Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Activity |
= |
94 |
% |
19453174 |
NPT1354 |
Cell Line |
TGBC11TKB |
Homo sapiens |
IC50 |
= |
374800.92 |
nM |
23354071 |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Activity |
= |
95 |
% |
8487254 |
NPT2283 |
Cell Line |
DK-MG |
Homo sapiens |
IC50 |
= |
617597.53 |
nM |
6195312 |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
349116.26 |
nM |
20363140 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
52707.09 |
nM |
20643902 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
14254.28 |
nM |
23707051 |
NPT2285 |
Cell Line |
COR-L105 |
Homo sapiens |
IC50 |
= |
667061.34 |
nM |
18298080 |
NPT2268 |
Cell Line |
DOK |
Homo sapiens |
IC50 |
= |
67535 |
nM |
11374975 |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
815568.16 |
nM |
19459694 |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
626391.77 |
nM |
19459694 |
NPT2403 |
Cell Line |
SBC-5 |
Homo sapiens |
IC50 |
= |
864644.12 |
nM |
19459694 |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
954235.03 |
nM |
24844534 |
NPT2328 |
Cell Line |
COLO-678 |
Homo sapiens |
IC50 |
= |
490591.1 |
nM |
12088440 |
NPT2401 |
Cell Line |
PANC-03-27 |
Homo sapiens |
IC50 |
= |
282056.95 |
nM |
1791475 |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
474826.75 |
nM |
22608855 |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
80575.05 |
nM |
9733489 |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
619029.54 |
nM |
20853847 |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
500443.65 |
nM |
18492609 |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
290899.25 |
nM |
25945867 |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
854077.55 |
nM |
20329739 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
393685.36 |
nM |
17958396 |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
431923.29 |
nM |
17988097 |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
41065.16 |
nM |
PubChem BioAssay data set |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
757456.42 |
nM |
22691179 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
436888.93 |
nM |
13678412 |
NPT2322 |
Cell Line |
CHL-1 |
Homo sapiens |
IC50 |
= |
42063.78 |
nM |
8946741 |
NPT2279 |
Cell Line |
COLO-792 |
Homo sapiens |
IC50 |
= |
736345.91 |
nM |
23985009 |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
354985.88 |
nM |
24195466 |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
59752.2 |
nM |
PubChem BioAssay data set |
NPT1653 |
Cell Line |
WM-115 |
Homo sapiens |
IC50 |
= |
413305.9 |
nM |
10.1016/j.cropro.2012.04.001 |
NPT2379 |
Cell Line |
P12-Ichikawa |
Homo sapiens |
IC50 |
= |
388167.91 |
nM |
18763827 |
NPT2474 |
Cell Line |
MDA-MB-415 |
Homo sapiens |
IC50 |
= |
474398.65 |
nM |
19874044 |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
103425.86 |
nM |
11678655 |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
139648 |
nM |
15084123 |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
16856.7 |
nM |
23964644 |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
22032.6 |
nM |
18479163 |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Activity |
= |
96 |
% |
10498214 |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
51974.23 |
nM |
26331426 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
423466.75 |
nM |
PubChem BioAssay data set |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
42196.36 |
nM |
PubChem BioAssay data set |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Activity |
= |
80 |
% |
16643054 |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Activity |
= |
95 |
% |
12932142 |
NPT2434 |
Cell Line |
TCC-SUP |
Homo sapiens |
IC50 |
= |
107842.52 |
nM |
18817444 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
582116.15 |
nM |
7528786 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
69931.56 |
nM |
22871217 |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
596264.29 |
nM |
8699183 |
NPT2369 |
Cell Line |
NCI-H2052 |
Homo sapiens |
IC50 |
= |
660912.86 |
nM |
17958396 |
NPT2450 |
Cell Line |
NCI-H2452 |
Homo sapiens |
IC50 |
= |
197086.95 |
nM |
17958396 |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
66048.94 |
nM |
17958396 |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
33819.11 |
nM |
17958396 |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
239034.76 |
nM |
17896816 |
NPT994 |
Cell Line |
ZR-75-30 |
Homo sapiens |
IC50 |
= |
444817.02 |
nM |
9514009 |
NPT2352 |
Cell Line |
MHH-ES-1 |
Homo sapiens |
IC50 |
= |
198540.28 |
nM |
19572611 |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Activity |
= |
110 |
% |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
IC50 |
= |
230529.08 |
nM |
11689077 |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
7649.48 |
nM |
19182783 |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Activity |
= |
77 |
% |
PubChem BioAssay data set |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
452412.78 |
nM |
8450319 |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
630639.89 |
nM |
18672931 |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
4771.72 |
nM |
8946745 |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
329140.27 |
nM |
22304344 |
NPT2377 |
Cell Line |
NCI-H2087 |
Homo sapiens |
IC50 |
= |
345544.7 |
nM |
23131412 |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
283366.18 |
nM |
23131412 |
NPT2387 |
Cell Line |
KYSE-410 |
Homo sapiens |
IC50 |
= |
247799.51 |
nM |
24461297 |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
82209.51 |
nM |
9873511 |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Activity |
= |
86 |
% |
18419154 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
IC50 |
= |
56608.21 |
nM |
12932130 |
NPT2407 |
Cell Line |
HCC1419 |
Homo sapiens |
IC50 |
= |
64736.23 |
nM |
19969457 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
886270.31 |
nM |
18247573 |
NPT1669 |
Cell Line |
NCI-H1792 |
Homo sapiens |
IC50 |
= |
479818.06 |
nM |
21856049 |
NPT2349 |
Cell Line |
HMV-2 cell line |
|
IC50 |
= |
250034.27 |
nM |
11325246 |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Activity |
= |
89 |
% |
18479163 |
NPT2365 |
Cell Line |
HO-1-N-1 |
Homo sapiens |
IC50 |
= |
363636.59 |
nM |
15043446 |
NPT3467 |
Cell Line |
SJRH30 |
Homo sapiens |
IC50 |
= |
732258.07 |
nM |
12852746 |
NPT2392 |
Cell Line |
S-117 |
Homo sapiens |
IC50 |
= |
755358.9 |
nM |
21907579 |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
516957.67 |
nM |
17043127 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
1257718.95 |
nM |
18674917 |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
120534.62 |
nM |
19231179 |
NPT2441 |
Cell Line |
NCI-H2347 |
Homo sapiens |
IC50 |
= |
1038457.79 |
nM |
17620378 |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
42716.96 |
nM |
17620378 |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
805730.24 |
nM |
18547811 |
NPT2311 |
Cell Line |
Calu-3 |
Homo sapiens |
IC50 |
= |
261759.2 |
nM |
20675019 |
NPT2389 |
Cell Line |
NCI-H1048 |
Homo sapiens |
IC50 |
= |
448659.39 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
35637.2 |
nM |
21093119 |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
104280.88 |
nM |
21481593 |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Activity |
= |
109 |
% |
DrugMatrix in vitro pharmacology data |
NPT2396 |
Cell Line |
KYSE-510 |
Homo sapiens |
IC50 |
= |
190025.26 |
nM |
DrugMatrix in vitro pharmacology data |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
45600 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2397 |
Cell Line |
KYSE-520 cell line |
|
IC50 |
= |
343988.42 |
nM |
DrugMatrix in vitro pharmacology data |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Activity |
= |
97 |
% |
22995772 |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Activity |
= |
71 |
% |
10.1007/s00044-011-9842-7 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
530277.26 |
nM |
10.1007/s00044-011-9842-7 |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
367484.08 |
nM |
10.1007/s00044-011-9605-5 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
426347.18 |
nM |
10.1007/s00044-012-0026-x |
NPT2368 |
Cell Line |
NCI-H2030 |
Homo sapiens |
IC50 |
= |
833902.93 |
nM |
10.1007/s00044-012-0320-7 |
NPT2316 |
Cell Line |
CFPAC-1 |
Homo sapiens |
IC50 |
= |
333270.68 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
111037.17 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
192109.4 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
109094.01 |
nM |
Open TG-GATES in vivo data: Organ Weight |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
780422.16 |
nM |
Open TG-GATES in vivo data: Organ Weight |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Activity |
= |
89 |
% |
Open TG-GATES in vivo data: Organ Weight |
NPT2497 |
Cell Line |
HEC-1 |
Homo sapiens |
IC50 |
= |
575901.13 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
214423.49 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3813 |
Individual Protein |
Tyrosine-protein kinase SRC |
Gallus gallus |
Activity |
= |
105 |
% |
Open TG-GATES in vivo data: Biochemistry |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
IC50 |
= |
89 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
573436.38 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
701043.54 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2420 |
Cell Line |
NCI-H2291 |
Homo sapiens |
IC50 |
= |
334496.03 |
nM |
DrugMatrix in vivo data: Pathology |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
120872.59 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2340 |
Cell Line |
KU-19-19 |
Homo sapiens |
IC50 |
= |
495973.25 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
86257.15 |
nM |
DrugMatrix in vivo data: Hematology |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
101139.42 |
nM |
24398288 |
NPT2476 |
Cell Line |
NCI-H441 |
Homo sapiens |
IC50 |
= |
423951.47 |
nM |
15646539 |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
609867.06 |
nM |
17844993 |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
IC50 |
= |
1065777.65 |
nM |
1336040 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
26520.92 |
nM |
16441059 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
584559.17 |
nM |
18288805 |
NPT2506 |
Cell Line |
RO82-W-1 |
Homo sapiens |
IC50 |
= |
150372.87 |
nM |
11473423 |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
17987.84 |
nM |
12617583 |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
282292.28 |
nM |
21106454 |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
224690.75 |
nM |
16933872 |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
49133.3 |
nM |
23501116 |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
211730.03 |
nM |
15165148 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
801272.43 |
nM |
23992864 |
NPT2451 |
Cell Line |
NCI-H28 |
Homo sapiens |
IC50 |
= |
822971.85 |
nM |
17685651 |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
60807.8 |
nM |
12932139 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
796836.09 |
nM |
8350093 |
NPT2465 |
Cell Line |
NCI-H1623 |
Homo sapiens |
IC50 |
= |
1297418.76 |
nM |
9722495 |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
714100.71 |
nM |
23734701 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
274315.53 |
nM |
12431048 |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
385877.51 |
nM |
14761187 |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
3014.12 |
nM |
3397991 |
NPT2175 |
Cell Line |
GAK |
Homo sapiens |
IC50 |
= |
754966.97 |
nM |
10757717 |
NPT2464 |
Cell Line |
MDA-MB-175-VII |
Homo sapiens |
IC50 |
= |
600078.21 |
nM |
20014752 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
138704.25 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2386 |
Cell Line |
KYSE-270 |
Homo sapiens |
IC50 |
= |
302765.02 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
654955.31 |
nM |
1356264 |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
62764.71 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
82388.18 |
nM |
DrugMatrix in vivo data: Hematology |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
606982.52 |
nM |
226705 |
NPT2504 |
Cell Line |
NCI-H1755 |
Homo sapiens |
IC50 |
= |
793271.08 |
nM |
12542359 |
NPT2388 |
Cell Line |
LU-135 |
Homo sapiens |
IC50 |
= |
34840.83 |
nM |
12713403 |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
1044949.67 |
nM |
16872137 |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
3837.08 |
nM |
23153007 |
NPT2492 |
Cell Line |
OAW-42 |
Homo sapiens |
IC50 |
= |
766826.06 |
nM |
22276679 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
407618.63 |
nM |
PubChem BioAssay data set |
NPT2443 |
Cell Line |
SNU-449 |
Homo sapiens |
IC50 |
= |
395122.56 |
nM |
16472241 |
NPT2427 |
Cell Line |
HCC1954 |
Homo sapiens |
IC50 |
= |
25661.66 |
nM |
PubChem BioAssay data set |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Activity |
= |
45 |
% |
23571415 |
NPT2310 |
Cell Line |
CaR-1 |
Homo sapiens |
IC50 |
= |
210950.39 |
nM |
PubChem BioAssay data set |
NPT2353 |
Cell Line |
NCI-H1993 |
Homo sapiens |
IC50 |
= |
828413.15 |
nM |
15730243 |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Activity |
= |
102 |
% |
15270579 |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
10043.19 |
nM |
23869482 |
NPT2207 |
Cell Line |
KP-N-YN |
Homo sapiens |
IC50 |
= |
97572.82 |
nM |
23859780 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
1091380.84 |
nM |
11325241 |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Activity |
= |
98 |
% |
10479293 |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
150043.61 |
nM |
PubChem BioAssay data set |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
47804.75 |
nM |
11434317 |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
80695.03 |
nM |
24216090 |
NPT2462 |
Cell Line |
HuO9 |
Homo sapiens |
IC50 |
= |
508459.72 |
nM |
24387625 |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
96740.29 |
nM |
PubChem BioAssay data set |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
80757.67 |
nM |
10.6019/CHEMBL1201861 |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
IC50 |
= |
157100.07 |
nM |
9392880 |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
82 |
% |
18163590 |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
235243.94 |
nM |
19783438 |
NPT2275 |
Cell Line |
EGI-1 |
Homo sapiens |
IC50 |
= |
56585.51 |
nM |
26351041 |
NPT2467 |
Cell Line |
RERF-LC-MS |
Homo sapiens |
IC50 |
= |
972626.36 |
nM |
24645629 |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Activity |
= |
99 |
% |
19702283 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
239301.68 |
nM |
24972328 |
NPT2304 |
Cell Line |
CAL-72 |
Homo sapiens |
IC50 |
= |
3885.27 |
nM |
1965654 |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
665558.81 |
nM |
10425121 |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
322608.01 |
nM |
23978065 |
NPT2458 |
Cell Line |
FTC-133 |
Homo sapiens |
IC50 |
= |
572594.05 |
nM |
10775404 |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
431357.41 |
nM |
24224843 |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
992099.1 |
nM |
9644083 |
NPT2294 |
Cell Line |
23132-87 |
Homo sapiens |
IC50 |
= |
452453.5 |
nM |
20949916 |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
289951.89 |
nM |
23819871 |
NPT2483 |
Cell Line |
SW13 |
Homo sapiens |
IC50 |
= |
112469.94 |
nM |
23819871 |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
614362.41 |
nM |
24593182 |
NPT2419 |
Cell Line |
HT-1376 |
Homo sapiens |
IC50 |
= |
943608.16 |
nM |
19716307 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
265661.78 |
nM |
PubChem BioAssay data set |
NPT2501 |
Cell Line |
MEL-HO |
Homo sapiens |
IC50 |
= |
659677.45 |
nM |
10924162 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
1067692.44 |
nM |
10924160 |
NPT2416 |
Cell Line |
UACC-893 |
Homo sapiens |
IC50 |
= |
767293.97 |
nM |
16933872 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
871526.26 |
nM |
16933872 |
NPT2302 |
Cell Line |
639-V |
Homo sapiens |
IC50 |
= |
45868.43 |
nM |
PubChem BioAssay data set |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
1023168.03 |
nM |
14738391 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
261516.92 |
nM |
8676127 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
482504.86 |
nM |
10924160 |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
359865.37 |
nM |
10924160 |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
87 |
% |
18723353 |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
1203629.68 |
nM |
23621840 |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
579387.2 |
nM |
8350085 |
NPT2490 |
Cell Line |
NCI-H1666 |
Homo sapiens |
IC50 |
= |
241665.85 |
nM |
15104503 |
NPT3460 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 3 |
Homo sapiens |
Activity |
= |
85 |
% |
25211032 |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Activity |
= |
101 |
% |
21044847 |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
592346.05 |
nM |
15043446 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
137335.39 |
nM |
10514310 |
NPT2512 |
Cell Line |
LCLC-97TM1 |
Homo sapiens |
IC50 |
= |
792336.36 |
nM |
20095629 |
NPT2445 |
Cell Line |
YH-13 |
Homo sapiens |
IC50 |
= |
680159.96 |
nM |
19902967 |
NPT2509 |
Cell Line |
SW1783 |
Homo sapiens |
IC50 |
= |
401797.81 |
nM |
19361174 |
NPT2319 |
Cell Line |
A204 |
Homo sapiens |
IC50 |
= |
81636.3 |
nM |
23911853 |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
260923.43 |
nM |
15270571 |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
634524.56 |
nM |
18278869 |
NPT2023 |
Cell Line |
NB7 |
Homo sapiens |
IC50 |
= |
278024.71 |
nM |
15568794 |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
505550.53 |
nM |
17346076 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
58888.45 |
nM |
8021914 |
NPT2362 |
Cell Line |
TYK-nu |
Homo sapiens |
IC50 |
= |
459340.61 |
nM |
23062825 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
544721.69 |
nM |
21314138 |
NPT2503 |
Cell Line |
NCI-H1703 |
Homo sapiens |
IC50 |
= |
164320.04 |
nM |
19943620 |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
201683.37 |
nM |
8496706 |
NPT2306 |
Cell Line |
Ca-Ski |
Homo sapiens |
IC50 |
= |
725600.8 |
nM |
16378364 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
IC50 |
= |
583 |
nM |
20384293 |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
192583.92 |
nM |
20061160 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
1081653.32 |
nM |
18800848 |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
40654.8 |
nM |
18712933 |
NPT2381 |
Cell Line |
SW900 |
Homo sapiens |
IC50 |
= |
106553.37 |
nM |
12852747 |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
274797.65 |
nM |
16792413 |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Activity |
= |
103 |
% |
PubChem BioAssay data set |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
50348.46 |
nM |
11473426 |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
494599.33 |
nM |
23822611 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
12668.57 |
nM |
24144848 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
88 |
% |
10514302 |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
940678.1 |
nM |
22916954 |
NPT2426 |
Cell Line |
HCC1806 |
Homo sapiens |
IC50 |
= |
122446.97 |
nM |
25871261 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
153572.38 |
nM |
25871261 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
1286400.13 |
nM |
PubChem BioAssay data set |
NPT2482 |
Cell Line |
SW 1116 |
Homo sapiens |
IC50 |
= |
446915.26 |
nM |
PubChem BioAssay data set |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
74319.62 |
nM |
21376582 |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
608924.33 |
nM |
21616566 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
902630.25 |
nM |
15921418 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
654537.58 |
nM |
PubChem BioAssay data set |
NPT2307 |
Cell Line |
769-P |
Homo sapiens |
IC50 |
= |
27783.91 |
nM |
9917297 |
NPT2470 |
Cell Line |
G-402 |
Homo sapiens |
IC50 |
= |
422909.83 |
nM |
11754602 |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
1449621.84 |
nM |
16420055 |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
191545.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2336 |
Cell Line |
OE19 |
Homo sapiens |
IC50 |
= |
885796.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
197260.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
406427.68 |
nM |
10.6019/CHEMBL1201861 |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
62328.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
386457.54 |
nM |
16643036 |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
167027.76 |
nM |
21839640 |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Activity |
= |
109 |
% |
21924800 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
IC50 |
= |
1040587.77 |
nM |
11170656 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
313295.55 |
nM |
23067550 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
1054945.09 |
nM |
15844934 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
630910.49 |
nM |
15043409 |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Activity |
= |
101 |
% |
15497933 |
NPT2508 |
Cell Line |
SW1710 |
Homo sapiens |
IC50 |
= |
170349.63 |
nM |
17253868 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
150005.36 |
nM |
22932311 |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
1138693.69 |
nM |
25468043 |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
587180.34 |
nM |
23031596 |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
723598.01 |
nM |
25946116 |
NPT2273 |
Cell Line |
EFO-21 |
Homo sapiens |
IC50 |
= |
227569.8 |
nM |
17432904 |
NPT2515 |
Cell Line |
MFE-280 |
Homo sapiens |
IC50 |
= |
109007.64 |
nM |
3039137 |
NPT2414 |
Cell Line |
SCC-25 |
Homo sapiens |
IC50 |
= |
524391.22 |
nM |
16040241 |
NPT1953 |
Cell Line |
D-336MG |
Homo sapiens |
IC50 |
= |
854735.44 |
nM |
17257839 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
601434.72 |
nM |
17420206 |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
116472.36 |
nM |
17438057 |
NPT2291 |
Cell Line |
CP50-MEL-B |
Homo sapiens |
IC50 |
= |
529495.15 |
nM |
18330977 |
NPT2384 |
Cell Line |
HPAF-II |
Homo sapiens |
IC50 |
= |
376592.61 |
nM |
18760509 |
NPT2325 |
Cell Line |
BPH-1 |
Homo sapiens |
IC50 |
= |
549795.83 |
nM |
17438050 |
NPT2305 |
Cell Line |
CAL-85-1 |
Homo sapiens |
IC50 |
= |
310724.29 |
nM |
17470649 |
NPT1995 |
Cell Line |
NB17 |
Homo sapiens |
IC50 |
= |
501865.92 |
nM |
17470649 |
NPT2115 |
Cell Line |
HCC2157 |
Homo sapiens |
IC50 |
= |
5652.01 |
nM |
17470660 |
NPT2364 |
Cell Line |
GP5d |
Homo sapiens |
IC50 |
= |
329881.67 |
nM |
19097894 |
NPT2456 |
Cell Line |
TE-11 |
Homo sapiens |
IC50 |
= |
61306.75 |
nM |
18316140 |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Activity |
= |
89 |
% |
18070962 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
IC50 |
= |
990 |
nM |
18070972 |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
68213.4 |
nM |
19540629 |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
186839.13 |
nM |
19926364 |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
97507.57 |
nM |
19884366 |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
385688.1 |
nM |
20558071 |
NPT2475 |
Cell Line |
NCI-H1651 |
Homo sapiens |
IC50 |
= |
354113.33 |
nM |
18299404 |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Activity |
= |
109 |
% |
18955529 |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
153919.85 |
nM |
18838581 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
IC50 |
= |
50500 |
nM |
18838581 |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
175225.9 |
nM |
18443128 |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
16855.67 |
nM |
18936192 |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
185139.02 |
nM |
19188377 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
1604155.93 |
nM |
19651910 |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
196922.65 |
nM |
19721064 |
NPT1944 |
Cell Line |
D-247MG |
Homo sapiens |
IC50 |
= |
391018.16 |
nM |
21273067 |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
67472.63 |
nM |
19581457 |
NPT2444 |
Cell Line |
YAPC |
Homo sapiens |
IC50 |
= |
602338.15 |
nM |
21524583 |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
64970.61 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
170193.16 |
nM |
PubChem BioAssay data set |
NPT2514 |
Cell Line |
LN-405 |
Homo sapiens |
IC50 |
= |
66592.77 |
nM |
10.1007/s00044-011-9861-4 |
NPT2271 |
Cell Line |
DoTc2-4510 |
Homo sapiens |
IC50 |
= |
163163.86 |
nM |
10.1007/s00044-009-9228-2 |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Activity |
= |
89 |
% |
10.1007/s00044-009-9206-8 |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
346316.12 |
nM |
10.1007/s00044-012-0437-8 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
455895.67 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2383 |
Cell Line |
ESS-1 |
Homo sapiens |
IC50 |
= |
689489.18 |
nM |
10.1039/C1MD00272D |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
154430.01 |
nM |
25495422 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
624325.58 |
nM |
10.1039/C4MD00124A |
NPT2300 |
Cell Line |
CAL-54 |
Homo sapiens |
IC50 |
= |
54104.81 |
nM |
26090896 |
NPT2494 |
Cell Line |
RMG-I |
Homo sapiens |
IC50 |
= |
221396.01 |
nM |
26497285 |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
206158.03 |
nM |
PubChem BioAssay data set |
NPT2298 |
Cell Line |
BALL-1 |
Homo sapiens |
IC50 |
= |
134456.67 |
nM |
15332867 |
NPT2412 |
Cell Line |
Panc1005 |
Homo sapiens |
IC50 |
= |
214654.34 |
nM |
21507644 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
807555.67 |
nM |
19132934 |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
IC50 |
= |
225352.54 |
nM |
8133298 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
IC50 |
= |
89 |
nM |
17157006 |
NPT1948 |
Cell Line |
A253 cell line |
|
IC50 |
= |
435625.1 |
nM |
9014350 |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
314824.08 |
nM |
12088447 |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
241567.76 |
nM |
19902967 |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
905741.55 |
nM |
19845338 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
62224.45 |
nM |
17378609 |
NPT2480 |
Cell Line |
RH-18 |
Homo sapiens |
IC50 |
= |
713561.77 |
nM |
17480100 |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
75947.02 |
nM |
16038541 |
NPT2366 |
Cell Line |
JEG-3 |
Homo sapiens |
IC50 |
= |
578482.33 |
nM |
17352491 |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
474850.97 |
nM |
16417306 |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Activity |
= |
98 |
% |
16417306 |
NPT2330 |
Cell Line |
D-566MG |
Homo sapiens |
IC50 |
= |
1003338.28 |
nM |
25737008 |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
245866.57 |
nM |
23611151 |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
1292668.54 |
nM |
11908959 |
NPT2286 |
Cell Line |
CAL-120 |
Homo sapiens |
IC50 |
= |
185989.09 |
nM |
21377877 |
NPT2446 |
Cell Line |
HCC38 |
Homo sapiens |
IC50 |
= |
517753.37 |
nM |
9514009 |
NPT2314 |
Cell Line |
BEN |
Homo sapiens |
IC50 |
= |
314946.88 |
nM |
1919592 |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Activity |
= |
105 |
% |
11858759 |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
105362.21 |
nM |
20627740 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
293060.48 |
nM |
20627740 |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
IC50 |
= |
246729.11 |
nM |
10.1584/jpestics.27.127 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
70866.87 |
nM |
23543830 |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
724808.88 |
nM |
PubChem BioAssay data set |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
176314.44 |
nM |
PubChem BioAssay data set |
NPT2334 |
Cell Line |
NCI-H1793 |
Homo sapiens |
IC50 |
= |
308606.19 |
nM |
12027733 |
NPT2303 |
Cell Line |
647-V |
Homo sapiens |
IC50 |
= |
1013659.17 |
nM |
20541427 |
NPT1969 |
Cell Line |
TGW |
Homo sapiens |
IC50 |
= |
86031.71 |
nM |
19902967 |
NPT2511 |
Cell Line |
HGC-27 |
Homo sapiens |
IC50 |
= |
224554.63 |
nM |
19902967 |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Activity |
= |
95 |
% |
19921834 |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
1177622.67 |
nM |
10924160 |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
1131743.9 |
nM |
21130542 |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Activity |
= |
88 |
% |
15497961 |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
102376.58 |
nM |
23434030 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
260540.68 |
nM |
23434030 |
NPT2350 |
Cell Line |
HN |
Homo sapiens |
IC50 |
= |
68561.49 |
nM |
23434131 |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
561991.65 |
nM |
16722644 |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
57031.69 |
nM |
PubChem BioAssay data set |
NPT2421 |
Cell Line |
PFSK-1 |
Homo sapiens |
IC50 |
= |
1279130.72 |
nM |
19095451 |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
85180.71 |
nM |
16643022 |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
222592.11 |
nM |
25136911 |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
73863.96 |
nM |
11741487 |
NPT2373 |
Cell Line |
KYSE-150 cell line |
|
IC50 |
= |
1267132.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
382452.32 |
nM |
10.6019/CHEMBL1201861 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
194425.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
178758.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2380 |
Cell Line |
SK-N-AS |
Homo sapiens |
IC50 |
= |
134604.25 |
nM |
16933872 |
NPT2422 |
Cell Line |
SCC-4 |
Homo sapiens |
IC50 |
= |
96129.86 |
nM |
24645629 |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Activity |
= |
105 |
% |
26034885 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
516803.13 |
nM |
26034885 |
NPT2425 |
Cell Line |
UMC-11 |
Homo sapiens |
IC50 |
= |
407590.5 |
nM |
11141110 |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
172678.24 |
nM |
12608849 |
NPT2455 |
Cell Line |
SNU-C2B |
Homo sapiens |
IC50 |
= |
314982.47 |
nM |
20102170 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
IC50 |
= |
370 |
nM |
10514334 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
252487.57 |
nM |
10514334 |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Activity |
= |
113 |
% |
17844994 |
NPT2390 |
Cell Line |
NCI-H2122 |
Homo sapiens |
IC50 |
= |
258358.72 |
nM |
25739048 |
NPT2293 |
Cell Line |
CAL-39 |
Homo sapiens |
IC50 |
= |
952998.19 |
nM |
24901800 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
9049.28 |
nM |
19555123 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
302444.87 |
nM |
12662106 |
NPT2437 |
Cell Line |
EW-22 |
Homo sapiens |
IC50 |
= |
445556.47 |
nM |
PubChem BioAssay data set |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
399954.98 |
nM |
25951057 |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
316685.45 |
nM |
25237727 |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
1123589.78 |
nM |
26341134 |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
426683.28 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
476727.95 |
nM |
10395485 |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
IC50 |
= |
27013.86 |
nM |
8389875 |
NPT6632 |
Cell Line |
CHP-134 |
Homo sapiens |
IC50 |
= |
11563.46 |
nM |
17493824 |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
103678.84 |
nM |
17188868 |
NPT2404 |
Cell Line |
SW982 |
Homo sapiens |
IC50 |
= |
364662.77 |
nM |
20739103 |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
76374.05 |
nM |
21419530 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
45856.23 |
nM |
21733601 |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Activity |
= |
86 |
% |
DrugMatrix in vitro pharmacology data |
NPT2348 |
Cell Line |
HLE |
Homo sapiens |
IC50 |
= |
693194.07 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
173036.92 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2406 |
Cell Line |
HCC1395 |
Homo sapiens |
IC50 |
= |
1311685.2 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2479 |
Cell Line |
OAW-28 |
Homo sapiens |
IC50 |
= |
133537.32 |
nM |
22104973 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
303500.73 |
nM |
22704923 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
461179.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2374 |
Cell Line |
KYSE-180 |
Homo sapiens |
IC50 |
= |
94839.12 |
nM |
10.6019/CHEMBL1201861 |
NPT890 |
Cell Line |
SNU-387 |
Homo sapiens |
IC50 |
= |
989827.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
550946.11 |
nM |
10.6019/CHEMBL1201861 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
63864.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2333 |
Cell Line |
DBTRG-05MG |
Homo sapiens |
IC50 |
= |
21709.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
300449.59 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT2428 |
Cell Line |
HT-3 |
Homo sapiens |
IC50 |
= |
862211.84 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT2354 |
Cell Line |
NCI-H2009 |
Homo sapiens |
IC50 |
= |
786384.61 |
nM |
Open TG-GATES in vivo data: Hematology |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
409009.34 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Activity |
= |
82 |
% |
Open TG-GATES in vivo data: Biochemistry |
NPT2498 |
Cell Line |
KOSC-2 |
Homo sapiens |
IC50 |
= |
226691.49 |
nM |
Open TG-GATES in vivo data: Biochemistry |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Activity |
= |
99 |
% |
Open TG-GATES in vivo data: Biochemistry |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
18313.45 |
nM |
Open TG-GATES in vivo data: Organ Weight |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
IC50 |
= |
20600 |
nM |
15646539 |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
745204 |
nM |
25062006 |
NPT2344 |
Cell Line |
SK-MEL-24 |
Homo sapiens |
IC50 |
= |
39224.2 |
nM |
24937209 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
725644.34 |
nM |
26010585 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
IC50 |
= |
527523.28 |
nM |
26160020 |
NPT2436 |
Cell Line |
VMRC-RCZ |
Homo sapiens |
IC50 |
= |
402636.03 |
nM |
26988298 |
NPT2457 |
Cell Line |
YKG-1 |
Homo sapiens |
IC50 |
= |
38257.59 |
nM |
22694318 |
NPT2339 |
Cell Line |
TGBC24TKB |
Homo sapiens |
IC50 |
= |
960753.62 |
nM |
17190463 |
NPT2485 |
Cell Line |
IA-LM |
Homo sapiens |
IC50 |
= |
266150.25 |
nM |
PubChem BioAssay data set |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
166603.21 |
nM |
19441852 |
NPT2317 |
Cell Line |
ChaGo-K-1 |
Homo sapiens |
IC50 |
= |
195428.97 |
nM |
24689881 |
NPT2278 |
Cell Line |
COLO-741 |
Homo sapiens |
IC50 |
= |
513157.59 |
nM |
24689881 |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Activity |
= |
95 |
% |
8105084 |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
534627.9 |
nM |
20570145 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
258763.11 |
nM |
26034885 |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
174102.99 |
nM |
14510611 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
11730.9 |
nM |
14664515 |
NPT3815 |
Individual Protein |
Tyrosine-protein kinase LCK |
Mus musculus |
Activity |
= |
88 |
% |
14640510 |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
91760.51 |
nM |
18314943 |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
55347.14 |
nM |
PubChem BioAssay data set |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Activity |
= |
108 |
% |
23398362 |
NPT2493 |
Cell Line |
OC-314 |
Homo sapiens |
IC50 |
= |
1643979.33 |
nM |
9548875 |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Activity |
= |
30 |
% |
20634081 |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Activity |
= |
127 |
% |
20624681 |
NPT2272 |
Cell Line |
EFM-19 |
Homo sapiens |
IC50 |
= |
433724.7 |
nM |
23819826 |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
453186.62 |
nM |
20035556 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
316226.27 |
nM |
20192247 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
803498.24 |
nM |
16448174 |
NPT2447 |
Cell Line |
HuCCT-1 |
Homo sapiens |
IC50 |
= |
504047.75 |
nM |
16448174 |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
18099.35 |
nM |
16448174 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
312854.43 |
nM |
19948405 |
NPT2507 |
Cell Line |
RPMI-2650 |
Homo sapiens |
IC50 |
= |
282787.01 |
nM |
8786361 |
NPT2460 |
Cell Line |
HCE-4 |
Homo sapiens |
IC50 |
= |
85569.17 |
nM |
2895165 |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
430662.62 |
nM |
17844994 |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
250702.26 |
nM |
17844994 |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
435167.93 |
nM |
17480098 |
NPT2487 |
Cell Line |
KNS-62 |
Homo sapiens |
IC50 |
= |
113873.82 |
nM |
11908979 |
NPT2440 |
Cell Line |
NCI-H1563 |
Homo sapiens |
IC50 |
= |
890236.36 |
nM |
19072209 |
NPT2363 |
Cell Line |
U-118-MG |
Homo sapiens |
IC50 |
= |
289593.73 |
nM |
15332848 |
NPT2274 |
Cell Line |
EFO-27 |
Homo sapiens |
IC50 |
= |
377591.91 |
nM |
11975490 |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Activity |
= |
116 |
% |
26900954 |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
676492.26 |
nM |
9871531 |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
977862.43 |
nM |
PubChem BioAssay data set |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
189229.96 |
nM |
15787442 |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
247337.8 |
nM |
24571273 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
815242 |
nM |
24571273 |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
142444.15 |
nM |
17609121 |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
11704.5 |
nM |
PubChem BioAssay data set |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
166093.35 |
nM |
12139460 |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
IC50 |
= |
22289.26 |
nM |
17064070 |
NPT2398 |
Cell Line |
MKN-7 |
Homo sapiens |
IC50 |
= |
806773.53 |
nM |
17242150 |
NPT2346 |
Cell Line |
TI-73 |
Homo sapiens |
IC50 |
= |
456497.4 |
nM |
19231182 |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Activity |
= |
92 |
% |
14510589 |
NPT2313 |
Cell Line |
BCPAP |
Homo sapiens |
IC50 |
= |
406137.19 |
nM |
12828469 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
161338.56 |
nM |
8450319 |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
33493.52 |
nM |
19196516 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
62951.34 |
nM |
17967917 |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
477927 |
nM |
19703776 |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
863537.22 |
nM |
20361799 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
IC50 |
= |
177750.17 |
nM |
20361799 |
NPT1184 |
Cell Line |
Daoy |
Homo sapiens |
IC50 |
= |
19393.91 |
nM |
20709557 |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Activity |
= |
103 |
% |
19651905 |
NPT2495 |
Cell Line |
SW1417 |
Homo sapiens |
IC50 |
= |
474085.18 |
nM |
21910466 |
NPT2359 |
Cell Line |
SK-MEL-30 |
Homo sapiens |
IC50 |
= |
14642.82 |
nM |
22269277 |
NPT2449 |
Cell Line |
NCI-H1573 |
Homo sapiens |
IC50 |
= |
72737.86 |
nM |
22464685 |
NPT2342 |
Cell Line |
NCI-H630 |
Homo sapiens |
IC50 |
= |
867571.56 |
nM |
21852132 |
NPT2343 |
Cell Line |
NCI-H650 |
Homo sapiens |
IC50 |
= |
273680.13 |
nM |
22683112 |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Activity |
= |
112 |
% |
22783984 |
NPT2391 |
Cell Line |
NCI-H810 |
Homo sapiens |
IC50 |
= |
643948.01 |
nM |
23270565 |
NPT2431 |
Cell Line |
NCI-H1437 |
Homo sapiens |
IC50 |
= |
162815.39 |
nM |
23896611 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
78834.05 |
nM |
24468411 |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
542288.96 |
nM |
10.1039/C1MD00127B |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
178481.51 |
nM |
24568587 |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
508206.06 |
nM |
137981 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
265182.43 |
nM |
24906512 |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
265346.1 |
nM |
25137549 |
NPT2438 |
Cell Line |
HTC-C3 |
Homo sapiens |
IC50 |
= |
21602.09 |
nM |
25137549 |
NPT2411 |
Cell Line |
NCI-H2228 |
Homo sapiens |
IC50 |
= |
166076.58 |
nM |
25593097 |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
IC50 |
= |
7738.35 |
nM |
25835647 |
NPT2321 |
Cell Line |
BHT-101 |
Homo sapiens |
IC50 |
= |
428791.59 |
nM |
15387651 |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Activity |
= |
49 |
% |
23398362 |
NPT2415 |
Cell Line |
SKG-IIIa |
Homo sapiens |
IC50 |
= |
978838.83 |
nM |
23398362 |
NPT2299 |
Cell Line |
CAL-51 |
Homo sapiens |
IC50 |
= |
64735.13 |
nM |
23398362 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
302126.56 |
nM |
10.1039/C2MD20076G |
NPT2472 |
Cell Line |
HuP-T4 |
Homo sapiens |
IC50 |
= |
953470.04 |
nM |
11374943 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
55.4 |
% |
15497938 |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
25601.58 |
nM |
14640569 |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
23896.88 |
nM |
23571415 |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
116831.65 |
nM |
17848089 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
500153.47 |
nM |
12639542 |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Activity |
= |
105 |
% |
11000036 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
232827.31 |
nM |
24697496 |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
678881.78 |
nM |
11975502 |
NPT2432 |
Cell Line |
NCI-H2342 |
Homo sapiens |
IC50 |
= |
1154755.6 |
nM |
10869203 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
479314.52 |
nM |
10869203 |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Activity |
= |
88 |
% |
10869203 |
NPT1216 |
Cell Line |
FaDu |
Homo sapiens |
IC50 |
= |
48827.42 |
nM |
19835393 |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Activity |
= |
23 |
% |
23734701 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
223369.42 |
nM |
20666364 |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
56086.49 |
nM |
24180210 |
NPT2496 |
Cell Line |
SW1463 |
Homo sapiens |
IC50 |
= |
95289.92 |
nM |
24044895 |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
1007659.91 |
nM |
24645629 |
NPT2281 |
Cell Line |
ABC-1 |
Homo sapiens |
IC50 |
= |
483529.83 |
nM |
15217281 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
120296.92 |
nM |
23354070 |
NPT2335 |
Cell Line |
NCI-H596 |
|
IC50 |
= |
626116.21 |
nM |
25245917 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Inhibition |
= |
60 |
% |
10843570 |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
336274.91 |
nM |
22901896 |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
451164.04 |
nM |
25856683 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
612240.39 |
nM |
21288727 |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
350437.02 |
nM |
25819096 |
NPT2372 |
Cell Line |
H-EMC-SS |
Homo sapiens |
IC50 |
= |
999391.91 |
nM |
20303767 |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Activity |
= |
82 |
% |
8133298 |
NPT2418 |
Cell Line |
HCC1569 |
Homo sapiens |
IC50 |
= |
570582.63 |
nM |
18640837 |
NPT2288 |
Cell Line |
AN3-CA |
Homo sapiens |
IC50 |
= |
248568.63 |
nM |
10479316 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
193121.78 |
nM |
26358281 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
97977.61 |
nM |
26358281 |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
11381.42 |
nM |
21643465 |
NPT2481 |
Cell Line |
SW1088 |
Homo sapiens |
IC50 |
= |
236698.22 |
nM |
22137934 |
NPT1313 |
Cell Line |
Capan-2 |
Homo sapiens |
IC50 |
= |
188316.87 |
nM |
12662097 |
NPT2486 |
Cell Line |
IGR-1 |
Homo sapiens |
IC50 |
= |
936890.11 |
nM |
23145909 |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
540099.29 |
nM |
15730238 |
NPT3465 |
Cell Line |
ECC10 |
Homo sapiens |
IC50 |
= |
52380.38 |
nM |
22445674 |
NPT2284 |
Cell Line |
C3A |
Homo sapiens |
IC50 |
= |
223539.92 |
nM |
9584401 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
79545.09 |
nM |
16309305 |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
575662.18 |
nM |
23691978 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
73749.78 |
nM |
14738391 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
166157.48 |
nM |
17353252 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
725066.23 |
nM |
19012394 |
NPT2442 |
Cell Line |
NCI-H2405 |
Homo sapiens |
IC50 |
= |
416498.97 |
nM |
20373816 |
NPT2510 |
Cell Line |
GCT |
Homo sapiens |
IC50 |
= |
316080.84 |
nM |
19805565 |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
5062.16 |
nM |
19805554 |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
321011.2 |
nM |
19933793 |
NPT2320 |
Cell Line |
BFTC-909 |
Homo sapiens |
IC50 |
= |
44913.26 |
nM |
20038618 |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
398363.94 |
nM |
18180356 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
183721.13 |
nM |
18644958 |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
62853.15 |
nM |
18710917 |
NPT2360 |
Cell Line |
SW756 |
Homo sapiens |
IC50 |
= |
966662.1 |
nM |
18725441 |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
38077.55 |
nM |
18285482 |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Activity |
= |
98 |
% |
18519722 |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Activity |
= |
94 |
% |
20970332 |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
52497.47 |
nM |
19349512 |
NPT2471 |
Cell Line |
HuP-T3 |
Homo sapiens |
IC50 |
= |
81189.99 |
nM |
19349512 |
NPT1505 |
Cell Line |
J82 |
Homo sapiens |
IC50 |
= |
253247.94 |
nM |
19258280 |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
7321.56 |
nM |
20231393 |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
113271.21 |
nM |
20805391 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
684698.09 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Activity |
= |
103 |
% |
23352268 |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
172234 |
nM |
DrugMatrix in vivo data: Biochemistry |
NPT2513 |
Cell Line |
LK-2 |
Homo sapiens |
IC50 |
= |
223963.7 |
nM |
DrugMatrix in vivo data: Hematology |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
218680.12 |
nM |
24927053 |
NPT2292 |
Cell Line |
CAL-33 |
Homo sapiens |
IC50 |
= |
471075.79 |
nM |
26476666 |
NPT1884 |
Cell Line |
HCC1937 |
Homo sapiens |
IC50 |
= |
606711.87 |
nM |
23268694 |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
239765.17 |
nM |
26295746 |
NPT2332 |
Cell Line |
COLO-680N |
Homo sapiens |
IC50 |
= |
80186.49 |
nM |
19228038 |
NPT2478 |
Cell Line |
NY |
Homo sapiens |
IC50 |
= |
14997.01 |
nM |
25510639 |
NPT2347 |
Cell Line |
GMS-10 |
Homo sapiens |
IC50 |
= |
508422.1 |
nM |
PubChem BioAssay data set |
NPT2500 |
Cell Line |
LCLC-103H cell line |
|
IC50 |
= |
344166.31 |
nM |
12762791 |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
14994.97 |
nM |
25397992 |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
359447.09 |
nM |
25397992 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
569710.31 |
nM |
20055495 |
NPT2502 |
Cell Line |
MEL-JUSO |
Homo sapiens |
IC50 |
= |
132028.13 |
nM |
21875800 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
104606.85 |
nM |
23587837 |
NPT2371 |
Cell Line |
SW837 |
Homo sapiens |
IC50 |
= |
174687.91 |
nM |
23587837 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
245592.58 |
nM |
17524651 |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
388404.37 |
nM |
19007286 |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
12796.25 |
nM |
25946116 |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
403413.46 |
nM |
25946116 |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
80 |
% |
25946116 |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
250828.64 |
nM |
PubChem BioAssay data set |
NPT2409 |
Cell Line |
LU-99A |
Homo sapiens |
IC50 |
= |
124848.62 |
nM |
19256529 |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
1063683.33 |
nM |
17190465 |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
559182.56 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
254274.65 |
nM |
DrugMatrix in vitro pharmacology data |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
161758.91 |
nM |
11430019 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
315574.25 |
nM |
2362268 |
NPT2324 |
Cell Line |
CHP-212 |
Homo sapiens |
IC50 |
= |
663168.43 |
nM |
PubChem BioAssay data set |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
82277.11 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
228893.54 |
nM |
PubChem BioAssay data set |
NPT2423 |
Cell Line |
SCC-9 |
Homo sapiens |
IC50 |
= |
776950 |
nM |
PubChem BioAssay data set |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Activity |
= |
72 |
% |
DrugMatrix in vivo data: Biochemistry |
NPT2270 |
Cell Line |
Detroit562 |
Homo sapiens |
IC50 |
= |
318920.87 |
nM |
24387683 |
NPT2367 |
Cell Line |
KYSE-140 |
Homo sapiens |
IC50 |
= |
443549.76 |
nM |
17118653 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
572066.93 |
nM |
23145909 |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
421705.41 |
nM |
16441070 |
NPT2370 |
Cell Line |
RVH-421 |
Homo sapiens |
IC50 |
= |
973677.36 |
nM |
16038541 |
NPT2329 |
Cell Line |
COLO-679 |
Homo sapiens |
IC50 |
= |
1230318.06 |
nM |
18847278 |
NPT2484 |
Cell Line |
GAMG |
Homo sapiens |
IC50 |
= |
186804.95 |
nM |
9917292 |
NPT2448 |
Cell Line |
KLE |
Homo sapiens |
IC50 |
= |
894808.74 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2357 |
Cell Line |
RT-112 |
Homo sapiens |
IC50 |
= |
92343.75 |
nM |
19674906 |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Activity |
= |
101 |
% |
11374948 |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
261808.68 |
nM |
15711537 |
NPT2323 |
Cell Line |
BHY |
Homo sapiens |
IC50 |
= |
55688.74 |
nM |
15711537 |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
145918.32 |
nM |
18077425 |
NPT2408 |
Cell Line |
KYSE-70 cell line |
|
IC50 |
= |
287628.87 |
nM |
18077425 |
NPT2395 |
Cell Line |
KYSE-450 |
Homo sapiens |
IC50 |
= |
131892.47 |
nM |
18077425 |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Activity |
= |
112 |
% |
18183025 |
NPT2499 |
Cell Line |
KP-4 |
Homo sapiens |
IC50 |
= |
158545.4 |
nM |
19654408 |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Activity |
= |
107 |
% |
21450463 |
NPT2269 |
Cell Line |
EPLC-272H |
Homo sapiens |
IC50 |
= |
35749.17 |
nM |
22037378 |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
26150.6 |
nM |
22037378 |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
62856.42 |
nM |
22037378 |
NPT2461 |
Cell Line |
HuO-3N1 |
Homo sapiens |
IC50 |
= |
2775.01 |
nM |
22560627 |
NPT2327 |
Cell Line |
D-423MG |
Homo sapiens |
IC50 |
= |
188858.49 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
100272.35 |
nM |
24960143 |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
121989.62 |
nM |
8759172 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
316355.95 |
nM |
23434636 |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
106 |
% |
20155971 |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
73547.83 |
nM |
14640511 |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
35102.38 |
nM |
21970540 |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
25059.35 |
nM |
25856683 |
NPT2167 |
Cell Line |
LB996-RCC |
Homo sapiens |
IC50 |
= |
74425.16 |
nM |
8463795 |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Activity |
= |
90 |
% |
19702283 |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
338840.33 |
nM |
1895288 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
531472.79 |
nM |
16472241 |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
1097655.7 |
nM |
16472241 |
NPT2491 |
Cell Line |
NCI-H1693 |
Homo sapiens |
IC50 |
= |
296645.26 |
nM |
DrugMatrix in vitro pharmacology data |
NPT2312 |
Cell Line |
8305C |
Homo sapiens |
IC50 |
= |
624848.99 |
nM |
DrugMatrix in vitro pharmacology data |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Activity |
= |
110 |
% |
15646539 |
NPT2376 |
Cell Line |
NBsusSR |
Homo sapiens |
IC50 |
= |
13316.91 |
nM |
10.6019/CHEMBL3301361 |
NPT2435 |
Cell Line |
VM-CUB-1 |
Homo sapiens |
IC50 |
= |
28192.73 |
nM |
24679044 |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
832808.73 |
nM |
18665642 |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Activity |
= |
100 |
% |
15482904 |
NPT2402 |
Cell Line |
PANC-08-13 |
Homo sapiens |
IC50 |
= |
138355.44 |
nM |
PubChem BioAssay data set |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
238962.11 |
nM |
8064806 |
NPT2439 |
Cell Line |
MC-IXC |
Homo sapiens |
IC50 |
= |
805206.69 |
nM |
18417256 |
NPT2453 |
Cell Line |
RCM-1 |
Homo sapiens |
IC50 |
= |
770675.19 |
nM |
17938184 |
NPT1980 |
Cell Line |
NB14 |
Homo sapiens |
IC50 |
= |
149546.14 |
nM |
20038624 |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
1822351.54 |
nM |
18694945 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
97 |
% |
19596880 |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
463979.33 |
nM |
DrugMatrix in vitro pharmacology data |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Activity |
= |
88 |
% |
22194678 |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
20564.12 |
nM |
22995771 |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Activity |
= |
98 |
% |
10.1007/s00044-011-9918-4 |
NPT3466 |
Cell Line |
MOLT-13 |
Homo sapiens |
IC50 |
= |
200745.91 |
nM |
23811259 |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
73572.7 |
nM |
DrugMatrix in vivo data: Pathology |
NPT2309 |
Cell Line |
CAPAN-1 |
Homo sapiens |
IC50 |
= |
50292.4 |
nM |
23992864 |
NPT2315 |
Cell Line |
BFTC-905 |
Homo sapiens |
IC50 |
= |
52498.73 |
nM |
12088429 |
NPT2290 |
Cell Line |
CAL-27 |
Homo sapiens |
IC50 |
= |
142027.54 |
nM |
18327911 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
98854.1 |
nM |
20655237 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
26766.12 |
nM |
3572419 |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
340178.34 |
nM |
17296744 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
177636.8 |
nM |
19721074 |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
296048.12 |
nM |
19721074 |
NPT1215 |
Cell Line |
8505C |
Homo sapiens |
IC50 |
= |
883379.59 |
nM |
22194678 |
NPT2282 |
Cell Line |
C32 |
Homo sapiens |
IC50 |
= |
17660.56 |
nM |
22459876 |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Activity |
= |
82 |
% |
23811085 |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
1122672.18 |
nM |
23811085 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
926994.84 |
nM |
24262883 |
NPT2301 |
Cell Line |
CAL-62 |
Homo sapiens |
IC50 |
= |
150508.11 |
nM |
26213786 |
NPT2289 |
Cell Line |
CAL-12T |
Homo sapiens |
IC50 |
= |
496486.35 |
nM |
21332115 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
IC50 |
= |
1529551.75 |
nM |
PubChem BioAssay data set |
NPT2399 |
Cell Line |
NCI-H2170 |
Homo sapiens |
IC50 |
= |
224405.12 |
nM |
15165138 |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Activity |
= |
99 |
% |
15165138 |
NPT2355 |
Cell Line |
NCI-H2029 |
Homo sapiens |
IC50 |
= |
269332.32 |
nM |
23999046 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
59533.43 |
nM |
21741249 |