Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
13000.0 |
nM |
PMID[16854069] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
10000.0 |
nM |
PMID[16854069] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
Activity |
= |
80.0 |
% |
PMID[16854069] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
9500.0 |
nM |
PMID[16854069] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
18000.0 |
nM |
PMID[16854069] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
Survival |
= |
5.0 |
% |
PMID[16854069] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[17665890] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50 |
= |
900.0 |
nM |
PMID[17665890] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
IC50 |
= |
200.0 |
nM |
PMID[17665890] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
9000.0 |
nM |
PMID[18816110] |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
1300.0 |
nM |
PMID[19783149] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
5200.0 |
nM |
PMID[19783149] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
5400.0 |
nM |
PMID[19783149] |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
6200.0 |
nM |
PMID[19783149] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
7.0 |
% |
PMID[19994845] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
66.0 |
% |
PMID[19994845] |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[19994845] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[19994845] |
NPT3369 |
Individual Protein |
Interferon-induced, double-stranded RNA-activated protein kinase |
Homo sapiens |
IC50 |
= |
600.0 |
nM |
PMID[21632247] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[23398362] |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[23398362] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
16.0 |
% |
PMID[23398362] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
28.0 |
% |
PMID[23398362] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
60.0 |
% |
PMID[23398362] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[23398362] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
54.0 |
% |
PMID[23398362] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
38.0 |
% |
PMID[23398362] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
16.0 |
% |
PMID[23398362] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
19.0 |
% |
PMID[23398362] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[23398362] |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
31.0 |
% |
PMID[23398362] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
51.0 |
% |
PMID[23398362] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
17.0 |
% |
PMID[23398362] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
46.0 |
% |
PMID[23398362] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
37.0 |
% |
PMID[23398362] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[23398362] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
67.0 |
% |
PMID[23398362] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
35.0 |
% |
PMID[23398362] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
16.0 |
% |
PMID[23398362] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[23398362] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[23398362] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
25.0 |
% |
PMID[23398362] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
50.0 |
% |
PMID[23398362] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
26.0 |
% |
PMID[23398362] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
25.0 |
% |
PMID[23398362] |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
127.0 |
% |
PMID[23398362] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[23398362] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
33.0 |
% |
PMID[23398362] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
34.0 |
% |
PMID[23398362] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
48.0 |
% |
PMID[23398362] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[23398362] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[23398362] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
20.0 |
% |
PMID[23398362] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
69.0 |
% |
PMID[23398362] |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[23398362] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
49.0 |
% |
PMID[23398362] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[23398362] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[23398362] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[23398362] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
57.0 |
% |
PMID[23398362] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[23398362] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[23398362] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[23398362] |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
83.0 |
% |
PMID[23398362] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[23398362] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[23398362] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[23398362] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[23398362] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
26.0 |
% |
PMID[23398362] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
14.0 |
% |
PMID[23398362] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
52.0 |
% |
PMID[23398362] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[23398362] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[23398362] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
37.0 |
% |
PMID[23398362] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
34.0 |
% |
PMID[23398362] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[23398362] |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
72.0 |
% |
PMID[23398362] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
65.0 |
% |
PMID[23398362] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
35.0 |
% |
PMID[23398362] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
39.0 |
% |
PMID[23398362] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[23398362] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[23398362] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
33.0 |
% |
PMID[23398362] |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
35.0 |
% |
PMID[23398362] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
69.0 |
% |
PMID[23398362] |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[23398362] |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[23398362] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[23398362] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Residual Activity |
= |
54.0 |
% |
PMID[23398362] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
22.0 |
% |
PMID[23398362] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
45.0 |
% |
PMID[23398362] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
34.0 |
% |
PMID[23398362] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
25.0 |
% |
PMID[23398362] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[23398362] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[23398362] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[23398362] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[23398362] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[23398362] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
32.0 |
% |
PMID[23398362] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[23398362] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[23398362] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[23398362] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
59.0 |
% |
PMID[23398362] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
12.0 |
% |
PMID[23398362] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
17.0 |
% |
PMID[23398362] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
22.0 |
% |
PMID[23398362] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
19.0 |
% |
PMID[23398362] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[23398362] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[23398362] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
45.0 |
% |
PMID[23398362] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
15.0 |
% |
PMID[23398362] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
66.0 |
% |
PMID[23398362] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[23398362] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
28.0 |
% |
PMID[23398362] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
9.0 |
% |
PMID[23398362] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
141.0 |
% |
PMID[23398362] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[23398362] |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
69.0 |
% |
PMID[23398362] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
13.0 |
% |
PMID[23398362] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
33.0 |
% |
PMID[23398362] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
19.0 |
% |
PMID[23398362] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
33.0 |
% |
PMID[23398362] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[23398362] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
59.0 |
% |
PMID[23398362] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
58.0 |
% |
PMID[23398362] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[23398362] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
83.0 |
% |
PMID[23398362] |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
45.0 |
% |
PMID[23398362] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
11.0 |
% |
PMID[23398362] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
12.0 |
% |
PMID[23398362] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[23398362] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
15.0 |
% |
PMID[23398362] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
20.0 |
% |
PMID[23398362] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[23398362] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[23398362] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[23398362] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
72.0 |
% |
PMID[23398362] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
64.0 |
% |
PMID[23398362] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
27.0 |
% |
PMID[23398362] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
20.0 |
% |
PMID[23398362] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[23398362] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[23398362] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Residual Activity |
= |
65.0 |
% |
PMID[23398362] |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[23398362] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
-4.0 |
% |
PMID[23398362] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[23398362] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
59.0 |
% |
PMID[23398362] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
25.0 |
% |
PMID[23398362] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
16.0 |
% |
PMID[23398362] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[23398362] |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
49.0 |
% |
PMID[23398362] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[23398362] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
60.0 |
% |
PMID[23398362] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[23398362] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[23398362] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
23.0 |
% |
PMID[23398362] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
54.0 |
% |
PMID[23398362] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[23398362] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
59.0 |
% |
PMID[23398362] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[23398362] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
37.0 |
% |
PMID[23398362] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[23398362] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT4094 |
Individual Protein |
Serine/threonine-protein kinase WNK3 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[23398362] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
72.0 |
% |
PMID[23398362] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
48.0 |
% |
PMID[23398362] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[23398362] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[23398362] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[23398362] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
4.0 |
% |
PMID[23398362] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[23398362] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[23398362] |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[23398362] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[23398362] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[23398362] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[23398362] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Residual Activity |
= |
83.0 |
% |
PMID[23398362] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
17.0 |
% |
PMID[23398362] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
28.0 |
% |
PMID[23398362] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
72.0 |
% |
PMID[23398362] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
15.0 |
% |
PMID[23398362] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
38.0 |
% |
PMID[23398362] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[23398362] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[23398362] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[23398362] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[23398362] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
36.0 |
% |
PMID[23398362] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
38.0 |
% |
PMID[23398362] |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[23398362] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
13.0 |
% |
PMID[23398362] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
67.0 |
% |
PMID[23398362] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[23398362] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Residual Activity |
= |
30.0 |
% |
PMID[23398362] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Residual Activity |
= |
25.0 |
% |
PMID[23398362] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[23398362] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[23398362] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[23398362] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[23398362] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
39.0 |
% |
PMID[23398362] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[23398362] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
83.0 |
% |
PMID[23398362] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
37.0 |
% |
PMID[23398362] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[23398362] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[23398362] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
51.0 |
% |
PMID[23398362] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
61.0 |
% |
PMID[23398362] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[23398362] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[23398362] |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[23398362] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[23398362] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[23398362] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[23398362] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
13.0 |
% |
PMID[23398362] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
18.0 |
% |
PMID[23398362] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[23398362] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
58.0 |
% |
PMID[23398362] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
23.0 |
% |
PMID[23398362] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3454 |
Individual Protein |
PAS domain-containing serine/threonine-protein kinase |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[23398362] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[23398362] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[23398362] |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[23398362] |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[23398362] |
NPT3454 |
Individual Protein |
PAS domain-containing serine/threonine-protein kinase |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[23398362] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
30.0 |
% |
PMID[23398362] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
28.0 |
% |
PMID[23398362] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
14.0 |
% |
PMID[23398362] |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[23398362] |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[23398362] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[23398362] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[23398362] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
47.0 |
% |
PMID[23398362] |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[23398362] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
8.0 |
% |
PMID[23398362] |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Residual Activity |
= |
16.0 |
% |
PMID[23398362] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Residual Activity |
= |
36.0 |
% |
PMID[23398362] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Residual Activity |
= |
11.0 |
% |
PMID[23398362] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[23398362] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
67.0 |
% |
PMID[23398362] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[23398362] |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
15.0 |
% |
PMID[23398362] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[23398362] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
30.0 |
% |
PMID[23398362] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
29.0 |
% |
PMID[23398362] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[23398362] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[23398362] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[23398362] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[23398362] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[23398362] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[23398362] |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
64.0 |
% |
PMID[23398362] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[23398362] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[23398362] |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[23398362] |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
IC50 |
= |
2100.0 |
nM |
PMID[23336033] |
NPT5455 |
Individual Protein |
Casein kinase I isoform alpha |
Sus scrofa |
IC50 |
= |
1200.0 |
nM |
PMID[23336033] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[23336033] |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
IC50 |
= |
3400.0 |
nM |
PMID[23688559] |
NPT540 |
Individual Protein |
Bile acid receptor FXR |
Homo sapiens |
Inhibition |
= |
96.3 |
% |
PMID[23688559] |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
IC50 |
= |
2100.0 |
nM |
PMID[24530227] |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
Inhibition |
= |
32.4 |
% |
PMID[24697244] |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
Inhibition |
= |
38.0 |
% |
PMID[24697244] |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
1500.0 |
nM |
PMID[24697244] |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
EC50 |
> |
30000.0 |
nM |
PMID[24697244] |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[24697244] |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[24798019] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
IC50 |
= |
85.0 |
nM |
PMID[24798019] |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
IC50 |
= |
2100.0 |
nM |
PMID[24798019] |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
IC50 |
= |
52.0 |
nM |
PMID[24798019] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50 |
= |
1500.0 |
nM |
PMID[27689729] |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
5300.0 |
nM |
PMID[28743492] |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
<= |
30.0 |
% |
PMID[30234987] |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[14761195] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[14761195] |
NPT1572 |
Protein Family |
Glycogen synthase kinase-3 |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[14761195] |
NPT1572 |
Protein Family |
Glycogen synthase kinase-3 |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[16854069] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[16854069] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
320.0 |
nM |
PMID[16854069] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[18077363] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
83.0 |
nM |
PMID[18077363] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
300.0 |
nM |
PMID[18077363] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
320.0 |
nM |
PMID[18077363] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000.0 |
nM |
PMID[18077363] |
NPT2 |
Others |
Unspecified |
|
IC50 |
>= |
10000.0 |
nM |
PMID[18077363] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[18816110] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
83.0 |
nM |
PMID[18816110] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.0 |
nM |
PMID[18816110] |
NPT1572 |
Protein Family |
Glycogen synthase kinase-3 |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[18816110] |
NPT610 |
Others |
Molecular identity unknown |
|
FC |
= |
2.7 |
n.a. |
PMID[19282173] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
1900.0 |
nM |
PMID[19783149] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Inhibition |
= |
70.0 |
% |
PMID[19783149] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Activity |
= |
6.0 |
% |
PMID[19994845] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
8.0 |
% |
PMID[19994845] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Activity |
= |
21.0 |
% |
PMID[19994845] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Activity |
= |
29.0 |
% |
PMID[19994845] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
55.0 |
% |
PMID[19994845] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Activity |
= |
85.0 |
% |
PMID[19994845] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.0 |
nM |
PMID[19994845] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10.0 |
nM |
PMID[15559249] |
NPT1570 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[15559249] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1995.26 |
nM |
PMID[19734910] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3162.28 |
nM |
PMID[19734910] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3981.07 |
nM |
PMID[19734910] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
10000.0 |
nM |
PMID[19734910] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
1584.89 |
nM |
PMID[19734910] |
NPT486 |
Organism |
Toxoplasma gondii |
Toxoplasma gondii |
ID50 |
= |
0.51 |
uM |
PMID[18824607] |
NPT27 |
Others |
Unspecified |
|
TD50 |
= |
16.0 |
uM |
PMID[18824607] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
38.0 |
% |
PMID[23398362] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[23398362] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[23398362] |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
7.0 |
% |
PMID[23398362] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[23398362] |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[23398362] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[23398362] |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
6.0 |
% |
PMID[23398362] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[23398362] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
9.0 |
% |
PMID[23398362] |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
40.0 |
% |
PMID[23398362] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[23398362] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[23398362] |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
34.0 |
% |
PMID[23398362] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
0.0 |
% |
PMID[23398362] |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
13.0 |
% |
PMID[23398362] |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[23398362] |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
32.0 |
% |
PMID[23398362] |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[23398362] |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[23398362] |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
10.0 |
% |
PMID[23398362] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Residual Activity |
= |
54.0 |
% |
PMID[23398362] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Residual Activity |
= |
12.0 |
% |
PMID[23398362] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
37.0 |
% |
PMID[23398362] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[23398362] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[23398362] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[23398362] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[23398362] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[23398362] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[23398362] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[23398362] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[23398362] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[23398362] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[23398362] |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[23398362] |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[23398362] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[23398362] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[23398362] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[23398362] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[23398362] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[23398362] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[23398362] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[23398362] |
NPT84 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
Rattus norvegicus |
IC50 |
= |
1700.0 |
nM |
PMID[23336033] |
NPT19056 |
SINGLE PROTEIN |
Glycogen synthase kinase 3 beta |
Sus scrofa |
IC50 |
= |
5.0 |
nM |
PMID[23336033] |
NPT84 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
Rattus norvegicus |
IC50 |
= |
520.0 |
nM |
PMID[24530227] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1900.0 |
nM |
PMID[24530227] |
NPT22078 |
PROTEIN FAMILY |
Glycogen synthase kinase-3 |
Sus scrofa |
IC50 |
= |
5.0 |
nM |
PMID[24530227] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[24530227] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5.0 |
nM |
PMID[24697244] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
500.0 |
nM |
PMID[24697244] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
1600.0 |
nM |
PMID[24697244] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
> |
3000.0 |
nM |
PMID[24697244] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
200.0 |
nM |
PMID[24697244] |
NPT1572 |
Protein Family |
Glycogen synthase kinase-3 |
Homo sapiens |
IC50 |
= |
5.0 |
nM |
PMID[24798019] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1900.0 |
nM |
PMID[24798019] |
NPT19059 |
TISSUE |
Spiral organ of cochlea |
Mus musculus |
EC50 |
= |
570.0 |
nM |
PMID[30091915] |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
192.0 |
nM |
PMID[30091915] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
-2.77 |
% |
DOI[10.21203/rs.3.rs-23951/v1] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
IC50 |
= |
270.0 |
nM |
PMID[30234987] |
NPT3944 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E1 |
Homo sapiens |
IC50 |
= |
14.0 |
nM |
PMID[30234987] |
NPT4158 |
Protein Complex |
CDK2/Cyclin A |
Homo sapiens |
IC50 |
= |
69.0 |
nM |
PMID[30234987] |
NPT1560 |
Protein Complex |
Cyclin-dependent kinase 4/cyclin D1 |
Homo sapiens |
IC50 |
= |
527.0 |
nM |
PMID[30234987] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
IC50 |
= |
41.0 |
nM |
PMID[30234987] |
NPT24345 |
PROTEIN COMPLEX |
CDK7/Cyclin H/MNAT1 |
Homo sapiens |
IC50 |
= |
3500.0 |
nM |
PMID[30234987] |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
IC50 |
= |
450.0 |
nM |
PMID[30234987] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
9.52 |
% |
DOI[10.6019/CHEMBL4495564] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
14.47 |
% |
DOI[10.6019/CHEMBL4495564] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
9.37 |
% |
DOI[10.6019/CHEMBL4495565] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
21.31 |
% |
DOI[10.6019/CHEMBL4495565] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
IC50 |
> |
33000.0 |
nM |
DOI[10.6019/CHEMBL4495565] |
NPT22224 |
CELL-LINE |
Vero C1008 |
Chlorocebus sabaeus |
CC50 |
> |
33000.0 |
nM |
DOI[10.6019/CHEMBL4495565] |
NPT2 |
Others |
Unspecified |
|
FC |
= |
0.758 |
n.a. |
PMID[31147141] |
NPT2 |
Others |
Unspecified |
|
FC |
= |
1.388 |
n.a. |
PMID[31147141] |
NPT27843 |
CELL-LINE |
KCL-22 |
Homo sapiens |
Activity |
> |
50.0 |
% |
PMID[27726390] |