Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
438800 |
Kb M-1 |
14643314 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
46.8 |
% |
10.1016/0960-894X(96)00092-3 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25.3 |
% |
10.1016/0960-894X(96)00092-3 |
NPT745 |
Individual Protein |
G-protein coupled bile acid receptor 1 |
Homo sapiens |
EC50 |
= |
580 |
nM |
18307294 |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
EC50 |
= |
20000 |
nM |
18307294 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
0.029 |
|
18307294 |
NPT2611 |
Cell Line |
GBM |
Homo sapiens |
LD50 |
>= |
0.05 |
nM |
18768321 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
LD50 |
> |
0.05 |
nM |
18768321 |
NPT2 |
Others |
Unspecified |
|
LD50 |
> |
0.05 |
nM |
18768321 |
NPT745 |
Individual Protein |
G-protein coupled bile acid receptor 1 |
Homo sapiens |
EC50 |
= |
5600 |
nM |
19911773 |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
EC50 |
= |
6700 |
nM |
19911773 |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT211 |
Individual Protein |
Hypoxia-inducible factor 1 alpha |
Homo sapiens |
Potency |
= |
50118.7 |
nM |
PubChem BioAssay data set |
NPT1226 |
Individual Protein |
Caspase-7 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
= |
44668.4 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
14125.4 |
nM |
PubChem BioAssay data set |
NPT53 |
Individual Protein |
4'-phosphopantetheinyl transferase ffp |
Bacillus subtilis |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT157 |
Individual Protein |
Breast cancer type 1 susceptibility protein |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT55 |
Individual Protein |
Putative fructose-1,6-bisphosphate aldolase |
Giardia intestinalis |
Potency |
= |
15811.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT58 |
Individual Protein |
Bloom syndrome protein |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT532 |
Individual Protein |
Lysine-specific demethylase 4A |
Homo sapiens |
Potency |
|
79432.8 |
nM |
PubChem BioAssay data set |
NPT443 |
Individual Protein |
Histone acetyltransferase GCN5 |
Homo sapiens |
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT4 |
Individual Protein |
Large T antigen |
Simian virus 40 |
IC50 |
|
26100 |
nM |
PubChem BioAssay data set |
NPT1139 |
Individual Protein |
Arachidonate 15-lipoxygenase, type II |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18100 |
nM |
21388808 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
10000 |
nM |
PubChem BioAssay data set |
NPT546 |
Individual Protein |
Retinoid X receptor alpha |
Homo sapiens |
Potency |
|
28183.8 |
nM |
PubChem BioAssay data set |
NPT546 |
Individual Protein |
Retinoid X receptor alpha |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT108 |
Individual Protein |
Estrogen receptor alpha |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT108 |
Individual Protein |
Estrogen receptor alpha |
Homo sapiens |
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT803 |
Individual Protein |
Flap endonuclease 1 |
Homo sapiens |
Potency |
|
28183.8 |
nM |
PubChem BioAssay data set |
NPT8 |
Individual Protein |
DNA polymerase iota |
Homo sapiens |
Potency |
|
794.3 |
nM |
PubChem BioAssay data set |
NPT3938 |
Individual Protein |
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
Homo sapiens |
IC50 |
= |
4823 |
nM |
PubChem BioAssay data set |
NPT98 |
Individual Protein |
HERG |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT199 |
Individual Protein |
DNA polymerase kappa |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT99 |
Individual Protein |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT249 |
Individual Protein |
Glucocorticoid receptor |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT249 |
Individual Protein |
Glucocorticoid receptor |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT699 |
Individual Protein |
UDP-glucuronosyltransferase 1-10 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT695 |
Individual Protein |
UDP-glucuronosyltransferase 1-8 |
Homo sapiens |
Activity |
= |
11 |
pm/min/mg |
10836148 |
NPT704 |
Individual Protein |
UDP-glucuronosyltransferase 2B15 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT904 |
Individual Protein |
UDP-glucuronosyltransferase 2B17 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT701 |
Individual Protein |
UDP-glucuronosyltransferase 2B4 |
Homo sapiens |
Activity |
= |
0 |
pm/min/mg |
10836148 |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
19952.62 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
20844.91 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
100000 |
nM |
PubChem BioAssay data set |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
60673.63 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
29308.93 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
17906.06 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
15631.48 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
37757.22 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
14288.94 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
22080.05 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
52360.04 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
34119.29 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
27989.81 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
15066.07 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
26001.6 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
44360.86 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
29991.63 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
27605.78 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
40271.7 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
100000 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
18281 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
100000 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
17378.01 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
32583.67 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
21978.6 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
19010.78 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
28183.83 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
37153.52 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
21527.82 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
29241.52 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
21281.39 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
54325.03 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
40179.08 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
41304.75 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
50003.45 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
20701.41 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
100000 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
56493.7 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
58748.94 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
24322.04 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
14621.77 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
42266.86 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
28248.8 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
23442.29 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
33573.76 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
26977.39 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
42364.3 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
68076.94 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
40457.59 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
24378.11 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
25468.3 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
17258.38 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
30408.85 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
28054.34 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
22855.99 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
58748.94 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
23604.78 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
31988.95 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
31332.86 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
29512.09 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
28444.61 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
28906.8 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
53951.06 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
28444.61 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
21527.82 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
18365.38 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
25292.98 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
22233.1 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
24603.68 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
66069.34 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
19815.27 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
30408.85 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
23496.33 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
46451.53 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
18365.38 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
35974.93 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
100000 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
44463.13 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
36559.48 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
19952.62 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
30199.52 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
26181.83 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
23878.11 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
33651.16 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
19952.62 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
40271.7 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
31045.6 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
35318.32 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
38636.7 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
18197.01 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
37497.3 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
22130.95 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
22594.36 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
26730.06 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
40738.03 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
37239.17 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
39994.47 |
nM |
PubChem BioAssay data set |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
|
33342.64 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
49317.38 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
28313.92 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
27669.42 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
31841.98 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
21877.62 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
63533.09 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
37068.07 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
21627.19 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
46131.76 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
27039.58 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
54325.03 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
23713.74 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
26001.6 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
46881.34 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
25527.01 |
nM |
PubChem BioAssay data set |
NPT745 |
Individual Protein |
G-protein coupled bile acid receptor 1 |
Homo sapiens |
EC50 |
= |
5000 |
nM |
24900463 |
NPT748 |
Individual Protein |
Bile acid transporter |
Homo sapiens |
Activity |
= |
63 |
% |
8132774 |
NPT1028 |
Individual Protein |
Multidrug resistance-associated protein 4 |
Homo sapiens |
Activity |
= |
68 |
% |
12883481 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
10322.5 |
nM |
PubChem BioAssay data set |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
19331.2 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
26603.2 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT102 |
Individual Protein |
Interleukin-8 |
Homo sapiens |
Potency |
|
74978 |
nM |
PubChem BioAssay data set |
NPT103 |
Individual Protein |
Nuclear receptor ROR-gamma |
Homo sapiens |
Potency |
|
74978 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
10000 |
nM |
23330053 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.6 |
|
23067554 |
NPT1210 |
Individual Protein |
T-cell protein-tyrosine phosphatase |
Homo sapiens |
IC50 |
= |
20450 |
nM |
23067554 |
NPT178 |
Individual Protein |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50 |
= |
12740 |
nM |
23067554 |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
IC50 |
= |
50000 |
nM |
23489211 |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
IC50 |
= |
57543.99 |
nM |
23489211 |
NPT920 |
Individual Protein |
Alpha-synuclein |
Homo sapiens |
Potency |
|
5011.9 |
nM |
PubChem BioAssay data set |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
60.21 |
% |
23571415 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
6.612 |
% |
23571415 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
> |
1000 |
|
24900622 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
1.1 |
|
24900622 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
13.9 |
|
24900622 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
0.6 |
|
24900622 |
NPT2 |
Others |
Unspecified |
|
Ratio EC50 |
= |
39.1 |
|
24900622 |
NPT745 |
Individual Protein |
G-protein coupled bile acid receptor 1 |
Homo sapiens |
EC50 |
= |
730 |
nM |
24900622 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
56000 |
nM |
24332653 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23000 |
nM |
24332653 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5 |
% |
24461290 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9 |
ug/ml |
24461290 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
19417.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
61652.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21786.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54947.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1949.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27195 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
27306 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54726 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
60882 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
61130.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
9731.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
54482.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
61130.6 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
60882 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30637.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48972.2 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
54947.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15423.9 |
nM |
PubChem BioAssay data set |
NPT106 |
Individual Protein |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
Potency |
|
19417.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17158.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
24544.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
68589.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
68310.7 |
nM |
PubChem BioAssay data set |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Potency |
|
21192.3 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
68589.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
43646.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
19496.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17305.9 |
nM |
PubChem BioAssay data set |
NPT162 |
Individual Protein |
Heat shock protein beta-1 |
Homo sapiens |
Potency |
|
61403.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
24445.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
4347 |
nM |
PubChem BioAssay data set |
NPT162 |
Individual Protein |
Heat shock protein beta-1 |
Homo sapiens |
Potency |
|
61652.4 |
nM |
PubChem BioAssay data set |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48557.7 |
nM |
PubChem BioAssay data set |
NPT446 |
Individual Protein |
Rap guanine nucleotide exchange factor 3 |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Inhibition |
= |
82.3 |
% |
24775917 |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
IC50 |
= |
18.3 |
nM |
24775917 |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Inhibition |
= |
16.1 |
% |
24775917 |
NPT2615 |
Cell Line |
HEK-293T |
Homo sapiens |
Inhibition |
< |
5 |
% |
24775917 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Kd |
= |
330 |
nM |
24818857 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Kd |
= |
9520 |
nM |
24818857 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Kd |
= |
18870 |
nM |
24818857 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Activity |
= |
48 |
% |
24818857 |
NPT745 |
Individual Protein |
G-protein coupled bile acid receptor 1 |
Homo sapiens |
EC50 |
= |
680 |
nM |
25735208 |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
54726 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
6889.6 |
nM |
PubChem BioAssay data set |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
61652.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
61403.5 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
|
19496.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
38743 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
76645.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48774.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
707.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
7761.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30513.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
21875.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
48360.3 |
nM |
PubChem BioAssay data set |
NPT757 |
Organism |
Plasmodium falciparum 3D7 |
Plasmodium falciparum 3D7 |
IC50 |
= |
26900 |
nM |
26063305 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
98 |
% |
26063305 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
22 |
% |
26063305 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
Inhibition |
= |
100 |
% |
26063305 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
Inhibition |
= |
5 |
% |
26063305 |
NPT757 |
Organism |
Plasmodium falciparum 3D7 |
Plasmodium falciparum 3D7 |
Inhibition |
= |
100 |
% |
26063305 |
NPT757 |
Organism |
Plasmodium falciparum 3D7 |
Plasmodium falciparum 3D7 |
Inhibition |
= |
85 |
% |
26063305 |
NPT5655 |
Individual Protein |
CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,3-sialyltransferase 1 |
Homo sapiens |
IC50 |
= |
21000 |
nM |
10.1039/C4MD00086B |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
81100 |
nM |
25685308 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
173100 |
nM |
25685308 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
97400 |
nM |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
8.88 |
% |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
11.54 |
% |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
13.15 |
% |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
10.21 |
% |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
18.79 |
% |
25685308 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
21.89 |
% |
25685308 |
NPT5656 |
Protein-Protein Interaction |
Tumour suppressor protein p53/Mdm4 |
Homo sapiens |
Kd |
= |
15000 |
nM |
10.1039/C4MD00328D |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
EC50 |
> |
50000 |
nM |
26774929 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
IC50 |
= |
13600 |
nM |
26774929 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
EC50 |
= |
2140 |
nM |
26774929 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
IC50 |
= |
46700 |
nM |
26774929 |
NPT2 |
Others |
Unspecified |
|
LD50 |
= |
55.9 |
nM |
26774929 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Activity |
= |
6 |
% |
26774929 |