Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
173 |
nM |
12190308 |
NPT274 |
Individual Protein |
Platelet activating factor receptor |
Homo sapiens |
IC50 |
> |
50000 |
nM |
1671420 |
NPT4293 |
Individual Protein |
Histamine H1 receptor |
Rattus norvegicus |
Ki |
= |
350 |
nM |
1671420 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
0.21 |
mg/kg |
7853343 |
NPT4292 |
Individual Protein |
Histamine H1 receptor |
Mus musculus |
ID50 |
= |
36 |
mg/kg |
7853343 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
Inhibition |
= |
80 |
% |
7853343 |
NPT419 |
Organism |
Oryctolagus cuniculus |
Oryctolagus cuniculus |
IC50 |
= |
135000 |
nM |
7914928 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ID50 |
> |
5 |
mg/kg |
7914928 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
> |
30 |
mg/kg |
7914928 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
IC50 |
= |
290 |
nM |
7914928 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
66.3 |
% |
7914928 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
= |
19 |
mg/kg |
7914928 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
> |
10 |
mg/kg |
7914928 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ID50 |
= |
2.4 |
mg/kg |
7914928 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
> |
50000 |
nM |
9934454 |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
169.82 |
nM |
12873512 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
1.8 |
mg/kg |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
1.6 |
mg/kg |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
2.7 |
mg/kg |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
6.2 |
mg/kg |
15771458 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
ED50 |
= |
0.08 |
mg/kg |
15771458 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
ED50 |
= |
0.32 |
mg/kg |
15771458 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
ED50 |
= |
2.2 |
mg/kg |
15771458 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
ED50 |
= |
0.42 |
mg/kg |
15771458 |
NPT1016 |
Organism |
Canis familiaris |
Canis lupus familiaris |
ED50 |
= |
0.2 |
mg/kg |
15771458 |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
Ki |
= |
37 |
nM |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.29 |
mg/kg |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.22 |
mg/kg |
15771458 |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
ED50 |
= |
0.074 |
mg/kg |
15771458 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.89 |
mg/kg |
15771458 |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
Ki |
= |
414 |
nM |
15482930 |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
169.82 |
nM |
15911273 |
NPT274 |
Individual Protein |
Platelet activating factor receptor |
Homo sapiens |
IC50 |
= |
135000 |
nM |
16220969 |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
IC50 |
= |
290 |
nM |
16220969 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
30 |
% |
15566302 |
NPT4292 |
Individual Protein |
Histamine H1 receptor |
Mus musculus |
ED50 |
= |
12.9 |
mg/kg |
15566302 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.75 |
mg/kg |
15566302 |
NPT156 |
Individual Protein |
Sphingomyelin phosphodiesterase |
Homo sapiens |
Activity |
= |
118.3 |
% |
18027916 |
NPT612 |
Individual Protein |
Canalicular multispecific organic anion transporter 1 |
Homo sapiens |
Activity |
= |
6 |
% |
18457386 |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
169.82 |
nM |
18448342 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
Inhibition |
= |
51.8 |
% |
18788725 |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
173.78 |
nM |
19110341 |
NPT4288 |
Individual Protein |
Histamine H1 receptor |
Cavia porcellus |
Inhibition |
= |
15.67 |
% |
20110173 |
NPT4288 |
Individual Protein |
Histamine H1 receptor |
Cavia porcellus |
Inhibition |
= |
33.36 |
% |
20110173 |
NPT4288 |
Individual Protein |
Histamine H1 receptor |
Cavia porcellus |
Inhibition |
= |
64.7 |
% |
20110173 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
13300 |
nM |
20180535 |
NPT580 |
Organism |
Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
= |
23000 |
nM |
20180535 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
6309.57 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
5011.87 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1995.26 |
nM |
19734910 |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT312 |
Organism |
Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Potency |
= |
17782.8 |
nM |
PubChem BioAssay data set |
NPT537 |
Individual Protein |
Ras-related protein Rab-9A |
Homo sapiens |
Potency |
= |
100000 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
11220.2 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT791 |
Individual Protein |
Cruzipain |
Trypanosoma cruzi |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT791 |
Individual Protein |
Cruzipain |
Trypanosoma cruzi |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT791 |
Individual Protein |
Cruzipain |
Trypanosoma cruzi |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
398.1 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT211 |
Individual Protein |
Hypoxia-inducible factor 1 alpha |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT796 |
Individual Protein |
Peripheral myelin protein 22 |
Homo sapiens |
Potency |
= |
42561.5 |
nM |
PubChem BioAssay data set |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT583 |
Individual Protein |
Inositol monophosphatase 1 |
Rattus norvegicus |
Potency |
= |
446.7 |
nM |
PubChem BioAssay data set |
NPT54 |
Individual Protein |
Nonstructural protein 1 |
Influenza A virus |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT54 |
Individual Protein |
Nonstructural protein 1 |
Influenza A virus |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Potency |
= |
23280.9 |
nM |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
2238.7 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
3548.1 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT45 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 2 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT538 |
Individual Protein |
Niemann-Pick C1 protein |
Homo sapiens |
Potency |
= |
58047.9 |
nM |
PubChem BioAssay data set |
NPT58 |
Individual Protein |
Bloom syndrome protein |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Potency |
= |
1258.9 |
nM |
PubChem BioAssay data set |
NPT96 |
Individual Protein |
Thrombopoietin |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT1416 |
Individual Protein |
Neuropeptide S receptor |
Homo sapiens |
Potency |
= |
7943.3 |
nM |
PubChem BioAssay data set |
NPT1416 |
Individual Protein |
Neuropeptide S receptor |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT1416 |
Individual Protein |
Neuropeptide S receptor |
Homo sapiens |
Potency |
= |
3981.1 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
6309.6 |
nM |
PubChem BioAssay data set |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
39.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT580 |
Organism |
Trypanosoma cruzi |
Trypanosoma cruzi |
EC50 |
= |
9000 |
nM |
20547819 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
1.9 |
|
20547819 |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
173.78 |
nM |
21185626 |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
25918.5 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
8199.5 |
nM |
PubChem BioAssay data set |
NPT800 |
Individual Protein |
M-phase phosphoprotein 8 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
56234.1 |
nM |
PubChem BioAssay data set |
NPT5 |
Individual Protein |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT135 |
Individual Protein |
Chromobox protein homolog 1 |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT63 |
Individual Protein |
Bromodomain adjacent to zinc finger domain protein 2B |
Homo sapiens |
Potency |
|
79432.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT1139 |
Individual Protein |
Arachidonate 15-lipoxygenase, type II |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
18526 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
11689.1 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
18348.9 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
20596.2 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
AC50 |
= |
12589.25 |
nM |
PubChem BioAssay data set |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
AC50 |
= |
15848.93 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
10417.9 |
nM |
PubChem BioAssay data set |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
|
446.7 |
nM |
PubChem BioAssay data set |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
8492.1 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
12990 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9196.2 |
nM |
PubChem BioAssay data set |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
56234.1 |
nM |
PubChem BioAssay data set |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
IC50 |
= |
16 |
nM |
DrugMatrix in vitro pharmacology data |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
IC50 |
= |
170 |
nM |
DrugMatrix in vitro pharmacology data |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
Ki |
= |
20 |
nM |
DrugMatrix in vitro pharmacology data |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
IC50 |
= |
39086.6 |
nM |
DrugMatrix in vitro pharmacology data |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
Ki |
= |
32022.8 |
nM |
DrugMatrix in vitro pharmacology data |
NPT291 |
Individual Protein |
Serotonin 2b (5-HT2b) receptor |
Homo sapiens |
IC50 |
= |
245 |
nM |
DrugMatrix in vitro pharmacology data |
NPT291 |
Individual Protein |
Serotonin 2b (5-HT2b) receptor |
Homo sapiens |
Ki |
= |
156 |
nM |
DrugMatrix in vitro pharmacology data |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
4549.88 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
10209.39 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
4149.54 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
15776.11 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
1636.82 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
10046.16 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
6123.5 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
11534.53 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
2084.49 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
13212.96 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
6123.5 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
5942.92 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
849.18 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
7780.37 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
4226.69 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
6561.45 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
15205.48 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
13995.87 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
12705.74 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
20844.91 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
18793.17 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
20044.72 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
13243.42 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
2636.33 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
11830.42 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
10592.54 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
12416.52 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
11142.95 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
40533.4 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
3828.25 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
3689.78 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
10864.26 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
11168.63 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
10023.05 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
13427.65 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
3265.88 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
7550.92 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
11220.18 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
10115.79 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
13899.53 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
10447.2 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
7396.05 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
15523.87 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
13335.21 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
3435.58 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
4731.51 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
7211.07 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
8830.8 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
1786.49 |
nM |
PubChem BioAssay data set |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
|
26915.35 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
15170.5 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
15031.42 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
4315.19 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
3176.87 |
nM |
PubChem BioAssay data set |
NPT861 |
Individual Protein |
Isocitrate dehydrogenase [NADP] cytoplasmic |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
14588.14 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
5571.86 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
6714.29 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
9141.13 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7500 |
nM |
22450132 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8400 |
nM |
22450132 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6200 |
nM |
22450132 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
11400 |
nM |
11454724 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
7500 |
nM |
22959205 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
8400 |
nM |
22959205 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6200 |
nM |
22959205 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
23109.3 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
5804.8 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
33498.3 |
nM |
PubChem BioAssay data set |
NPT501 |
Individual Protein |
Alpha-galactosidase A |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT100 |
Individual Protein |
Glutaminase kidney isoform, mitochondrial |
Homo sapiens |
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10000 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
326.4 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT478 |
Individual Protein |
Ataxin-2 |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT101 |
Individual Protein |
Glucagon-like peptide 1 receptor |
Homo sapiens |
Potency |
|
14125.4 |
nM |
PubChem BioAssay data set |
NPT755 |
Individual Protein |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
Homo sapiens |
Potency |
|
100000 |
nM |
PubChem BioAssay data set |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Inhibition |
= |
28.1 |
% |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
45 |
% |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
43.2 |
% |
22541068 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
2 |
|
22506484 |
NPT616 |
Cell Line |
MDCK |
Canis lupus familiaris |
Ratio |
= |
1.9 |
|
22506484 |
NPT857 |
Cell Line |
LLC-PK1 |
Sus scrofa |
Ratio |
= |
0.5 |
|
24900570 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
20596.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
12995.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11885.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2660.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14963.1 |
nM |
PubChem BioAssay data set |
NPT861 |
Individual Protein |
Isocitrate dehydrogenase [NADP] cytoplasmic |
Homo sapiens |
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
IC50 |
= |
3070 |
nM |
23688559 |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Inhibition |
= |
72.5 |
% |
23688559 |
NPT543 |
Individual Protein |
Pregnane X receptor |
Homo sapiens |
EC50 |
= |
3000 |
nM |
23688559 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
83.88 |
% |
23571415 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
101.04 |
% |
23571415 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11883.2 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
17373.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29847 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
61130.6 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
29849.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27535.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
38895.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
61644.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54482.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29849.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21117.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
61130.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48966.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
23710.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43641.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10682.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3348.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
26603.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8412 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
33488.9 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
76958.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27306 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
26601.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21872.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
13332.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17373.9 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
61644.8 |
nM |
PubChem BioAssay data set |
NPT104 |
Individual Protein |
Cerebroside-sulfatase |
Homo sapiens |
Potency |
|
213.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9688.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33488.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30637.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
68589.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43277.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33491.5 |
nM |
PubChem BioAssay data set |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
|
43641.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6740 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54941 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30106.5 |
nM |
PubChem BioAssay data set |
NPT162 |
Individual Protein |
Heat shock protein beta-1 |
Homo sapiens |
Potency |
|
26601.1 |
nM |
PubChem BioAssay data set |
NPT162 |
Individual Protein |
Heat shock protein beta-1 |
Homo sapiens |
Potency |
|
54941 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7497.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21313.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
26832.5 |
nM |
PubChem BioAssay data set |
NPT11 |
Individual Protein |
Guanine nucleotide-binding protein G(s), subunit alpha |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8412.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10870.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
10590.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9439.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
8634.9 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
54941 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16785.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5623.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
14125.4 |
nM |
PubChem BioAssay data set |
NPT251 |
Individual Protein |
Histamine H1 receptor |
Homo sapiens |
Ki |
= |
311 |
nM |
25318072 |
NPT4342 |
Individual Protein |
Sodium-dependent neutral amino acid transporter B(0)AT2 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
25318072 |
NPT1418 |
Individual Protein |
Anandamide amidohydrolase |
Homo sapiens |
Inhibition |
= |
11 |
% |
25752982 |
NPT4288 |
Individual Protein |
Histamine H1 receptor |
Cavia porcellus |
Kd |
= |
72.44 |
nM |
25752982 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11400 |
nM |
23812503 |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
IC50 |
= |
2800 |
nM |
22328583 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
IC50 |
> |
30000 |
nM |
22328583 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
IC50 |
> |
30000 |
nM |
22328583 |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
IC50 |
> |
30000 |
nM |
22328583 |
NPT1463 |
Individual Protein |
Cytochrome P450 2J2 |
Homo sapiens |
Activity |
= |
11.4 |
% |
22328583 |
NPT1463 |
Individual Protein |
Cytochrome P450 2J2 |
Homo sapiens |
Activity |
= |
4 |
% |
22328583 |
NPT628 |
Individual Protein |
Cytochrome P450 2C8 |
Homo sapiens |
IC50 |
= |
2950 |
nM |
22328583 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
IC50 |
< |
100 |
nM |
22328583 |
NPT543 |
Individual Protein |
Pregnane X receptor |
Homo sapiens |
EC50 |
= |
10000 |
nM |
20966043 |
NPT543 |
Individual Protein |
Pregnane X receptor |
Homo sapiens |
EC50 |
= |
12600 |
nM |
20966043 |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
19960 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
23914.5 |
nM |
PubChem BioAssay data set |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
16930.1 |
nM |
PubChem BioAssay data set |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
48966.2 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
7562.4 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
12299.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
2511.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
436.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
19493.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21131.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6859 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
AC50 |
|
6309.6 |
nM |
PubChem BioAssay data set |