MIC |
> |
2500 |
nM |
10411476 |
NPT186 |
Organism |
Candida tropicalis |
Candida tropicalis |
MIC |
> |
2500 |
nM |
10411476 |
NPT188 |
Organism |
Candida parapsilosis |
Candida parapsilosis |
MIC |
> |
2500 |
nM |
10411476 |
NPT85 |
Organism |
Filobasidiella neoformans |
Cryptococcus neoformans |
MIC |
> |
2500 |
nM |
10411476 |
NPT3173 |
Organism |
Arthroderma benhamiae |
Arthroderma benhamiae |
MIC |
> |
2500 |
nM |
10411476 |
NPT87 |
Organism |
Aspergillus fumigatus |
Aspergillus fumigatus |
MIC |
> |
2500 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
40 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
500 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
400 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
650 |
nM |
10411476 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
60 |
nM |
10411476 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CC50 |
= |
40 |
nM |
10411476 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
CC50 |
= |
90 |
nM |
10411476 |
NPT347 |
Cell Line |
Lymphoblastoid cells |
Homo sapiens |
CC50 |
= |
60 |
nM |
10411476 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.8 |
ug/ml |
9873640 |
NPT5509 |
Cell Line |
BRO melanoma cell line |
|
IC50 |
= |
0.2 |
ug/ml |
9873640 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
9873640 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.5 |
ug/ml |
9873640 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
9873640 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ID50 |
= |
0.01 |
ug/ml |
10602713 |
NPT2046 |
Cell Line |
EVSA-T |
Homo sapiens |
ID50 |
= |
0.008 |
ug/ml |
10602713 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
ID50 |
= |
0.011 |
ug/ml |
10602713 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
ID50 |
= |
0.06 |
ug/ml |
10602713 |
NPT2 |
Others |
Unspecified |
|
ID50 |
= |
0.016 |
ug/ml |
10602713 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ID50 |
= |
0.09 |
ug/ml |
10602713 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
ID50 |
= |
0.199 |
ug/ml |
10602713 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
0.0064 |
ug/ml |
11551772 |
NPT5193 |
Cell Line |
RPTEC |
Homo sapiens |
GI50 |
= |
0.072 |
ug/ml |
11551772 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
0.029 |
ug/ml |
11551772 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.0046 |
ug/ml |
11551772 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
0.092 |
ug/ml |
11551772 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
0.071 |
ug/ml |
11551772 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
0.073 |
ug/ml |
11551772 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
0.059 |
ug/ml |
11551772 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
23 |
nM |
11755363 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
56 |
nM |
11755363 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
13 |
nM |
11755363 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
16700 |
nM |
11755363 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
100 |
nM |
11606141 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
5000 |
nM |
11606141 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
100 |
nM |
11606141 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
50 |
nM |
11606141 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
7000 |
nM |
11606141 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
11606141 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
11606141 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
20 |
nM |
11606141 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
> |
10000 |
nM |
11606141 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
50 |
nM |
11606141 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
80 |
nM |
11606141 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
8 |
nM |
11606141 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
80 |
nM |
11606141 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
60 |
nM |
11606141 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
140 |
nM |
11606141 |
NPT933 |
Cell Line |
U373 MG |
Homo sapiens |
IC50 |
= |
10 |
nM |
11606141 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
11606141 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.0346 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.43 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0896 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.0335 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.33 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT5510 |
Cell Line |
PAC-2 cell line |
|
ED50 |
= |
0.031 |
ug/ml |
10.1016/0960-894X(95)00309-H |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.9 |
nM |
1613753 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.1 |
nM |
1613753 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
5.5 |
nM |
1613753 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
ED50 |
= |
3.2 |
nM |
1613753 |
NPT3958 |
Cell Line |
MLM |
|
ED50 |
= |
1.3 |
nM |
1613753 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
15 |
nM |
11806725 |
NPT4463 |
Cell Line |
LL |
|
IC50 |
= |
22 |
nM |
11806725 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9.6 |
nM |
11806725 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
4.39 |
|
11806725 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
12.7 |
|
11806725 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
27 |
nM |
11806725 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
137 |
nM |
11806725 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
EC50 |
= |
2500 |
nM |
10.1016/S0960-894X(96)00243-0 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.00844 |
ug/ml |
10.1016/0960-894X(95)00004-D |
NPT5511 |
Cell Line |
MCF9 |
Homo sapiens |
ED50 |
= |
0.0673 |
ug/ml |
10.1016/0960-894X(95)00004-D |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0261 |
ug/ml |
10.1016/0960-894X(95)00004-D |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
7.8 |
nM |
10479282 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
15.6 |
nM |
10479282 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2474 |
nM |
10479282 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
52.8 |
nM |
10479282 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
102.8 |
nM |
10479282 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
56.4 |
nM |
10479282 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
231.2 |
nM |
10479282 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
19.9 |
nM |
10479282 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
466 |
nM |
10479282 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
2.7 |
|
15012986 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
5.4 |
|
15012986 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
60 |
nM |
14761187 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1800 |
nM |
14761187 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3000 |
nM |
14761187 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
400 |
nM |
14761187 |
NPT5512 |
Cell Line |
TRAMP-C1A |
Mus musculus |
IC50 |
= |
75.9 |
nM |
14971910 |
NPT5513 |
Cell Line |
C2D cell line |
|
IC50 |
= |
46.5 |
nM |
14971910 |
NPT5514 |
Cell Line |
C2G cell line |
|
IC50 |
= |
28.7 |
nM |
14971910 |
NPT5515 |
Cell Line |
TRAMP-C2H |
Mus musculus |
IC50 |
= |
30.3 |
nM |
14971910 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1016/S0960-894X(01)80594-1 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
40 |
nM |
10.1016/S0960-894X(01)81264-6 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10.1016/S0960-894X(01)81264-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
100 |
nM |
10.1016/S0960-894X(01)81264-6 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.028 |
ug/ml |
10612603 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
2.97 |
ug/ml |
10612603 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.88 |
ug/ml |
10612603 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.339 |
ug/ml |
10612603 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.988 |
ug/ml |
10612603 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.16 |
ug/ml |
8632402 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.76 |
ug/ml |
8632402 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.9 |
ug/ml |
8632402 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.87 |
ug/ml |
8632402 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
6.37 |
ug/ml |
8632402 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.63 |
ug/ml |
8632402 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.00021 |
ug/ml |
11551759 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.0058 |
ug/ml |
11551759 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0013 |
ug/ml |
11551759 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.00046 |
ug/ml |
11551759 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.00024 |
ug/ml |
11551759 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
0.00018 |
ug/ml |
11551759 |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Survival |
= |
0.37 |
|
6685770 |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Survival |
< |
0.1 |
|
6685770 |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Survival |
= |
0.18 |
|
6685770 |
NPT5516 |
Cell Line |
EBV-positive nasopharyngealcell lines |
|
Survival |
= |
0.69 |
|
6685770 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.26 |
ug/ml |
8627602 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.0262 |
ug/ml |
8627602 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.194 |
ug/ml |
8627602 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0494 |
ug/ml |
8627602 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.0663 |
ug/ml |
8627602 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.287 |
ug/ml |
8627602 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
0.034 |
ug/ml |
8627602 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
300 |
nM |
9548820 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
10000 |
nM |
9548820 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.06 |
nM |
3806575 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Ratio |
= |
0.96 |
|
3806575 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
0.27 |
ug/ml |
10.1016/0960-894X(96)00156-4 |
NPT789 |
Cell Line |
SNU-354 |
Homo sapiens |
IC50 |
= |
0.54 |
ug/ml |
10.1016/0960-894X(96)00156-4 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.15 |
ug/ml |
10.1016/0960-894X(96)00156-4 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
37.57 |
ug/ml |
10.1016/0960-894X(96)00156-4 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
200 |
ug/ml |
3018245 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
20 |
ug/ml |
3018245 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
10 |
ug/ml |
3018245 |
NPT17 |
Organism |
Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
< |
5 |
ug/ml |
3018245 |
NPT1228 |
Organism |
Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
< |
5 |
ug/ml |
3018245 |
NPT314 |
Organism |
Bacillus cereus |
Bacillus cereus |
MIC |
= |
10 |
ug/ml |
3018245 |
NPT79 |
Organism |
Bacillus subtilis |
Bacillus subtilis |
MIC |
= |
20 |
ug/ml |
3018245 |
NPT4068 |
Organism |
Corynebacterium diphtheriae |
Corynebacterium diphtheriae |
MIC |
= |
20 |
ug/ml |
3018245 |
NPT5504 |
Cell Line |
UACC-375 |
|
IC50 |
= |
112 |
nM |
8648600 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
35 |
nM |
8648600 |
NPT5517 |
Cell Line |
Tumor cell lines |
|
IC50 |
= |
74 |
nM |
8648600 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
35 |
nM |
8648600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
28 |
nM |
8648600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
8648600 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
53 |
nM |
8648600 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
130 |
nM |
8648600 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22 |
nM |
8648600 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
61 |
nM |
8648600 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
10151 |
|
8648600 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
TGI |
= |
120 |
% |
8648600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
250 |
nM |
8784443 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
30 |
nM |
8784443 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
IC50 |
= |
620 |
nM |
8784443 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
Inhibition |
< |
50 |
% |
11591511 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.066 |
nM |
7057426 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.05 |
nM |
3839851 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
37.84 |
nM |
15115402 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
39.56 |
nM |
15115402 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Ratio |
= |
0.9 |
|
15115402 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
28 |
nM |
8151613 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
57 |
nM |
7996544 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
7600 |
nM |
7996544 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
50 |
nM |
7996544 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
60 |
nM |
7996544 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
830 |
nM |
9733489 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.6 |
nM |
3806572 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
3806572 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
34.3 |
nM |
10377224 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
7.6 |
nM |
10377224 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ID50 |
= |
0.9 |
nM |
9022792 |
NPT5518 |
Cell Line |
MCF7-VP16 |
Homo sapiens |
ID50 |
= |
14.2 |
nM |
9022792 |
NPT5499 |
Cell Line |
H2981 cell line |
|
IC50 |
= |
500 |
nM |
7731023 |
NPT673 |
Organism |
Gallus gallus |
Gallus gallus |
ED50 |
= |
0.9 |
nM |
6302253 |
NPT673 |
Organism |
Gallus gallus |
Gallus gallus |
ED50 |
= |
2.5 |
nM |
6302253 |
NPT673 |
Organism |
Gallus gallus |
Gallus gallus |
ED50 |
= |
0.1 |
nM |
6302253 |
NPT673 |
Organism |
Gallus gallus |
Gallus gallus |
ED50 |
= |
0.18 |
nM |
6302253 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
330 |
nM |
8576914 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
36 |
nM |
8576914 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
= |
5600 |
nM |
8576914 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
160 |
|
8576914 |
NPT5504 |
Cell Line |
UACC-375 |
|
IC50 |
= |
112 |
nM |
7699715 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
35 |
nM |
7699715 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
35 |
nM |
7699715 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
3884 |
nM |
7699715 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
0.0247 |
ug/ml |
1875336 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
3.841 |
ug/ml |
1875336 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
148.7 |
|
1875336 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
179 |
nM |
12570384 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50 |
nM |
12459020 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
40 |
nM |
12459020 |
NPT731 |
Cell Line |
LXFL 529 |
Homo sapiens |
IC50 |
= |
40 |
nM |
12459020 |
NPT2842 |
Cell Line |
EMT6 |
Mus musculus |
ED50 |
= |
0.012 |
nM |
7452674 |
NPT2842 |
Cell Line |
EMT6 |
Mus musculus |
ED50 |
< |
0.0001 |
nM |
7452674 |
NPT2 |
Others |
Unspecified |
|
Ratio |
> |
120 |
|
7452674 |
NPT5519 |
Cell Line |
SBC-3 |
Homo sapiens |
IC50 |
= |
0.0112 |
ug/ml |
11311062 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.129 |
ug/ml |
11311062 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
0.275 |
ug/ml |
11311062 |
NPT3858 |
Cell Line |
KATO III stomach cancer cell lines |
|
IC50 |
= |
0.905 |
ug/ml |
11311062 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
0.00639 |
ug/ml |
11311062 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
0.0121 |
ug/ml |
11311062 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
0.136 |
ug/ml |
11311062 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.09 |
ug/ml |
12161130 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
12161130 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
870 |
nM |
1479585 |
NPT2943 |
Cell Line |
NCI-H417 |
Homo sapiens |
IC50 |
= |
230 |
nM |
1479585 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
230 |
nM |
1479585 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
620 |
nM |
1479585 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
400 |
nM |
11606134 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
10780911 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
63 |
nM |
1447730 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3100 |
nM |
1447730 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
33 |
nM |
1447730 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
560 |
nM |
1447730 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.11 |
ug/ml |
11354370 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.17 |
ug/ml |
11354370 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
0.21 |
ug/ml |
11354370 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
11354370 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
11354370 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.53 |
ug/ml |
11354370 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
11354370 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
0.17 |
ug/ml |
11354370 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
0.17 |
ug/ml |
11354370 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.21 |
ug/ml |
11354370 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
0.32 |
ug/ml |
11354370 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
11354370 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
0.06 |
ug/ml |
11354370 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.24 |
ug/ml |
11354370 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.13 |
ug/ml |
11354370 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
0.3 |
ug/ml |
11354370 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
IC50 |
= |
0.29 |
ug/ml |
11354370 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
11354370 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
15 |
nM |
12620081 |
NPT4264 |
Cell Line |
Lewis lung carcinoma cell line |
|
IC50 |
= |
22 |
nM |
12620081 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
12620081 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
4.4 |
|
12620081 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
13 |
|
12620081 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
69 |
nM |
3397990 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.053 |
ug/ml |
2002477 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
2002477 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.017 |
ug/ml |
2002477 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
12 |
nM |
10395490 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
33 |
nM |
10395490 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
18 |
nM |
10395490 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
290 |
nM |
9822542 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
3130 |
nM |
9822542 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.066 |
nM |
6827523 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
25 |
nM |
12443763 |
NPT1178 |
Cell Line |
KB 3-1 |
Homo sapiens |
IC50 |
= |
21 |
nM |
12443763 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
7010 |
nM |
12443763 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
250 |
nM |
12443763 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
12000 |
nM |
12443763 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
9703471 |
NPT4595 |
Cell Line |
CH1 |
Homo sapiens |
IC50 |
= |
6.3 |
nM |
9703471 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
78 |
nM |
9703471 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15 |
nM |
9207945 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22 |
nM |
9207945 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9.6 |
nM |
9207945 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
31 |
nM |
10395479 |
NPT4264 |
Cell Line |
Lewis lung carcinoma cell line |
|
IC50 |
= |
22 |
nM |
10395479 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
10395479 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Ratio |
= |
4.4 |
|
10395479 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Ratio |
= |
13 |
|
10395479 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
6.2 |
nM |
10498214 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
ED50 |
= |
150 |
nM |
10498214 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
37 |
nM |
10498214 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
3.5 |
nM |
10498214 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
57 |
nM |
10498214 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
6.3 |
nM |
10498214 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
ED50 |
= |
18.7 |
nM |
10498214 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.028 |
ug/ml |
1992140 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
48 |
nM |
1992140 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15 |
nM |
2547068 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
TD50 |
= |
0.015 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
TD50 |
= |
0.03 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TD50 |
= |
0.15 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
TD50 |
= |
0.006 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT4464 |
Cell Line |
L1210/Adr |
Mus musculus |
TD50 |
= |
0.4 |
ug/ml |
10.1016/0960-894X(95)00538-5 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
20 |
day |
14971908 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
9.8 |
day |
14971908 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ID50 |
= |
0.019 |
ug/ml |
3761328 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.6 |
nM |
3761328 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
3761328 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
68 |
nM |
3761328 |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
8200 |
nM |
3761328 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
121 |
|
3761328 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
ID50 |
= |
0.066 |
nM |
6951049 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.0031 |
ug/ml |
10.1016/S0960-894X(97)00191-1 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.0031 |
ug/ml |
10.1016/S0960-894X(97)00191-1 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.0031 |
ug/ml |
10.1016/S0960-894X(97)00191-1 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.0031 |
ug/ml |
10.1016/S0960-894X(97)00191-1 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
0.52 |
ug/ml |
10698460 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
48.9 |
ug/ml |
10698460 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.0096 |
ug/ml |
9871531 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.54 |
ug/ml |
9871531 |
NPT2090 |
Cell Line |
SNU-16 |
Homo sapiens |
IC50 |
= |
0.16 |
ug/ml |
9871531 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.004 |
ug/ml |
12459024 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
EC50 |
= |
700 |
nM |
11708923 |
NPT5520 |
Cell Line |
DuPro |
Homo sapiens |
EC50 |
= |
1800 |
nM |
11708923 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.6 |
nM |
3761325 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
3761325 |
NPT2831 |
Cell Line |
P388/S |
Mus musculus |
IC50 |
= |
68 |
nM |
3761325 |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
8200 |
nM |
3761325 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
120 |
|
3761325 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.05 |
|
2296017 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.03 |
|
2296017 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.1 |
|
2296017 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.032 |
|
2296017 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.33 |
|
2296017 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.039 |
|
2296017 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.09 |
ug/ml |
12113817 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.11 |
ug/ml |
12113817 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
0.117 |
ug/ml |
12113817 |
NPT4460 |
Cell Line |
L2987 |
Homo sapiens |
IC50 |
= |
300 |
nM |
12798317 |
NPT2827 |
Cell Line |
Human breast cancer cell lines |
|
IC50 |
= |
0.9 |
ug/ml |
11514168 |
NPT5502 |
Cell Line |
Human melanoma cell line |
|
IC50 |
> |
5 |
ug/ml |
11514168 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
30 |
ug/ml |
11514168 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
25 |
nM |
11128630 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
80 |
% |
11128630 |
NPT5522 |
Cell Line |
NCI-H647 |
|
IC50 |
< |
1 |
nM |
10780913 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4 |
nM |
10780913 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
8 |
nM |
10780913 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
130 |
nM |
10780913 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
10780913 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
IC50 |
= |
30 |
nM |
10780913 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10780913 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10 |
nM |
10780913 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
6 |
nM |
10780913 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
7 |
nM |
10780913 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
9 |
nM |
10780913 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
5 |
nM |
10780913 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
4 |
nM |
10780913 |
NPT5523 |
Cell Line |
F460pv8/eto |
|
IC50 |
= |
20 |
nM |
10780913 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
26 |
nM |
11806721 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
860 |
nM |
11806721 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
9700 |
nM |
11806721 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
24 |
nM |
11806721 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
2400 |
nM |
11806721 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
Inhibition |
= |
29 |
% |
3351854 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
Inhibition |
= |
70 |
% |
3351854 |
NPT730 |
Cell Line |
MC-38 |
Mus musculus |
Inhibition |
= |
93 |
% |
3351854 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
25.1 |
nM |
9003520 |
NPT934 |
Cell Line |
SK-VLB |
Homo sapiens |
IC50 |
= |
6540 |
nM |
9003520 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
280 |
nM |
9003520 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
15 |
nM |
9003520 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
32000 |
nM |
12039588 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
90 |
nM |
12039588 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
280 |
nM |
12039588 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
230 |
nM |
12039588 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
140 |
nM |
12039588 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
25 |
nM |
10890167 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
1.17 |
mg/kg |
10698441 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
20 |
nM |
10.1016/S0960-894X(97)10122-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1016/S0960-894X(97)10122-6 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1016/S0960-894X(97)10122-6 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1016/S0960-894X(97)10122-6 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
900 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
100 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
50 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
IC50 |
= |
200 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
80 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
50 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
50 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
50 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT913 |
Cell Line |
CHO-K1 |
Cricetulus griseus |
IC50 |
= |
1200 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT4350 |
Cell Line |
HEL 299 |
|
IC50 |
= |
1700 |
nM |
10.1016/0960-894X(96)00216-8 |
NPT3871 |
Cell Line |
N592 |
|
IC50 |
= |
40 |
nM |
8258835 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
8258835 |
NPT5524 |
Cell Line |
PAM |
Mus musculus |
IC50 |
= |
156000 |
nM |
9554873 |
NPT5524 |
Cell Line |
PAM |
Mus musculus |
IC50 |
= |
150000 |
nM |
9554873 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
12431049 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431049 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431049 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431049 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
10 |
nM |
12431049 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431049 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
30 |
nM |
12431049 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
90 |
nM |
12431049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
50 |
nM |
12431049 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
120 |
nM |
12431049 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
40 |
nM |
12431049 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
20 |
nM |
12431049 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
150 |
nM |
12431049 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
12431049 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
40 |
nM |
12431049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
300 |
nM |
9258351 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
10000 |
nM |
9258351 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
61.8 |
nM |
12392727 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
49.8 |
nM |
12392727 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.95 |
nM |
12392727 |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
9.2 |
nM |
12392727 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8.7 |
nM |
12392727 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2.7 |
nM |
12392727 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
52.8 |
nM |
12392727 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.2 |
nM |
12392727 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
9873394 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
300 |
|
9873394 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
340 |
nM |
9873394 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
15 |
nM |
9191970 |
NPT5525 |
Cell Line |
LLTC cell line |
|
IC50 |
= |
22 |
nM |
9191970 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
9.6 |
nM |
9191970 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Ratio |
= |
4.39 |
|
9191970 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Ratio |
= |
12.7 |
|
9191970 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
EC50 |
= |
700 |
nM |
14667208 |
NPT5520 |
Cell Line |
DuPro |
Homo sapiens |
EC50 |
= |
1800 |
nM |
14667208 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Ki |
= |
2000000 |
M-1 |
10.1016/0960-894X(95)00070-A |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
8145234 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
4 |
ug/ml |
8145234 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
133 |
|
8145234 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD10 |
= |
7.5 |
mg/kg/day |
8145234 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
15715467 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
93.55 |
% |
15715467 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
22 |
nM |
15715481 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
290 |
nM |
15715481 |
NPT571 |
Cell Line |
A2780cisR |
Homo sapiens |
IC50 |
= |
6 |
nM |
15715481 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
15715481 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
178 |
nM |
15715481 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
15715481 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
64 |
nM |
15715481 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
33 |
nM |
15715481 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
820 |
nM |
15715481 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
21 |
nM |
15715481 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
59 |
nM |
15715481 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7 |
nM |
15715481 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
11.3 |
nM |
15743178 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
15743178 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
CC50 |
= |
470 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
233000 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
414000 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
> |
400000 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
> |
235000 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
680 |
nM |
15745812 |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
CC50 |
= |
2900 |
nM |
15745812 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
1900 |
nM |
15745812 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10 |
nM |
15225700 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
90 |
nM |
15225700 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
15225700 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
100 |
nM |
15546712 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
30 |
nM |
15317455 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
330 |
nM |
15317455 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
400 |
nM |
15317455 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
23940 |
nM |
15317455 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
810 |
nM |
15456268 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
22 |
nM |
15456268 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
9100 |
nM |
15456268 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
2300 |
nM |
15456268 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
15922597 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.09 |
ug/ml |
15922597 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.07 |
ug/ml |
15922597 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
0.09 |
ug/ml |
15922597 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.28 |
ug/ml |
15922597 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
80 |
nM |
16169719 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
320 |
nM |
16169719 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
16 |
nM |
16169719 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
1560 |
nM |
16169719 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.4 |
nM |
16168652 |
NPT5526 |
Cell Line |
AT3B-1 |
Rattus norvegicus |
IC50 |
= |
42400 |
nM |
16168650 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
6700 |
nM |
16168650 |
NPT5526 |
Cell Line |
AT3B-1 |
Rattus norvegicus |
IC50 |
= |
167500 |
nM |
16168650 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
45200 |
nM |
16168650 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
250 |
nM |
16168650 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LD50 |
= |
1.8 |
nM |
16203143 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
LD50 |
= |
1.1 |
nM |
16203143 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
LD50 |
= |
14.2 |
nM |
16203143 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
LD50 |
= |
1.2 |
nM |
16203143 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LD50 |
= |
1.3 |
nM |
16203143 |
NPT320 |
Protein Family |
DNA topoisomerase II |
Homo sapiens |
Activity |
= |
0.001 |
nmol |
16242325 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
91.61 |
% |
16504508 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
Inhibition |
= |
51.26 |
% |
16504508 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
76.96 |
% |
16504508 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
150 |
nM |
16563756 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-19 |
% |
16563756 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-7 |
% |
16563756 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-10 |
% |
16563756 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
35 |
% |
16563756 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
53 |
% |
16563756 |
NPT4470 |
Cell Line |
Panel (10 carcinoma cell lines) |
|
Inhibition |
= |
91 |
% |
16621542 |
NPT4471 |
Cell Line |
Panel (12 tumour cell lines) |
Homo sapiens |
IC70 |
= |
39 |
nM |
16621542 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
150 |
nM |
16913700 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
20 |
nM |
16913700 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
1 |
nM |
16913700 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
40 |
nM |
16913700 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
16913700 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
150 |
nM |
16913700 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
90 |
nM |
16913700 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
30 |
nM |
16913700 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
20 |
nM |
16913700 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
10 |
nM |
16913700 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
20 |
nM |
16913700 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
IC50 |
= |
20 |
nM |
16913700 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
16913700 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2370 |
nM |
16777412 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
153 |
nM |
16824751 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
9.7 |
nM |
16824751 |
NPT2829 |
Cell Line |
MES-SA/DxS |
Homo sapiens |
IC50 |
= |
704 |
nM |
16824751 |
NPT2829 |
Cell Line |
MES-SA/DxS |
Homo sapiens |
Ratio IC50 |
= |
72.6 |
|
16824751 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
67 |
% |
17034133 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Activity |
= |
36 |
% |
17064069 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
4690 |
nM |
17154505 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Ratio IC50 |
= |
14 |
|
17154505 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
550 |
nM |
17154505 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
300 |
nM |
17154505 |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
1738 |
nM |
17154505 |
NPT552 |
Cell Line |
P388/ADR |
Mus musculus |
IC50 |
= |
123 |
nM |
17154505 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Ratio IC50 |
= |
16 |
|
17154505 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Ratio IC50 |
= |
9 |
|
17154505 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
22 |
nM |
17154505 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
316.23 |
nM |
17125253 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
6309.57 |
nM |
17125253 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12.59 |
nM |
17125253 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
2511.89 |
nM |
17125253 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17125253 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
50.12 |
nM |
17125253 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
199.53 |
nM |
17125253 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
31.62 |
nM |
17125253 |
NPT1635 |
Cell Line |
H9c2 |
Rattus norvegicus |
IC50 |
= |
31.62 |
nM |
17125253 |
NPT1635 |
Cell Line |
H9c2 |
Rattus norvegicus |
IC50 |
= |
19.95 |
nM |
17125253 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
1000 |
nM |
17125253 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
501.19 |
nM |
17125253 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
125.89 |
nM |
17125253 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
31.62 |
nM |
17125253 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7.5 |
nM |
17125254 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
61 |
nM |
17125254 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
3 |
nM |
17125254 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
8.1 |
|
17125254 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
0.4 |
|
17125254 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
GI50 |
= |
210 |
nM |
17181155 |
NPT980 |
Individual Protein |
Apoptosis regulator Bcl-2 |
Homo sapiens |
GI50 |
= |
26000 |
nM |
17181155 |
NPT2796 |
Individual Protein |
Apoptosis regulator Bcl-X |
Homo sapiens |
GI50 |
= |
24000 |
nM |
17181155 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
17253840 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
17253840 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
17253840 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
17253840 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
17253840 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17181164 |
NPT5512 |
Cell Line |
TRAMP-C1A |
Mus musculus |
GI50 |
= |
20.4 |
nM |
17181166 |
NPT5515 |
Cell Line |
TRAMP-C2H |
Mus musculus |
GI50 |
= |
15.8 |
nM |
17181166 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
GI50 |
= |
45.3 |
nM |
17181166 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7.5 |
ug/ml |
17181171 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
0.65 |
ug/ml |
17181171 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Inhibition |
= |
69 |
% |
17181166 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
29 |
nM |
17228871 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
480 |
nM |
17228871 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
86 |
% |
17228871 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
300 |
nM |
16919455 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
15 |
% |
16962775 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
Inhibition |
= |
9 |
% |
16962775 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Inhibition |
= |
3 |
% |
16962775 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
12 |
% |
16962775 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
11 |
% |
16962775 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
7 |
% |
16962775 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
6 |
% |
16962775 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
Inhibition |
= |
10 |
% |
16962775 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
5 |
% |
16962775 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Inhibition |
= |
10 |
% |
16962775 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
Inhibition |
= |
11 |
% |
16962775 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
100 |
nM |
17256903 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17286429 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17286429 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
17286429 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17286429 |
NPT1183 |
Cell Line |
WiDr |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
17315955 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.21 |
ug/ml |
17315955 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
17315955 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
60 |
nM |
17323939 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
62 |
|
17323939 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
9 |
|
17323939 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
900 |
nM |
17378530 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
EC50 |
= |
2000 |
nM |
17378530 |
NPT309 |
Cell Line |
1A9 |
Homo sapiens |
EC50 |
= |
100 |
nM |
17378530 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
= |
200 |
nM |
17378530 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
EC50 |
= |
400 |
nM |
17378530 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
22 |
nM |
17375902 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
178 |
nM |
17375902 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
7 |
nM |
17375902 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17375902 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
33 |
nM |
17375902 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
17375902 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
286 |
|
17375902 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
290 |
nM |
17375902 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
41 |
|
17375902 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
15588086 |
NPT3844 |
Protein Complex |
Anti-estrogen binding site (AEBS) |
Homo sapiens |
IC50 |
= |
200 |
nM |
15588086 |
NPT3844 |
Protein Complex |
Anti-estrogen binding site (AEBS) |
Homo sapiens |
IC50 |
= |
10000 |
nM |
15588086 |
NPT3844 |
Protein Complex |
Anti-estrogen binding site (AEBS) |
Homo sapiens |
IC50 |
= |
300 |
nM |
15588086 |
NPT3844 |
Protein Complex |
Anti-estrogen binding site (AEBS) |
Homo sapiens |
IC50 |
= |
150 |
nM |
15588086 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
0.76 |
ug/ml |
17358082 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
0.08 |
ug/ml |
17358082 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.48 |
ug/ml |
17358082 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7.5 |
ug/ml |
17070063 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
0.65 |
ug/ml |
17070063 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17049252 |
NPT2 |
Others |
Unspecified |
|
ID50 |
= |
0.35 |
ug/ml |
17035027 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
260 |
nM |
17107806 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17107806 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.46 |
ug/ml |
17417907 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.34 |
ug/ml |
17417907 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.42 |
ug/ml |
17417907 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.19 |
ug/ml |
17417907 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
0.77 |
ug/ml |
17417907 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
13 |
nM |
17069934 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
17069934 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
112 |
nM |
17070967 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
118 |
nM |
17070967 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
181 |
nM |
17070967 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
97 |
nM |
17070967 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
225 |
nM |
17070967 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
140 |
nM |
17276690 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
17276690 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
14.3 |
|
17276690 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
17276690 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4400 |
nM |
17276690 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.1 |
|
17276690 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.008 |
nM |
17482824 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
ED50 |
= |
0.102 |
nM |
17482824 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.274 |
nM |
17482824 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.152 |
nM |
17482824 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.173 |
nM |
17482824 |
NPT2 |
Others |
Unspecified |
|
ED50 |
> |
0.5 |
nM |
17482824 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LC50 |
= |
1400 |
nM |
17512741 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
100 |
nM |
17512741 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
TGI |
= |
300 |
nM |
17512741 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
100 |
nM |
17512741 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
TGI |
= |
200 |
nM |
17512741 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1000 |
nM |
17512741 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
100 |
nM |
17512741 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
300 |
nM |
17512741 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
400 |
nM |
17512741 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
0.71 |
ug/ml |
17547458 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
0.39 |
ug/ml |
17547458 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.41 |
ug/ml |
17547458 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7.1 |
nM |
17601739 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17000 |
nM |
17601739 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
17614292 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
17614292 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93 |
nM |
17614292 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
94 |
nM |
17614292 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
22 |
nM |
17141923 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
350 |
nM |
17141923 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17141923 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17175071 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17175071 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
420 |
nM |
17175071 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
830 |
nM |
17175071 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
36 |
% |
17175071 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
16.3 |
% |
17175071 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
17175071 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.5 |
% |
17175071 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.3 |
% |
17175071 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
17567069 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.13 |
ug/ml |
17567069 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
0.048 |
ug/ml |
17567069 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
750 |
nM |
17583953 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
350 |
nM |
17583953 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
580 |
nM |
17583953 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
180 |
nM |
17585747 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
180 |
nM |
17585747 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
130 |
nM |
17585747 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17585747 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
4000 |
nM |
17585747 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
400000 |
nM |
17595134 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1300000 |
nM |
17595134 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
17622129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
620 |
nM |
17622129 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
140 |
nM |
17622129 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
740 |
nM |
17622129 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
360 |
nM |
17622129 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
> |
1000 |
nM |
17696516 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
199.53 |
nM |
17696516 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
316.23 |
nM |
17696516 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
158.49 |
nM |
17696516 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
316.23 |
nM |
17696516 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
316.23 |
nM |
17696516 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
58.88 |
nM |
17696516 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
6.026 |
nM |
17696516 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
70.79 |
nM |
17696516 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
91.2 |
nM |
17696516 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
208.93 |
nM |
17696516 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
109.65 |
nM |
17696516 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
177.83 |
nM |
17696516 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
109.65 |
nM |
17696516 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13182.57 |
nM |
17696516 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1380 |
nM |
17418916 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
17400463 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17400463 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
420 |
nM |
17400463 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5 |
% |
17696516 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
15510 |
nM |
17400463 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
29 |
% |
17696516 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
150 |
nM |
17194596 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
60 |
nM |
17194596 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
620 |
nM |
17194596 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
60 |
nM |
17194596 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17194596 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
290 |
nM |
17194596 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
70 |
nM |
17194596 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17194596 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
78 |
% |
17194596 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2670 |
nM |
17194596 |
NPT5192 |
Cell Line |
U-937/GTB |
Homo sapiens |
IC50 |
= |
110 |
nM |
17442577 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
17442577 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
180 |
nM |
17442577 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
14200 |
nM |
17442577 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
4600 |
nM |
17194586 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
17194586 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
7700 |
nM |
17194586 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
17600 |
nM |
17194586 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3300 |
nM |
17194586 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.1 |
nM |
17591444 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
4.97 |
nM |
17591444 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.18 |
nM |
17591444 |
NPT309 |
Cell Line |
1A9 |
Homo sapiens |
ED50 |
= |
0.02 |
nM |
17591444 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
ED50 |
= |
1.2 |
nM |
17591444 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.26 |
nM |
17591444 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
ED50 |
= |
0.15 |
nM |
17591444 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
ED50 |
= |
0.04 |
nM |
17591444 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
ED50 |
= |
0.04 |
nM |
17591444 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
3.7 |
nM |
17656091 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
27 |
nM |
17656091 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17656091 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
35 |
nM |
17656091 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
200 |
nM |
17656091 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17656091 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
37 |
nM |
17656091 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17656091 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1920 |
nM |
17723301 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
2320 |
nM |
17723301 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24900 |
nM |
17723301 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
170 |
nM |
17723301 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
17723301 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2260 |
nM |
17723301 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.28 |
ug/ml |
17764956 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.34 |
ug/ml |
17764956 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.54 |
ug/ml |
17764956 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.48 |
ug/ml |
17764956 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
17764956 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
17764956 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
17822905 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
17822905 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
17822905 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
600 |
nM |
17822905 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
500 |
nM |
17822905 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
17822905 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
500 |
nM |
17822905 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
17827021 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
17827021 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.47 |
ug/ml |
17827021 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.25 |
ug/ml |
17827021 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.03 |
ug/ml |
17827021 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
0.24 |
ug/ml |
17827021 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.031 |
nM |
17904839 |
NPT2 |
Others |
Unspecified |
|
Activity |
> |
3.4 |
nM |
17904839 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
0.52 |
nM |
17904839 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
> |
3.4 |
nM |
17904839 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
0.221 |
nM |
17904839 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
> |
3.4 |
nM |
17904839 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17935309 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
40 |
nM |
17935309 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17935309 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17935309 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17935309 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
17935309 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
5 |
% |
17950603 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Inhibition |
= |
36 |
% |
17950603 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
74 |
% |
17950603 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
56 |
% |
17950603 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
Inhibition |
= |
62 |
% |
17950603 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
13 |
nM |
17239597 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
909 |
nM |
17239597 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
100 |
nM |
17448574 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
200 |
nM |
17448574 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
380 |
nM |
17490878 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
17490878 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
5.7 |
nM |
17490878 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
298 |
nM |
17490878 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
970 |
nM |
17827007 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
17827007 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1170 |
nM |
17827007 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
4780 |
nM |
17827007 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
347 |
nM |
17888666 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1550 |
nM |
17888666 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13489.63 |
nM |
17890094 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
93.33 |
nM |
17890094 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
59.5 |
nM |
17655260 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
ED50 |
= |
59.5 |
nM |
17655260 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.8 |
ug/ml |
17918910 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1.2 |
ug/ml |
17918910 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1.41 |
ug/ml |
17918910 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.06 |
ug/ml |
17970595 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.38 |
ug/ml |
17970595 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.22 |
ug/ml |
18052129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100 |
ug/ml |
18052129 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.45 |
ug/ml |
18052129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15.27 |
ug/ml |
18052129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1260 |
nM |
18052324 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
18052326 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
18052326 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
18052326 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
158.49 |
nM |
18173233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
199.53 |
nM |
18173233 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
2360000 |
nM |
18023182 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
1450000 |
nM |
18023182 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
8540000 |
nM |
18023182 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
5480000 |
nM |
18023182 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
200 |
nM |
18063366 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18063366 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
70 |
nM |
18063366 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
100 |
nM |
18063366 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
600 |
nM |
18063366 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18063366 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1570 |
nM |
18178085 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
18178085 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3090 |
nM |
18178085 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1390 |
nM |
18178085 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
720 |
nM |
18178085 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
100 |
% |
17962022 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
55 |
% |
17962022 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
IC50 |
= |
35 |
ug/ml |
17962022 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
20 |
% |
17962022 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
17981462 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17981462 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
LC50 |
= |
2500 |
nM |
17981462 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
Survival |
= |
72.2 |
% |
17993275 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
Survival |
= |
4.4 |
% |
17993275 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
Survival |
= |
3.5 |
% |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
115.5 |
% |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
100.1 |
% |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
22.1 |
% |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
9.5 |
% |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
7.5 |
% |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
110 |
% |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
105.6 |
% |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
8.6 |
% |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
2.5 |
% |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
1.1 |
% |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
97.5 |
% |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
81.4 |
% |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
20.2 |
% |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
7 |
% |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
6.1 |
% |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Survival |
= |
86.5 |
% |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Survival |
= |
82.2 |
% |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Survival |
= |
37.71 |
% |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Survival |
= |
16.8 |
% |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
Survival |
= |
6.6 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
85.6 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
23.1 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
5.8 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
1.5 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
107.6 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
105.4 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
56.9 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
13.8 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
7.4 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
121.3 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
96.8 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
50.48 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
11.8 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
5 |
% |
17993275 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15000 |
nM |
17993275 |
NPT464 |
Cell Line |
Daudi |
Homo sapiens |
IC50 |
= |
300 |
nM |
17993275 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
17993275 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2000 |
nM |
17993275 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
17993275 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9000 |
nM |
17993275 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2000 |
nM |
17993275 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
500 |
nM |
17993275 |
NPT433 |
Subcellular |
Liver microsomes |
Homo sapiens |
Activity |
= |
4.63 |
% |
18024139 |
NPT1574 |
Tissue |
Liver |
Homo sapiens |
Activity |
= |
15.1 |
% |
18024139 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
28 |
nM |
18077173 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
100 |
% |
18086527 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
75 |
% |
18086527 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
64 |
% |
18086527 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
55 |
% |
18086527 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
Activity |
= |
20 |
% |
18086527 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
81500 |
nM |
18086527 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
18207392 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
18207392 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
18207392 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
18207392 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
170 |
nM |
18207392 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
150 |
nM |
18207392 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
18207392 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
18207392 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
180 |
nM |
18207392 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
180 |
nM |
18207392 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
6.2 |
nM |
18243696 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
1460 |
nM |
18251492 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
44890 |
nM |
18251492 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
30740 |
nM |
18251492 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
5 |
% |
17936633 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
150 |
|
17964170 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
47800 |
nM |
17964170 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
300 |
nM |
17964170 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
17964791 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
17964791 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93 |
nM |
17964791 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
17976995 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.9 |
ug/ml |
17976995 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
17976995 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.75 |
ug/ml |
17976995 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7.5 |
ug/ml |
17976995 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.16 |
ug/ml |
17981473 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
17981473 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
17981473 |
NPT885 |
Cell Line |
PBL |
|
IC50 |
= |
0.97 |
ug/ml |
18053728 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
18164206 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
180 |
nM |
18313307 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
31980 |
nM |
18313307 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
178000 |
nM |
18313307 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18313307 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
36740 |
nM |
18313307 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
334000 |
nM |
18313307 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
240 |
nM |
18313307 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
24140 |
nM |
18313307 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
101000 |
nM |
18313307 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22 |
nM |
18321715 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
41 |
nM |
18321715 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
19 |
nM |
18321715 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
44 |
nM |
18321715 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
251 |
nM |
18321715 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
52 |
nM |
18321715 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
22 |
nM |
18321715 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
44 |
nM |
18321715 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IC50 |
= |
10000 |
nM |
18040043 |
NPT5527 |
Individual Protein |
Botulinum neurotoxin type B |
Clostridium botulinum |
Activity |
= |
9.4 |
nM |
18075579 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
> |
400000 |
nM |
18181575 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
> |
400000 |
nM |
18181575 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
90 |
nM |
18181575 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
60 |
nM |
18181575 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI |
= |
66.9 |
% |
18198839 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
51.6 |
% |
18198839 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
66.6 |
% |
18198839 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
73.2 |
% |
18198839 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
18247573 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
18247573 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
18247573 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1110 |
nM |
18247573 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.17 |
ug |
18502125 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LC50 |
= |
0.088 |
ppm |
1602301 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.8 |
ug/ml |
1602301 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
5.1 |
ug/ml |
1602301 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.2 |
ug/ml |
1602301 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
6.96 |
ug/ml |
2348205 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.9 |
ug/ml |
2348205 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.01 |
ug/ml |
2348205 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
0.04 |
ug/ml |
11000028 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.2 |
ug/ml |
11000028 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.06 |
ug/ml |
11000028 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
0.03 |
ug/ml |
11000028 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
0.1 |
ug/ml |
11000028 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.00622 |
ug/ml |
11087592 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.953 |
ug/ml |
11087592 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0287 |
ug/ml |
11087592 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.00286 |
ug/ml |
11087592 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.0577 |
ug/ml |
11087592 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
0.0061 |
ug/ml |
11087592 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI50 |
= |
12 |
nM |
10691710 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.7 |
ug/ml |
10869194 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13.4 |
ug/ml |
10869194 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
10869194 |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
10869194 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
11678655 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
11678655 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
11678655 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
11678655 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
11678655 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
7.2 |
nM |
11170674 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
8 |
nM |
11754602 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2200 |
nM |
11754602 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
63 |
day |
17626183 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.13 |
ug/ml |
11325235 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.82 |
ug/ml |
11325235 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.28 |
ug/ml |
11325235 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
2.26 |
ug/ml |
11325235 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
5.02 |
ug/ml |
11325235 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
2.62 |
ug/ml |
11325235 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
11325244 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
11325244 |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
11325244 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
11325244 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
11325244 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
91.8 |
% |
18375126 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
94.6 |
% |
18375126 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18375126 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
< |
1.1 |
ug/ml |
11374943 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
< |
1.1 |
ug/ml |
11374943 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
< |
1.1 |
ug/ml |
11374943 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
< |
1.1 |
ug/ml |
11374943 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.058 |
ug/ml |
11374944 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
200000 |
nM |
11430001 |
NPT4476 |
Individual Protein |
DNA topoisomerase |
Bos taurus |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4451 |
Individual Protein |
DNA topoisomerase I |
Mus musculus |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4477 |
Individual Protein |
DNA topoisomerase 1 |
Chlorocebus aethiops |
IC50 |
> |
200000 |
nM |
11430001 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
> |
200000 |
nM |
11430001 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
IC50 |
= |
1000 |
nM |
11430001 |
NPT908 |
Individual Protein |
Ribonuclease pancreatic |
Bos taurus |
IC50 |
= |
25000 |
nM |
11430001 |
NPT4478 |
Individual Protein |
Deoxyribonuclease-1 |
Bos taurus |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4479 |
Individual Protein |
Deoxyribonuclease-2-alpha |
Sus scrofa |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4480 |
Individual Protein |
DNA ligase |
Enterobacteria phage T4 |
IC50 |
> |
200000 |
nM |
11430001 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24000 |
nM |
11430001 |
NPT4481 |
Individual Protein |
Type-2 restriction enzyme BamHI |
Bacillus amyloliquefaciens |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4482 |
Individual Protein |
Type-2 restriction enzyme EcoRI |
Escherichia coli |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4483 |
Individual Protein |
Type-2 restriction enzyme HindIII |
Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) |
IC50 |
= |
96000 |
nM |
11430001 |
NPT4484 |
Individual Protein |
Type-2 restriction enzyme PstI |
Providencia stuartii |
IC50 |
> |
200000 |
nM |
11430001 |
NPT4485 |
Individual Protein |
Type-2 restriction enzyme ScaI |
Streptomyces caespitosus |
IC50 |
= |
25000 |
nM |
11430001 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
IC50 |
= |
73000 |
nM |
11430001 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
LD50 |
= |
2.5 |
ug/ml |
12502329 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.3 |
ug/ml |
12502336 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.3 |
ug/ml |
12502336 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
80 |
nM |
18258442 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
410 |
nM |
18258442 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
5.1 |
|
18258442 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
180 |
nM |
18262426 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
180 |
nM |
18262426 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
18262426 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
18262426 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
18262426 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
18262426 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
110 |
nM |
18262426 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
170 |
nM |
18262426 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
18262426 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.241 |
ug/ml |
11473425 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.45 |
ug/ml |
11473425 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
11 |
ug/ml |
11473441 |
NPT1881 |
Uncleic Acid |
Calf thymus DNA |
Bos taurus |
Activity |
= |
100 |
% |
1812211 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Activity |
= |
100 |
% |
1812211 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
11520227 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
11520227 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
11520227 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
11520227 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
11520227 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
20 |
nM |
17227762 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
90 |
nM |
17227762 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
17227762 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
200 |
nM |
11575949 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
55 |
nM |
11678649 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
570 |
nM |
11678649 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
94 |
nM |
11678649 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
8.1 |
nM |
11678649 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93 |
nM |
11678649 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.02 |
ug/ml |
17618015 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.002 |
ug/ml |
17618015 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
17618015 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.02 |
ug/ml |
17618015 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.07 |
ug/ml |
17618015 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
17618015 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
17618015 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
17618015 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
120 |
nM |
17673337 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
230 |
nM |
17673337 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
160 |
nM |
17673337 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
270 |
nM |
17673337 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
17692432 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93 |
nM |
17692432 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
17692432 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
18 |
nM |
18357994 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.007 |
nM |
18314958 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.056 |
nM |
18314958 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.117 |
nM |
18314958 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.164 |
nM |
18314958 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Activity |
= |
37.67 |
% |
17512094 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Activity |
= |
61.33 |
% |
17512094 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Activity |
= |
1 |
% |
17512094 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Inhibition |
= |
37.67 |
% |
17512094 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Ratio |
= |
0.57 |
|
17512094 |
NPT1490 |
Cell Line |
Ehrlich |
Mus musculus |
IC50 |
> |
10000 |
nM |
18281125 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
10 |
nM |
18281125 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
420 |
nM |
18281125 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
15510 |
nM |
18281125 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
21 |
nM |
19028425 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
25 |
nM |
19028425 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
18 |
nM |
19028425 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19093883 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2210 |
nM |
19093883 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
Ratio IC50 |
= |
93 |
|
19093883 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
17949859 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.4 |
nM |
17949859 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
25 |
|
17949859 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
18 |
nM |
17949859 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.7 |
nM |
17949859 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
25.7 |
|
17949859 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
EC50 |
= |
570 |
nM |
19282188 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
EC50 |
= |
290 |
nM |
19282188 |
NPT4783 |
Cell Line |
SNU-398 |
Homo sapiens |
GI50 |
= |
390 |
nM |
19282188 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
Activity |
= |
50 |
% |
19282188 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5820 |
nM |
11473418 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
4350 |
nM |
11473418 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
400 |
nM |
11473418 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
2550 |
nM |
11473418 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1690 |
nM |
11473418 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1820 |
nM |
11473418 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.0008 |
nM |
14640532 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
0.0003 |
nM |
14640532 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
0.00085 |
nM |
14640532 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.16 |
ug/ml |
10.1021/np50124a024 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
10.1021/np50124a024 |
NPT5528 |
Cell Line |
MOLT-4F |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
10.1021/np50124a024 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
10.1021/np50124a024 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
ED50 |
= |
0.3 |
ug/ml |
10.1021/np50124a024 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
LD50 |
= |
13 |
ug/ml |
8594149 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.48 |
ug/ml |
1593281 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.47 |
ug/ml |
1593281 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
6.69 |
ug/ml |
1593281 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Inhibition |
= |
33 |
% |
1791470 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Inhibition |
= |
91 |
% |
1791470 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Inhibition |
= |
100 |
% |
1791470 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.08 |
ug/ml |
1791471 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
6.84 |
ug/ml |
1791471 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.77 |
ug/ml |
1791471 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.16 |
ug/ml |
1791471 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
4.05 |
ppm |
1665173 |
NPT141 |
Organism |
Agrobacterium tumefaciens |
Agrobacterium tumefaciens |
Inhibition |
= |
68.8 |
% |
1665173 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.92 |
ug/ml |
1665173 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.15 |
ug/ml |
1665173 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.44 |
ug/ml |
1665173 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
12662097 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.17 |
ug/ml |
12662097 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
12662097 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
12662097 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
12662097 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
12662102 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
12662102 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
12662102 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
12662102 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.07 |
ug/ml |
12662102 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
12762820 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
12762820 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
12762820 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.19 |
ug/ml |
12762820 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.29 |
ug/ml |
12762820 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.16 |
ug/ml |
8991957 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
2.49 |
ug/ml |
8991957 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
3.42 |
ug/ml |
8991957 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
3.17 |
ug/ml |
8991957 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.57 |
ug/ml |
8778247 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
9.68 |
ug/ml |
8778247 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.93 |
ug/ml |
8778247 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.9 |
ug/ml |
8778247 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.81 |
ug/ml |
8778247 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
2.24 |
ug/ml |
8778247 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.52 |
ug/ml |
8882434 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.37 |
ug/ml |
8882434 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.23 |
ug/ml |
8882434 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
3.79 |
ug/ml |
8882434 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
8882434 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
5.06 |
ug/ml |
8882434 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.67 |
ug/ml |
9599253 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.12 |
ug/ml |
9599253 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
9.66 |
ug/ml |
9599253 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.98 |
ug/ml |
9599253 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.27 |
ug/ml |
9599253 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.45 |
ug/ml |
9599253 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.91 |
ug/ml |
9599260 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.79 |
ug/ml |
9599260 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.78 |
ug/ml |
9599260 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
6.2 |
ug/ml |
9599260 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
4.6 |
ug/ml |
9599260 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.53 |
ug/ml |
9599260 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.22 |
ug/ml |
9134750 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
1.19 |
ug/ml |
9134750 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
3.92 |
ug/ml |
9134750 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.2 |
ug/ml |
9051915 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
< |
0.1 |
ug/ml |
9051915 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
= |
16 |
ug/ml |
9051915 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42800 |
nM |
15165162 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94000 |
nM |
15165162 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93000 |
nM |
15165162 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
10.1021/np960188t |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
10.1021/np960188t |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
10.1021/np960188t |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
10.1021/np960188t |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
1.8 |
ug/ml |
10.1021/np960188t |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
8882437 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
8882437 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
8882437 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.0022 |
ug/ml |
9644064 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.081 |
ug/ml |
9644064 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.0053 |
ug/ml |
9644064 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
0.0049 |
ug/ml |
9644064 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
0.011 |
ug/ml |
9644064 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
0.0024 |
ug/ml |
9644064 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.005 |
ug/ml |
8759170 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1.5 |
ug/ml |
8759170 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.26 |
ug/ml |
9214729 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
5.3 |
ug/ml |
9214729 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
9214729 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
9214729 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
9214729 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
3.2 |
ug/ml |
9214729 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.8 |
ug/ml |
9214729 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
0.09 |
ug/ml |
9249977 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.09 |
ug/ml |
9249977 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.55 |
ug/ml |
9249977 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.97 |
ug/ml |
9249977 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
0.01 |
ug/ml |
9249977 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
0.11 |
ug/ml |
9249977 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
15270579 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
15270579 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
15270579 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
15270579 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
15270579 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
15270581 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
15270581 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
94 |
nM |
15270581 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.43 |
ug/ml |
8904848 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.09 |
ug/ml |
8904848 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.46 |
ug/ml |
8904848 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
6.49 |
ug/ml |
8904848 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.62 |
ug/ml |
8904848 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
7.9 |
ug/ml |
8904848 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.78 |
ug/ml |
8946743 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.28 |
ug/ml |
8946743 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.7 |
ug/ml |
8946743 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.78 |
ug/ml |
8946743 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LC50 |
= |
8 |
10'-2ppm |
8946743 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
1.89 |
ug/ml |
8946743 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
2.43 |
ug/ml |
8946743 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
Survival |
= |
21 |
% |
9834149 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Survival |
= |
19 |
% |
9834149 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.14 |
ug/ml |
14738384 |
NPT5192 |
Cell Line |
U-937/GTB |
Homo sapiens |
IC50 |
= |
100 |
nM |
14987049 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
100 |
nM |
14987049 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.012 |
ug/ml |
16252909 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
16252909 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.003 |
ug/ml |
16252909 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
16252909 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.35 |
ug/ml |
16252909 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.1 |
ug/ml |
16252910 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.79 |
ug/ml |
16252914 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.65 |
ug/ml |
16252914 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.56 |
ug/ml |
16252914 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
16252914 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
2.57 |
10'-1ppm |
8946744 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.28 |
ug/ml |
8946744 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
4.95 |
ug/ml |
8946744 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.98 |
ug/ml |
8946744 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
4.62 |
ug/ml |
8946744 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
5.83 |
ug/ml |
8946744 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
4.23 |
ug/ml |
8946744 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
70 |
nM |
16309317 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
170 |
nM |
16309317 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
170 |
nM |
16309317 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6.50E-07 |
ug/ml |
15043429 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
7.20E-07 |
ug/ml |
15043429 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
8.60E-07 |
ug/ml |
15043429 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.99 |
ug/ml |
9461654 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.53 |
ug/ml |
9461654 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.51 |
ug/ml |
9461654 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
4.24 |
ug/ml |
9461654 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.76 |
ug/ml |
9461654 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.33 |
ug/ml |
9461654 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
15104487 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
15104487 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
15104487 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
15104487 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
15104487 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.47 |
ug/ml |
15104488 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.25 |
ug/ml |
15104488 |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
ED50 |
= |
0.29 |
ug/ml |
15104488 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.41 |
ug/ml |
15104488 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
ED50 |
= |
0.57 |
ug/ml |
15104488 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED50 |
= |
0.22 |
ug/ml |
15104488 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.035 |
ug/ml |
8984156 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
8984156 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
0.008 |
ug/ml |
8984156 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
8984156 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
1.5 |
ug/ml |
8984156 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.1 |
ug/ml |
8984151 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.8 |
ug/ml |
8984151 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
2.7 |
ug/ml |
8984151 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
4.7 |
ug/ml |
8984151 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.0004 |
ug/ml |
8991944 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.027 |
ug/ml |
8991944 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
0.00051 |
ug/ml |
8991944 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.99 |
ug/ml |
9014350 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.89 |
ug/ml |
9014350 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.57 |
ug/ml |
9014350 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1.57 |
ug/ml |
15165136 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1.7 |
ug/ml |
15165136 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1 |
ug/ml |
15165136 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1.53 |
ug/ml |
15165136 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
8991955 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.3 |
ug/ml |
8991955 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.007 |
ug/ml |
8991955 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LC50 |
= |
0.257 |
ug/ml |
8991957 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.84 |
ug/ml |
8991957 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.47 |
ug/ml |
8991957 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
18440233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8050 |
nM |
18440233 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8040 |
nM |
18440233 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7880 |
nM |
18440233 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
680 |
nM |
18440233 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
9320 |
nM |
18440233 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
22 |
nM |
18429610 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
178 |
nM |
18429610 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
31 |
nM |
18429610 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
64 |
nM |
18429610 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
820 |
nM |
18429610 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1009 |
nM |
18429610 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5300 |
nM |
18429610 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
60 |
% |
18429610 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
100 |
% |
18429610 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
130 |
% |
18429610 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
22 |
% |
18429610 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
28 |
% |
18429610 |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
Activity |
= |
87 |
% |
18457386 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
180 |
nM |
18419154 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
900 |
nM |
18419154 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
860 |
nM |
18419154 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
640 |
nM |
18419154 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
590 |
nM |
18419154 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
18439831 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
18439831 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
94 |
nM |
18439831 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
47 |
% |
18707881 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI |
= |
69 |
% |
18707881 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
54 |
% |
18707881 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
64 |
% |
18707881 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
54 |
% |
18707881 |
NPT1514 |
Uncleic Acid |
DNA |
Bos taurus |
FC |
= |
2 |
|
18788722 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10 |
nM |
19220018 |
NPT1893 |
Cell Line |
MEF |
Mus musculus |
IC50 |
= |
3400 |
nM |
19186946 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
0.45 |
ug/ml |
18586355 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.47 |
ug/ml |
18586355 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
18586355 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
18586355 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
18586355 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
18586355 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.03 |
ug/ml |
18586355 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
100 |
% |
18586355 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16 |
nM |
19285863 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.7 |
nM |
19285863 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
13 |
nM |
19285863 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
49 |
nM |
19285863 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26 |
nM |
19285863 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
9.2 |
ug/ml |
7623031 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.3 |
ug/ml |
7623031 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.92 |
ug/ml |
7623031 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.01 |
ug/ml |
7673926 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.26 |
ug/ml |
7673926 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.75 |
ug/ml |
7673926 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.56 |
ug/ml |
7673935 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.42 |
ug/ml |
7673935 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.01 |
ug/ml |
7673935 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.94 |
ug/ml |
7673936 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.06 |
ug/ml |
7673936 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.48 |
ug/ml |
7673936 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.19 |
ug/ml |
15387653 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.31 |
ug/ml |
15387653 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.21 |
ug/ml |
15387653 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.19 |
ug/ml |
15387653 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.73 |
ug/ml |
15387653 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
30 |
nM |
7561901 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LD50 |
= |
1.13 |
ug/ml |
14575439 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LD50 |
= |
1.82 |
ug/ml |
14575439 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LD50 |
= |
1.28 |
ug/ml |
14575439 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
LD50 |
= |
2.26 |
ug/ml |
14575439 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LD50 |
= |
5.02 |
ug/ml |
14575439 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
LD50 |
= |
2.62 |
ug/ml |
14575439 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
20 |
nM |
15387664 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.41 |
ug/ml |
7494147 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.29 |
ug/ml |
7494147 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.16 |
ug/ml |
7494147 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.97 |
ug/ml |
7494147 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
6.24 |
ug/ml |
7494147 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.95 |
ug/ml |
7494147 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.313 |
ug/ml |
7494150 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.56 |
ug/ml |
7494150 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.42 |
ug/ml |
7494150 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.01 |
ug/ml |
7494150 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
59 |
nM |
14640513 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
14640517 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
14640517 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
14640517 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.19 |
ug/ml |
14640517 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.24 |
ug/ml |
14640517 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.09 |
ug/ml |
14640526 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
14640526 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
14640526 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
14640526 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
14640526 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
15497935 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
15497935 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
15497935 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
15497935 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.18 |
ug/ml |
15497935 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
14640527 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.09 |
ug/ml |
14640527 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
14640527 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
14640527 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.79 |
ug/ml |
14640527 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.07 |
ug/ml |
15104515 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.24 |
ug/ml |
15104515 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
15104515 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
15104515 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.17 |
ug/ml |
15104515 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
37 |
nM |
2778449 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IZ |
= |
5 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
74 |
nM |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
25 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
17.5 |
mm |
2778449 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IZ |
= |
5 |
mm |
2778449 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
15620238 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
15620238 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
15620238 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.45 |
ug/ml |
12608866 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.45 |
ug/ml |
12608866 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
15620238 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
43 |
nM |
15620248 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
15620248 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
93 |
nM |
15620248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
26.02 |
% |
15620248 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.12 |
ug/ml |
9392887 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
9392887 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
9392887 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.23 |
ug/ml |
9392887 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
2.4 |
ug/ml |
9392887 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
0.04 |
ug/ml |
12762806 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.066 |
ug/ml |
12762806 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.93 |
ug/ml |
9322367 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.69 |
ug/ml |
9322367 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
7.25 |
ug/ml |
9322367 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.13 |
ug/ml |
9322367 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
1.46 |
ug/ml |
9322367 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.42 |
ug/ml |
9322367 |
NPT2 |
Others |
Unspecified |
|
ID50 |
= |
0.2 |
ug/ml |
3819736 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ID50 |
= |
0.0055 |
ug/ml |
3819736 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
ID50 |
= |
0.5 |
ug/ml |
3819736 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6.20E-07 |
ug/ml |
12828475 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
3.60E-07 |
ug/ml |
12828475 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
5.30E-07 |
ug/ml |
12828475 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1.7 |
ug/ml |
12880315 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1.57 |
ug/ml |
12880315 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1 |
ug/ml |
12880315 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1.53 |
ug/ml |
12880315 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.08 |
ug/ml |
8201311 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.48 |
ug/ml |
8201311 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.47 |
ug/ml |
8201311 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
6.69 |
ug/ml |
8201311 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
90 |
nM |
12608854 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
140 |
nM |
12608854 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
230 |
nM |
12608854 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
280 |
nM |
12608854 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
320 |
nM |
12608854 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.1 |
ug/ml |
8021648 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.28 |
ug/ml |
8021648 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.79 |
ug/ml |
8021648 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
350 |
nM |
8350087 |
NPT2 |
Others |
Unspecified |
|
IC80 |
= |
0.001 |
nM |
8350087 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.08 |
ug/ml |
8350089 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.98 |
ug/ml |
8350089 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.02 |
ug/ml |
8350089 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.32 |
ug/ml |
8350089 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
2.5 |
ug/ml |
12608856 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
1.8 |
ug/ml |
12608856 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
> |
40 |
ug/ml |
12608856 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
40 |
ug/ml |
12608856 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.3 |
ug/ml |
8377016 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
9.13 |
ug/ml |
8377016 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.08 |
ug/ml |
8377016 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
130 |
nM |
18513976 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
820 |
nM |
18547115 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
480 |
nM |
18547115 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
400 |
nM |
18547115 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
70 |
nM |
18547115 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
650 |
nM |
18547115 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
160 |
nM |
18585035 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
60 |
nM |
18585035 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
210 |
nM |
18585035 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
110 |
nM |
18585035 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
120 |
nM |
18585035 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
182 |
nM |
18508273 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
85 |
% |
18508273 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
82 |
% |
18508273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
-25 |
% |
18508273 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
Activity |
= |
-4 |
% |
18508273 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
TGI |
= |
39 |
% |
18508273 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8600 |
nM |
18512984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
170 |
nM |
18512984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
0.9 |
% |
18512984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
4.9 |
% |
18512984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
8.9 |
% |
18512984 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
76.6 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.4 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
51.3 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
7.7 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
33.5 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.4 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
24.8 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
6.9 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60.8 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.9 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.6 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
12 |
% |
18512984 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
73.4 |
% |
18512984 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3.9 |
nM |
18829316 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
92.13 |
% |
18829316 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
100 |
nM |
19007287 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
100 |
nM |
19007287 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
100 |
nM |
19007287 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Activity |
= |
58 |
% |
18762427 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Activity |
= |
53.7 |
% |
18762427 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
13.1 |
% |
18762427 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
920 |
nM |
18783950 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
30 |
nM |
18783950 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
18783950 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
18783950 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
18783950 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
18 |
nM |
19136263 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2840 |
nM |
19140665 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
32 |
nM |
19140665 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
GI50 |
= |
0.07 |
ug/ml |
18023932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
0.39 |
ug/ml |
18023932 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
GI50 |
= |
0.11 |
ug/ml |
18023932 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
EC50 |
= |
0.01 |
ug/ml |
18990572 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
EC50 |
= |
0.01 |
ug/ml |
18990572 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
EC50 |
= |
0.01 |
ug/ml |
18990572 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
EC50 |
= |
0.03 |
ug/ml |
18990572 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
EC50 |
= |
0.03 |
ug/ml |
18990572 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8300 |
nM |
19329312 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
10200 |
nM |
19329312 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
14300 |
nM |
19329312 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
0.088 |
ug/ml |
1453182 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
5.04 |
ug/ml |
1453182 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.31 |
ug/ml |
1453182 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.45 |
ug/ml |
1453182 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI |
= |
38 |
% |
1479379 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI |
= |
105 |
% |
1479379 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
GI |
= |
99 |
% |
1479379 |
NPT140 |
Organism |
Artemia |
Artemia |
LC50 |
= |
8 |
ug/ml |
1479382 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.37 |
ug/ml |
1479382 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.08 |
ug/ml |
1479382 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
4.83 |
ug/ml |
1479382 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.09 |
ug/ml |
1294696 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.05 |
ug/ml |
1294696 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.12 |
ug/ml |
1294696 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.1 |
ug/ml |
7714532 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.28 |
ug/ml |
7714532 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.7 |
ug/ml |
7714532 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
ED50 |
= |
1.2 |
ug/ml |
7714533 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
3.2 |
ug/ml |
7714533 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
3.1 |
ug/ml |
7714533 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
5.6 |
ug/ml |
7714533 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
7714533 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
7714533 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
ED50 |
= |
2.8 |
ug/ml |
7714533 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
2.5 |
ug/ml |
7714533 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.01 |
ug/ml |
8676130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.03 |
ug/ml |
8676130 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.62 |
ug/ml |
8676130 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
3.66 |
ug/ml |
8676130 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
1.96 |
ug/ml |
8676130 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.32 |
ug/ml |
8676130 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.241 |
ug/ml |
11975482 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.45 |
ug/ml |
11975482 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
12193011 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
12193011 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
ED50 |
= |
0.002 |
ug/ml |
12193011 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
12193011 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
ED50 |
= |
0.003 |
ug/ml |
12193011 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.006 |
ug/ml |
12193011 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
12193011 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
12193011 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
12350153 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.16 |
ug/ml |
12350153 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
12350153 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
12350153 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
12350153 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
Inhibition |
= |
52 |
% |
16989517 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.27 |
ug/ml |
16989536 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.17 |
ug/ml |
16989536 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
15921415 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
15921415 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
15921415 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
15921415 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
15921415 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
15921417 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
15921417 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
15921417 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
15921417 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
170 |
nM |
15921419 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
50000 |
nM |
15921419 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
ED50 |
= |
0.15 |
ug/ml |
15921421 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
ED50 |
= |
0.14 |
ug/ml |
15921421 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.19 |
ug/ml |
15921421 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
16643027 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
16643027 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
16643027 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
16643027 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.06 |
ug/ml |
16643027 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
1.1 |
ug/ml |
10479316 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
5.6 |
ug/ml |
10479316 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
8.3 |
ug/ml |
10479316 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.7 |
ug/ml |
10479316 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
3.6 |
ug/ml |
10479316 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
8.9 |
ug/ml |
10479316 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
17067159 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2.7 |
ug/ml |
17067159 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
17067159 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
15921426 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
15921426 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
15921426 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
15921426 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.08 |
ug/ml |
15921426 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
270 |
nM |
15921436 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LD50 |
= |
0.09 |
ug/ml |
10514301 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LD50 |
= |
0.19 |
ug/ml |
10514301 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
LD50 |
= |
0.02 |
ug/ml |
10514301 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.0043 |
ug/ml |
10514307 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.129 |
ug/ml |
10514307 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.0168 |
ug/ml |
10514307 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
0.0156 |
ug/ml |
10514307 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.0499 |
ug/ml |
10514307 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
0.00101 |
ug/ml |
10514307 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.2 |
ug/ml |
17125220 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.3 |
ug/ml |
17125220 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
17125220 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
17125220 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
320 |
nM |
17125233 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
280 |
nM |
17125233 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
430 |
nM |
17125240 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
660 |
nM |
17125240 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
1550 |
nM |
17125240 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
310 |
nM |
17125240 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
410 |
nM |
17125240 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
100 |
nM |
15974615 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
100 |
nM |
15974615 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
800 |
nM |
17190442 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
17190442 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
17190442 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
200 |
nM |
17190442 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
100 |
nM |
17190442 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
699 |
nM |
16724842 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2210 |
nM |
16724842 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.3 |
ug/ml |
16724859 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
16724859 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
16724859 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
16724859 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
17190456 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.19 |
ug/ml |
17190456 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.08 |
ug/ml |
17190456 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.07 |
ug/ml |
17190456 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.13 |
ug/ml |
17190456 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.7 |
ug/ml |
9917277 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
2.1 |
ug/ml |
9917277 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.1 |
ug/ml |
9917277 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.9 |
ug/ml |
9917277 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
6.2 |
ug/ml |
9917277 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
2.3 |
ug/ml |
9917277 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.45 |
ug/ml |
10654411 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
10 |
nM |
17190470 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
17190470 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
40 |
nM |
17190470 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
17190470 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
7 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
158 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
137 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
61 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
29 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
10 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
3 |
% |
541685 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
8 |
% |
541685 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
40 |
% |
541685 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
38 |
% |
541685 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
29 |
% |
541685 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
20 |
% |
541685 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Activity |
= |
158 |
% |
541685 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Activity |
= |
166 |
% |
541685 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Activity |
= |
160 |
% |
541685 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Activity |
= |
127 |
% |
541685 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
6.22 |
ug/ml |
15730242 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
9.53 |
ug/ml |
15730242 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
2.87 |
ug/ml |
15730242 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
5.77 |
ug/ml |
15730242 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
6.1 |
ug/ml |
15730242 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
2.86 |
ug/ml |
15730242 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
380 |
nM |
15730243 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
15730243 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6.20E-07 |
ug/ml |
15730249 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
3.60E-07 |
ug/ml |
15730249 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
5.30E-07 |
ug/ml |
15730249 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
4.47 |
ug/ml |
10.1021/np970510f |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
8.97 |
ug/ml |
10.1021/np970510f |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
1.62 |
ug/ml |
10.1021/np970510f |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.1 |
ug/ml |
10.1021/np970510f |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
2.13 |
ug/ml |
10.1021/np970510f |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
2.88 |
ug/ml |
10.1021/np970510f |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
2.94 |
ug/ml |
9584396 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
1.24 |
ug/ml |
9584396 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
3.81 |
ug/ml |
9584396 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.58 |
ug/ml |
9584396 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
3.55 |
ug/ml |
9584396 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
4.56 |
ug/ml |
9584396 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
16441084 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
16441084 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
16441084 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
16441084 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.05 |
ug/ml |
16441084 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
15730260 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
220 |
nM |
16499322 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
7 |
nM |
16872155 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.11 |
ug/ml |
15787431 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.09 |
ug/ml |
15787431 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.04 |
ug/ml |
15787431 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
690 |
nM |
16499322 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
10217707 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
10217707 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
10217707 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
10217707 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.9 |
ug/ml |
10217707 |
NPT1475 |
Cell Line |
WI-38 VA13 |
Homo sapiens |
IC50 |
= |
380 |
nM |
16933868 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
16933868 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.07 |
ug/ml |
15787431 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
ED50 |
= |
0.17 |
ug/ml |
15787431 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
6.50E-07 |
ug/ml |
15787438 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
7.20E-07 |
ug/ml |
15787438 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
8.60E-07 |
ug/ml |
15787438 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
15787450 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
15787450 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
15787450 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
15787450 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
0.03 |
ug/ml |
15787450 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
10346965 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
10346965 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
10346965 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
ED50 |
= |
0.3 |
ug/ml |
10346965 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
ED50 |
= |
0 |
ug/ml |
10346965 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.4 |
ug/ml |
10346965 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
ED50 |
= |
0.1 |
ug/ml |
10346965 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.6 |
ug/ml |
10346965 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
ED50 |
= |
0.2 |
ug/ml |
10346965 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
1.3 |
ug/ml |
10395501 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.09 |
ug/ml |
10395501 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
= |
0.01 |
ug/ml |
10395501 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
ED50 |
= |
1.9 |
ug/ml |
10395501 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
10395501 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
ED50 |
= |
4.3 |
ug/ml |
10395501 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
219 |
nM |
16933890 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
288 |
nM |
16933890 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
40.5 |
nM |
16933890 |
NPT5192 |
Cell Line |
U-937/GTB |
Homo sapiens |
IC50 |
= |
110 |
nM |
16562840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
16562840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
180 |
nM |
16562840 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
14200 |
nM |
16562840 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.38 |
ug/ml |
16562847 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
0.42 |
ug/ml |
16562847 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
0.5 |
ug/ml |
16562847 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
18656370 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
18656370 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
18656370 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
IC50 |
= |
600 |
nM |
18656370 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
500 |
nM |
18656370 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
18656370 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
500 |
nM |
18656370 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
18657979 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
18657979 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
18657979 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
18657979 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
18657979 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
18657979 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
1720 |
nM |
18657979 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
18657979 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
180 |
nM |
18657979 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
18657979 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
18657979 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.011 |
ug/ml |
18590312 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
18590312 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC |
= |
0.025 |
ug/ml |
18590312 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.025 |
ug/ml |
18590312 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.17 |
ug/ml |
18590313 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.27 |
ug/ml |
18590313 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.15 |
ug/ml |
18590313 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.32 |
ug/ml |
18590313 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.52 |
ug/ml |
18590313 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
0.09 |
ug/ml |
18590313 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.003 |
ug/ml |
18590313 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
IC50 |
= |
3 |
nM |
19053767 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2 |
nM |
19053767 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
20 |
nM |
19053767 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
IC50 |
= |
30 |
nM |
19053767 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
50 |
nM |
19053767 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
19053767 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
40 |
nM |
19053767 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
200 |
nM |
19053767 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
160 |
nM |
19053767 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19053767 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
GI50 |
= |
1200 |
nM |
19188072 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
1000 |
nM |
19188072 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
CC50 |
= |
2000 |
nM |
19188072 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
51 |
|
19208482 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio IC50 |
= |
3.1 |
|
19208482 |
NPT2757 |
Individual Protein |
Purinergic receptor P2Y12 |
Homo sapiens |
Inhibition |
= |
7 |
% |
19463000 |
NPT2757 |
Individual Protein |
Purinergic receptor P2Y12 |
Homo sapiens |
Ki |
> |
10000 |
nM |
19463000 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
760 |
nM |
19473028 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1150 |
nM |
19473028 |
NPT1160 |
Cell Line |
BJ |
Homo sapiens |
IC50 |
= |
2700 |
nM |
19473028 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
78 |
nM |
19394829 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
19394829 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
200 |
nM |
19394829 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
200 |
nM |
19394829 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
90 |
nM |
19394829 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
19394829 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
4.16 |
nM |
19345581 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.13 |
nM |
19345581 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
4.45 |
nM |
19345581 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
6.66 |
nM |
19345581 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
4.73 |
nM |
19345581 |
NPT2196 |
Cell Line |
NB1 |
Homo sapiens |
IC50 |
= |
5.15 |
nM |
19345581 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5.1 |
nM |
19394218 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
930 |
nM |
19394218 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
190 |
nM |
19394218 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
7920 |
nM |
19394218 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
21 |
nM |
19394218 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
1.2 |
nM |
19394218 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
3 |
nM |
19394218 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
190 |
nM |
18692939 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
160 |
nM |
18692939 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
310 |
nM |
18692939 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
Activity |
= |
60 |
% |
19610651 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42800 |
nM |
19070942 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94000 |
nM |
19070942 |
NPT5530 |
Cell Line |
CNS cells |
Homo sapiens |
GI50 |
= |
94000 |
nM |
19070942 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
19084293 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
19084293 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.25 |
ug/ml |
19084293 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.5 |
ug/ml |
19296616 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
19159272 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
19159272 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.47 |
ug/ml |
19159272 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.25 |
ug/ml |
19159272 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
120 |
nM |
19405508 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
100 |
nM |
19405508 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
60 |
nM |
19405508 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7 |
nM |
19405508 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
16 |
nM |
19341288 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
330 |
nM |
19341288 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
120 |
nM |
19341288 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
410 |
nM |
19072548 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
< |
0.55 |
ug/ml |
19105653 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
< |
0.55 |
ug/ml |
19105653 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
< |
0.55 |
ug/ml |
19105653 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
< |
0.55 |
ug/ml |
19105653 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
3.2 |
ug/ml |
19105653 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
< |
0.55 |
ug/ml |
19105653 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
40 |
nM |
19278239 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7 |
nM |
19435339 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
56 |
nM |
19435339 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
117 |
nM |
19435339 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
164 |
nM |
19435339 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4180 |
nM |
19128861 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3240 |
nM |
19128861 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1600 |
nM |
19583252 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
19583252 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2500 |
nM |
19585998 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
19585998 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
19585998 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
19585998 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IG50 |
= |
3.73 |
nM |
19501507 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IG50 |
= |
0.019 |
nM |
19501507 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25280 |
nM |
19523827 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
530 |
nM |
19523827 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
47.7 |
|
19523827 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
577 |
nM |
19725578 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
9.2 |
|
19725578 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
63 |
nM |
19725578 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.144 |
ug/ml |
19456117 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.899 |
ug/ml |
19456117 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
0.058 |
ug/ml |
19456117 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
19555123 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
0.042 |
ug/ml |
19555123 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
60 |
nM |
19482476 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
19482476 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
EC50 |
= |
465.4 |
nM |
19743858 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
3078 |
nM |
19743858 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
EC50 |
= |
1508 |
nM |
19743858 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
8046 |
nM |
19743858 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
320 |
nM |
19422203 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.36 |
ug/ml |
19456120 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.98 |
ug/ml |
19456120 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.45 |
ug/ml |
19456120 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
8.92 |
ug/ml |
19456120 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
> |
10 |
ug/ml |
19456120 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
1640 |
nM |
19596579 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
610 |
nM |
19596579 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
510 |
nM |
19596579 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
GI50 |
= |
250 |
nM |
19596579 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
730 |
nM |
19596579 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
410 |
nM |
19596579 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1 |
nM |
19655762 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6 |
nM |
19655762 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12 |
nM |
19655762 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
13 |
nM |
19655762 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
58 |
nM |
19655762 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
81 |
nM |
19655762 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
240 |
nM |
19655762 |
NPT1635 |
Cell Line |
H9c2 |
Rattus norvegicus |
FC |
= |
3 |
|
19655762 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
FC |
= |
14 |
|
19655762 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC30 |
= |
2.13 |
ug/ml |
19371979 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC30 |
= |
1.51 |
ug/ml |
19371979 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
19342127 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.024 |
ug/ml |
19342127 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.015 |
ug/ml |
19342127 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
0.19 |
ug/ml |
19342127 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
19342127 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
100 |
nM |
19361894 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
150 |
nM |
19361894 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
80 |
nM |
19361894 |
NPT1723 |
Cell Line |
HBL-100 |
Homo sapiens |
IC50 |
= |
240 |
nM |
19361894 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
80 |
nM |
19361894 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3000 |
nM |
19361894 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
100 |
nM |
19361894 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
630 |
nM |
19361894 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
Inhibition |
= |
34 |
% |
19615898 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
19406535 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
480 |
nM |
19406535 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
20 |
nM |
19406535 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
960 |
nM |
19406535 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
600 |
nM |
19406535 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
720 |
nM |
19406535 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
510 |
nM |
19406535 |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
19406535 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1320 |
nM |
19406535 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
1770 |
nM |
19406535 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
4.9 |
ug/ml |
18973387 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
18973388 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.2 |
ug/ml |
18973388 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
18973388 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
18973388 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
18973388 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
0.1 |
ug/ml |
18973388 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.7 |
ug/ml |
19540022 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19457675 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
19457675 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
1.81 |
|
19457675 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5 |
ug/ml |
19700322 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6.71 |
ug/ml |
19932530 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8.72 |
ug/ml |
19932530 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
19939522 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
55 |
% |
19939522 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
57 |
% |
19939522 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
93 |
% |
19939522 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
19 |
% |
19944497 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
68 |
% |
19944497 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32 |
% |
19944497 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
19944497 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38 |
ug/ml |
19944497 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
48 |
% |
19926172 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
55 |
% |
19926172 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
34 |
% |
19926172 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
28 |
% |
19926172 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI |
= |
93 |
% |
19926172 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
44 |
% |
19926172 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
86 |
% |
19926172 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
60 |
nM |
19926173 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
19926173 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
19853327 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
75 |
% |
19853327 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
55 |
% |
19853327 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
20 |
% |
19853327 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
52 |
ug/ml |
19853327 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68130 |
nM |
19879135 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
19879135 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
68 |
% |
19879135 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
30 |
% |
19879135 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
24 |
% |
19879135 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Ratio IC50 |
= |
7 |
|
19947600 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Ratio IC50 |
= |
0.48 |
|
19947600 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Ratio IC50 |
= |
14 |
|
19947600 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
420 |
nM |
19947600 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
410 |
nM |
19947600 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
60 |
nM |
19947600 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
880 |
nM |
19947600 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
19947600 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Ratio IC50 |
= |
1.02 |
|
19947600 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
Inhibition |
= |
82.28 |
% |
19679380 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
65.47 |
% |
19679380 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Inhibition |
= |
66.66 |
% |
19679380 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
75 |
nM |
19819696 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
46 |
nM |
19819696 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
28 |
nM |
19819696 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
350 |
nM |
19819696 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
37 |
nM |
19819696 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
730 |
nM |
19819703 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1030 |
nM |
19819703 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
240 |
nM |
19647439 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
190 |
nM |
19647439 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
290 |
nM |
19647439 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
27 |
nM |
19647439 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
420 |
nM |
19910192 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
20000 |
nM |
19910192 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
72 |
% |
19913412 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2040 |
nM |
19879765 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2040 |
nM |
19879765 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1960 |
nM |
19879765 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1730 |
nM |
19879765 |
NPT5531 |
Tissue |
Bone marrow |
Mus musculus |
Activity |
= |
0.2 |
% |
20060717 |
NPT5531 |
Tissue |
Bone marrow |
Mus musculus |
Activity |
= |
0.3 |
% |
20060717 |
NPT5531 |
Tissue |
Bone marrow |
Mus musculus |
Activity |
= |
0.1 |
% |
20060717 |
NPT5531 |
Tissue |
Bone marrow |
Mus musculus |
Activity |
= |
0.4 |
% |
20060717 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.34 |
ug/ml |
20036537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.56 |
ug/ml |
20036537 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1.05 |
ug/ml |
20036537 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.42 |
ug/ml |
20036537 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.32 |
ug/ml |
20036537 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
20036537 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
0.55 |
ug/ml |
20022253 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.42 |
ug/ml |
20022253 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
330 |
nM |
20171108 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2230 |
nM |
20171108 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
90 |
nM |
20171108 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1760 |
nM |
20171108 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
Activity |
= |
0.817 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
27.28 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.32 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.15 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
2.00E-06 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.11 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.19 |
ug |
20171109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.046 |
ug |
20171109 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
20 |
|
20151639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
nM |
20151639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3100 |
nM |
20151639 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
0.1 |
ug/ml |
20153202 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
1 |
ug/ml |
20153202 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
CC50 |
= |
2 |
ug/ml |
20153202 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
160 |
nM |
20176479 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
380 |
nM |
20176479 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
40 |
nM |
20176479 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
820 |
nM |
20176479 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
20035557 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
240 |
nM |
20038128 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300 |
nM |
20038128 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
80 |
nM |
20038128 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
180 |
nM |
20045222 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
130 |
nM |
20045222 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
850 |
nM |
20138760 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Inhibition |
= |
60.89 |
% |
20138760 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
62.79 |
% |
20138760 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
350 |
nM |
20138760 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
8500 |
nM |
20055495 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
50 |
nM |
19914747 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
530 |
nM |
19919052 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
38 |
nM |
20014800 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
TGI |
= |
310 |
nM |
20014800 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LC50 |
= |
2410 |
nM |
20014800 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
66 |
nM |
20014800 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
400 |
nM |
20014800 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
> |
17200 |
nM |
20014800 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
62 |
nM |
20014800 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
TGI |
= |
260 |
nM |
20014800 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1570 |
nM |
20014800 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1.3 |
ug/ml |
19928902 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.9 |
ug/ml |
19928902 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.6 |
ug/ml |
19928902 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
19928902 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
19928902 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
19783438 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
ED50 |
= |
0.003 |
ug/ml |
19783438 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
ED50 |
= |
0.001 |
ug/ml |
19783438 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
ED50 |
= |
0.029 |
ug/ml |
19783438 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
ED50 |
= |
0.071 |
ug/ml |
19783438 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
70 |
nM |
19788290 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
19788290 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
120 |
nM |
19788290 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
750 |
nM |
19788290 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
250 |
nM |
19739600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
19739600 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
920 |
nM |
19795842 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
280 |
nM |
19739600 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
50 |
nM |
19748781 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
837 |
nM |
19860383 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
70 |
% |
19634903 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
370 |
nM |
19824618 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
640 |
nM |
19824618 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
400 |
nM |
19824618 |
NPT793 |
Cell Line |
MOLT-3 |
Homo sapiens |
IC50 |
= |
40 |
nM |
19824618 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
800 |
nM |
19658408 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1200 |
nM |
19658408 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
19658408 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6300 |
nM |
19658408 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
19778068 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.13 |
ug/ml |
19778068 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.2 |
ug/ml |
19778068 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
410 |
nM |
19689125 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
50 |
nM |
19780590 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
19780590 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
370 |
nM |
19780590 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
90 |
nM |
19780590 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
500 |
nM |
19780590 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
840 |
nM |
19689125 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
620 |
nM |
19689125 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3120 |
nM |
19689125 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3070 |
nM |
19689125 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
94 |
nM |
19428155 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
19428155 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
19428155 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
10.86 |
nM |
19428155 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.16 |
ug/ml |
19691312 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.41 |
ug/ml |
19691312 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.46 |
ug/ml |
19691312 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.43 |
ug/ml |
19691312 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
0.14 |
ug/ml |
19691312 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.35 |
ug/ml |
19691312 |
NPT682 |
Cell Line |
SK-N-MC |
Homo sapiens |
IC50 |
= |
120 |
nM |
20303768 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5950 |
nM |
20303768 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18 |
nM |
20210346 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
10 |
nM |
20210346 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
11 |
nM |
20210346 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
30.8 |
% |
20210346 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
8.9 |
% |
20210346 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
59.9 |
% |
20210346 |
NPT191 |
Organism |
Hepatitis C virus |
Hepatitis C virus |
IC50 |
= |
2600 |
nM |
20363140 |
NPT191 |
Organism |
Hepatitis C virus |
Hepatitis C virus |
EC50 |
< |
300 |
nM |
20363140 |
NPT2 |
Others |
Unspecified |
|
Ratio CC50/EC50 |
< |
0.1 |
|
20363140 |
NPT191 |
Organism |
Hepatitis C virus |
Hepatitis C virus |
IC50 |
= |
12000 |
nM |
20363140 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
20329738 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.25 |
ug/ml |
20329738 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.57 |
ug/ml |
20329738 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
0.12 |
% |
20022146 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
912 |
nM |
20356064 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2620 |
nM |
20056520 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3240 |
nM |
20056520 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
14350 |
nM |
20064676 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3610 |
nM |
20064676 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
37 |
nM |
20180542 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
55 |
nM |
20180542 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37.5 |
ug/ml |
20149941 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
20 |
% |
20149941 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
39 |
% |
20149941 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60 |
% |
20149941 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
20149941 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2050 |
nM |
20405844 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
20405844 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
3160 |
nM |
20405844 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
3700 |
nM |
20405844 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
6100 |
nM |
20455578 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
5600 |
nM |
20455578 |
NPT2 |
Others |
Unspecified |
|
EC50 |
> |
10000 |
nM |
20455578 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
> |
10000 |
nM |
20455578 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
40 |
nM |
20207049 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
10 |
nM |
20207049 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20207049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
40 |
nM |
20207049 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
Inhibition |
= |
30 |
% |
20471276 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
Inhibition |
= |
0 |
% |
20471276 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
33 |
nM |
20471276 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
520 |
nM |
20471276 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
1 |
ug/ml |
20207452 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
20207452 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
15.9 |
|
20471276 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
20334960 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
20334960 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
700 |
nM |
20334960 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
400 |
nM |
20334960 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
20334960 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
100 |
nM |
20334960 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
580 |
nM |
20149494 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
4160 |
nM |
20356655 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
1.13 |
nM |
20356655 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
4.45 |
nM |
20356655 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
6.12 |
nM |
20356655 |
NPT2196 |
Cell Line |
NB1 |
Homo sapiens |
IC50 |
= |
5.15 |
nM |
20356655 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
4.73 |
nM |
20356655 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
20413187 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
70 |
% |
20413187 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25 |
% |
20413187 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17 |
% |
20413187 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
69900 |
nM |
20413187 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
180 |
nM |
20413188 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
40 |
nM |
20413188 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5990 |
nM |
20413188 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
50 |
nM |
20413188 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
20413188 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
70 |
nM |
20413188 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
180 |
nM |
20413188 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
30 |
nM |
20413188 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
330 |
nM |
20413188 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
1840 |
nM |
20413188 |
NPT2 |
Others |
Unspecified |
|
TGI |
> |
100000 |
nM |
20413188 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
1420 |
nM |
20413188 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
2300 |
nM |
20413188 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
= |
8110 |
nM |
20413188 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
46000 |
nM |
20413188 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
550 |
nM |
20413188 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
LC50 |
= |
460 |
nM |
20413188 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
46000 |
nM |
20413188 |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
100000 |
nM |
20413188 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
37900 |
nM |
20413188 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
20413188 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
20413188 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
20413188 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
20359789 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
920 |
nM |
20359789 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
30 |
nM |
20359789 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
20359789 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
20359789 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
20359789 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7400 |
nM |
20362359 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
410 |
nM |
20362359 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.59 |
ug/ml |
20399544 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.72 |
ug/ml |
20399544 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.65 |
ug/ml |
20399544 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC90 |
= |
6.82 |
ug/ml |
20399544 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC90 |
= |
8.77 |
ug/ml |
20399544 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC90 |
= |
7.32 |
ug/ml |
20399544 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
400 |
nM |
20570145 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
20 |
nM |
20570145 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
280 |
nM |
20538470 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
324 |
nM |
20538470 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
264 |
nM |
20538470 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
220 |
nM |
20538470 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
36.9 |
nM |
20527917 |
NPT2251 |
Cell Line |
ADR5000 cell line |
|
IC50 |
> |
5200 |
nM |
20527917 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
52 |
nM |
20545334 |
NPT2 |
Others |
Unspecified |
|
IC50 |
<= |
52 |
nM |
20545334 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
5 |
ug/ml |
20550123 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
20550123 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1.35 |
ug/ml |
20550123 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
0.8 |
ug/ml |
20550123 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1.2 |
ug/ml |
20550123 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.6 |
ug/ml |
20550123 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
20593838 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
170 |
nM |
20593838 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
120 |
nM |
20593838 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
20537433 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
20537433 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
20537433 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
0.96 |
ug/ml |
20537433 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
178 |
nM |
20579876 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
317 |
nM |
20579876 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
182 |
nM |
20579876 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
2177 |
nM |
20579876 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
194 |
nM |
20579876 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
GI50 |
= |
202 |
nM |
20579876 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
21 |
nM |
20594848 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
3 |
nM |
20594848 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
12 |
nM |
20594848 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
38 |
nM |
20594848 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
5120 |
nM |
20634081 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
70 |
nM |
20638854 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
240 |
nM |
20718475 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
590 |
nM |
20718475 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
190 |
nM |
20718475 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
140 |
nM |
20718475 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
360 |
nM |
20718475 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10 |
nM |
20719504 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1 |
nM |
20719504 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
2 |
nM |
20719504 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
28 |
nM |
20719504 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
0.0248 |
ug/ml |
20722446 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.457 |
ug/ml |
20722446 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
0.001 |
ug/ml |
20722446 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
0.286 |
ug/ml |
20722446 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
GI |
= |
91.19 |
% |
20722446 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI |
= |
94.69 |
% |
20722446 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
96.38 |
% |
20722446 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI |
= |
93.1 |
% |
20722446 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
20732817 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
20732817 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
20732817 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
20732817 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
20732817 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
20732817 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
20732817 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
20732817 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
20732817 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
20732817 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
170 |
nM |
20732817 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
330 |
nM |
20815366 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2180 |
nM |
20815366 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
20 |
nM |
20675130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
210 |
nM |
20675130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
740 |
nM |
20675130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.461 |
|
20684857 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.494 |
|
20684857 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.546 |
|
20684857 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.721 |
|
20684857 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
71800 |
nM |
20684857 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
81 |
nM |
20690624 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
> |
1000 |
nM |
20690624 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3.76 |
ug/ml |
20599299 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3.64 |
ug/ml |
20599299 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4.57 |
ug/ml |
20599299 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
320 |
nM |
20729093 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
10990 |
nM |
20729093 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
2830 |
nM |
20729093 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
= |
7860 |
nM |
20729093 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
2370 |
nM |
20729093 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
4030 |
nM |
20729093 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
= |
10250 |
nM |
20729093 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
16400 |
nM |
20729093 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
= |
1420 |
nM |
20729093 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
42.7 |
% |
20729093 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
34.7 |
% |
20729093 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
28 |
% |
20729093 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
2.5 |
ug |
20729093 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
290 |
nM |
20619940 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
260 |
nM |
20619940 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
300 |
nM |
20619940 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
IC50 |
= |
20000 |
nM |
20662543 |
NPT143 |
Individual Protein |
DNA topoisomerase I |
Homo sapiens |
Inhibition |
= |
35 |
% |
20662543 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
85 |
% |
20662543 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1900 |
nM |
20662543 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
8 |
nM |
20833057 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
< |
100000 |
nM |
20667627 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
35481.34 |
nM |
20667627 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
2570.4 |
nM |
20667627 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
2089.3 |
nM |
20667627 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
2089.3 |
nM |
20667627 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
158.49 |
nM |
20667627 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
141.25 |
nM |
20667627 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
134.9 |
nM |
20667627 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
131.83 |
nM |
20667627 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
109.65 |
nM |
20667627 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
107.15 |
nM |
20667627 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
107.15 |
nM |
20667627 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
> |
100 |
nM |
20667627 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
> |
100 |
nM |
20667627 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
28.5 |
nM |
20732810 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
16.5 |
nM |
20732810 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI |
= |
12.3 |
nM |
20732810 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
280 |
nM |
20732810 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
180 |
nM |
20732810 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
220 |
nM |
20732810 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.12 |
ug/ml |
20732814 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.45 |
ug/ml |
20732814 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.33 |
ug/ml |
20732814 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
0.28 |
ug/ml |
20732814 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
250 |
nM |
20800481 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
Activity |
= |
50 |
% |
20800481 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5230 |
nM |
20850308 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3220 |
nM |
20850308 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
370 |
nM |
20846862 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
49 |
nM |
20846862 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
1060 |
nM |
20846862 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
750 |
nM |
20846862 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9200 |
nM |
20846862 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
370 |
nM |
20846862 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
70 |
nM |
20846862 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
600 |
nM |
20846862 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
20850305 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
ED50 |
> |
0 |
ug/ml |
20850305 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
ED50 |
= |
0.03 |
ug/ml |
20850305 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.02 |
ug/ml |
20850305 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
ED50 |
= |
0.02 |
ug/ml |
20850305 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2570 |
nM |
20873721 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
6060 |
nM |
20873721 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6400 |
nM |
20873721 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
3140 |
nM |
20873721 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2030 |
nM |
20932754 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
900 |
nM |
20932754 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Inhibition |
= |
30 |
% |
20884207 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
= |
4 |
mm |
20739103 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
= |
3 |
mm |
20739103 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
< |
2940 |
nM |
20810194 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
< |
2940 |
nM |
20810194 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
Inhibition |
= |
93.8 |
% |
20817326 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
36.4 |
% |
20817326 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
89.4 |
% |
20817326 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
98 |
% |
20817326 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
100 |
% |
20817326 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
3300 |
nM |
20817326 |
NPT3998 |
Cell Line |
LLC cell line |
|
IC50 |
= |
3.7 |
ug/ml |
20813435 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.3 |
ug/ml |
20813435 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.97 |
ug/ml |
20739102 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4.19 |
ug/ml |
20739102 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.73 |
ug/ml |
20739102 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.73 |
ug/ml |
20739102 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2300 |
nM |
20832916 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
1100 |
nM |
20832916 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
954 |
nM |
20832916 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
20832916 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1230 |
nM |
20931970 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
740 |
nM |
20931970 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
950 |
nM |
20931970 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1630 |
nM |
20931970 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1540 |
nM |
20931970 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
850 |
nM |
20931970 |
NPT1160 |
Cell Line |
BJ |
Homo sapiens |
IC50 |
= |
2330 |
nM |
20931970 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
4.2 |
% |
20943401 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
59.2 |
% |
20943401 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
77.6 |
nM |
20936874 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
0.09 |
ug/ml |
21041092 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.03 |
ug/ml |
21041092 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
0.33 |
ug/ml |
21041092 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
0.04 |
ug/ml |
21041092 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
0.03 |
ug/ml |
21041092 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
0.28 |
ug/ml |
21041092 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
0.08 |
ug/ml |
21041092 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.07 |
ug/ml |
21041092 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
0.4 |
ug/ml |
21041092 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
0.33 |
ug/ml |
21041092 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
3.3 |
ug/ml |
21041092 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
TGI |
= |
6.6 |
ug/ml |
21041092 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
= |
2.67 |
ug/ml |
21041092 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
0.9 |
ug/ml |
21041092 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
5.85 |
ug/ml |
21041092 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
TGI |
= |
2.95 |
ug/ml |
21041092 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
3.9 |
ug/ml |
21041092 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
20.48 |
ug/ml |
21041092 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
220 |
nM |
21071221 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
520 |
nM |
21071221 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
610 |
nM |
21071221 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
820 |
nM |
21071221 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
21106454 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.42 |
ug/ml |
21106454 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
14.47 |
ug/ml |
21106454 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.63 |
ug/ml |
21106454 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.35 |
ug/ml |
21106454 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1.32 |
ug/ml |
21106454 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
0.23 |
nM |
21067930 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
0.38 |
nM |
21067930 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
0.19 |
nM |
21067930 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
900 |
nM |
21058726 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21058726 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21058726 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21035234 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
21035234 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3300 |
nM |
21035234 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
57.9 |
% |
21035921 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
48.8 |
% |
21035921 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
54.6 |
% |
21035921 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
31.8 |
% |
21035921 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI |
= |
60 |
% |
21035921 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
65 |
nM |
20884089 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
3600 |
nM |
20961671 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
20971532 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
480 |
nM |
20971532 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
20 |
nM |
20971532 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
960 |
nM |
20971532 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
1660 |
nM |
20971532 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
43.3 |
nM |
20934235 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
130.2 |
nM |
20934235 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
35.6 |
nM |
20934235 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
21115246 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1330 |
nM |
21115246 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1750 |
nM |
21115246 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1250 |
nM |
21115246 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
92 |
nM |
20949916 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
67 |
nM |
20949916 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
170 |
nM |
20949916 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
52.8 |
% |
21146994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
45.9 |
% |
21146994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
1.2 |
% |
21146994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
5.2 |
% |
21146994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
89.2 |
% |
21146994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
5.6 |
% |
21146994 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
8 |
% |
21094049 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
43 |
% |
21094049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
47 |
% |
21094049 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
1.3 |
% |
21094049 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
5 |
% |
21094049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3.3 |
% |
21094049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16800 |
nM |
21094049 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
10400 |
nM |
21094049 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21094049 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
600 |
nM |
21094049 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
4780 |
nM |
21095131 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
970 |
nM |
21095131 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1170 |
nM |
21095131 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
21095131 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21142180 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
990 |
nM |
21142180 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
40 |
nM |
21142180 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
22 |
nM |
21142180 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.047 |
nM |
21142180 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.5 |
nM |
21142180 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
41 |
nM |
21142180 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
186 |
nM |
21142180 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
540 |
nM |
21087017 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
21087017 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12 |
nM |
21087017 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
450 |
nM |
21087017 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
370 |
nM |
21087017 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
170 |
nM |
21087017 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
98 |
nM |
21090800 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
370 |
nM |
21090800 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2300 |
nM |
21090800 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
19 |
% |
21112675 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32 |
% |
21112675 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
68 |
% |
21112675 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
21112675 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38 |
ug/ml |
21112675 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
19950 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
25400 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
19950 |
nM |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
3160 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.721 |
|
21093116 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.546 |
|
21093116 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.461 |
|
21093116 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.494 |
|
21093116 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
32020 |
nM |
21093116 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
43.3 |
nM |
21138784 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
130.2 |
nM |
21138784 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
35.6 |
nM |
21138784 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
370 |
nM |
21144624 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
21144624 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
60 |
nM |
21144624 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
120 |
nM |
21144624 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9700 |
nM |
21144624 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
81 |
|
21144624 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
110 |
nM |
21144624 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
520 |
nM |
21144624 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
4.7 |
|
21144624 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
5010 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
25400 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
5010 |
nM |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
250 |
nM |
21115210 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
100 |
nM |
21115210 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
200 |
nM |
21115210 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
20 |
nM |
21115210 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
= |
19950 |
nM |
21115210 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
420 |
nM |
21115213 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21115213 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
880 |
nM |
21115213 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
60 |
nM |
21115213 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
410 |
nM |
21115213 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
5120 |
nM |
21256013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
90 |
nM |
21215623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
21215623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
1.2 |
|
21215623 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
6.6 |
|
21215623 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
670 |
nM |
21174408 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
290 |
nM |
21174408 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
340 |
nM |
21174408 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.163 |
ug/ml |
21158422 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
6.25 |
ug/ml |
18591276 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
1.56 |
ug/ml |
18591276 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
69000 |
nM |
20547797 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
78 |
% |
20606071 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26.4 |
nM |
21324686 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
153.95 |
nM |
21324686 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2702.33 |
nM |
21324686 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
134 |
|
21324686 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26.4 |
nM |
21324692 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
134 |
|
21324692 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
153.95 |
nM |
21324692 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2702.33 |
nM |
21324692 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
820 |
nM |
21353544 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
44 |
nM |
21354800 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
100 |
nM |
21354800 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17.9 |
nM |
21296467 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
19 |
nM |
21296467 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
30.3 |
nM |
21296467 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
37.5 |
nM |
21296467 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
419.8 |
nM |
21296467 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
46 |
% |
21376582 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
89 |
% |
21376582 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
79 |
% |
21376582 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
6300 |
nM |
21429743 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
12300 |
nM |
21429743 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
124000 |
nM |
21429743 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
66200 |
nM |
21429743 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
6800 |
nM |
21429743 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
25300 |
nM |
21429743 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.69 |
ug/ml |
21334795 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
21334795 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.06 |
ug/ml |
21334795 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.41 |
ug/ml |
21334795 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42.8 |
nM |
21435889 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94 |
nM |
21435889 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
94 |
nM |
21435889 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
160 |
nM |
21444205 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
21444205 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2398 |
nM |
21444205 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
79.93 |
|
21444205 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
86.5 |
% |
21507635 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
55 |
% |
21507635 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
Activity |
= |
31.8 |
% |
21507635 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
42800 |
nM |
21504224 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
94000 |
nM |
21504224 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
94000 |
nM |
21504224 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
94000 |
nM |
21504224 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
9700 |
nM |
21341710 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
55 |
% |
21482109 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
96 |
% |
21482109 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
21381705 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
830 |
nM |
21381705 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
20 |
nM |
21381705 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21381705 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
53300 |
nM |
20884091 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
4800 |
nM |
20884091 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
20884091 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
5800 |
nM |
20884091 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
130 |
nM |
21496972 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
130 |
nM |
21496972 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
140 |
nM |
21496972 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
190 |
nM |
21496972 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
190 |
nM |
21496972 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
21425785 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
21425785 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
21425785 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
21425785 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
21425785 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.97 |
ug/ml |
21429629 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
Activity |
= |
72.5 |
% |
21440337 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
76.6 |
% |
21440337 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
Activity |
= |
60.79 |
% |
21440337 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
65.33 |
% |
21440337 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
Activity |
= |
50.97 |
% |
21440337 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
33.88 |
% |
21440337 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
19900 |
nM |
21440337 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
2 |
nM |
19632833 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
100 |
nM |
19632833 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
19632833 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
300 |
nM |
19632833 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
600 |
nM |
19632833 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
700 |
nM |
19632833 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
900 |
nM |
19632833 |
NPT4490 |
Cell Line |
IMR-90 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
19632833 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1000 |
nM |
19632833 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
19632833 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
19632833 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2400 |
nM |
19632833 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
19632833 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
6 |
% |
21531049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
15 |
% |
21531049 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
50 |
% |
21531049 |
NPT1182 |
Cell Line |
J774.A1 |
Mus musculus |
IC50 |
= |
20 |
nM |
21555166 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
100 |
nM |
20673627 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
< |
100 |
nM |
20673627 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
110 |
nM |
20673627 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
170 |
nM |
20673627 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
2100 |
nM |
20673627 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
120 |
nM |
20673627 |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
100 |
nM |
20673627 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
< |
100 |
nM |
20673627 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
20673627 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
130 |
nM |
20673627 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
150 |
nM |
20673627 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1640 |
nM |
21534590 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1130 |
nM |
21553829 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
120 |
nM |
21553829 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
930 |
nM |
21553829 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
21553829 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
600 |
nM |
21553829 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1300 |
nM |
21553829 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
4400 |
nM |
21553829 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21553829 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
21553829 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
21553829 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
6700 |
nM |
21553829 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
600 |
nM |
21553829 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Ratio IC50 |
= |
11.1 |
|
21553829 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21563750 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
120 |
nM |
21663319 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
13150 |
nM |
21663319 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
109.6 |
|
21663319 |
NPT1357 |
Cell Line |
H22 |
Mus musculus |
IC50 |
= |
36510 |
nM |
21620529 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
17540 |
nM |
21620529 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.61 |
ug |
21620529 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.25 |
ug |
21620529 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.15 |
ug |
21620529 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.12 |
ug |
21620529 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
7.31 |
|
21620529 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
GI |
= |
48.22 |
% |
21620529 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
477 |
nM |
21570750 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21570750 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4380 |
nM |
21570750 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
198 |
nM |
21570750 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2947 |
nM |
21570750 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
338 |
nM |
21570750 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-1.6 |
ug |
21570750 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-2.3 |
ug |
21570750 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
TGI |
= |
39.6 |
% |
21570750 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
TGI |
= |
45 |
% |
21570750 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5.5 |
ug/ml |
21723735 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
3.73 |
ug/ml |
21723735 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
21684168 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
0.05 |
ug/ml |
21684168 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
0.08 |
ug/ml |
21684168 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
0.09 |
ug/ml |
21684168 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21601964 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21601964 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1030 |
nM |
21600678 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
21601964 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
700 |
nM |
21601964 |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
Inhibition |
= |
72.1 |
% |
21741833 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2010 |
nM |
21741833 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
42520 |
nM |
21741833 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
30 |
nM |
21741833 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
230 |
nM |
21741833 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
21741833 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
830 |
nM |
21741833 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
70 |
nM |
21741833 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
260 |
nM |
21741833 |
NPT1317 |
Cell Line |
CCRF S-180 |
Mus musculus |
IC50 |
= |
29200 |
nM |
21620529 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
17230 |
nM |
21620529 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
21500 |
nM |
21620529 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.16 |
ug/ml |
21708464 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.51 |
ug/ml |
21708464 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1.6 |
ug/ml |
21708464 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2.3 |
ug/ml |
21708464 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
0.24 |
ug/ml |
21708464 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
110 |
nM |
21737288 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
130 |
nM |
21737288 |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
100 |
nM |
21737288 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
< |
100 |
nM |
21737288 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
100 |
nM |
21737288 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
150 |
nM |
21737288 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
< |
100 |
nM |
21737288 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
310 |
nM |
21704523 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
12200 |
nM |
21704523 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21705223 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
16 |
nM |
21711054 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
5 |
nM |
21711054 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
21 |
nM |
21711054 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
11 |
nM |
21711054 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
6 |
nM |
21711054 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
10 |
nM |
21711054 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
20031423 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
20031423 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
20031423 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
20031423 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
170 |
nM |
20031423 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
20031423 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
20031423 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
20031423 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
20031423 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
20031423 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
20031423 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
21721519 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
21721519 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
< |
10 |
ug/ml |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
TGI |
= |
32.4 |
ug/ml |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
LC50 |
= |
60.9 |
ug/ml |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
Activity |
= |
-66.9 |
% |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
Activity |
= |
-39.5 |
% |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
Activity |
= |
8.2 |
% |
21802797 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
Activity |
= |
10.7 |
% |
21802797 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3700 |
nM |
21704436 |
NPT5532 |
Cell Line |
HCT-29 |
|
IC50 |
= |
2500 |
nM |
21704436 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
21704436 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
21704436 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21704436 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
13000 |
nM |
21827183 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
450 |
nM |
21641694 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
21641694 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
360 |
nM |
21641694 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
60 |
nM |
21641694 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
230 |
nM |
21641694 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Ratio IC50 |
= |
80 |
|
21780800 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
32 |
|
21780800 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
6.1 |
|
21780800 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
10 |
ug/ml |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
TGI |
= |
41.3 |
ug/ml |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
> |
80 |
ug/ml |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
-66.9 |
% |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
-39.5 |
% |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
8.2 |
% |
21802797 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
10.7 |
% |
21802797 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
740 |
nM |
21797280 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
850 |
nM |
21797280 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
500 |
nM |
21797280 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1540 |
nM |
21797280 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
950 |
nM |
21797280 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1630 |
nM |
21797280 |
NPT1160 |
Cell Line |
BJ |
Homo sapiens |
IC50 |
= |
2330 |
nM |
21797280 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
21741131 |
NPT859 |
Cell Line |
HFF |
Homo sapiens |
CC50 |
= |
30 |
nM |
21741131 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
250 |
nM |
21761866 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
43440 |
nM |
21761866 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
173.77 |
|
21761866 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
21676506 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
21676506 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
21676506 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
21676506 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
21676506 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
21676506 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
21676506 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
170 |
nM |
21676506 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
21676506 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
21676506 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
21676506 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
1.2 |
nM |
21774499 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
194 |
nM |
21774499 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5 |
nM |
21774499 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2170 |
nM |
21868138 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
2030 |
nM |
21868138 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
3092 |
nM |
21868138 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3600 |
nM |
21868138 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
3137 |
nM |
21868138 |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
IC50 |
= |
40 |
nM |
21664013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio |
= |
0.291 |
|
21664013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio |
= |
0.42 |
|
21664013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio |
= |
0.439 |
|
21664013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio |
= |
0.523 |
|
21664013 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1.3 |
ug/ml |
21664013 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
490 |
nM |
21885166 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
660 |
nM |
21885166 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
1130 |
nM |
21885166 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1290 |
nM |
21784631 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1570 |
nM |
21784631 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
71800 |
nM |
21890248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.721 |
|
21890248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.546 |
|
21890248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.461 |
|
21890248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.494 |
|
21890248 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
21794959 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
TGI |
> |
100000 |
nM |
21794959 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
< |
100 |
nM |
21794959 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
53.26 |
% |
21885273 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1510 |
nM |
21885273 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8940 |
nM |
21885273 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13600 |
nM |
21885273 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
20000 |
nM |
21885273 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1220 |
nM |
21885273 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
4100 |
nM |
21885273 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
580 |
nM |
21885273 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
6240 |
nM |
21885273 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
1660 |
nM |
21885273 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
7420 |
nM |
21885273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
21.92 |
% |
21885273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
24.62 |
% |
21885273 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
300 |
nM |
21999655 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
600 |
nM |
21999655 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21999655 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
500 |
nM |
21999655 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
300 |
nM |
21999655 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300 |
nM |
21999655 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
21999655 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
800 |
nM |
21999655 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
425 |
nM |
21843940 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17840 |
nM |
21843940 |
NPT199 |
Individual Protein |
DNA polymerase kappa |
Homo sapiens |
Potency |
|
26679.5 |
nM |
PubChem BioAssay data set |
NPT901 |
Individual Protein |
UDP-glucuronosyltransferase 1-1 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT703 |
Individual Protein |
UDP-glucuronosyltransferase 1-9 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT257 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Oryctolagus cuniculus |
IC50 |
= |
13590 |
nM |
DrugMatrix in vitro pharmacology data |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
15336 |
nM |
DrugMatrix in vitro pharmacology data |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ki |
= |
3693 |
nM |
DrugMatrix in vitro pharmacology data |
NPT277 |
Individual Protein |
Caspase-1 |
Homo sapiens |
IC50 |
= |
12192 |
nM |
DrugMatrix in vitro pharmacology data |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
IC50 |
= |
5147 |
nM |
DrugMatrix in vitro pharmacology data |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
IC50 |
= |
2485 |
nM |
DrugMatrix in vitro pharmacology data |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
IC50 |
= |
31913 |
nM |
DrugMatrix in vitro pharmacology data |
NPT289 |
Individual Protein |
Serotonin 1b (5-HT1b) receptor |
Rattus norvegicus |
IC50 |
= |
34464 |
nM |
DrugMatrix in vitro pharmacology data |
NPT289 |
Individual Protein |
Serotonin 1b (5-HT1b) receptor |
Rattus norvegicus |
Ki |
= |
15666 |
nM |
DrugMatrix in vitro pharmacology data |
NPT293 |
Individual Protein |
Serotonin 4 (5-HT4) receptor |
Cavia porcellus |
IC50 |
= |
12468 |
nM |
DrugMatrix in vitro pharmacology data |
NPT293 |
Individual Protein |
Serotonin 4 (5-HT4) receptor |
Cavia porcellus |
Ki |
= |
2078 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15245 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
13668 |
nM |
DrugMatrix in vitro pharmacology data |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
270 |
nM |
21875046 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
GI50 |
= |
10 |
nM |
21875046 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
120 |
nM |
21875046 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
90 |
nM |
21875046 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
EC50 |
= |
2500 |
nM |
21882827 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
477 |
nM |
21983438 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
400 |
nM |
21983438 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
456 |
nM |
21983438 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
FC |
= |
6 |
|
21882827 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21996519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
21996519 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
< |
1000 |
nM |
21996519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
1000 |
nM |
21996519 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
21996519 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
180 |
nM |
22000924 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
GI50 |
= |
130 |
nM |
22000924 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
700 |
nM |
22014995 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
8700 |
nM |
22014995 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
710 |
nM |
22014995 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4700 |
nM |
21721528 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
140 |
nM |
21721528 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
= |
9300 |
nM |
21721528 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21721528 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
420 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2020 |
nM |
21721528 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
390 |
nM |
21721528 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3060 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
50 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
80 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
690 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
2700 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
530 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
17480 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
380 |
nM |
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
1580 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
240 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
870 |
nM |
21721528 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
10 |
nM |
21721528 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
240 |
nM |
21721528 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
200 |
nM |
21721528 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
19720 |
nM |
21721528 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
80 |
nM |
21721528 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
9700 |
nM |
21721528 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
235 |
|
21721528 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
Ratio IC50 |
= |
66.4 |
|
21721528 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Ratio IC50 |
= |
46.9 |
|
21721528 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
56 |
|
21721528 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Ratio IC50 |
= |
7.8 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
1.7 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
13.8 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
59.7 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
11.7 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
386.7 |
|
21721528 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
55.4 |
|
21721528 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
27.14 |
|
21721528 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
Ratio IC50 |
= |
17.5 |
|
21721528 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
Ratio IC50 |
= |
98.6 |
|
21721528 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
Ratio IC50 |
= |
129.3 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
8.5 |
|
21721528 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
Ratio IC50 |
= |
34.9 |
|
21721528 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
770 |
nM |
21800859 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1930 |
nM |
21800859 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
590 |
nM |
21800859 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
260 |
nM |
21800859 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1030 |
nM |
21800859 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
630 |
nM |
21800859 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
120 |
nM |
22027100 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
109.6 |
|
22027100 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
13100 |
nM |
22027100 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4500 |
nM |
22000946 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
22000946 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
GI |
= |
51.18 |
% |
22004723 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
GI |
= |
6.53 |
% |
22004723 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI |
= |
45.13 |
% |
22004723 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
420 |
nM |
22070654 |
NPT181 |
Cell Line |
Bel-7402 |
Homo sapiens |
IC50 |
= |
530 |
nM |
22070654 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
720 |
nM |
22070654 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
980 |
nM |
22070654 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
330 |
nM |
22070654 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
960 |
nM |
22000949 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
20 |
nM |
22000949 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
22000949 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
22000949 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6860 |
nM |
22119131 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5460 |
nM |
22119131 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7360 |
nM |
22119131 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6860 |
nM |
22119132 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5460 |
nM |
22119132 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7360 |
nM |
22119132 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
68.8 |
nM |
22177409 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
86 |
nM |
22177409 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
91.5 |
nM |
22177409 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2180 |
nM |
22136907 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
5510 |
nM |
22136907 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1020 |
nM |
22209733 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
30 |
nM |
22209733 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
22209733 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2510 |
nM |
22209733 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
250 |
nM |
22100139 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2020 |
nM |
22136907 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1060 |
nM |
22136907 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
790 |
nM |
22136907 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
13600 |
nM |
22148280 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
430 |
nM |
22119124 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
56830 |
nM |
22119124 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
132.2 |
|
22119124 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
5230 |
nM |
22123320 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11670 |
nM |
22123320 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3070 |
nM |
22123320 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
15650 |
nM |
22123320 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
18230 |
nM |
22123320 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
62260 |
nM |
22123320 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
88 |
% |
22123322 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
72 |
% |
22123322 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
81 |
% |
22123322 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
64 |
% |
22123322 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI |
= |
90 |
% |
22123322 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
86 |
% |
22123322 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.73 |
ug/ml |
22178093 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
6610 |
nM |
22182926 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8650 |
nM |
22182926 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1120 |
nM |
22182926 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
65250 |
nM |
22182926 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
100 |
nM |
22104151 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
< |
100 |
nM |
22104151 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
< |
100 |
nM |
22104151 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
14700 |
nM |
22104151 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
1900 |
nM |
22104151 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
13010 |
nM |
22104151 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
160 |
nM |
22104151 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
22197145 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
22197145 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
83200 |
nM |
22197145 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
22197145 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
330 |
nM |
22004007 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2290 |
nM |
22004007 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
110 |
nM |
22004007 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
81 |
% |
22257529 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
17.8 |
% |
22257529 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
0.9 |
% |
22257529 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
29.8 |
% |
22257529 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
68 |
% |
22257529 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
1.9 |
% |
22257529 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
22044164 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
22044164 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
22044164 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
22044164 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
31 |
% |
22209415 |
NPT76 |
Cell Line |
C6 |
Rattus norvegicus |
Inhibition |
= |
27 |
% |
22209415 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
7000 |
nM |
22182501 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
85 |
% |
22245048 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
76 |
% |
22245048 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Activity |
= |
20 |
% |
22304849 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
20 |
% |
22304849 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1280 |
nM |
22318164 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2850 |
nM |
22318164 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
860 |
nM |
22318164 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3690 |
nM |
22318164 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1450 |
nM |
22318164 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17900 |
nM |
22280818 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
160 |
nM |
22280818 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
900 |
nM |
22280818 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
28810 |
nM |
22280818 |
NPT317 |
Uncleic Acid |
Nucleic Acid |
|
Inhibition |
= |
83 |
% |
22257890 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
22357112 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
5 |
% |
22357112 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
13 |
% |
22357112 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17 |
% |
22357112 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
33 |
% |
22357112 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
22361684 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
22361684 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
22361684 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
22361684 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
22361684 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
22361684 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
22361684 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
22361684 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
22361684 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1810 |
nM |
22361684 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
140 |
nM |
22361684 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
22364746 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
22364746 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
22364746 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
22364746 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
22364746 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
22364746 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
22364746 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
22364746 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
5800 |
nM |
22326399 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
22326399 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22330634 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
< |
100 |
nM |
22330634 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.73 |
ug/ml |
22370339 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.97 |
ug/ml |
22370339 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
1700 |
nM |
22304344 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7100 |
nM |
22304344 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
22304344 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5300 |
nM |
22304344 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
22304344 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6900 |
nM |
22304344 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8140 |
nM |
22386528 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
970 |
nM |
22386528 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
15070 |
nM |
22386528 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
14840 |
nM |
22386528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
46690 |
nM |
22405646 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
430 |
nM |
22405646 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
108 |
|
22405646 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
0.27 |
ug/ml |
22410248 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
0.24 |
ug/ml |
22410248 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
22410248 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
0.18 |
ug/ml |
22410248 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.14 |
ug/ml |
22410248 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
0.068 |
ug/ml |
22410248 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.27 |
ug/ml |
22410248 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2500 |
nM |
22272829 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
6060 |
nM |
22272829 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6040 |
nM |
22272829 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
3140 |
nM |
22272829 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
19510 |
nM |
22276650 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
23480 |
nM |
22276650 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
16020 |
nM |
22276650 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8090 |
nM |
22444025 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
22444025 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6860 |
nM |
22444025 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5000 |
nM |
22283451 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7000 |
nM |
22283451 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7000 |
nM |
22283451 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
22283451 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
22283451 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
172000 |
nM |
22283451 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
65 |
% |
22472045 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2 |
nM |
22483395 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2 |
nM |
22483395 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
2 |
nM |
22483395 |
NPT574 |
Cell Line |
XF498 |
Homo sapiens |
IC50 |
= |
15 |
nM |
22483395 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
35 |
nM |
22483395 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
46690 |
nM |
22429509 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
430 |
nM |
22429509 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
108 |
|
22429509 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2500000 |
nM |
22440624 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5000000 |
nM |
22440624 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
2500000 |
nM |
22440624 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
190 |
nM |
22414612 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
22414612 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
22464458 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3690 |
nM |
22472043 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1180 |
nM |
22472043 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Ratio IC50 |
= |
3.1 |
|
22472043 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
22276998 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
45 |
nM |
22276998 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
Inhibition |
= |
69.1 |
% |
22276998 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
Activity |
= |
51.5 |
% |
22276998 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1540 |
nM |
22316168 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1900 |
nM |
22316168 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
210 |
nM |
22316168 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
546 |
nM |
22316168 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
180 |
nM |
22316168 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
98320 |
nM |
22316168 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
64300 |
nM |
22316168 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
24900344 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
Activity |
= |
63 |
% |
24900344 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
83 |
% |
24900344 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
Activity |
= |
61 |
% |
24900344 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
24900344 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
24900344 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
24900344 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
> |
20000 |
nM |
24900344 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
200 |
nM |
24900344 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2 |
% |
24900344 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
100 |
nM |
22250891 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
420 |
nM |
22264149 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
620 |
nM |
22264149 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
420 |
nM |
22264149 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
240 |
nM |
22264149 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
580 |
nM |
22264149 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
540 |
nM |
22537362 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
50000 |
nM |
22537362 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
12 |
nM |
22537362 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
450 |
nM |
22537362 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
370 |
nM |
22537362 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
170 |
nM |
22537362 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI |
= |
2.4 |
nM |
22537680 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
3.7 |
nM |
22537680 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
13.5 |
nM |
22537680 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI |
= |
2.1 |
nM |
22537680 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI |
= |
1.3 |
nM |
22537680 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI |
= |
6.3 |
nM |
22537680 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
13.9 |
nM |
22537680 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
22413887 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.31 |
ug/ml |
22413887 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.8 |
ug/ml |
22413887 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1.4 |
ug/ml |
22413887 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
0.31 |
ug/ml |
22413887 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1.39 |
ug/ml |
22413887 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
GI |
= |
0.8 |
nM |
22537680 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2820 |
nM |
22542958 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3280 |
nM |
22542958 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5220 |
nM |
22542958 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1700 |
nM |
22482432 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16800 |
nM |
22482432 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
100 |
nM |
22482432 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
114 |
nM |
24900437 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1300 |
nM |
22555152 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
IC50 |
= |
40 |
nM |
22555152 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
30 |
nM |
22555152 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
40 |
nM |
22555152 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
50 |
nM |
22555152 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
22555152 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
60 |
nM |
22555152 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.551 |
% |
22583778 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.48 |
% |
22583778 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.139 |
% |
22583778 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.13 |
% |
22583778 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
32000 |
nM |
22583778 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
390 |
nM |
22555152 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
22520152 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
22520152 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
8000 |
nM |
22520152 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
22647719 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
3200 |
nM |
22647719 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5570 |
nM |
22647723 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
17670 |
nM |
22647723 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
168 |
nM |
22647723 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.2 |
ug/ml |
22658083 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.36 |
ug/ml |
22658083 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
5900 |
nM |
22668451 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
19300 |
nM |
22668451 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
30 |
nM |
22668451 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
5600 |
nM |
22668451 |
NPT5192 |
Cell Line |
U-937/GTB |
Homo sapiens |
IC50 |
= |
160 |
nM |
21434649 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
21852132 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1410 |
nM |
22677031 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
310 |
nM |
22677031 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
330 |
nM |
22677031 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Survival |
= |
11.9 |
% |
22677031 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
23.6 |
% |
22677031 |
NPT1182 |
Cell Line |
J774.A1 |
Mus musculus |
CC50 |
= |
20 |
nM |
22608675 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
22608675 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
320 |
nM |
22770744 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1170 |
nM |
22770744 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
95610 |
nM |
22770744 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
120 |
nM |
22770744 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
750 |
nM |
22770744 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
120 |
nM |
22770744 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
22632935 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Activity |
= |
78.2 |
% |
22633832 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
78.2 |
% |
22633832 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
430 |
nM |
22450134 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
46690 |
nM |
22450134 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
= |
108 |
|
22450134 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1600 |
nM |
22530813 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2600 |
nM |
22530813 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
2600 |
nM |
22530813 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
22530813 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1600 |
nM |
22530813 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
1630 |
nM |
22738641 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
1660 |
nM |
22738641 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
22738641 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
1340 |
nM |
22738641 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
GI50 |
= |
1000 |
nM |
22738641 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1650 |
nM |
22738641 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
3300 |
nM |
22652254 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
6400 |
nM |
22766218 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
320 |
nM |
22515366 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
340 |
nM |
22515366 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
790 |
nM |
22515366 |
NPT3998 |
Cell Line |
LLC cell line |
|
IC50 |
= |
207 |
nM |
22515366 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-21 |
% |
22515366 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
700 |
nM |
22749279 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
600 |
nM |
22749279 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
22749279 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
900 |
nM |
22749279 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
300 |
nM |
22749279 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
3400 |
nM |
22749279 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
60 |
nM |
22616554 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4600 |
nM |
22616554 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1820 |
nM |
22819942 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1760 |
nM |
22819942 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1570 |
nM |
22819942 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
22819942 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
8460 |
nM |
22687747 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
13240 |
nM |
22687747 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
3790 |
nM |
22687747 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1370 |
nM |
22687747 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
22889559 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8620 |
nM |
22818039 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
2760 |
nM |
22818039 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
19010 |
nM |
22818039 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10860 |
nM |
22818039 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
20930 |
nM |
22818039 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
10530 |
nM |
22818039 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Ratio IC50 |
= |
2 |
|
22931300 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2140 |
nM |
22663190 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
4700 |
nM |
22742761 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1700 |
nM |
22742761 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
60 |
nM |
22858298 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
14 |
nM |
22858298 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
5 |
nM |
22858298 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
6.7 |
nM |
22858298 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Ratio IC50 |
> |
5 |
|
22931300 |
NPT1422 |
Individual Protein |
ATP-binding cassette sub-family G member 2 |
Homo sapiens |
Activity |
= |
72 |
% |
12682043 |
NPT957 |
Individual Protein |
Multidrug resistance-associated protein 7 |
Homo sapiens |
Activity |
= |
18.2 |
% |
12527806 |
NPT2850 |
Individual Protein |
Multidrug resistance associated protein |
Homo sapiens |
Activity |
= |
80 |
% |
11585759 |
NPT1594 |
Individual Protein |
Multidrug resistance-associated protein 1 |
Homo sapiens |
IC50 |
= |
50000 |
nM |
8621644 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
Ki |
= |
8500 |
nM |
11405287 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
40 |
nM |
22944121 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5270 |
nM |
22944121 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
131.8 |
|
22944121 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
22944121 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
250 |
nM |
22944121 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
25 |
|
22944121 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1 |
nM |
22951040 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
4 |
nM |
22951040 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
4 |
nM |
22951040 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
82 |
nM |
22951040 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
8600 |
nM |
24900509 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1050 |
nM |
24900509 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
24900509 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
FC |
= |
1.2 |
|
22612652 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
52 |
% |
22982122 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI |
= |
26 |
% |
22982122 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
GI |
= |
83 |
% |
22982122 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
GI |
= |
73 |
% |
22982122 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
45 |
% |
22982122 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
GI |
= |
56 |
% |
22982122 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
75 |
% |
22982122 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
37 |
nM |
22884578 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
5200 |
nM |
22884578 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
> |
140 |
|
22884578 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5.4 |
nM |
23085106 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
11100 |
nM |
22586124 |
NPT474 |
Organism |
Plasmodium berghei |
Plasmodium berghei |
IC50 |
= |
886 |
nM |
22586124 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
58 |
nM |
22586124 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
37.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6676.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3317.3 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
22582991 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
440 |
nM |
22582991 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
110 |
nM |
22582991 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
5.3 |
|
22582991 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
15 |
|
22582991 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
50 |
|
22582991 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
100 |
|
22582991 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
> |
10 |
|
22582991 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Ratio IC50 |
> |
20 |
|
22582991 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
6.7 |
|
22582991 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
> |
15 |
|
22582991 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
Ratio IC50 |
= |
6.1 |
|
22582991 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
22946634 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
22946634 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
30 |
nM |
23039861 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
23043498 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
2700 |
nM |
23043498 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2700 |
nM |
23043498 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
GI |
= |
92.1 |
% |
23124210 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
GI |
= |
92.1 |
% |
23124210 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
GI |
= |
99.2 |
% |
23124210 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
700 |
nM |
23124210 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1280 |
nM |
23124210 |
NPT26 |
Individual Protein |
Reverse transcriptase |
Human immunodeficiency virus 1 |
IC50 |
= |
52000 |
nM |
22695131 |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Ki |
= |
230000 |
nM |
22541068 |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
IC50 |
= |
240000 |
nM |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Ki |
= |
38000 |
nM |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
IC50 |
= |
41000 |
nM |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Ki |
= |
150000 |
nM |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
IC50 |
= |
160000 |
nM |
22541068 |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Inhibition |
= |
49.9 |
% |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
26.6 |
% |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
-5.8 |
% |
22541068 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
400 |
nM |
23148652 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
40 |
nM |
23148652 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
FC |
= |
50 |
|
21348461 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
> |
5000 |
nM |
21348461 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
GI50 |
> |
5000 |
nM |
21348461 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
GI |
= |
40 |
% |
22916727 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
1340 |
nM |
22503656 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1050 |
nM |
22503656 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
22503656 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1030 |
nM |
22503656 |
NPT683 |
Individual Protein |
Aldehyde reductase |
Homo sapiens |
Activity |
= |
11 |
nmol/min |
22982121 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
22 |
nM |
23072299 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
40 |
nM |
23072299 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
990 |
nM |
23072299 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
23072299 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
Ratio IC50 |
= |
0.15 |
|
23079523 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
5.03 |
|
23079523 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
Ratio IC50 |
= |
2.09 |
|
23079523 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
Ratio IC50 |
= |
31.83 |
|
23079523 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
1910 |
nM |
23079523 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
31.95 |
|
23079523 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12140 |
nM |
23079523 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
380 |
nM |
23079523 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
15.17 |
|
23079523 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
910 |
nM |
23079523 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
60 |
nM |
23079523 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
23079527 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
23079527 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
23079527 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
< |
1000 |
nM |
23079527 |
NPT2 |
Others |
Unspecified |
|
Survival |
= |
22 |
day |
22985027 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
100 |
|
22985027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6700 |
nM |
22985027 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
50 |
nM |
22985027 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
115 |
% |
22985027 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.5 |
% |
22985027 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
49.1 |
% |
22985027 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
37.6 |
% |
22985027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
2.75 |
ug/ml |
23123017 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.003 |
ug/ml |
23123017 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3.2 |
ug/ml |
23123017 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
3.4 |
ug/ml |
23123017 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
629 |
nM |
23123017 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1700 |
nM |
23145909 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
4700 |
nM |
23145909 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
Ratio IC50 |
= |
109.6 |
|
23117171 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13150 |
nM |
23117171 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
120 |
nM |
23117171 |
NPT1377 |
Individual Protein |
Carnitine palmitoyltransferase 2 |
Rattus norvegicus |
IC50 |
> |
100000 |
nM |
21504156 |
NPT5534 |
Individual Protein |
Carnitine palmitoyltransferase 1A |
Rattus norvegicus |
IC50 |
= |
250000 |
nM |
21504156 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.48 |
ug/ml |
10.1007/s00044-011-9894-8 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
10.1007/s00044-011-9894-8 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.01 |
ug/ml |
10.1007/s00044-011-9894-8 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
10.1007/s00044-011-9894-8 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
63000 |
nM |
10.1007/s00044-011-9761-7 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
10.1007/s00044-011-9903-y |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.39 |
ug/ml |
10.1007/s00044-011-9903-y |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.45 |
ug/ml |
10.1007/s00044-011-9903-y |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
2 |
|
10.1007/s00044-011-9832-9 |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
1 |
|
10.1007/s00044-011-9832-9 |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
0.2 |
cm |
10.1007/s00044-011-9832-9 |
NPT2640 |
Organism |
Bacopa monnieri |
Bacopa monnieri |
Activity |
= |
0 |
|
10.1007/s00044-011-9832-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2970 |
nM |
10.1007/s00044-011-9874-z |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7.5 |
ug/ml |
23024574 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.16 |
ug/ml |
10.1007/s00044-011-9882-z |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
< |
1000 |
nM |
10.1007/s00044-011-9884-x |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
1000 |
nM |
10.1007/s00044-011-9884-x |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
10.1007/s00044-011-9884-x |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
10.1007/s00044-011-9884-x |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
32000 |
nM |
10.1007/s00044-011-9751-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.125 |
|
10.1007/s00044-011-9751-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.122 |
|
10.1007/s00044-011-9751-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.479 |
|
10.1007/s00044-011-9751-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.537 |
|
10.1007/s00044-011-9751-9 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
TGI |
= |
169.82 |
nM |
10.1007/s00044-011-9561-0 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
TGI |
= |
2089.3 |
nM |
10.1007/s00044-011-9561-0 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
199.53 |
nM |
10.1007/s00044-011-9561-0 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
TGI |
= |
2344.23 |
nM |
10.1007/s00044-011-9561-0 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
GI50 |
= |
112.2 |
nM |
10.1007/s00044-011-9561-0 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
131.83 |
nM |
10.1007/s00044-011-9561-0 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
120.23 |
nM |
10.1007/s00044-011-9561-0 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
123.03 |
nM |
10.1007/s00044-011-9561-0 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
39 |
nM |
10.1007/s00044-010-9340-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
211 |
nM |
10.1007/s00044-010-9340-3 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
10.1007/s00044-010-9340-3 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
53 |
nM |
10.1007/s00044-010-9340-3 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
100 |
nM |
10.1007/s00044-010-9517-9 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
70 |
nM |
10.1007/s00044-010-9517-9 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
90 |
nM |
10.1007/s00044-010-9517-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
71800 |
nM |
10.1007/s00044-010-9332-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.494 |
|
10.1007/s00044-010-9332-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.461 |
|
10.1007/s00044-010-9332-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.546 |
|
10.1007/s00044-010-9332-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
0.721 |
|
10.1007/s00044-010-9332-3 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1007/s00044-009-9222-8 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
17 |
ug/ml |
10.1007/s00044-010-9433-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Survival |
= |
35.87 |
% |
10.1007/s00044-010-9433-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Survival |
= |
51.22 |
% |
10.1007/s00044-010-9433-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Survival |
= |
74.21 |
% |
10.1007/s00044-010-9433-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Survival |
= |
90.02 |
% |
10.1007/s00044-010-9433-z |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
750 |
nM |
10.1007/s00044-011-9587-3 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
5000 |
nM |
10.1007/s00044-011-9587-3 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
800 |
nM |
10.1007/s00044-011-9587-3 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
< |
550 |
nM |
10.1007/s00044-011-9587-3 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
< |
550 |
nM |
10.1007/s00044-011-9587-3 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
550 |
nM |
10.1007/s00044-011-9587-3 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
19 |
ug/ml |
10.1007/s00044-010-9436-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.97 |
ug/ml |
10.1007/s00044-011-9636-y |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3220 |
nM |
10.1007/s00044-011-9653-x |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5230 |
nM |
10.1007/s00044-011-9653-x |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
GI50 |
< |
100 |
nM |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
TGI |
< |
100 |
nM |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
LC50 |
= |
170 |
nM |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
Activity |
= |
-70.7 |
% |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
Activity |
= |
-64.2 |
% |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
Activity |
= |
-62.5 |
% |
10.1007/s00044-012-0084-0 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
Activity |
= |
-24 |
% |
10.1007/s00044-012-0084-0 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
3170 |
nM |
10.1007/s00044-012-0150-7 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
16 |
nM |
10.1007/s00044-012-0051-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1080 |
nM |
10.1007/s00044-012-0057-3 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1190 |
nM |
10.1007/s00044-012-0057-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1280 |
nM |
10.1007/s00044-012-0057-3 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
10.1007/s00044-012-0150-7 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2670 |
nM |
10.1007/s00044-012-0150-7 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.12 |
ug/ml |
10.1007/s00044-012-0168-x |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1.81 |
ug/ml |
10.1007/s00044-012-0168-x |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
43.13 |
% |
10.1007/s00044-012-0168-x |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
22.85 |
% |
10.1007/s00044-012-0168-x |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
10.1007/s00044-012-0098-7 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1760 |
nM |
10.1007/s00044-013-0584-6 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10900 |
nM |
10.1007/s00044-013-0584-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1880 |
nM |
10.1007/s00044-013-0584-6 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
640 |
nM |
10.1007/s00044-013-0584-6 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
19000 |
nM |
10.1007/s00044-013-0586-4 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
24270 |
nM |
10.1007/s00044-012-0018-x |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
19900 |
nM |
10.1007/s00044-012-0018-x |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
18 |
ug/ml |
10.1007/s00044-012-0071-5 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
30 |
nM |
10.1007/s00044-012-0232-6 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1760 |
nM |
10.1007/s00044-012-0232-6 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
110 |
nM |
10.1007/s00044-012-0232-6 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
90 |
nM |
10.1007/s00044-012-0232-6 |
NPT5198 |
Cell Line |
OVCAR |
Homo sapiens |
GI50 |
= |
950 |
nM |
10.1007/s00044-012-0232-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.38 |
ug/ml |
10.1007/s00044-012-0025-y |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.23 |
ug/ml |
10.1007/s00044-012-0025-y |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.35 |
ug/ml |
10.1007/s00044-012-0025-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
330 |
nM |
10.1007/s00044-012-0232-6 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
GI50 |
= |
20 |
nM |
10.1007/s00044-012-0232-6 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
0.24 |
ug/ml |
10.1007/s00044-012-0236-2 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
10.1007/s00044-012-0236-2 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
0.48 |
ug/ml |
10.1007/s00044-012-0236-2 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.02 |
ug/ml |
10.1007/s00044-012-0236-2 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI |
= |
93.6 |
% |
10.1007/s00044-012-0236-2 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
GI |
= |
95.2 |
% |
10.1007/s00044-012-0236-2 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI |
= |
91.1 |
% |
10.1007/s00044-012-0236-2 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
4890 |
nM |
10.1007/s00044-013-0558-8 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3270 |
nM |
10.1007/s00044-013-0558-8 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
99.5 |
% |
10.1007/s00044-013-0534-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
88.9 |
% |
10.1007/s00044-013-0534-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
70.3 |
% |
10.1007/s00044-013-0534-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
50.8 |
% |
10.1007/s00044-013-0534-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7200 |
nM |
10.1007/s00044-013-0534-3 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
350 |
nM |
10.1007/s00044-012-0428-9 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
30 |
nM |
10.1007/s00044-012-0428-9 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1007/s00044-012-0428-9 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
4490 |
nM |
10.1007/s00044-012-0436-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
10.1007/s00044-012-0436-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7360 |
nM |
10.1007/s00044-013-0497-4 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
840 |
nM |
10.1007/s00044-013-0497-4 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5460 |
nM |
10.1007/s00044-013-0497-4 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
6860 |
nM |
10.1007/s00044-013-0497-4 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
10.1007/s00044-012-0450-y |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
< |
1000 |
nM |
10.1007/s00044-012-0450-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
710 |
nM |
10.1007/s00044-012-0370-x |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
8700 |
nM |
10.1007/s00044-012-0370-x |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1007/s00044-012-0370-x |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
6.33 |
% |
10.1007/s00044-012-0373-7 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
12 |
% |
10.1007/s00044-012-0373-7 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Activity |
= |
9 |
% |
10.1007/s00044-012-0373-7 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
90 |
nM |
10.1007/s00044-012-0213-9 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
90 |
nM |
10.1007/s00044-012-0213-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
40 |
nM |
10.1007/s00044-012-0213-9 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1007/s00044-012-0272-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
EC50 |
= |
2500 |
nM |
10.1007/s00044-012-0294-5 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
78.2 |
% |
10.1007/s00044-012-0294-5 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
420 |
nM |
10.1007/s00044-012-0402-6 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1007/s00044-012-0402-6 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
640 |
nM |
10.1007/s00044-012-0402-6 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
2840 |
nM |
23245571 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
30 |
nM |
23245571 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
23940 |
nM |
23313636 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
960 |
nM |
23313636 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
85460 |
nM |
23290052 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
290 |
nM |
23290052 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
190 |
nM |
23290052 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
200 |
nM |
23218718 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
200 |
nM |
23218718 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
330 |
nM |
23218718 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23218718 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2200 |
nM |
23218718 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
630 |
nM |
23291120 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10 |
nM |
23470139 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
60.52 |
|
23360284 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2300 |
nM |
23360284 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38 |
nM |
23360284 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
161 |
nM |
23360521 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
23360521 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
93 |
nM |
23360521 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
300 |
nM |
23360521 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
43 |
nM |
23360521 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3 |
|
24900668 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
730 |
nM |
24900668 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
24900668 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
12 |
% |
24900668 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
60000 |
nM |
24900668 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4000 |
nM |
24900668 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
60000 |
nM |
24900668 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
55700 |
nM |
24900668 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Ratio IC50 |
= |
3 |
|
23168081 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
23353747 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
550 |
nM |
23806072 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
49 |
nM |
23544451 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
280 |
nM |
23544451 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11296 |
nM |
23445496 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
118 |
|
23445496 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
95.6 |
nM |
23445496 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
1330 |
nM |
23434227 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1650 |
nM |
23434227 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
540 |
nM |
23434227 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
680 |
nM |
23434227 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
9200 |
nM |
23547843 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
1600 |
nM |
23547843 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3900 |
nM |
23547843 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1500 |
nM |
23547843 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
2600 |
nM |
23547843 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
3700 |
nM |
23547843 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3800 |
nM |
23547843 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
200 |
nM |
23547843 |
NPT2268 |
Cell Line |
DOK |
Homo sapiens |
IC50 |
= |
1017.62 |
nM |
10.6019/CHEMBL1201861 |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
372.72 |
nM |
10.6019/CHEMBL1201861 |
NPT4600 |
Cell Line |
DV-90 |
Homo sapiens |
IC50 |
= |
329.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1184 |
Cell Line |
Daoy |
Homo sapiens |
IC50 |
= |
8.073 |
nM |
10.6019/CHEMBL1201861 |
NPT464 |
Cell Line |
Daudi |
Homo sapiens |
IC50 |
= |
68.96 |
nM |
10.6019/CHEMBL1201861 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
73.73 |
nM |
10.6019/CHEMBL1201861 |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
12.1 |
nM |
10.6019/CHEMBL1201861 |
NPT4601 |
Cell Line |
EHEB |
Homo sapiens |
IC50 |
= |
112.59 |
nM |
10.6019/CHEMBL1201861 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
871.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
325.41 |
nM |
10.6019/CHEMBL1201861 |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
13.72 |
nM |
10.6019/CHEMBL1201861 |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
6.109 |
nM |
10.6019/CHEMBL1201861 |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
39.22 |
nM |
10.6019/CHEMBL1201861 |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
89.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2270 |
Cell Line |
Detroit562 |
Homo sapiens |
IC50 |
= |
230.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2271 |
Cell Line |
DoTc2-4510 |
Homo sapiens |
IC50 |
= |
36.25 |
nM |
10.6019/CHEMBL1201861 |
NPT1906 |
Cell Line |
EB-3 |
Homo sapiens |
IC50 |
= |
771.02 |
nM |
10.6019/CHEMBL1201861 |
NPT1907 |
Cell Line |
EB2 |
Homo sapiens |
IC50 |
= |
33.73 |
nM |
10.6019/CHEMBL1201861 |
NPT1908 |
Cell Line |
EC-GI-10 |
Homo sapiens |
IC50 |
= |
8686.86 |
nM |
10.6019/CHEMBL1201861 |
NPT1910 |
Cell Line |
ECC4 |
Homo sapiens |
IC50 |
= |
4765.41 |
nM |
10.6019/CHEMBL1201861 |
NPT4602 |
Cell Line |
EFE-184 |
Homo sapiens |
IC50 |
= |
8372.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2272 |
Cell Line |
EFM-19 |
Homo sapiens |
IC50 |
= |
478.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2273 |
Cell Line |
EFO-21 |
Homo sapiens |
IC50 |
= |
361.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2274 |
Cell Line |
EFO-27 |
Homo sapiens |
IC50 |
= |
97.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2275 |
Cell Line |
EGI-1 |
Homo sapiens |
IC50 |
= |
598.27 |
nM |
10.6019/CHEMBL1201861 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
18297.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
215.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
32.89 |
nM |
10.6019/CHEMBL1201861 |
NPT4603 |
Cell Line |
C-4-II |
Homo sapiens |
IC50 |
= |
472.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2279 |
Cell Line |
COLO-792 |
Homo sapiens |
IC50 |
= |
3028.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
171.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1189 |
Cell Line |
DG-75 |
Homo sapiens |
IC50 |
= |
665.83 |
nM |
10.6019/CHEMBL1201861 |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
102.25 |
nM |
10.6019/CHEMBL1201861 |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
2291.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2281 |
Cell Line |
ABC-1 |
Homo sapiens |
IC50 |
= |
83.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
2513.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2282 |
Cell Line |
C32 |
Homo sapiens |
IC50 |
= |
32872.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2284 |
Cell Line |
C3A |
Homo sapiens |
IC50 |
= |
415.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
3573.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2283 |
Cell Line |
DK-MG |
Homo sapiens |
IC50 |
= |
50681.55 |
nM |
10.6019/CHEMBL1201861 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
396.31 |
nM |
10.6019/CHEMBL1201861 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
49.34 |
nM |
10.6019/CHEMBL1201861 |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
31.12 |
nM |
10.6019/CHEMBL1201861 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
33.31 |
nM |
10.6019/CHEMBL1201861 |
NPT1917 |
Cell Line |
CA46 |
Homo sapiens |
IC50 |
= |
136.88 |
nM |
10.6019/CHEMBL1201861 |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
1274.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2285 |
Cell Line |
COR-L105 |
Homo sapiens |
IC50 |
= |
188.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
31.96 |
nM |
10.6019/CHEMBL1201861 |
NPT1918 |
Cell Line |
DMS-79 |
Homo sapiens |
IC50 |
= |
2909.88 |
nM |
10.6019/CHEMBL1201861 |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
19.99 |
nM |
10.6019/CHEMBL1201861 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
13.27 |
nM |
10.6019/CHEMBL1201861 |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
65.03 |
nM |
10.6019/CHEMBL1201861 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
IC50 |
= |
375.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2286 |
Cell Line |
CAL-120 |
Homo sapiens |
IC50 |
= |
777.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2289 |
Cell Line |
CAL-12T |
Homo sapiens |
IC50 |
= |
20.65 |
nM |
10.6019/CHEMBL1201861 |
NPT1921 |
Cell Line |
COR-L279 |
Homo sapiens |
IC50 |
= |
56.95 |
nM |
10.6019/CHEMBL1201861 |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
4395.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1923 |
Cell Line |
DMS-153 |
Homo sapiens |
IC50 |
= |
698.15 |
nM |
10.6019/CHEMBL1201861 |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
IC50 |
= |
78.9 |
nM |
10.6019/CHEMBL1201861 |
NPT4604 |
Cell Line |
DMS-53 |
Homo sapiens |
IC50 |
= |
6171.06 |
nM |
10.6019/CHEMBL1201861 |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
281.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2288 |
Cell Line |
AN3-CA |
Homo sapiens |
IC50 |
= |
72.32 |
nM |
10.6019/CHEMBL1201861 |
NPT1925 |
Cell Line |
CAL-148 |
Homo sapiens |
IC50 |
= |
26.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2290 |
Cell Line |
CAL-27 |
Homo sapiens |
IC50 |
= |
32.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2291 |
Cell Line |
CP50-MEL-B |
Homo sapiens |
IC50 |
= |
3987.03 |
nM |
10.6019/CHEMBL1201861 |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
2017.67 |
nM |
10.6019/CHEMBL1201861 |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
21.24 |
nM |
10.6019/CHEMBL1201861 |
NPT1927 |
Cell Line |
ARH-77 |
Homo sapiens |
IC50 |
= |
109.99 |
nM |
10.6019/CHEMBL1201861 |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
127.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
104.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2292 |
Cell Line |
CAL-33 |
Homo sapiens |
IC50 |
= |
67.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2293 |
Cell Line |
CAL-39 |
Homo sapiens |
IC50 |
= |
98.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2299 |
Cell Line |
CAL-51 |
Homo sapiens |
IC50 |
= |
17.32 |
nM |
10.6019/CHEMBL1201861 |
NPT1929 |
Cell Line |
CPC-N |
Homo sapiens |
IC50 |
= |
68.4 |
nM |
10.6019/CHEMBL1201861 |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
64.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2294 |
Cell Line |
23132-87 |
Homo sapiens |
IC50 |
= |
15.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
31.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2302 |
Cell Line |
639-V |
Homo sapiens |
IC50 |
= |
15.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
855.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2300 |
Cell Line |
CAL-54 |
Homo sapiens |
IC50 |
= |
300.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2301 |
Cell Line |
CAL-62 |
Homo sapiens |
IC50 |
= |
32.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
16.07 |
nM |
10.6019/CHEMBL1201861 |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
213278.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2303 |
Cell Line |
647-V |
Homo sapiens |
IC50 |
= |
18.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
19.09 |
nM |
10.6019/CHEMBL1201861 |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
29.85 |
nM |
10.6019/CHEMBL1201861 |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
7417.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2304 |
Cell Line |
CAL-72 |
Homo sapiens |
IC50 |
= |
840.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2305 |
Cell Line |
CAL-85-1 |
Homo sapiens |
IC50 |
= |
44.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
159.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2306 |
Cell Line |
Ca-Ski |
Homo sapiens |
IC50 |
= |
44.84 |
nM |
10.6019/CHEMBL1201861 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
50.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2310 |
Cell Line |
CaR-1 |
Homo sapiens |
IC50 |
= |
1783.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2307 |
Cell Line |
769-P |
Homo sapiens |
IC50 |
= |
20.76 |
nM |
10.6019/CHEMBL1201861 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
8.472 |
nM |
10.6019/CHEMBL1201861 |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
149.31 |
nM |
10.6019/CHEMBL1201861 |
NPT929 |
Cell Line |
BC1 cell line |
|
IC50 |
= |
86.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2309 |
Cell Line |
CAPAN-1 |
Homo sapiens |
IC50 |
= |
51.76 |
nM |
10.6019/CHEMBL1201861 |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
238.31 |
nM |
10.6019/CHEMBL1201861 |
NPT1307 |
Cell Line |
Calu-1 |
Homo sapiens |
IC50 |
= |
73.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2311 |
Cell Line |
Calu-3 |
Homo sapiens |
IC50 |
= |
55.98 |
nM |
10.6019/CHEMBL1201861 |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
22.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2312 |
Cell Line |
8305C |
Homo sapiens |
IC50 |
= |
63.12 |
nM |
10.6019/CHEMBL1201861 |
NPT1936 |
Cell Line |
BC-3 |
Homo sapiens |
IC50 |
= |
165.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2313 |
Cell Line |
BCPAP |
Homo sapiens |
IC50 |
= |
52.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
51.02 |
nM |
10.6019/CHEMBL1201861 |
NPT4605 |
Cell Line |
CCF-STTG1 |
Homo sapiens |
IC50 |
= |
35.5 |
nM |
10.6019/CHEMBL1201861 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
24.52 |
nM |
10.6019/CHEMBL1201861 |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
253.55 |
nM |
10.6019/CHEMBL1201861 |
NPT4458 |
Cell Line |
Caov-3 cell line |
|
IC50 |
= |
406.19 |
nM |
10.6019/CHEMBL1201861 |
NPT1313 |
Cell Line |
Capan-2 |
Homo sapiens |
IC50 |
= |
898.11 |
nM |
10.6019/CHEMBL1201861 |
NPT1215 |
Cell Line |
8505C |
Homo sapiens |
IC50 |
= |
19.56 |
nM |
10.6019/CHEMBL1201861 |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
51.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2314 |
Cell Line |
BEN |
Homo sapiens |
IC50 |
= |
1237.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2315 |
Cell Line |
BFTC-905 |
Homo sapiens |
IC50 |
= |
16.18 |
nM |
10.6019/CHEMBL1201861 |
NPT1942 |
Cell Line |
CESS |
Homo sapiens |
IC50 |
= |
39.36 |
nM |
10.6019/CHEMBL1201861 |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
53.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2317 |
Cell Line |
ChaGo-K-1 |
Homo sapiens |
IC50 |
= |
107.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
80.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2319 |
Cell Line |
A204 |
Homo sapiens |
IC50 |
= |
12.88 |
nM |
10.6019/CHEMBL1201861 |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
17.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2320 |
Cell Line |
BFTC-909 |
Homo sapiens |
IC50 |
= |
118.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2321 |
Cell Line |
BHT-101 |
Homo sapiens |
IC50 |
= |
395.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2323 |
Cell Line |
BHY |
Homo sapiens |
IC50 |
= |
28.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2322 |
Cell Line |
CHL-1 |
Homo sapiens |
IC50 |
= |
37.73 |
nM |
10.6019/CHEMBL1201861 |
NPT1945 |
Cell Line |
CHP-126 |
Homo sapiens |
IC50 |
= |
59.24 |
nM |
10.6019/CHEMBL1201861 |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
305.52 |
nM |
10.6019/CHEMBL1201861 |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
250.13 |
nM |
10.6019/CHEMBL1201861 |
NPT1948 |
Cell Line |
A253 cell line |
|
IC50 |
= |
46.12 |
nM |
10.6019/CHEMBL1201861 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
68.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1949 |
Cell Line |
BL-41 |
Homo sapiens |
IC50 |
= |
122.22 |
nM |
10.6019/CHEMBL1201861 |
NPT1950 |
Cell Line |
BL-70 |
Homo sapiens |
IC50 |
= |
342.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2324 |
Cell Line |
CHP-212 |
Homo sapiens |
IC50 |
= |
34.96 |
nM |
10.6019/CHEMBL1201861 |
NPT1951 |
Cell Line |
CMK |
Homo sapiens |
IC50 |
= |
77.42 |
nM |
10.6019/CHEMBL1201861 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
26.99 |
nM |
10.6019/CHEMBL1201861 |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
248.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
40.14 |
nM |
10.6019/CHEMBL1201861 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
9.168 |
nM |
10.6019/CHEMBL1201861 |
NPT4606 |
Cell Line |
BOKU |
Homo sapiens |
IC50 |
= |
110.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2325 |
Cell Line |
BPH-1 |
Homo sapiens |
IC50 |
= |
22.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
1740.68 |
nM |
10.6019/CHEMBL1201861 |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
513.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
84.47 |
nM |
10.6019/CHEMBL1201861 |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
5242.62 |
nM |
10.6019/CHEMBL1201861 |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
28.46 |
nM |
10.6019/CHEMBL1201861 |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
162.48 |
nM |
10.6019/CHEMBL1201861 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
778.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
250.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2328 |
Cell Line |
COLO-678 |
Homo sapiens |
IC50 |
= |
427.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2329 |
Cell Line |
COLO-679 |
Homo sapiens |
IC50 |
= |
15.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2332 |
Cell Line |
COLO-680N |
Homo sapiens |
IC50 |
= |
33.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
1653.05 |
nM |
10.6019/CHEMBL1201861 |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
161.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
11.81 |
nM |
10.6019/CHEMBL1201861 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
20.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
521.83 |
nM |
10.6019/CHEMBL1201861 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
210.96 |
nM |
10.6019/CHEMBL1201861 |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
219.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2278 |
Cell Line |
COLO-741 |
Homo sapiens |
IC50 |
= |
194.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2333 |
Cell Line |
DBTRG-05MG |
Homo sapiens |
IC50 |
= |
67.11 |
nM |
10.6019/CHEMBL1201861 |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
38.44 |
nM |
10.6019/CHEMBL1201861 |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
405.05 |
nM |
10.6019/CHEMBL1201861 |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
49.96 |
nM |
10.6019/CHEMBL1201861 |
NPT2335 |
Cell Line |
NCI-H596 |
|
IC50 |
= |
108.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
426.02 |
nM |
10.6019/CHEMBL1201861 |
NPT1968 |
Cell Line |
OMC-1 |
Homo sapiens |
IC50 |
= |
172.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2200 |
Cell Line |
RPMI-6666 |
Homo sapiens |
IC50 |
= |
65.99 |
nM |
10.6019/CHEMBL1201861 |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
IC50 |
= |
130.14 |
nM |
10.6019/CHEMBL1201861 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
213.37 |
nM |
10.6019/CHEMBL1201861 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
36754.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
201.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
49.72 |
nM |
10.6019/CHEMBL1201861 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
26.63 |
nM |
10.6019/CHEMBL1201861 |
NPT1969 |
Cell Line |
TGW |
Homo sapiens |
IC50 |
= |
1459.42 |
nM |
10.6019/CHEMBL1201861 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
989.42 |
nM |
10.6019/CHEMBL1201861 |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
69.65 |
nM |
10.6019/CHEMBL1201861 |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
93.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
241.46 |
nM |
10.6019/CHEMBL1201861 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
62.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2348 |
Cell Line |
HLE |
Homo sapiens |
IC50 |
= |
35.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
517.42 |
nM |
10.6019/CHEMBL1201861 |
NPT1974 |
Cell Line |
IST-SL2 |
Homo sapiens |
IC50 |
= |
73.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
3.443 |
nM |
10.6019/CHEMBL1201861 |
NPT2340 |
Cell Line |
KU-19-19 |
Homo sapiens |
IC50 |
= |
2269.17 |
nM |
10.6019/CHEMBL1201861 |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
204.47 |
nM |
10.6019/CHEMBL1201861 |
NPT1977 |
Cell Line |
LOUCY |
Homo sapiens |
IC50 |
= |
21.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
3.987 |
nM |
10.6019/CHEMBL1201861 |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
328304.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
22.08 |
nM |
10.6019/CHEMBL1201861 |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
134.55 |
nM |
10.6019/CHEMBL1201861 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
493.21 |
nM |
10.6019/CHEMBL1201861 |
NPT1981 |
Cell Line |
NCI-H1882 |
Homo sapiens |
IC50 |
= |
215 |
nM |
10.6019/CHEMBL1201861 |
NPT1982 |
Cell Line |
NCI-H1963 |
Homo sapiens |
IC50 |
= |
430.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2353 |
Cell Line |
NCI-H1993 |
Homo sapiens |
IC50 |
= |
1000.76 |
nM |
10.6019/CHEMBL1201861 |
NPT1983 |
Cell Line |
NCI-H64 |
Homo sapiens |
IC50 |
= |
132.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2343 |
Cell Line |
NCI-H650 |
Homo sapiens |
IC50 |
= |
217.61 |
nM |
10.6019/CHEMBL1201861 |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
18.91 |
nM |
10.6019/CHEMBL1201861 |
NPT1986 |
Cell Line |
RPMI 8402 |
Homo sapiens |
IC50 |
= |
53.86 |
nM |
10.6019/CHEMBL1201861 |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
192.13 |
nM |
10.6019/CHEMBL1201861 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
230.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2344 |
Cell Line |
SK-MEL-24 |
Homo sapiens |
IC50 |
= |
914.35 |
nM |
10.6019/CHEMBL1201861 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
35537.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
111.71 |
nM |
10.6019/CHEMBL1201861 |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
34156.06 |
nM |
10.6019/CHEMBL1201861 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
114.6 |
nM |
10.6019/CHEMBL1201861 |
NPT4607 |
Cell Line |
TT |
Homo sapiens |
IC50 |
= |
9069.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2347 |
Cell Line |
GMS-10 |
Homo sapiens |
IC50 |
= |
2397.38 |
nM |
10.6019/CHEMBL1201861 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
285.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2349 |
Cell Line |
HMV-2 cell line |
|
IC50 |
= |
22.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2350 |
Cell Line |
HN |
Homo sapiens |
IC50 |
= |
354.27 |
nM |
10.6019/CHEMBL1201861 |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
96.31 |
nM |
10.6019/CHEMBL1201861 |
NPT1505 |
Cell Line |
J82 |
Homo sapiens |
IC50 |
= |
21.34 |
nM |
10.6019/CHEMBL1201861 |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
33.24 |
nM |
10.6019/CHEMBL1201861 |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
126.76 |
nM |
10.6019/CHEMBL1201861 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
389.19 |
nM |
10.6019/CHEMBL1201861 |
NPT1993 |
Cell Line |
LP-1 |
Homo sapiens |
IC50 |
= |
67928.39 |
nM |
10.6019/CHEMBL1201861 |
NPT1994 |
Cell Line |
MHH-CALL-2 |
Homo sapiens |
IC50 |
= |
359.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2352 |
Cell Line |
MHH-ES-1 |
Homo sapiens |
IC50 |
= |
21.58 |
nM |
10.6019/CHEMBL1201861 |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
359.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2354 |
Cell Line |
NCI-H2009 |
Homo sapiens |
IC50 |
= |
51.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2368 |
Cell Line |
NCI-H2030 |
Homo sapiens |
IC50 |
= |
28.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
49.03 |
nM |
10.6019/CHEMBL1201861 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
568.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1985 |
Cell Line |
OPM-2 |
Homo sapiens |
IC50 |
= |
501.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
182.49 |
nM |
10.6019/CHEMBL1201861 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
470.41 |
nM |
10.6019/CHEMBL1201861 |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
19.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2357 |
Cell Line |
RT-112 |
Homo sapiens |
IC50 |
= |
32.92 |
nM |
10.6019/CHEMBL1201861 |
NPT4608 |
Cell Line |
RT-4 |
Homo sapiens |
IC50 |
= |
1844.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
IC50 |
= |
147.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2359 |
Cell Line |
SK-MEL-30 |
Homo sapiens |
IC50 |
= |
35.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2360 |
Cell Line |
SW756 |
Homo sapiens |
IC50 |
= |
274.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
59092.09 |
nM |
10.6019/CHEMBL1201861 |
NPT1999 |
Cell Line |
TUR |
Homo sapiens |
IC50 |
= |
76.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2362 |
Cell Line |
TYK-nu |
Homo sapiens |
IC50 |
= |
662.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2363 |
Cell Line |
U-118-MG |
Homo sapiens |
IC50 |
= |
856.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2364 |
Cell Line |
GP5d |
Homo sapiens |
IC50 |
= |
49.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
255.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2365 |
Cell Line |
HO-1-N-1 |
Homo sapiens |
IC50 |
= |
222.83 |
nM |
10.6019/CHEMBL1201861 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
35.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
625.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2366 |
Cell Line |
JEG-3 |
Homo sapiens |
IC50 |
= |
95.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
1494.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2367 |
Cell Line |
KYSE-140 |
Homo sapiens |
IC50 |
= |
50.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
384.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
18.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
220.22 |
nM |
10.6019/CHEMBL1201861 |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
229.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
2185 |
nM |
10.6019/CHEMBL1201861 |
NPT2369 |
Cell Line |
NCI-H2052 |
Homo sapiens |
IC50 |
= |
160.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2009 |
Cell Line |
NCI-H2081 |
Homo sapiens |
IC50 |
= |
234.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2010 |
Cell Line |
NCI-H716 |
Homo sapiens |
IC50 |
= |
69511.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2011 |
Cell Line |
NCI-H719 |
Homo sapiens |
IC50 |
= |
39.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
41972.64 |
nM |
10.6019/CHEMBL1201861 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
156.78 |
nM |
10.6019/CHEMBL1201861 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
IC50 |
= |
116.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2370 |
Cell Line |
RVH-421 |
Homo sapiens |
IC50 |
= |
169.13 |
nM |
10.6019/CHEMBL1201861 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
335.43 |
nM |
10.6019/CHEMBL1201861 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
31.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2013 |
Cell Line |
SK-MM-2 |
Homo sapiens |
IC50 |
= |
942.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2380 |
Cell Line |
SK-N-AS |
Homo sapiens |
IC50 |
= |
2730.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2371 |
Cell Line |
SW837 |
Homo sapiens |
IC50 |
= |
117.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
120.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
9813.93 |
nM |
10.6019/CHEMBL1201861 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
451.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
137.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
51.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
67.19 |
nM |
10.6019/CHEMBL1201861 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
IC50 |
= |
290.7 |
nM |
10.6019/CHEMBL1201861 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
45.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2384 |
Cell Line |
HPAF-II |
Homo sapiens |
IC50 |
= |
527.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
242.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
4606.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2373 |
Cell Line |
KYSE-150 cell line |
|
IC50 |
= |
27.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2374 |
Cell Line |
KYSE-180 |
Homo sapiens |
IC50 |
= |
59.75 |
nM |
10.6019/CHEMBL1201861 |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
99.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
18609.27 |
nM |
10.6019/CHEMBL1201861 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
34.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
9.862 |
nM |
10.6019/CHEMBL1201861 |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
79.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2377 |
Cell Line |
NCI-H2087 |
Homo sapiens |
IC50 |
= |
49.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
48.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
22.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
135.02 |
nM |
10.6019/CHEMBL1201861 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
61.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2379 |
Cell Line |
P12-Ichikawa |
Homo sapiens |
IC50 |
= |
49.27 |
nM |
10.6019/CHEMBL1201861 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
334.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
294.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
2565.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
52325.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
16.93 |
nM |
10.6019/CHEMBL1201861 |
NPT2030 |
Cell Line |
U-698-M |
Homo sapiens |
IC50 |
= |
139.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
346.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
21.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2383 |
Cell Line |
ESS-1 |
Homo sapiens |
IC50 |
= |
11.09 |
nM |
10.6019/CHEMBL1201861 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
IC50 |
= |
71.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
313.44 |
nM |
10.6019/CHEMBL1201861 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
26.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
IC50 |
= |
74.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2033 |
Cell Line |
JIYOYE |
Homo sapiens |
IC50 |
= |
137.8 |
nM |
10.6019/CHEMBL1201861 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
385.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2386 |
Cell Line |
KYSE-270 |
Homo sapiens |
IC50 |
= |
7.211 |
nM |
10.6019/CHEMBL1201861 |
NPT2387 |
Cell Line |
KYSE-410 |
Homo sapiens |
IC50 |
= |
103.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2395 |
Cell Line |
KYSE-450 |
Homo sapiens |
IC50 |
= |
44.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
67.68 |
nM |
10.6019/CHEMBL1201861 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
31.91 |
nM |
10.6019/CHEMBL1201861 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
81.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2398 |
Cell Line |
MKN-7 |
Homo sapiens |
IC50 |
= |
689.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2035 |
Cell Line |
NCCIT |
Homo sapiens |
IC50 |
= |
20.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
737.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2390 |
Cell Line |
NCI-H2122 |
Homo sapiens |
IC50 |
= |
37.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
192.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2038 |
Cell Line |
NCI-H748 |
Homo sapiens |
IC50 |
= |
147.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2391 |
Cell Line |
NCI-H810 |
Homo sapiens |
IC50 |
= |
18.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
57.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2041 |
Cell Line |
P31-FUJ |
Homo sapiens |
IC50 |
= |
44328.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
44.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2392 |
Cell Line |
S-117 |
Homo sapiens |
IC50 |
= |
1705.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
114.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
5228.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
116.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
69.95 |
nM |
10.6019/CHEMBL1201861 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
353.87 |
nM |
10.6019/CHEMBL1201861 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
64.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
83.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2046 |
Cell Line |
EVSA-T |
Homo sapiens |
IC50 |
= |
2300.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2047 |
Cell Line |
HC-1 |
Homo sapiens |
IC50 |
= |
37.32 |
nM |
10.6019/CHEMBL1201861 |
NPT4609 |
Cell Line |
HCC1143 |
Homo sapiens |
IC50 |
= |
10479.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
591.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2394 |
Cell Line |
HSC-4 |
Homo sapiens |
IC50 |
= |
75.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
405.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2050 |
Cell Line |
K052 |
Homo sapiens |
IC50 |
= |
21441.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
96.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2396 |
Cell Line |
KYSE-510 |
Homo sapiens |
IC50 |
= |
15.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2397 |
Cell Line |
KYSE-520 cell line |
|
IC50 |
= |
260.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
344.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2054 |
Cell Line |
LU-165 |
Homo sapiens |
IC50 |
= |
639.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
135.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
122.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
579.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
37.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2059 |
Cell Line |
NCI-H2141 |
Homo sapiens |
IC50 |
= |
573.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2399 |
Cell Line |
NCI-H2170 |
Homo sapiens |
IC50 |
= |
109.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
1570.26 |
nM |
10.6019/CHEMBL1201861 |
NPT4610 |
Cell Line |
NCI-H838 |
Homo sapiens |
IC50 |
= |
224.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2061 |
Cell Line |
NCI-H889 |
Homo sapiens |
IC50 |
= |
1938.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2401 |
Cell Line |
PANC-03-27 |
Homo sapiens |
IC50 |
= |
28.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2402 |
Cell Line |
PANC-08-13 |
Homo sapiens |
IC50 |
= |
1630.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
156.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2403 |
Cell Line |
SBC-5 |
Homo sapiens |
IC50 |
= |
20.74 |
nM |
10.6019/CHEMBL1201861 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
50.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
25.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2404 |
Cell Line |
SW982 |
Homo sapiens |
IC50 |
= |
6.051 |
nM |
10.6019/CHEMBL1201861 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
329.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
23337.11 |
nM |
10.6019/CHEMBL1201861 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
362.05 |
nM |
10.6019/CHEMBL1201861 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
1321.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2064 |
Cell Line |
UACC-812 |
Homo sapiens |
IC50 |
= |
3337.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
61.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
341.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2406 |
Cell Line |
HCC1395 |
Homo sapiens |
IC50 |
= |
8151.22 |
nM |
10.6019/CHEMBL1201861 |
NPT2407 |
Cell Line |
HCC1419 |
Homo sapiens |
IC50 |
= |
631.74 |
nM |
10.6019/CHEMBL1201861 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
14.82 |
nM |
10.6019/CHEMBL1201861 |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
212.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2419 |
Cell Line |
HT-1376 |
Homo sapiens |
IC50 |
= |
189.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
29.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
1478.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2408 |
Cell Line |
KYSE-70 cell line |
|
IC50 |
= |
224.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
324.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
346.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2409 |
Cell Line |
LU-99A |
Homo sapiens |
IC50 |
= |
146.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
106.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
321.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2060 |
Cell Line |
NCI-H2171 |
Homo sapiens |
IC50 |
= |
440.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2075 |
Cell Line |
NCI-H2196 |
Homo sapiens |
IC50 |
= |
229.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2076 |
Cell Line |
NCI-H2227 |
Homo sapiens |
IC50 |
= |
5362.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2411 |
Cell Line |
NCI-H2228 |
Homo sapiens |
IC50 |
= |
13.48 |
nM |
10.6019/CHEMBL1201861 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
479.92 |
nM |
10.6019/CHEMBL1201861 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
65.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2412 |
Cell Line |
Panc1005 |
Homo sapiens |
IC50 |
= |
88.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
236.12 |
nM |
10.6019/CHEMBL1201861 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
957.22 |
nM |
10.6019/CHEMBL1201861 |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
188.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2414 |
Cell Line |
SCC-25 |
Homo sapiens |
IC50 |
= |
153.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
19.96 |
nM |
10.6019/CHEMBL1201861 |
NPT2415 |
Cell Line |
SKG-IIIa |
Homo sapiens |
IC50 |
= |
311.14 |
nM |
10.6019/CHEMBL1201861 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
245.48 |
nM |
10.6019/CHEMBL1201861 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
469.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2416 |
Cell Line |
UACC-893 |
Homo sapiens |
IC50 |
= |
521.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
86.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2425 |
Cell Line |
UMC-11 |
Homo sapiens |
IC50 |
= |
331.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
9.626 |
nM |
10.6019/CHEMBL1201861 |
NPT2418 |
Cell Line |
HCC1569 |
Homo sapiens |
IC50 |
= |
109.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2081 |
Cell Line |
HCC1599 |
Homo sapiens |
IC50 |
= |
72.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2426 |
Cell Line |
HCC1806 |
Homo sapiens |
IC50 |
= |
74.96 |
nM |
10.6019/CHEMBL1201861 |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
3.509 |
nM |
10.6019/CHEMBL1201861 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
36.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2083 |
Cell Line |
KARPAS-422 |
Homo sapiens |
IC50 |
= |
193.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
1267.63 |
nM |
10.6019/CHEMBL1201861 |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
790.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2087 |
Cell Line |
L-540 |
Homo sapiens |
IC50 |
= |
213.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
109.24 |
nM |
10.6019/CHEMBL1201861 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
81.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
31.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
605.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
290.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
152.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
51433 |
nM |
10.6019/CHEMBL1201861 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
416.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2090 |
Cell Line |
SNU-16 |
Homo sapiens |
IC50 |
= |
31183.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
570.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2093 |
Cell Line |
PF-382 |
Homo sapiens |
IC50 |
= |
67.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2421 |
Cell Line |
PFSK-1 |
Homo sapiens |
IC50 |
= |
678.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2077 |
Cell Line |
SCC-3 |
Homo sapiens |
IC50 |
= |
67.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2422 |
Cell Line |
SCC-4 |
Homo sapiens |
IC50 |
= |
183.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2423 |
Cell Line |
SCC-9 |
Homo sapiens |
IC50 |
= |
3913.09 |
nM |
10.6019/CHEMBL1201861 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
IC50 |
= |
394.87 |
nM |
10.6019/CHEMBL1201861 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
148.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
57.06 |
nM |
10.6019/CHEMBL1201861 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
2804.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
33.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2435 |
Cell Line |
VM-CUB-1 |
Homo sapiens |
IC50 |
= |
75.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
1.912 |
nM |
10.6019/CHEMBL1201861 |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
250.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1884 |
Cell Line |
HCC1937 |
Homo sapiens |
IC50 |
= |
115.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2427 |
Cell Line |
HCC1954 |
Homo sapiens |
IC50 |
= |
540.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2428 |
Cell Line |
HT-3 |
Homo sapiens |
IC50 |
= |
133.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2429 |
Cell Line |
HT55 |
Homo sapiens |
IC50 |
= |
1471.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
21.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
361.52 |
nM |
10.6019/CHEMBL1201861 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
437.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
315.11 |
nM |
10.6019/CHEMBL1201861 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
905.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2102 |
Cell Line |
MC-CAR |
Homo sapiens |
IC50 |
= |
48.74 |
nM |
10.6019/CHEMBL1201861 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
22.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2104 |
Cell Line |
NCI-H1417 |
Homo sapiens |
IC50 |
= |
370.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2105 |
Cell Line |
NCI-H1436 |
Homo sapiens |
IC50 |
= |
71637.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2431 |
Cell Line |
NCI-H1437 |
Homo sapiens |
IC50 |
= |
64.64 |
nM |
10.6019/CHEMBL1201861 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
283.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2432 |
Cell Line |
NCI-H2342 |
Homo sapiens |
IC50 |
= |
22.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
33.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
76 |
nM |
10.6019/CHEMBL1201861 |
NPT4611 |
Cell Line |
PLC-PRF-5 |
Homo sapiens |
IC50 |
= |
901.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
11.22 |
nM |
10.6019/CHEMBL1201861 |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
177109.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2110 |
Cell Line |
SCLC-21H |
Homo sapiens |
IC50 |
= |
2006.24 |
nM |
10.6019/CHEMBL1201861 |
NPT4612 |
Cell Line |
SNG-M |
Homo sapiens |
IC50 |
= |
18.32 |
nM |
10.6019/CHEMBL1201861 |
NPT890 |
Cell Line |
SNU-387 |
Homo sapiens |
IC50 |
= |
236.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2433 |
Cell Line |
SNU-423 |
Homo sapiens |
IC50 |
= |
155.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2095 |
Cell Line |
TALL-1 |
Homo sapiens |
IC50 |
= |
7968.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2434 |
Cell Line |
TCC-SUP |
Homo sapiens |
IC50 |
= |
1230.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
76.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2436 |
Cell Line |
VMRC-RCZ |
Homo sapiens |
IC50 |
= |
93.26 |
nM |
10.6019/CHEMBL1201861 |
NPT1653 |
Cell Line |
WM-115 |
Homo sapiens |
IC50 |
= |
51038.39 |
nM |
10.6019/CHEMBL1201861 |
NPT2113 |
Cell Line |
EW-24 |
Homo sapiens |
IC50 |
= |
970.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2115 |
Cell Line |
HCC2157 |
Homo sapiens |
IC50 |
= |
63.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
181.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2438 |
Cell Line |
HTC-C3 |
Homo sapiens |
IC50 |
= |
703.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
2.118 |
nM |
10.6019/CHEMBL1201861 |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
6.336 |
nM |
10.6019/CHEMBL1201861 |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
35.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
235.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2439 |
Cell Line |
MC-IXC |
Homo sapiens |
IC50 |
= |
67.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
391.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2103 |
Cell Line |
MONO-MAC-6 |
Homo sapiens |
IC50 |
= |
154.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
392.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2124 |
Cell Line |
MRK-nu-1 |
Homo sapiens |
IC50 |
= |
43.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2125 |
Cell Line |
NCI-H1522 |
Homo sapiens |
IC50 |
= |
1431.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2440 |
Cell Line |
NCI-H1563 |
Homo sapiens |
IC50 |
= |
556.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2449 |
Cell Line |
NCI-H1573 |
Homo sapiens |
IC50 |
= |
1717.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2441 |
Cell Line |
NCI-H2347 |
Homo sapiens |
IC50 |
= |
158.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2442 |
Cell Line |
NCI-H2405 |
Homo sapiens |
IC50 |
= |
234.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2450 |
Cell Line |
NCI-H2452 |
Homo sapiens |
IC50 |
= |
1371.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
29.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
139.13 |
nM |
10.6019/CHEMBL1201861 |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
20.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
30061.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
104.58 |
nM |
10.6019/CHEMBL1201861 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
92.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2443 |
Cell Line |
SNU-449 |
Homo sapiens |
IC50 |
= |
548.01 |
nM |
10.6019/CHEMBL1201861 |
NPT4613 |
Cell Line |
SNU-475 |
Homo sapiens |
IC50 |
= |
2925.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2129 |
Cell Line |
SNU-C1 |
Homo sapiens |
IC50 |
= |
32417.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
112.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2131 |
Cell Line |
WSU-NHL |
Homo sapiens |
IC50 |
= |
154.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2444 |
Cell Line |
YAPC |
Homo sapiens |
IC50 |
= |
3328.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
279.89 |
nM |
10.6019/CHEMBL1201861 |
NPT4614 |
Cell Line |
EW-7 |
Homo sapiens |
IC50 |
= |
30.63 |
nM |
10.6019/CHEMBL1201861 |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
27.78 |
nM |
10.6019/CHEMBL1201861 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
17.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2446 |
Cell Line |
HCC38 |
Homo sapiens |
IC50 |
= |
42.5 |
nM |
10.6019/CHEMBL1201861 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
2017.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2447 |
Cell Line |
HuCCT-1 |
Homo sapiens |
IC50 |
= |
72.93 |
nM |
10.6019/CHEMBL1201861 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
258.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
1019 |
nM |
10.6019/CHEMBL1201861 |
NPT2448 |
Cell Line |
KLE |
Homo sapiens |
IC50 |
= |
175.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
413.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
344.64 |
nM |
10.6019/CHEMBL1201861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2136 |
Cell Line |
MDA-MB-134-VI |
Homo sapiens |
IC50 |
= |
1617.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
499.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
252.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
214955.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
981.31 |
nM |
10.6019/CHEMBL1201861 |
NPT4615 |
Cell Line |
NCI-H1618 |
Homo sapiens |
IC50 |
= |
104.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2451 |
Cell Line |
NCI-H28 |
Homo sapiens |
IC50 |
= |
1740.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
43.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
224.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
79.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2453 |
Cell Line |
RCM-1 |
Homo sapiens |
IC50 |
= |
4492.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
180.1 |
nM |
10.6019/CHEMBL1201861 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
49.08 |
nM |
10.6019/CHEMBL1201861 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
121.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2455 |
Cell Line |
SNU-C2B |
Homo sapiens |
IC50 |
= |
460.97 |
nM |
10.6019/CHEMBL1201861 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
IC50 |
= |
24.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2456 |
Cell Line |
TE-11 |
Homo sapiens |
IC50 |
= |
240.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
81.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2457 |
Cell Line |
YKG-1 |
Homo sapiens |
IC50 |
= |
18.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2146 |
Cell Line |
YT |
Homo sapiens |
IC50 |
= |
1045.68 |
nM |
10.6019/CHEMBL1201861 |
NPT1216 |
Cell Line |
FaDu |
Homo sapiens |
IC50 |
= |
102.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2458 |
Cell Line |
FTC-133 |
Homo sapiens |
IC50 |
= |
229.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
2054.63 |
nM |
10.6019/CHEMBL1201861 |
NPT2460 |
Cell Line |
HCE-4 |
Homo sapiens |
IC50 |
= |
18.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2461 |
Cell Line |
HuO-3N1 |
Homo sapiens |
IC50 |
= |
2365.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
90.68 |
nM |
10.6019/CHEMBL1201861 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
218.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2147 |
Cell Line |
LB647-SCLC |
Homo sapiens |
IC50 |
= |
123.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
6468.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2464 |
Cell Line |
MDA-MB-175-VII |
Homo sapiens |
IC50 |
= |
971.53 |
nM |
10.6019/CHEMBL1201861 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1530.55 |
nM |
10.6019/CHEMBL1201861 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
10.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
23.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2465 |
Cell Line |
NCI-H1623 |
Homo sapiens |
IC50 |
= |
604.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
131.94 |
nM |
10.6019/CHEMBL1201861 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
IC50 |
= |
194396.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2151 |
Cell Line |
NCI-H345 |
Homo sapiens |
IC50 |
= |
4011.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
41.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
1.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
45.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2142 |
Cell Line |
REH |
Homo sapiens |
IC50 |
= |
8.115 |
nM |
10.6019/CHEMBL1201861 |
NPT2467 |
Cell Line |
RERF-LC-MS |
Homo sapiens |
IC50 |
= |
425.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
6.733 |
nM |
10.6019/CHEMBL1201861 |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
92.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
9902.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2143 |
Cell Line |
ST486 |
Homo sapiens |
IC50 |
= |
15.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2156 |
Cell Line |
SU-DHL-1 |
Homo sapiens |
IC50 |
= |
102.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2157 |
Cell Line |
SUP-T1 |
Homo sapiens |
IC50 |
= |
79.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2481 |
Cell Line |
SW1088 |
Homo sapiens |
IC50 |
= |
2069.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2145 |
Cell Line |
TE-15 |
Homo sapiens |
IC50 |
= |
24.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2158 |
Cell Line |
TE-441-T |
Homo sapiens |
IC50 |
= |
89.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
37.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
160.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
321.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
27.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
IC50 |
= |
30.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2470 |
Cell Line |
G-402 |
Homo sapiens |
IC50 |
= |
99.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
164.87 |
nM |
10.6019/CHEMBL1201861 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
207.39 |
nM |
10.6019/CHEMBL1201861 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
2354.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2471 |
Cell Line |
HuP-T3 |
Homo sapiens |
IC50 |
= |
165.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2472 |
Cell Line |
HuP-T4 |
Homo sapiens |
IC50 |
= |
52.22 |
nM |
10.6019/CHEMBL1201861 |
NPT2485 |
Cell Line |
IA-LM |
Homo sapiens |
IC50 |
= |
63.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2163 |
Cell Line |
KMOE-2 |
Homo sapiens |
IC50 |
= |
576.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2164 |
Cell Line |
KMS-12-PE |
Homo sapiens |
IC50 |
= |
418.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
206.25 |
nM |
10.6019/CHEMBL1201861 |
NPT2167 |
Cell Line |
LB996-RCC |
Homo sapiens |
IC50 |
= |
78.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
292.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2474 |
Cell Line |
MDA-MB-415 |
Homo sapiens |
IC50 |
= |
7573.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
4851.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
33.92 |
nM |
10.6019/CHEMBL1201861 |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
78.62 |
nM |
10.6019/CHEMBL1201861 |
NPT2475 |
Cell Line |
NCI-H1651 |
Homo sapiens |
IC50 |
= |
11.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2476 |
Cell Line |
NCI-H441 |
Homo sapiens |
IC50 |
= |
28.42 |
nM |
10.6019/CHEMBL1201861 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
1337.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2478 |
Cell Line |
NY |
Homo sapiens |
IC50 |
= |
228.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2479 |
Cell Line |
OAW-28 |
Homo sapiens |
IC50 |
= |
178.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
22.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2171 |
Cell Line |
SIG-M5 |
Homo sapiens |
IC50 |
= |
25.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2172 |
Cell Line |
SIMA |
Homo sapiens |
IC50 |
= |
381.86 |
nM |
10.6019/CHEMBL1201861 |
NPT3467 |
Cell Line |
SJRH30 |
Homo sapiens |
IC50 |
= |
172.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2483 |
Cell Line |
SW13 |
Homo sapiens |
IC50 |
= |
115.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2495 |
Cell Line |
SW1417 |
Homo sapiens |
IC50 |
= |
363.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
469.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
7.503 |
nM |
10.6019/CHEMBL1201861 |
NPT2175 |
Cell Line |
GAK |
Homo sapiens |
IC50 |
= |
256.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2484 |
Cell Line |
GAMG |
Homo sapiens |
IC50 |
= |
59.96 |
nM |
10.6019/CHEMBL1201861 |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
272.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2486 |
Cell Line |
IGR-1 |
Homo sapiens |
IC50 |
= |
33.88 |
nM |
10.6019/CHEMBL1201861 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
7.205 |
nM |
10.6019/CHEMBL1201861 |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
242.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
160.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2179 |
Cell Line |
LC-1F |
Homo sapiens |
IC50 |
= |
1662.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
5.074 |
nM |
10.6019/CHEMBL1201861 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
76.18 |
nM |
10.6019/CHEMBL1201861 |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
186.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
112.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
3460.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2491 |
Cell Line |
NCI-H1693 |
Homo sapiens |
IC50 |
= |
290.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2183 |
Cell Line |
NCI-H1694 |
Homo sapiens |
IC50 |
= |
200.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2503 |
Cell Line |
NCI-H1703 |
Homo sapiens |
IC50 |
= |
126.42 |
nM |
10.6019/CHEMBL1201861 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
12.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2184 |
Cell Line |
NCI-H510A |
Homo sapiens |
IC50 |
= |
359.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2492 |
Cell Line |
OAW-42 |
Homo sapiens |
IC50 |
= |
153.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
45.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2186 |
Cell Line |
RL |
Homo sapiens |
IC50 |
= |
1420.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2494 |
Cell Line |
RMG-I |
Homo sapiens |
IC50 |
= |
513.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
111.05 |
nM |
10.6019/CHEMBL1201861 |
NPT4616 |
Cell Line |
SK-CO-1 |
Homo sapiens |
IC50 |
= |
129.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2496 |
Cell Line |
SW1463 |
Homo sapiens |
IC50 |
= |
1957.01 |
nM |
10.6019/CHEMBL1201861 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
IC50 |
= |
82.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
257.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
212.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
725.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
568.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2497 |
Cell Line |
HEC-1 |
Homo sapiens |
IC50 |
= |
182.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2193 |
Cell Line |
IM-9 |
Homo sapiens |
IC50 |
= |
51.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2194 |
Cell Line |
IMR-5 |
Homo sapiens |
IC50 |
= |
34.68 |
nM |
10.6019/CHEMBL1201861 |
NPT4617 |
Cell Line |
IPC-298 |
Homo sapiens |
IC50 |
= |
196.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2498 |
Cell Line |
KOSC-2 |
Homo sapiens |
IC50 |
= |
248.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2499 |
Cell Line |
KP-4 |
Homo sapiens |
IC50 |
= |
40.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2195 |
Cell Line |
LC4-1 |
Homo sapiens |
IC50 |
= |
240.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2500 |
Cell Line |
LCLC-103H cell line |
|
IC50 |
= |
20.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2512 |
Cell Line |
LCLC-97TM1 |
Homo sapiens |
IC50 |
= |
11.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
176.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2501 |
Cell Line |
MEL-HO |
Homo sapiens |
IC50 |
= |
18.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2502 |
Cell Line |
MEL-JUSO |
Homo sapiens |
IC50 |
= |
14.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
804.65 |
nM |
10.6019/CHEMBL1201861 |
NPT623 |
Cell Line |
NALM-6 |
Homo sapiens |
IC50 |
= |
18.63 |
nM |
10.6019/CHEMBL1201861 |
NPT4618 |
Cell Line |
NCI-H1734 |
Homo sapiens |
IC50 |
= |
53 |
nM |
10.6019/CHEMBL1201861 |
NPT2504 |
Cell Line |
NCI-H1755 |
Homo sapiens |
IC50 |
= |
873.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
266.61 |
nM |
10.6019/CHEMBL1201861 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
IC50 |
= |
51.93 |
nM |
10.6019/CHEMBL1201861 |
NPT2198 |
Cell Line |
NCI-H524 |
Homo sapiens |
IC50 |
= |
48824.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
15.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2336 |
Cell Line |
OE19 |
Homo sapiens |
IC50 |
= |
200.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2506 |
Cell Line |
RO82-W-1 |
Homo sapiens |
IC50 |
= |
1343.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2507 |
Cell Line |
RPMI-2650 |
Homo sapiens |
IC50 |
= |
13.69 |
nM |
10.6019/CHEMBL1201861 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
25.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
53.22 |
nM |
10.6019/CHEMBL1201861 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
12.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2508 |
Cell Line |
SW1710 |
Homo sapiens |
IC50 |
= |
17.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2509 |
Cell Line |
SW1783 |
Homo sapiens |
IC50 |
= |
97.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
1060.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2339 |
Cell Line |
TGBC24TKB |
Homo sapiens |
IC50 |
= |
2414.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2510 |
Cell Line |
GCT |
Homo sapiens |
IC50 |
= |
861.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2203 |
Cell Line |
GDM-1 |
Homo sapiens |
IC50 |
= |
159.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
175.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2511 |
Cell Line |
HGC-27 |
Homo sapiens |
IC50 |
= |
13.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
44.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
323.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2207 |
Cell Line |
KP-N-YN |
Homo sapiens |
IC50 |
= |
1663.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
218.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2513 |
Cell Line |
LK-2 |
Homo sapiens |
IC50 |
= |
581.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2514 |
Cell Line |
LN-405 |
Homo sapiens |
IC50 |
= |
1801.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2844 |
Cell Line |
MES-SA |
Homo sapiens |
IC50 |
= |
99.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2515 |
Cell Line |
MFE-280 |
Homo sapiens |
IC50 |
= |
1668.12 |
nM |
10.6019/CHEMBL1201861 |
NPT3882 |
Cell Line |
MFE-296 |
Homo sapiens |
IC50 |
= |
70.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2196 |
Cell Line |
NB1 |
Homo sapiens |
IC50 |
= |
45.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
188.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
277.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
133.21 |
nM |
10.6019/CHEMBL1201861 |
NPT1669 |
Cell Line |
NCI-H1792 |
Homo sapiens |
IC50 |
= |
572.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2334 |
Cell Line |
NCI-H1793 |
Homo sapiens |
IC50 |
= |
900.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
EC50 |
= |
390 |
nM |
23600925 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
110 |
nM |
23600925 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
270 |
nM |
23600925 |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
140 |
nM |
23600925 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
240 |
nM |
23600925 |
NPT3555 |
Cell Line |
HOS-TE85 |
Homo sapiens |
IC50 |
= |
590 |
nM |
23600925 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
23600925 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
670 |
nM |
23600925 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
65 |
nM |
23600925 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
170 |
nM |
23600925 |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
76 |
nM |
23600925 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
100 |
nM |
23600925 |
NPT3554 |
Cell Line |
SK-ES1 |
|
IC50 |
= |
42 |
nM |
23600925 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
90 |
nM |
23600925 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
170 |
nM |
23600925 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.38 |
ug/ml |
23511021 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.26 |
ug/ml |
23511021 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.29 |
ug/ml |
23511021 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.24 |
ug/ml |
23511021 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
23511021 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
130 |
nM |
23634786 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23634786 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
10 |
nM |
23634786 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
23634786 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
410 |
nM |
23548547 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
120 |
nM |
23548547 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
23501113 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
23501113 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.9 |
|
23578690 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
86 |
nM |
23578690 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
76 |
nM |
23578690 |
NPT2548 |
Cell Line |
SNU-638 |
Homo sapiens |
IC50 |
= |
840 |
nM |
23608763 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
2910 |
nM |
23608763 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
940 |
nM |
23806110 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
590 |
nM |
23806110 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
740 |
nM |
23806110 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
1200 |
nM |
23806110 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5000000 |
nM |
23685942 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
2500000 |
nM |
23685942 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2500000 |
nM |
23685942 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5000000 |
nM |
23685942 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.2 |
nM |
23484434 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1100 |
nM |
23484434 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
144.8 |
nM |
23623253 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
65.4 |
nM |
23623253 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
64.1 |
nM |
23623253 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
28 |
nM |
23623253 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
82 |
nM |
23664877 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
500 |
nM |
23664877 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
750 |
nM |
23639650 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
560 |
nM |
23639650 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
900 |
nM |
23639650 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
28.2 |
|
23673218 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
271 |
nM |
23673218 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9.6 |
nM |
23673218 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
23802716 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
70 |
nM |
23802716 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
80 |
nM |
23802716 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1810 |
nM |
23802716 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
120 |
nM |
23802716 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
750 |
nM |
23802716 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23802716 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
42 |
% |
23643901 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7360 |
nM |
23708013 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5460 |
nM |
23708013 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4100 |
nM |
23748152 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
23748152 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
23748152 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1210 |
nM |
23764302 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
23764302 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
501 |
nM |
23764302 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
451 |
nM |
23764302 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.4 |
ug/ml |
23831694 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.1 |
ug/ml |
23831694 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
120 |
nM |
23795891 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15880 |
nM |
23795891 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
380 |
nM |
23795891 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
500 |
nM |
23799303 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
700 |
nM |
23799303 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
19950 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
25400 |
nM |
23831811 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
5010 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
6310 |
nM |
23831811 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
200 |
nM |
23831811 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
20 |
nM |
23831811 |
NPT639 |
Cell Line |
NCI-H187 |
Homo sapiens |
IC50 |
= |
140 |
nM |
23806014 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7660 |
nM |
23806014 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
560 |
nM |
23806014 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
630 |
nM |
23810282 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
440 |
nM |
23810282 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
23810282 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
130 |
nM |
23815260 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
10 |
nM |
23815260 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
10 |
nM |
23815260 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
23815260 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
210 |
nM |
23848233 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
65 |
nM |
23777898 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
72 |
nM |
23777898 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
3240 |
nM |
23850203 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
= |
37700 |
nM |
23792351 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
28300 |
nM |
23792351 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
26100 |
nM |
23792351 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
LC50 |
= |
21400 |
nM |
23792351 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1020 |
nM |
23871222 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
5720 |
nM |
23871222 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
TGI |
= |
45500 |
nM |
23876338 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
10300 |
nM |
23876338 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
4900 |
nM |
23876338 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
TGI |
= |
3600 |
nM |
23876338 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
TGI |
= |
2500 |
nM |
23876338 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
TGI |
= |
2100 |
nM |
23876338 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
= |
1000 |
nM |
23876338 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
TGI |
= |
400 |
nM |
23876338 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
TGI |
= |
200 |
nM |
23876338 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
23 |
nM |
23886686 |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
23849207 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
170 |
nM |
23849207 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
170 |
nM |
23849207 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
23849207 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
23849207 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
23849207 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
23849207 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
23849207 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
100 |
nM |
23849207 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
LC50 |
= |
2520 |
nM |
23871905 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
GI50 |
= |
50 |
nM |
23871905 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
LC50 |
= |
85700 |
nM |
23871905 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
= |
60 |
nM |
23871905 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
LC50 |
= |
21330 |
nM |
23871905 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
= |
230 |
nM |
23871905 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
LC50 |
= |
85700 |
nM |
23871905 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
= |
330 |
nM |
23871905 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
LC50 |
= |
34750 |
nM |
23871905 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
510 |
nM |
23871905 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
51290 |
nM |
23871905 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
30 |
nM |
23871905 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
110 |
nM |
23871905 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
LC50 |
= |
87100 |
nM |
23871905 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
320 |
nM |
23871905 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
LC50 |
= |
26180 |
nM |
23871905 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
= |
490 |
nM |
23871905 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
LC50 |
= |
86700 |
nM |
23871905 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
= |
180 |
nM |
23871905 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
LC50 |
= |
72440 |
nM |
23871905 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
= |
70 |
nM |
23871905 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
LC50 |
= |
4690 |
nM |
23871905 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
= |
950 |
nM |
23871905 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
80 |
nM |
23871905 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
LC50 |
= |
1900 |
nM |
23871905 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
LC50 |
= |
51640 |
nM |
23871905 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
130 |
nM |
23871905 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
13510 |
nM |
23932340 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
910 |
nM |
23932340 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
509 |
nM |
23932340 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
459 |
nM |
23932340 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
1900 |
nM |
23964644 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
GI50 |
= |
510 |
nM |
23964644 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
1800 |
nM |
23964644 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
2000 |
nM |
23964644 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
520 |
nM |
23964644 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
1400 |
nM |
23964644 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
520 |
nM |
24025124 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
700 |
nM |
24025124 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
= |
220 |
nM |
23871905 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
7160 |
nM |
23871905 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
LC50 |
= |
43250 |
nM |
23871905 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
= |
410 |
nM |
23871905 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
LC50 |
= |
74300 |
nM |
23871905 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
= |
370 |
nM |
23871905 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
LC50 |
= |
84330 |
nM |
23871905 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
= |
390 |
nM |
23871905 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
= |
170 |
nM |
23871905 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
LC50 |
= |
740 |
nM |
23871905 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
= |
120 |
nM |
23871905 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
LC50 |
= |
8150 |
nM |
23871905 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
= |
140 |
nM |
23871905 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
LC50 |
= |
490 |
nM |
23871905 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
= |
80 |
nM |
23871905 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
LC50 |
= |
15920 |
nM |
23871905 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
= |
210 |
nM |
23871905 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
LC50 |
= |
1060 |
nM |
23871905 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
= |
170 |
nM |
23871905 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
LC50 |
= |
9570 |
nM |
23871905 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
= |
250 |
nM |
23871905 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
LC50 |
= |
4050 |
nM |
23871905 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
= |
180 |
nM |
23871905 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
LC50 |
= |
3970 |
nM |
23871905 |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
= |
120 |
nM |
23871905 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
LC50 |
= |
50350 |
nM |
23871905 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
= |
70 |
nM |
23871905 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
LC50 |
= |
30620 |
nM |
23871905 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
= |
40 |
nM |
23871905 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
LC50 |
= |
3300 |
nM |
23871905 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
= |
70 |
nM |
23871905 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
LC50 |
= |
49770 |
nM |
23871905 |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
= |
40 |
nM |
23871905 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
LC50 |
= |
27230 |
nM |
23871905 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
= |
120 |
nM |
23871905 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
LC50 |
= |
69980 |
nM |
23871905 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
= |
30480 |
nM |
23871905 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
LC50 |
= |
58610 |
nM |
23871905 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
90 |
nM |
23871905 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
LC50 |
= |
92680 |
nM |
23871905 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
= |
270 |
nM |
23871905 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
LC50 |
= |
67450 |
nM |
23871905 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
120 |
nM |
23871905 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
= |
6460 |
nM |
23871905 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LC50 |
= |
54580 |
nM |
23871905 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
80 |
nM |
23871905 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
LC50 |
= |
21680 |
nM |
23871905 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
= |
260 |
nM |
23871905 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
LC50 |
= |
4330 |
nM |
23871905 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
180 |
nM |
23871905 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
LC50 |
= |
2800 |
nM |
23871905 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
= |
30 |
nM |
23871905 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
51290 |
nM |
23871905 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
20 |
nM |
23871905 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
LC50 |
= |
67760 |
nM |
23871905 |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
= |
540 |
nM |
23871905 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
LC50 |
= |
13150 |
nM |
23871905 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
150 |
nM |
23871905 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
LC50 |
= |
6400 |
nM |
23871905 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
= |
50 |
nM |
23871905 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
LC50 |
= |
42270 |
nM |
23871905 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
= |
100 |
nM |
23871905 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
LC50 |
= |
67610 |
nM |
23871905 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
70 |
nM |
23871905 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
47970 |
nM |
23871905 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
410 |
nM |
23871905 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
60 |
nM |
23871905 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
= |
30 |
nM |
23871905 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
= |
80 |
nM |
23871905 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
= |
30 |
nM |
23871905 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
450 |
nM |
23911578 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1210 |
nM |
23911578 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
500 |
nM |
23911578 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
23911578 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
190 |
nM |
23871905 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
LC50 |
= |
89330 |
nM |
23871905 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
120 |
nM |
23871905 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
LC50 |
= |
100000 |
nM |
23871905 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
= |
80 |
nM |
23871905 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.7 |
ug/ml |
23891181 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.9 |
ug/ml |
23891181 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
5 |
ug/ml |
23891181 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3240 |
nM |
23835482 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
LC50 |
= |
4300 |
nM |
23869452 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
23849207 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
IC50 |
= |
2800 |
nM |
24044895 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
900 |
nM |
24044895 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
700 |
nM |
24044895 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24.4 |
ug/ml |
24012683 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.18 |
ug/ml |
24012683 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
8830 |
nM |
23994327 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7710 |
nM |
23994327 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
7360 |
nM |
23994327 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
EC50 |
= |
40 |
nM |
23988351 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
EC50 |
= |
290 |
nM |
23988351 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
250 |
nM |
23988351 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
< |
100 |
nM |
10.1007/s00044-013-0855-2 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
TGI |
> |
100 |
nM |
10.1007/s00044-013-0855-2 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
100 |
nM |
10.1007/s00044-013-0855-2 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
> |
100 |
nM |
10.1007/s00044-013-0855-2 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
LC50 |
> |
100000 |
nM |
10.1007/s00044-013-0855-2 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
> |
100000 |
nM |
10.1007/s00044-013-0855-2 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
10.1007/s00044-013-0854-3 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1010 |
nM |
10.1007/s00044-013-0854-3 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
24021462 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
24021462 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
24021462 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
30 |
nM |
24021462 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
920 |
nM |
24021462 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
24021462 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Ratio IC50 |
= |
14 |
|
24028446 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1560 |
nM |
24028446 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
150 |
nM |
24028446 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
1100 |
nM |
24028446 |
NPT2257 |
Cell Line |
MCF-10A |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24028446 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
21900 |
nM |
24028446 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24028446 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24028446 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
90 |
nM |
10.1007/s00044-013-0712-3 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
90 |
nM |
10.1007/s00044-013-0712-3 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
40 |
nM |
10.1007/s00044-013-0712-3 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
850 |
nM |
23992864 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
730 |
nM |
23992864 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
310 |
nM |
23992864 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
410 |
nM |
23992864 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
100 |
nM |
24050254 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
24050254 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
Inhibition |
= |
81.36 |
% |
10.1007/s00044-013-0730-1 |
NPT180 |
Cell Line |
HCT-8 |
Homo sapiens |
Inhibition |
= |
97.07 |
% |
10.1007/s00044-013-0730-1 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
Inhibition |
= |
94.64 |
% |
10.1007/s00044-013-0730-1 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
440 |
nM |
10.1007/s00044-013-0777-z |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
790 |
nM |
10.1007/s00044-013-0777-z |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
830 |
nM |
10.1007/s00044-013-0777-z |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
1006 |
nM |
10.1007/s00044-013-0784-0 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3980 |
nM |
10.1007/s00044-013-0784-0 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
190 |
nM |
10.1007/s00044-013-0788-9 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
220 |
nM |
10.1007/s00044-013-0788-9 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
300 |
nM |
10.1007/s00044-013-0788-9 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
28 |
nM |
10.1007/s00044-013-0788-9 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
2560 |
nM |
10.1007/s00044-013-0795-x |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2680 |
nM |
10.1007/s00044-013-0795-x |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2440 |
nM |
10.1007/s00044-013-0795-x |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
90 |
nM |
24128115 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
350 |
nM |
24128115 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
< |
2 |
|
10.1007/s00044-013-0854-3 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
740 |
nM |
10.1007/s00044-013-0854-3 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
30210 |
nM |
24077528 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
32780 |
nM |
24077528 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
24330 |
nM |
24077528 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
27110 |
nM |
24077528 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
19220 |
nM |
24077528 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
33980 |
nM |
24077528 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
24099994 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
= |
28 |
nM |
24113365 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
144.8 |
nM |
24113365 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
64.1 |
nM |
24113365 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
65.4 |
nM |
24113365 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1210 |
nM |
24113366 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
24113366 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
501 |
nM |
24113366 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
451 |
nM |
24113366 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
14.1 |
ug/ml |
24090920 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Inhibition |
= |
82 |
% |
24095746 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Inhibition |
= |
88 |
% |
24095746 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
91 |
% |
24095746 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4.11 |
ug/ml |
24095746 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3.9 |
ug/ml |
24095746 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2.8 |
ug/ml |
24095746 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3.2 |
nM |
24013411 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2.5 |
nM |
24013411 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
3070 |
nM |
24013413 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2680 |
nM |
24013413 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1380 |
nM |
24013413 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
410 |
nM |
24013413 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
Inhibition |
= |
21 |
% |
24095089 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
Inhibition |
= |
13 |
% |
24095089 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
300 |
nM |
24095089 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1500 |
nM |
24095089 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
200 |
nM |
24095089 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
200 |
nM |
24095089 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
24095089 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24095089 |
NPT2 |
Others |
Unspecified |
|
IC50 |
< |
100 |
nM |
24095089 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
IC50 |
> |
20000 |
nM |
24095089 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
< |
100 |
nM |
24095089 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
400 |
nM |
24095089 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Inhibition |
= |
90 |
% |
24095089 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
83.5 |
% |
24095089 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Inhibition |
= |
85.8 |
% |
24095089 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
80.6 |
% |
24095089 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
6.9 |
% |
24095089 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
Inhibition |
= |
86 |
% |
24095089 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
92.6 |
% |
24095089 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
Inhibition |
= |
41 |
% |
24095089 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
Inhibition |
= |
88.1 |
% |
24095089 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
Inhibition |
= |
96.2 |
% |
24095089 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
80.7 |
nM |
24012378 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.04 |
|
24012378 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.9 |
|
24012378 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Ratio IC50 |
= |
0.4 |
|
24012378 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.4 |
|
24012378 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
0.16 |
|
24012378 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.03 |
|
24012378 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
24012378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7800 |
nM |
24095093 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
70 |
nM |
24095093 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
90 |
nM |
24012378 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
200 |
nM |
24012378 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
200 |
nM |
24012378 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24012378 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
78 |
nM |
24012378 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
24080103 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
20 |
nM |
24080103 |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
FC |
> |
100 |
|
24141203 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.87 |
ug/ml |
24177357 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.6 |
ug/ml |
24177357 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.8 |
ug/ml |
24177357 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
1380 |
nM |
24182355 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
970 |
nM |
24182355 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
980 |
nM |
24182355 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24182355 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1480 |
nM |
24182355 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11 |
nM |
24195466 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
100 |
nM |
24158013 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
70 |
nM |
24158013 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
90 |
nM |
24158013 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
2750 |
nM |
24161704 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3130 |
nM |
24161704 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
411 |
nM |
24231309 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
24231309 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
877 |
nM |
24231309 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
90 |
nM |
24215890 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
400000 |
nM |
24184076 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
310 |
nM |
24184076 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
GI50 |
= |
320 |
nM |
24184076 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
240 |
nM |
24184076 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
120 |
nM |
24148837 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
320 |
nM |
24148837 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1170 |
nM |
24148837 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
95610 |
nM |
24148837 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
120 |
nM |
24148837 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
750 |
nM |
24148837 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
790 |
nM |
24251417 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
680 |
nM |
24251417 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
270 |
nM |
24251417 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
350 |
nM |
24251417 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
310 |
nM |
24251417 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
50 |
nM |
24251417 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1070 |
nM |
24287557 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
910 |
nM |
24287557 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
509 |
nM |
24287557 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
459 |
nM |
24287557 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
62 |
% |
24287561 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
69 |
% |
24332623 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24300737 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24300737 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24300737 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24300737 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
700 |
nM |
24300737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.89 |
ug/ml |
24269165 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
3.26 |
ug/ml |
24269165 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
24287557 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
1510 |
nM |
24387625 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
24387625 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
700 |
nM |
24387625 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
410 |
nM |
24387625 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
50 |
nM |
24387625 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
24387625 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
34.07 |
nM |
24411197 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
59.77 |
nM |
24411197 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
136.2 |
nM |
24411197 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
170 |
nM |
24370114 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
24370114 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
160 |
nM |
24370114 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
210 |
nM |
24370114 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
20 |
nM |
24370114 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3170 |
nM |
23792352 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
23792352 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LD50 |
= |
1.2 |
nM |
24437979 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
990 |
nM |
24437979 |
NPT3171 |
Cell Line |
V79 |
Cricetulus griseus |
IC50 |
= |
240 |
nM |
24530030 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
160 |
nM |
24530030 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
420 |
nM |
24530030 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
370 |
nM |
24530030 |
NPT3881 |
Cell Line |
MX1 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24530030 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
130 |
nM |
24530030 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
530 |
nM |
24530030 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
440 |
nM |
24530030 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
20 |
nM |
24530030 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
24530030 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
400 |
nM |
24530030 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
830 |
nM |
24530030 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
350 |
nM |
24530030 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
24530030 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1760 |
nM |
24487188 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
190 |
nM |
24487188 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
24487188 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
1990 |
nM |
24487188 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
360 |
nM |
24487188 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10900 |
nM |
24487188 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
390 |
nM |
24487188 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
10 |
nM |
23827179 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
23827179 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
23827179 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3510 |
nM |
24418772 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
2430 |
nM |
24418772 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1650 |
nM |
24418772 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
423 |
nM |
24398294 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
37 |
nM |
24398294 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
488 |
nM |
24398294 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
230 |
nM |
24398294 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
440 |
nM |
24513041 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
650 |
nM |
24513041 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
1700 |
nM |
24485783 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
Activity |
= |
5 |
% |
24051300 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
Activity |
= |
14 |
% |
24051300 |
NPT144 |
Individual Protein |
Telomerase reverse transcriptase |
Homo sapiens |
Activity |
= |
34 |
% |
24051300 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
24051300 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17 |
% |
24051300 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
> |
10000 |
nM |
24484281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4800 |
nM |
24484281 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
24484281 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500 |
nM |
24484281 |
NPT2 |
Others |
Unspecified |
|
GI50 |
> |
1000 |
nM |
24502276 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
676.08 |
nM |
24502276 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
0.26 |
ug/ml |
24589485 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
0.03 |
ug/ml |
24589485 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
0.02 |
ug/ml |
24589485 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.34 |
ug/ml |
24589485 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6940 |
nM |
24607876 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
7410 |
nM |
24607876 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
8190 |
nM |
24607876 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7470 |
nM |
24607876 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24507927 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
800 |
nM |
24507927 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
700 |
nM |
24507927 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
24507927 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23270 |
nM |
24561670 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2585 |
|
24561670 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
9 |
nM |
24561670 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
1060 |
nM |
24582982 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1310 |
nM |
24582982 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1150 |
nM |
24582982 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
530 |
nM |
10.1039/C3MD00149K |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
1800 |
nM |
10.1039/C3MD00149K |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
215000 |
nM |
10.1039/C3MD00149K |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
179000 |
nM |
10.1039/C3MD00149K |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1100 |
nM |
10.1039/C3MD00166K |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
10.1039/C3MD00166K |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
900 |
nM |
10.1039/C3MD00166K |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
10900 |
nM |
10.1039/C2MD20270K |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
8700 |
nM |
10.1039/C2MD20270K |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6300 |
nM |
10.1039/C2MD20270K |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
< |
1000 |
nM |
10.1039/C3MD00097D |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
7000 |
nM |
10.1039/C3MD00097D |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
10.1039/C3MD00097D |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
GI50 |
= |
85 |
nM |
24163729 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
150 |
nM |
24163729 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
354.8 |
nM |
PubChem BioAssay data set |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
281.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
525.8 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
477 |
nM |
10.1039/C0MD00219D |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
400 |
nM |
10.1039/C0MD00219D |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
456 |
nM |
10.1039/C0MD00219D |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
110 |
nM |
10.1039/C1MD00234A |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
700 |
nM |
10.1039/C1MD00234A |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
6.4 |
|
10.1039/C1MD00234A |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60 |
% |
10.1039/C0MD00252F |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
94.85 |
% |
10.1039/C0MD00116C |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
4 |
% |
10.1039/C0MD00116C |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
1.15 |
% |
10.1039/C0MD00116C |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1400 |
nM |
10.1039/C1MD00038A |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
10.1039/C1MD00038A |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2600 |
nM |
10.1039/C1MD00038A |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
88.2 |
% |
10.1039/C1MD00038A |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI |
= |
94.7 |
% |
10.1039/C1MD00038A |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
GI |
= |
84.2 |
% |
10.1039/C1MD00038A |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
GI |
= |
93.1 |
% |
10.1039/C1MD00038A |
NPT2 |
Others |
Unspecified |
|
GI |
= |
90.7 |
% |
10.1039/C1MD00038A |
NPT2 |
Others |
Unspecified |
|
GI |
= |
95.9 |
% |
10.1039/C1MD00038A |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
164 |
nM |
10.1039/C1MD00155H |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10.1039/C1MD00155H |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
154 |
nM |
10.1039/C1MD00155H |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
16 |
% |
10.1039/C2MD20302B |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
2 |
% |
10.1039/C2MD20302B |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
82 |
% |
10.1039/C2MD20302B |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Inhibition |
= |
79 |
% |
10.1039/C3MD00193H |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
70 |
nM |
10.1039/C0MD00179A |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
109 |
nM |
10.1039/C0MD00179A |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
223 |
nM |
10.1039/C0MD00179A |
NPT1059 |
Cell Line |
HMEC |
Homo sapiens |
GI50 |
= |
276 |
nM |
10.1039/C0MD00179A |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
GI50 |
= |
462 |
nM |
10.1039/C0MD00179A |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
7250 |
nM |
10.1039/C1MD00072A |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI50 |
= |
170 |
nM |
10.1039/C1MD00072A |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
160 |
nM |
10.1039/C1MD00072A |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
160 |
nM |
10.1039/C1MD00072A |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
= |
170 |
nM |
10.1039/C1MD00072A |
NPT133 |
Cell Line |
ZR-75-1 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
10.1039/C1MD00072A |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
250 |
nM |
10.1039/C1MD00193K |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
13 |
|
10.1039/C2MD20302B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
31000 |
nM |
10.1039/C2MD20302B |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
370 |
nM |
10.1039/C2MD20302B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
140 |
nM |
10.1039/C2MD20302B |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
730 |
nM |
10.1039/C2MD20302B |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
160 |
nM |
10.1039/C2MD20302B |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
100 |
nM |
10.1039/C2MD20302B |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
95610 |
nM |
10.1039/C2MD20327H |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1170 |
nM |
10.1039/C2MD20327H |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
750 |
nM |
10.1039/C2MD20327H |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
360 |
nM |
10.1039/C2MD20327H |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
320 |
nM |
10.1039/C2MD20327H |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10.1039/C2MD20327H |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
120 |
nM |
10.1039/C2MD20327H |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
= |
140 |
nM |
10.1039/C1MD00072A |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
= |
140 |
nM |
10.1039/C1MD00072A |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
170 |
nM |
10.1039/C1MD00072A |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1830 |
nM |
10.1039/C1MD00072A |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
970 |
nM |
10.1039/C2MD20023F |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8140 |
nM |
10.1039/C2MD20023F |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
14840 |
nM |
10.1039/C2MD20023F |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
15070 |
nM |
10.1039/C2MD20023F |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
10550 |
nM |
10.1039/C3MD00013C |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
10880 |
nM |
10.1039/C3MD00013C |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
10.1039/C3MD00013C |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
950 |
nM |
10.1039/C3MD00013C |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1120 |
nM |
10.1039/C3MD00013C |
NPT566 |
Organism |
Salmonella typhimurium |
Salmonella enterica subsp. enterica serovar Typhimurium |
Activity |
= |
108 |
nmol |
423181 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.5 |
nM |
423181 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.7 |
nM |
423181 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.5 |
nM |
423182 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
423182 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
4.4 |
mg/kg |
423191 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
460 |
nM |
24742385 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
510 |
nM |
24742385 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
910 |
nM |
24742385 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1070 |
nM |
24742385 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
> |
200000 |
nM |
24742385 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
13600 |
nM |
24681979 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
16000 |
nM |
24681979 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15400 |
nM |
24681979 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
16900 |
nM |
24681979 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
550 |
nM |
23932070 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
20.2 |
nM |
24211639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
578.2 |
nM |
24211639 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
40 |
nM |
24631190 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
24631190 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
170 |
nM |
24631190 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6500 |
nM |
24631190 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
500 |
nM |
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
12 |
|
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.27 |
|
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
44.5 |
|
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.82 |
|
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.07 |
|
24631190 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
37.94 |
|
24631190 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
77 |
nM |
24684844 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68434 |
nM |
24684844 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
888.75 |
|
24684844 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
150 |
nM |
24650643 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
180 |
nM |
24650643 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
330 |
nM |
24650643 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
550 |
nM |
24650643 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
550 |
nM |
24686011 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
= |
150 |
nM |
24686011 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
330 |
nM |
24686011 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
200 |
nM |
24650715 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
50 |
nM |
24650715 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
0.257 |
|
24686014 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
0.158 |
|
24686014 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
0.098 |
|
24686014 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio |
= |
0.125 |
|
24686014 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6100 |
nM |
24686014 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.002 |
nM |
490537 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.7 |
nM |
490537 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
176 |
mg/kg |
490545 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
Activity |
= |
104 |
mg/kg |
490545 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.5 |
nM |
490536 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.58 |
nM |
490536 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Ratio ED50 |
= |
2.6 |
|
490536 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
1.5 |
% |
628003 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
0.58 |
% |
628003 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
80 |
nM |
24717154 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
120 |
nM |
24717154 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
120 |
nM |
24717154 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
980 |
nM |
24717154 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
1870 |
nM |
24717154 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2000 |
nM |
24592993 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
178 |
nM |
24792464 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
830 |
nM |
24836071 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
790 |
nM |
24836071 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
440 |
nM |
24836071 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10890 |
nM |
24793880 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
6700 |
nM |
24793880 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8400 |
nM |
24793880 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8620 |
nM |
24793880 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
480 |
nM |
24852278 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
640 |
nM |
24852278 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
220 |
nM |
24852278 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24852278 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
24780595 |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
IC50 |
= |
700 |
nM |
24780595 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
800 |
nM |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
600 |
nM |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
3033.7 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
3331.1 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
3791.8 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4007.5 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4794.2 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
4994.1 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
6690.3 |
FU/min |
24780595 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
7240.4 |
FU/min |
24780595 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
70 |
nM |
24780599 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
20 |
nM |
24780599 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
24780599 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
28.9 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
34.5 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
52.2 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
22.5 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
50.8 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Inhibition |
= |
56.9 |
% |
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Ratio |
= |
152 |
|
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Ratio |
= |
121 |
|
1271407 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
32 |
nM |
915894 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.67 |
nM |
915894 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
Activity |
= |
1 |
mg/kg |
915894 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
1.5 |
nM |
915894 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.8 |
nM |
176359 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
ED50 |
= |
0.9 |
nM |
176359 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
390 |
nM |
24953027 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
840 |
nM |
24904965 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
930 |
nM |
24904965 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3760 |
nM |
24904965 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
4880 |
nM |
24904965 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10900 |
nM |
24953027 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
360 |
nM |
24953027 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
1990 |
nM |
24953027 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
24953027 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
190 |
nM |
24953027 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1760 |
nM |
24953027 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
85.13 |
% |
24844196 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
Inhibition |
= |
69.2 |
% |
24844196 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
90.66 |
% |
24844196 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
56.93 |
% |
24844196 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
73.92 |
% |
24844196 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
73.22 |
% |
24844196 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
67.63 |
% |
24844196 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Inhibition |
= |
69.05 |
% |
24844196 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
912 |
nM |
24844756 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
24910974 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
500 |
nM |
24910974 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
130 |
nM |
24824796 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1360 |
nM |
24941129 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
24941129 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1500 |
nM |
24941129 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
12500 |
nM |
24974349 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
90 |
nM |
24858544 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11300 |
nM |
24858544 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
118 |
|
24858544 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
-35.58 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
-27.62 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
-18.52 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
-12.52 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
-10.35 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0.25 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0.95 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
1.56 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
3.35 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
6350 |
nM |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
11.4 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
11.62 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13250 |
nM |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
18.38 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
24.25 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
30.15 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
30.25 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
32.31 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1000 |
nM |
24835787 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1340 |
nM |
24835787 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
1630 |
nM |
24835787 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
= |
1650 |
nM |
24835787 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
1660 |
nM |
24835787 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
1790 |
nM |
24835787 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
50.62 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
69.86 |
% |
24929289 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
76.31 |
% |
24929289 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Inhibition |
= |
88.36 |
% |
24929289 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
455 |
nM |
24996140 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.1 |
nM |
24996140 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
24946216 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.314 |
% |
24878360 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.309 |
% |
24878360 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.251 |
% |
24878360 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.266 |
% |
24878360 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8020 |
nM |
24878360 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
330 |
nM |
24941130 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
310 |
nM |
24941130 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
350 |
nM |
24941130 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
330 |
nM |
24941130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
350 |
nM |
24941130 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
340 |
nM |
24941130 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
2 |
% |
24941130 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
5 |
% |
24941130 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
4 |
% |
24941130 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2 |
% |
24941130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
1 |
% |
24941130 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
2 |
% |
24941130 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
45 |
% |
24941130 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
49 |
% |
24941130 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
Activity |
= |
47 |
% |
24941130 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
34 |
% |
24941130 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
44 |
% |
24941130 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
28 |
% |
24941130 |
NPT3901 |
Tissue |
Chorioallantoic membrane |
Gallus gallus |
IC50 |
= |
0.04 |
nM |
24890652 |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
IC50 |
= |
1.35 |
nM |
24890652 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
0.7 |
ug/ml |
24828374 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
0.8 |
ug/ml |
24828374 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
24828374 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3240 |
nM |
24856067 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
620 |
nM |
25537271 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
770 |
nM |
25537271 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2780 |
nM |
25462233 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
500 |
nM |
25554367 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
25554367 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
300 |
nM |
25554367 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2900 |
nM |
25554367 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
900 |
nM |
25462233 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3820 |
nM |
25462233 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
4060 |
nM |
25462233 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2120 |
nM |
25462233 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
73 |
nM |
25462234 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
97 |
nM |
25462234 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
85 |
nM |
25462234 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
23 |
nM |
25462234 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
360 |
nM |
25462264 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.3 |
10'-11uM |
25468043 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
14000 |
nM |
25468043 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17000 |
nM |
25468043 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.302 |
ug/ml |
25468043 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
450 |
nM |
25462264 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
530 |
nM |
25462264 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
52500 |
nM |
25462264 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
67600 |
nM |
25462264 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3450 |
nM |
25462265 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7700 |
nM |
25462265 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1170 |
nM |
25462265 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
25478997 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.5 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.15 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
14.7 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
81.65 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
23 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.5 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40 |
% |
25462273 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.5 |
% |
25462273 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
400 |
nM |
25481396 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1000 |
nM |
25481396 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
860 |
nM |
25481396 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1080 |
nM |
25481396 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
25453798 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1500 |
nM |
25453799 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
390 |
nM |
25453799 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
360 |
nM |
25453799 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
124 |
nM |
25462279 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
69 |
nM |
25462279 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
154 |
nM |
25462279 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
6000 |
nM |
25453802 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3400 |
nM |
25453802 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
25453802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3500 |
nM |
25453802 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25490132 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
25490132 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
400 |
nM |
25490132 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
500 |
nM |
25490132 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
5 |
% |
25466181 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40.7 |
% |
25466181 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
123 |
nM |
25497963 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
414 |
nM |
25497963 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
210 |
nM |
25529742 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
180 |
nM |
25529742 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
25499433 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19.9 |
nM |
25499433 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
13.52 |
nM |
24973030 |
NPT1523 |
Cell Line |
NFF |
Homo sapiens |
IC50 |
= |
125.6 |
nM |
24973030 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
8.97 |
|
24973030 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1.21 |
ug/ml |
25042338 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1.09 |
ug/ml |
25042338 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10 |
nM |
25059501 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
10 |
nM |
25059501 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10 |
nM |
25059501 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
660 |
nM |
25059501 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
79 |
% |
25062007 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
84 |
% |
25062007 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
830 |
nM |
25078311 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
790 |
nM |
25078311 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
440 |
nM |
25078311 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
690 |
nM |
25089733 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
470 |
nM |
25089733 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1220 |
nM |
25089733 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
= |
0.54 |
ug/ml |
25062010 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.038 |
ug/ml |
25062010 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
GI50 |
= |
0.039 |
ug/ml |
25062010 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
0.15 |
ug/ml |
25062010 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
25062010 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
3.8 |
ug/ml |
25062010 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.43 |
ug/ml |
25062010 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
GI50 |
= |
0.11 |
ug/ml |
25062010 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2900 |
nM |
25105722 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1.4 |
nM |
25098650 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
21.7 |
nM |
25098650 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
2.5 |
nM |
25098650 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
107.7 |
nM |
25098650 |
NPT176 |
Organism |
Artemia salina |
Artemia salina |
LD50 |
= |
0.434 |
ug/ml |
25036793 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
15530 |
nM |
25064350 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6750 |
nM |
25064350 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7040 |
nM |
25064350 |
NPT2738 |
Cell Line |
Ishikawa |
Homo sapiens |
IC50 |
= |
9020 |
nM |
25064350 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3000 |
nM |
25096298 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
25096298 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5490000 |
nM |
24583357 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4230 |
nM |
24969014 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
420 |
nM |
24969014 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1530 |
nM |
24969014 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1250 |
nM |
24969014 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
9360 |
nM |
24969014 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
7.5 |
|
24969014 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
570 |
nM |
25019480 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
239 |
nM |
25019480 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
258 |
nM |
25019480 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
95.6 |
nM |
25025853 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11296 |
nM |
25025853 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
118 |
|
25025853 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
340 |
nM |
25247771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
840 |
nM |
25247771 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1470 |
nM |
25247771 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
nM |
25247772 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220 |
nM |
25247772 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
25247772 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
210 |
nM |
25247772 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
180 |
nM |
25247772 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
2040 |
nM |
25160837 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
330 |
nM |
25160837 |
NPT2609 |
Cell Line |
BeWo |
Homo sapiens |
IC50 |
= |
1070 |
nM |
25160837 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
420 |
nM |
25160837 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220 |
nM |
25163667 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
220 |
nM |
25163667 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
250 |
nM |
25163667 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
400 |
nM |
25163667 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
140 |
nM |
25353976 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
540 |
nM |
25127463 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
320 |
nM |
25127463 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
310 |
nM |
25127463 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7860 |
nM |
25127463 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
73 |
nM |
25264072 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
97 |
nM |
25264072 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
85 |
nM |
25264072 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
23 |
nM |
25264072 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI |
= |
79.8 |
% |
25409491 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
5960 |
nM |
25140752 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8050 |
nM |
25140752 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
8500 |
nM |
25140752 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2600 |
nM |
25300819 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
690 |
nM |
25300819 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
25147145 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
880 |
nM |
25147145 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
25147145 |
NPT2 |
Others |
Unspecified |
|
EC50 |
> |
200 |
ug/ml |
25147145 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
600 |
nM |
25172418 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
600 |
nM |
25172418 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
700 |
nM |
25172418 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
600 |
nM |
25172418 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
450 |
nM |
25172420 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.314 |
% |
25255434 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.309 |
% |
25255434 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.251 |
% |
25255434 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
0.266 |
% |
25255434 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8.02 |
nM |
25255434 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
10 |
nM |
25282267 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
20 |
nM |
25282267 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
200 |
nM |
25300820 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
700 |
nM |
25300820 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
> |
10000 |
nM |
25300820 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
700 |
nM |
25300820 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
25300820 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
109 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
83 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
91 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
36.9 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
52 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
55.8 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
16 |
% |
25302569 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
28.3 |
% |
25302569 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
500 |
nM |
25172420 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
25172420 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1210 |
nM |
25172420 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
360 |
nM |
25314138 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
740 |
nM |
25314138 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
25314138 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
650 |
nM |
25314138 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
460 |
nM |
25314138 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1574200 |
nM |
25314138 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
0.1 |
ug/ml |
25372601 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
= |
1 |
ug/ml |
25372601 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
CC50 |
= |
2 |
ug/ml |
25372601 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.21 |
|
25375258 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2400 |
nM |
25375258 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
19600 |
nM |
25375258 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.12 |
|
25375258 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1100 |
nM |
25375258 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5400 |
nM |
25375258 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
25241926 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
700 |
nM |
25241926 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
800 |
nM |
25241926 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
600 |
nM |
25241926 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
170 |
nM |
25215856 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28200 |
nM |
25215856 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
166 |
|
25215856 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
920 |
nM |
25259516 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
25259516 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
30 |
nM |
25259516 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
25259516 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
25259516 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
90 |
nM |
25259516 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
65 |
nM |
25259516 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25259516 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7000 |
nM |
25244612 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1400 |
nM |
25244612 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
25244612 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
370 |
nM |
25244612 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
800 |
nM |
25244612 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4400 |
nM |
25244612 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
8.8 |
|
25244612 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.1 |
|
25244612 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
GI50 |
= |
120 |
nM |
25317694 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
13500 |
nM |
25317694 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
112.5 |
|
25317694 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
880 |
nM |
25419616 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
740 |
nM |
25419616 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
870 |
nM |
25419616 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
912 |
nM |
25245672 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
TGI |
= |
0.92 |
ug/ml |
25510639 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
3.3 |
ug/ml |
25510639 |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
TGI |
= |
1.6 |
ug/ml |
25510639 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
TGI |
> |
25 |
ug/ml |
25510639 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
4.9 |
ug/ml |
25510639 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
11.7 |
ug/ml |
25510639 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
7.6 |
ug/ml |
25510639 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
TGI |
= |
2.3 |
ug/ml |
25510639 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
TGI |
= |
4.1 |
ug/ml |
25510639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
0.02 |
ug/ml |
25534608 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
0.04 |
ug/ml |
25534608 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3130 |
nM |
25563891 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25563891 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
7200 |
nM |
25563891 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24000 |
nM |
25563891 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
10.33 |
% |
25563891 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
53 |
% |
25563891 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
630 |
nM |
25461322 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6 |
% |
25563891 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
30.66 |
% |
25563891 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
25061803 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3400 |
nM |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
290 |
nM |
25061803 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
25061803 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
25061803 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
106 |
|
25061803 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1170 |
nM |
25619894 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Activity |
= |
11 |
% |
25619894 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25619894 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
95610 |
nM |
25619894 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
750 |
nM |
25619894 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25619894 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
460 |
nM |
25868743 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
750 |
nM |
25737400 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25737400 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
95610 |
nM |
25737400 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1170 |
nM |
25737400 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
320 |
nM |
25737400 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
7860 |
nM |
25737400 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25737400 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
< |
10 |
nM |
25827522 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
20 |
nM |
25827522 |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
10 |
nM |
25827522 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
10 |
nM |
25827522 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2200 |
nM |
25881821 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
4300 |
nM |
25881821 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
25881821 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
300 |
nM |
25765907 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
25765907 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
25846065 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
60 |
nM |
25846065 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
8 |
nM |
25846065 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1.359 |
ug/ml |
25862199 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3.118 |
ug/ml |
25862199 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2.684 |
ug/ml |
25862199 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
53.6 |
% |
25618019 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
12 |
% |
25618019 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI |
= |
89.34 |
% |
25703298 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI |
= |
84.9 |
% |
25703298 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI |
= |
92.03 |
% |
25703298 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
79.01 |
% |
25703298 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI |
= |
82.01 |
% |
25703298 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1280 |
nM |
25703298 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1546 |
nM |
25703298 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
477 |
nM |
25703298 |
NPT3998 |
Cell Line |
LLC cell line |
|
TGI |
= |
52.5 |
% |
25703298 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3570 |
nM |
25594739 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3030 |
nM |
25594739 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
25559208 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
25594739 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2240 |
nM |
25594739 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
2780 |
nM |
25594739 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
CC50 |
= |
8 |
nM |
25559208 |
NPT3891 |
Cell Line |
S180 |
Mus musculus |
IC50 |
= |
9250 |
nM |
25648297 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
9700 |
nM |
25655719 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
800 |
nM |
25655719 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3500 |
nM |
25655719 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
500 |
nM |
25655719 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
990 |
nM |
25615796 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1900 |
nM |
25615796 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
25615796 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2290 |
nM |
25615796 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1610 |
nM |
25615796 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.721 |
|
25618015 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.546 |
|
25618015 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
550 |
nM |
25686590 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.461 |
|
25618015 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.494 |
|
25618015 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
36300 |
nM |
25618015 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
5 |
ug/ml |
25686593 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
700 |
nM |
25874331 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
25874331 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
25874331 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
25874331 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1350 |
nM |
25874331 |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
CC50 |
= |
600 |
nM |
25791675 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
25791675 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
880 |
nM |
25644674 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
150 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5460 |
nM |
25644674 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
890 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
90 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
180 |
nM |
25644674 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
180 |
nM |
25644674 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
22 |
|
25644674 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
36.4 |
|
25644674 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2630 |
nM |
25743216 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
17670 |
nM |
25743216 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
44400 |
nM |
25743216 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
69330 |
nM |
25743216 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1050 |
nM |
25743216 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
Activity |
= |
37.13 |
% |
25747499 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2390 |
nM |
25747499 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
229.98 |
|
25747499 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
400 |
nM |
25747499 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
> |
91990 |
nM |
25747499 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
38.49 |
|
25747499 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
980 |
nM |
25747499 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
93.87 |
|
25747499 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
1190 |
nM |
25812966 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1220 |
nM |
25812966 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1450 |
nM |
25812966 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
870 |
nM |
25812966 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
9 |
nM |
25817774 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9260 |
nM |
25817774 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16 |
nM |
25817774 |
NPT3998 |
Cell Line |
LLC cell line |
|
TGI |
= |
40 |
% |
25668341 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
26810 |
nM |
25912674 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
33130 |
nM |
25912674 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
2010 |
nM |
25965778 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
2870 |
nM |
25965778 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
80 |
% |
26005022 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
3110 |
nM |
25933593 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1110 |
nM |
25933593 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2310 |
nM |
25933593 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1430 |
nM |
25933593 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5910 |
nM |
25933593 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
25611519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
25611519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3500 |
nM |
25965778 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
3220 |
nM |
25965778 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
40 |
nM |
25611519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
25611519 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
500 |
nM |
25611519 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
nM |
25984840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220 |
nM |
25984840 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
25984840 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
210 |
nM |
25984840 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
180 |
nM |
25984840 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1100 |
nM |
25634623 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
LC50 |
= |
1500 |
nM |
25634623 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
2600 |
nM |
26005918 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
1100 |
nM |
26005918 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
2600 |
nM |
26005918 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
26005918 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
1600 |
nM |
26005918 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
9000 |
nM |
26005918 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
200 |
nM |
25953156 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
450 |
nM |
25953156 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
560 |
nM |
25953156 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
400 |
nM |
25953156 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
190 |
nM |
25953156 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
910 |
nM |
25953156 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
0.74 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
1.7 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
1.6 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
1.8 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
4.7 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2.9 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
0.7 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
0.5 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2.5 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
1.9 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2.8 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
4.5 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2.2 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
1.3 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
2.7 |
|
22867862 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Ratio |
= |
3.5 |
|
22867862 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
59 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
186.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16626.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11.8 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1830 |
nM |
25581396 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1460 |
nM |
25581396 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
630 |
nM |
25966052 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1300 |
nM |
25966052 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300 |
nM |
25966052 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1780 |
nM |
25966052 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
3180 |
nM |
25966052 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
460 |
nM |
26052884 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2 |
nM |
25466198 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
12 |
nM |
25466198 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
1 |
nM |
25466198 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
129 |
nM |
25466198 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
910 |
nM |
25734623 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
11520 |
nM |
25734623 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
58 |
nM |
25781655 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
200 |
nM |
25781655 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
25781655 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1026 |
nM |
26005543 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
663 |
nM |
26005543 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
43.4 |
% |
26005543 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
34.1 |
% |
26005543 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
21.4 |
% |
26005543 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.1 |
% |
26005543 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7211 |
nM |
26005543 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
100 |
nM |
25932671 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
25932671 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
200 |
nM |
25932671 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25932671 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
520 |
nM |
25936262 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1230 |
nM |
25936262 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1340 |
nM |
25936262 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
880 |
nM |
25936262 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50 |
nM |
25937235 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
25937235 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
150 |
nM |
25937235 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
20 |
nM |
25937235 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Ratio IC50 |
= |
3.5 |
|
25937235 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
10 |
nM |
25937235 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
30 |
nM |
25937235 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
100 |
nM |
25937235 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
500 |
nM |
25993619 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
26083682 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23 |
nM |
26083682 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
26071861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2 |
nM |
25981688 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
12 |
nM |
25981688 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
1 |
nM |
25981688 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
109 |
nM |
25981688 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
930 |
nM |
25981689 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
IC50 |
= |
2200 |
nM |
25981689 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1130 |
nM |
25981689 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
1330 |
nM |
25981689 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
Activity |
= |
20.15 |
% |
25981689 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
Activity |
= |
11.02 |
% |
25981689 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
Activity |
= |
31.17 |
% |
25981689 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
Activity |
= |
68.23 |
% |
25981689 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
Activity |
= |
0.6 |
% |
25981689 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
180 |
nM |
25998504 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
337 |
nM |
25998504 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
123 |
nM |
25998504 |
NPT2738 |
Cell Line |
Ishikawa |
Homo sapiens |
IC50 |
= |
100 |
nM |
25998504 |
NPT464 |
Cell Line |
Daudi |
Homo sapiens |
IC50 |
= |
127 |
nM |
25998504 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
35 |
nM |
25998504 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2807 |
nM |
25998504 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
80.2 |
|
25998504 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12340 |
nM |
26022842 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10780 |
nM |
26022842 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
6130 |
nM |
26022842 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
7360 |
nM |
26022842 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
2000 |
nM |
26287401 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
17670 |
nM |
26200396 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
23220 |
nM |
26200396 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
34520 |
nM |
26200396 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
22 |
nM |
25937236 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5300 |
nM |
25937236 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Ratio IC50 |
= |
241 |
|
25937236 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
790 |
nM |
25975638 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
920 |
nM |
25975638 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
200 |
nM |
25975638 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
170 |
nM |
25975638 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
220 |
nM |
25975638 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
140 |
nM |
25975638 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
8.5 |
ug/ml |
26048808 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
31 |
nM |
26067381 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
10 |
nM |
26067381 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10 |
nM |
26067381 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
10 |
nM |
26067381 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
26252628 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
600 |
nM |
26252628 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
1300 |
nM |
26252628 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5200 |
nM |
26252628 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
26252628 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
6300 |
nM |
26252628 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1610 |
nM |
26260339 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
3 |
nM |
26260339 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
536.67 |
|
26260339 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
850 |
nM |
26263187 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
250 |
nM |
26305181 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
320 |
nM |
26305181 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
50 |
nM |
26305181 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
450 |
nM |
26305181 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1580 |
nM |
26264845 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
960 |
nM |
26264845 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1380 |
nM |
26264845 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2630 |
nM |
26264845 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7260 |
nM |
26163197 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
90 |
nM |
26163197 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
50 |
nM |
26163197 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
310 |
nM |
26163197 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.44 |
|
26163197 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.04 |
|
26163197 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
80.67 |
|
26163197 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
6.2 |
|
26163197 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
950 |
nM |
26163220 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
1600 |
nM |
26163220 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
1900 |
nM |
26163220 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
1400 |
nM |
26163220 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
510 |
nM |
26356746 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
910 |
nM |
26356746 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
600 |
nM |
26356746 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
26356746 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
5.4 |
ug/ml |
26371504 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
0.4 |
ug/ml |
26371504 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
60 |
nM |
26142490 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
20 |
nM |
26142490 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
150 |
nM |
26142490 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
190 |
nM |
26142490 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
20 |
nM |
26142490 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
40 |
nM |
26142490 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
320 |
nM |
26142490 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
410 |
nM |
26142490 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
510 |
nM |
26142490 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
960 |
nM |
26142490 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
550 |
nM |
26142490 |
NPT3171 |
Cell Line |
V79 |
Cricetulus griseus |
IC50 |
= |
280 |
nM |
26142490 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
230 |
nM |
26142490 |
NPT616 |
Cell Line |
MDCK |
Canis lupus familiaris |
IC50 |
= |
430 |
nM |
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
10 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
5.4 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
4.4 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
8.4 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
53 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
27 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
22 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
42 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.7 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.9 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.5 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.9 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.2 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
2.3 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
17 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
9 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
7.3 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
14 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.7 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.8 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.7 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.3 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.6 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.5 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.4 |
|
26142490 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.2 |
|
26142490 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1000 |
nM |
26291474 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1500 |
nM |
26291474 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
2000 |
nM |
26291474 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
690 |
nM |
26295905 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
470 |
nM |
26295905 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1220 |
nM |
26295905 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5400 |
nM |
26317881 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6200 |
nM |
26317881 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
10900 |
nM |
26317881 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
26256032 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
950 |
nM |
26361737 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
1080 |
nM |
26361737 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1880 |
nM |
26361737 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1230 |
nM |
26361737 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
6.75 |
|
26123642 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
6000 |
nM |
26222449 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
500 |
nM |
26222449 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1909 |
nM |
26301558 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1258 |
nM |
26301558 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1986 |
nM |
26301558 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1054 |
nM |
26301558 |
NPT3140 |
Cell Line |
MGC-803 |
Homo sapiens |
IC50 |
= |
700 |
nM |
26280921 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
600 |
nM |
26280921 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
26280921 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
26280921 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1350 |
nM |
26280921 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5.58 |
nM |
26291039 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
0.294 |
nM |
26291039 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
4.16 |
nM |
26291039 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
0.414 |
nM |
26291039 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
CC50 |
= |
20 |
nM |
26119992 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
CC50 |
= |
20 |
nM |
26119992 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
CC50 |
= |
30 |
nM |
26119992 |
NPT2615 |
Cell Line |
HEK-293T |
Homo sapiens |
IC50 |
= |
750 |
nM |
26298501 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
570 |
nM |
26298501 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
430 |
nM |
26298501 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
9800 |
nM |
26298501 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
6290 |
nM |
26298501 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
7400 |
nM |
26298501 |
NPT2615 |
Cell Line |
HEK-293T |
Homo sapiens |
IC50 |
= |
840 |
nM |
26298501 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1020 |
nM |
26298501 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
450 |
nM |
26298501 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
7650 |
nM |
26298501 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
6030 |
nM |
26298501 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
6460 |
nM |
26298501 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
280 |
nM |
26338363 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6730 |
nM |
26338363 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
50 |
nM |
26338363 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
530 |
nM |
26338363 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.89 |
|
26338363 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.08 |
|
26338363 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
23.62 |
|
26338363 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
10.6 |
|
26338363 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1690 |
nM |
26381063 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
510 |
nM |
26381063 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
920 |
nM |
26381063 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
EC50 |
= |
30 |
nM |
26320088 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
EC50 |
= |
20 |
nM |
26320088 |
NPT4473 |
Cell Line |
WIL2-NS |
Homo sapiens |
EC50 |
= |
40 |
nM |
26320088 |
NPT4474 |
Cell Line |
CCRF-SB |
Homo sapiens |
EC50 |
= |
10 |
nM |
26320088 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
EC50 |
= |
300 |
nM |
26320088 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
900 |
nM |
26320088 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
EC50 |
= |
700 |
nM |
26320088 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
100 |
nM |
26320088 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
EC50 |
= |
200 |
nM |
26320088 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
300 |
nM |
26320088 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
EC50 |
= |
300 |
nM |
26320088 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
9.00E-05 |
ug/ml |
26420384 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
4.00E-05 |
ug/ml |
26420384 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
9.00E-05 |
ug/ml |
26420384 |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
10.9 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
16.1 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
64.8 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
7.7 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
500 |
nM |
10.1039/C4MD00219A |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
IC50 |
= |
1200 |
nM |
10.1039/C4MD00219A |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
10.1039/C4MD00219A |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1100 |
nM |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
67.5 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
0.7 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
15.1 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
Activity |
= |
16.8 |
% |
10.1039/C4MD00219A |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
FC |
= |
3 |
|
10.1039/C4MD00219A |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
2450 |
nM |
10.1039/C4MD00228H |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
3410 |
nM |
10.1039/C4MD00228H |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3120 |
nM |
10.1039/C4MD00228H |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
10.1039/C4MD00228H |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Activity |
= |
92 |
% |
10.1039/C4MD00228H |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Activity |
= |
5 |
% |
10.1039/C4MD00228H |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Activity |
= |
3 |
% |
10.1039/C4MD00228H |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
30 |
nM |
10.1039/C4MD00371C |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
20 |
nM |
10.1039/C4MD00371C |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
90 |
nM |
10.1039/C4MD00371C |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
480 |
nM |
10.1039/C4MD00371C |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
370 |
nM |
10.1039/C4MD00371C |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
12 |
|
10.1039/C4MD00371C |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
18.5 |
|
10.1039/C4MD00371C |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
4.1 |
|
10.1039/C4MD00371C |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.7 |
|
10.1039/C4MD00371C |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
120 |
mg/dl |
26253231 |
NPT1635 |
Cell Line |
H9c2 |
Rattus norvegicus |
Activity |
= |
53 |
% |
26253231 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1780 |
nM |
26253231 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2250 |
nM |
26253231 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
130 |
nM |
26253231 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1110 |
nM |
26253231 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
20 |
nM |
26280922 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
180 |
nM |
26280922 |
NPT659 |
Cell Line |
SMMC-7721 |
Homo sapiens |
IC50 |
= |
570 |
nM |
26280922 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
170 |
nM |
26280922 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
140 |
nM |
26280922 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
60 |
nM |
26280922 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
420 |
nM |
26397393 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
570 |
nM |
26397393 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
370 |
nM |
26397393 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
930 |
nM |
26330077 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
1940 |
nM |
26330077 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1510 |
nM |
26330077 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1580 |
nM |
26330077 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
630 |
nM |
26330077 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
630 |
nM |
25799376 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
120 |
nM |
25799376 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.1 |
nM |
26360048 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
GI50 |
= |
26.8 |
nM |
26462052 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
3330 |
nM |
26334499 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
1900 |
nM |
26334499 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
520 |
nM |
26334499 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1120 |
nM |
26494582 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
620 |
nM |
26494582 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
290 |
nM |
26494582 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
260 |
nM |
26494582 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
170 |
nM |
26494582 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
90 |
nM |
26494582 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
89900 |
nM |
26494582 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1680 |
nM |
26494582 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
100 |
nM |
26494582 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7520 |
nM |
26494582 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
110 |
nM |
26494582 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
424 |
nM |
26494582 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1400 |
nM |
26398312 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1200 |
nM |
26398312 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
680 |
nM |
26398312 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
830 |
nM |
26398312 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
440 |
nM |
26496013 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
330 |
nM |
26496013 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
110 |
nM |
26496013 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
840 |
nM |
26496013 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
1080 |
nM |
26496013 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
210 |
nM |
26454648 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
50 |
nM |
26454648 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
130 |
nM |
26454648 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
300 |
nM |
26454648 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
GI50 |
< |
46 |
nM |
26454648 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
43.7 |
% |
26454648 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
55.6 |
% |
26454648 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
69.8 |
% |
26454648 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
39.6 |
% |
26454648 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
97.9 |
% |
26454648 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
8140 |
nM |
26513642 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
7510 |
nM |
26513642 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
4450 |
nM |
26513642 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
26561719 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1.28 |
ug/ml |
10.1039/C4MD00566J |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2.6 |
ug/ml |
10.1039/C4MD00566J |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
2.08 |
ug/ml |
10.1039/C4MD00566J |
NPT319 |
Cell Line |
B16 |
Mus musculus |
IC50 |
= |
3.16 |
ug/ml |
10.1039/C4MD00566J |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3.2 |
ug/ml |
10.1039/C4MD00566J |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
910 |
nM |
26433616 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1080 |
nM |
26433616 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
> |
100000 |
nM |
26433616 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2490 |
nM |
26542964 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
3180 |
nM |
26542964 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
3920 |
nM |
26542964 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
5.4 |
ug/ml |
26469557 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
IC50 |
= |
0.5 |
ug/ml |
26469557 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
0.4 |
ug/ml |
26469557 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
77.4 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
65.3 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
51.6 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
44.9 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
91 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
83 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
75 |
% |
26560050 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
48 |
% |
26560050 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
460 |
nM |
26690914 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.1 |
nM |
26690914 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
23.6 |
|
26646219 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
30.4 |
|
26646219 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
26.6 |
|
26646219 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
21300 |
nM |
26646219 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
900 |
nM |
26646219 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
26646219 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
26646219 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
26586599 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
800 |
nM |
26586599 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
800 |
nM |
26586599 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
700 |
nM |
26586599 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1600 |
nM |
26551342 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
26551342 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
0.15 |
ug/ml |
26561866 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.85 |
ug/ml |
26561866 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
0.07 |
ug/ml |
26561866 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
5100 |
nM |
26561866 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
GI50 |
= |
0.25 |
ug/ml |
26561866 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.22 |
ug/ml |
26561866 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
4000 |
nM |
26561866 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
120 |
nM |
26633734 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
110 |
nM |
26633734 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
200 |
nM |
26633734 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
60 |
nM |
26633734 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
370 |
nM |
26633734 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9750 |
nM |
26633734 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
81.25 |
|
26633734 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23 |
nM |
26711144 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
26711144 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1172 |
nM |
10.1039/C5MD00127G |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
900 |
nM |
26711890 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
530 |
nM |
10.1039/C5MD00163C |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1700 |
nM |
10.1039/C5MD00163C |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
300 |
nM |
10.1039/C5MD00163C |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
500 |
nM |
26631318 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
150 |
nM |
26639764 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7200 |
nM |
26639764 |
NPT2711 |
Cell Line |
BALB/3T3 |
Mus musculus |
IC50 |
= |
110 |
nM |
26639764 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
48 |
|
26639764 |
NPT2 |
Others |
Unspecified |
|
TGI |
= |
36.1 |
ug/ml |
10.1039/C5MD00224A |
NPT2 |
Others |
Unspecified |
|
LC50 |
> |
80 |
ug/ml |
10.1039/C5MD00224A |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
10 |
ug/ml |
10.1039/C5MD00224A |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
TGI |
< |
10 |
ug/ml |
10.1039/C5MD00224A |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
LC50 |
= |
36.9 |
ug/ml |
10.1039/C5MD00224A |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
< |
10 |
ug/ml |
10.1039/C5MD00224A |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3560 |
nM |
26706352 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2570 |
nM |
26706352 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3700 |
nM |
26706352 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
900 |
nM |
26774921 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
79600 |
nM |
26774921 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
700 |
nM |
26774921 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
800 |
nM |
26774921 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
26649907 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
26649907 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0 |
|
26649907 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
21900 |
nM |
26649907 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
6900 |
nM |
26649907 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
834 |
nM |
26638041 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
12 |
nM |
26638041 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
77 |
nM |
26638041 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
1930 |
nM |
26638041 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1780 |
nM |
26708114 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
1060 |
nM |
26708114 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1820 |
nM |
26708114 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1160 |
nM |
26708114 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
1670 |
nM |
26708114 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40 |
nM |
26810263 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
LC50 |
= |
1170 |
nM |
26681508 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
1560 |
nM |
26681508 |
NPT2 |
Others |
Unspecified |
|
LC50 |
= |
370 |
nM |
26681508 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5730 |
nM |
26873414 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
10150 |
nM |
26873414 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
140 |
nM |
26873414 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
9030 |
nM |
26873414 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16370 |
nM |
26873414 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2120 |
nM |
26874744 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3820 |
nM |
26874744 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2780 |
nM |
26874744 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3000 |
nM |
26874744 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
924 |
nM |
26972921 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
150 |
nM |
26972921 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
300 |
nM |
26972921 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
112 |
nM |
26840362 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
2.40E-05 |
ug |
26386603 |
NPT3891 |
Cell Line |
S180 |
Mus musculus |
Activity |
= |
0.401 |
ug |
26386603 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1360 |
nM |
26386603 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
130 |
nM |
26386603 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
270 |
nM |
26386603 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
580 |
nM |
26386603 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
160 |
nM |
26386603 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
600 |
nM |
26386603 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
26859070 |
NPT75 |
Cell Line |
U251 |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
26859070 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.14 |
ug/ml |
26859070 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
= |
0.025 |
ug/ml |
26859070 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
26859070 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
0.085 |
ug/ml |
26859070 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
0.13 |
ug/ml |
26859070 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
GI50 |
< |
0.025 |
ug/ml |
26859070 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
26720155 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
400 |
nM |
26890118 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
100 |
nM |
26890118 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4300 |
nM |
26890118 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
43 |
|
26890118 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
26890118 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
26890118 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
5 |
|
26890118 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
340 |
nM |
26890119 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
380 |
nM |
26890119 |
NPT3190 |
Cell Line |
NHDF |
Homo sapiens |
IC50 |
= |
3380 |
nM |
26890119 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
26720155 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4910 |
nM |
26720155 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
26720155 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
90 |
nM |
26720155 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
26720155 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
26720155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
26720155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
920 |
nM |
26720155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7310 |
nM |
26874404 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
980 |
nM |
26874404 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1480 |
nM |
26874404 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
720 |
nM |
26874404 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
960 |
nM |
26874404 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
740 |
nM |
26874404 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
46.25 |
% |
10.1039/C5MD00459D |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
33.78 |
% |
10.1039/C5MD00459D |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
15.5 |
% |
10.1039/C5MD00459D |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.59 |
% |
10.1039/C5MD00459D |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
870 |
nM |
26900656 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1120 |
nM |
26900656 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1010 |
nM |
26900656 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
1340 |
nM |
26900656 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Survival |
= |
4 |
% |
26947606 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70 |
nM |
26947606 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
380 |
nM |
26947606 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
100 |
nM |
26947606 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
450 |
nM |
26947606 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
350 |
nM |
26947606 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
Activity |
= |
3.93 |
nM |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
0.473 |
nM |
26948540 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
1.25 |
nM |
26948540 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.5 |
nM |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
1 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
44 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
8 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
48 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
4 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
37 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
9 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
50 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
6 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
34 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
11 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
49 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
36 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
10 |
% |
26948540 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
46 |
% |
26948540 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
1590 |
nM |
26948541 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1330 |
nM |
26948541 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2340 |
nM |
26948541 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1080 |
nM |
26948541 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1490 |
nM |
26807545 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1010 |
nM |
26807545 |
NPT1872 |
Cell Line |
Bcap37 |
Homo sapiens |
IC50 |
= |
1190 |
nM |
26807545 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
800 |
nM |
26807545 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2810 |
nM |
27015609 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
2570 |
nM |
27015609 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1130 |
nM |
27015609 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1410 |
nM |
27015609 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3010 |
nM |
27015609 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
950 |
nM |
27016707 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100 |
nM |
27016707 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
450 |
nM |
27016707 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
380 |
nM |
27080182 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
27080182 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
300 |
nM |
27080187 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
380 |
nM |
27080187 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
130 |
nM |
27080187 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
8020 |
nM |
26907155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4750 |
nM |
26907155 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2100 |
nM |
27055942 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
3300 |
nM |
27055942 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
27055942 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
90 |
nM |
27060757 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
810 |
nM |
27060757 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
780 |
nM |
27060757 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
70 |
nM |
27060757 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
52 |
nM |
27060757 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
10 |
nM |
26994690 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
90 |
nM |
26994690 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
< |
10 |
nM |
26994690 |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
10 |
nM |
26994690 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
230 |
nM |
27036521 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
3390 |
nM |
27036521 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1940 |
nM |
27036521 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25040 |
nM |
27036521 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
89680 |
nM |
27036521 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
2 |
|
27036521 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
6100 |
nM |
10.1039/C5MD00513B |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
7200 |
nM |
10.1039/C5MD00513B |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
7100 |
nM |
10.1039/C5MD00513B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5400 |
nM |
10.1039/C5MD00513B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10100 |
nM |
10.1039/C5MD00513B |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37400 |
nM |
10.1039/C5MD00515A |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
3.2 |
% |
10.1039/C5MD00515A |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
16.7 |
% |
10.1039/C5MD00515A |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
32.4 |
% |
10.1039/C5MD00515A |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2590 |
nM |
10.1039/C5MD00581G |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1730 |
nM |
10.1039/C5MD00581G |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
930 |
nM |
10.1039/C5MD00581G |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2480 |
nM |
10.1039/C5MD00581G |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
2960 |
nM |
10.1039/C5MD00581G |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
30 |
nM |
27080175 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
160 |
nM |
27080175 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
27080175 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1170 |
nM |
27080175 |
NPT5420 |
Cell Line |
MCF10 |
Homo sapiens |
IC50 |
= |
160 |
nM |
27080175 |
NPT2452 |
Cell Line |
NCI-H292 |
|
Activity |
= |
94.1 |
% |
27142752 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
74.8 |
% |
27142752 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
79.4 |
% |
27142752 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
91.7 |
% |
27142752 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
92.9 |
% |
27142752 |
NPT1182 |
Cell Line |
J774.A1 |
Mus musculus |
Activity |
= |
96 |
% |
27142752 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Activity |
= |
96.5 |
% |
27142752 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
27112448 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4800 |
nM |
27112448 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.48 |
|
27085944 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.551 |
|
27085944 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.139 |
|
27085944 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
0.13 |
|
27085944 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
32000 |
nM |
27085944 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
51 |
nM |
27089210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
73 |
nM |
27089210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8800 |
nM |
27089210 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
= |
72.6 |
nM |
27096046 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
= |
99.5 |
nM |
27096046 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
112 |
nM |
27096046 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
92.3 |
nM |
27096046 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
125 |
nM |
27096046 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
85.4 |
nM |
27096046 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3100 |
nM |
27173802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1850 |
nM |
27173802 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
5000 |
nM |
27173802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9500 |
nM |
27173802 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
6750 |
nM |
27173802 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13000 |
nM |
27173802 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
97.98 |
% |
27234888 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
92.68 |
% |
27234888 |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
Inhibition |
= |
98.07 |
% |
27234888 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
73 |
nM |
27209232 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
GI50 |
= |
73.11 |
nM |
27209232 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
97 |
nM |
27209232 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
97.05 |
nM |
27209232 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
85 |
nM |
27209232 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
= |
85.11 |
nM |
27209232 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
23 |
nM |
27209232 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
23.01 |
nM |
27209232 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1000 |
nM |
27265687 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
20 |
% |
27265687 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
0 |
% |
27265687 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
Activity |
= |
10 |
% |
27265687 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
2100 |
nM |
26821210 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
360 |
nM |
26904921 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
250 |
nM |
27231128 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
920 |
nM |
27231128 |
NPT15 |
Cell Line |
Jurkat |
Homo sapiens |
IC50 |
= |
30 |
nM |
27231128 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
IC50 |
= |
2980 |
nM |
27231128 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
200 |
nM |
27231128 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
90 |
nM |
27231128 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
70 |
nM |
27231128 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4910 |
nM |
27231128 |
NPT171 |
Cell Line |
MRC5 |
Homo sapiens |
IC50 |
= |
100 |
nM |
27231128 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
TGI |
= |
50 |
% |
27241692 |
NPT168 |
Cell Line |
P388 |
Mus musculus |
IC50 |
= |
900 |
nM |
27256910 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
870 |
nM |
27256910 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
940 |
nM |
27256910 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
550 |
nM |
27256910 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2780 |
nM |
27256910 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
95.6 |
% |
27096049 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
94.3 |
% |
27096049 |
NPT2 |
Others |
Unspecified |
|
GI |
= |
99.6 |
% |
27096049 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
GI50 |
< |
10 |
nM |
10.1039/C6MD00097E |
NPT2 |
Others |
Unspecified |
|
GI50 |
< |
10 |
nM |
10.1039/C6MD00097E |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
< |
10 |
nM |
10.1039/C6MD00097E |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
< |
10 |
nM |
10.1039/C6MD00097E |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
2170 |
nM |
27149641 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
1020 |
nM |
27149641 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
980 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1170 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3290 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.35 |
|
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1510 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.29 |
|
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3140 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.44 |
|
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50400 |
nM |
27149641 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
49.4 |
|
27149641 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7190 |
nM |
27108400 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
68900 |
nM |
27108400 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5500 |
nM |
27108400 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
50 |
nM |
27363939 |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
IC50 |
= |
830 |
nM |
27363939 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
390 |
nM |
27363939 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
IC50 |
= |
44400 |
nM |
27108400 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4210 |
nM |
27108400 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
8.07 |
|
27108400 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
0.06 |
|
27108400 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
CC50 |
= |
200 |
nM |
27155463 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
30 |
nM |
27363939 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1290 |
nM |
27116711 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20 |
nM |
27116711 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
370 |
nM |
27116711 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
550 |
nM |
27116711 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
1060 |
nM |
27311894 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15690 |
nM |
27311894 |