Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
41 |
% |
2769683 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.9 |
% |
15808480 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.9 |
% |
16500101 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.1 |
% |
16500101 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
134.8 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
136 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
115.5 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
124.1 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
116.3 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
126.4 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
113.1 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
105.6 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
119.8 |
mg/dl |
17249729 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18.7 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
24.5 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
15.9 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
29.2 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18.2 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
21.1 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
20.7 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
30 |
% |
17336063 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.9 |
% |
17095211 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.1 |
% |
17095211 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26.5 |
% |
17197179 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
23.5 |
% |
17197179 |
NPT1592 |
Individual Protein |
Dipeptidyl peptidase IV |
Homo sapiens |
IC50 |
= |
29000 |
nM |
18068977 |
NPT1592 |
Individual Protein |
Dipeptidyl peptidase IV |
Homo sapiens |
Inhibition |
= |
12.7 |
% |
18068977 |
NPT1592 |
Individual Protein |
Dipeptidyl peptidase IV |
Homo sapiens |
Inhibition |
= |
21.9 |
% |
18068977 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
20.5 |
% |
18353644 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
19.1 |
% |
18353644 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.9 |
% |
18353644 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
1 |
% |
19243175 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
48 |
% |
9214733 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-11 |
% |
18465847 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-22 |
% |
18465847 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
Inhibition |
= |
19.6 |
% |
18788725 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
20.9 |
% |
19303291 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
21.9 |
% |
19303291 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
27.2 |
% |
19282172 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
23.9 |
% |
19282172 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
263.2 |
mg/dl |
11858757 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
232.7 |
mg/dl |
11858757 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
38.9 |
ug |
11858757 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
5.4 |
ug |
11858757 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
23.5 |
% |
18947904 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26.5 |
% |
18947904 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-127.6 |
mg/dl |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
18.6 |
mg/dl |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
45.4 |
ug |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
4.1 |
ug |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-151.8 |
mg/dl |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
76.1 |
mg/dl |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
43.2 |
ug |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
4.5 |
ug |
10479309 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-132 |
mg/dl |
10075783 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
40.9 |
ug |
10075783 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
7.3 |
ug |
10075783 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
-160 |
mg/dl |
10075783 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26.4 |
% |
18952419 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
17.1 |
% |
18952419 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
18.6 |
% |
18952419 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
24.8 |
% |
18952419 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.9 |
% |
18436346 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.1 |
% |
18436346 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
20.2 |
% |
18436346 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
11.2 |
% |
18436346 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
31.2 |
% |
19362832 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26.9 |
% |
19362832 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
21.4 |
% |
19362832 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
-23.5 |
% |
19515563 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
-26.5 |
% |
19515563 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
11 |
% |
19261478 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
53 |
% |
19261478 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
0.53 |
% |
20022146 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
13.5 |
% |
20471838 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18 |
% |
20471838 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
20.2 |
% |
20471838 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
32 |
% |
20518543 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
42 |
% |
20797859 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
28 |
% |
20797859 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
29.8 |
% |
20797859 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
3.5 |
nM |
PubChem BioAssay data set |
NPT442 |
Individual Protein |
Ferritin light chain |
Equus caballus |
Potency |
= |
7943.3 |
nM |
PubChem BioAssay data set |
NPT839 |
Cell Line |
L6 |
Rattus norvegicus |
Activity |
= |
19.4 |
% |
21129962 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
27.2 |
% |
21129962 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
24.1 |
% |
21129962 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
16.12 |
umol/ml |
21215628 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
17.09 |
umol/ml |
21215628 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
16.97 |
umol/ml |
21215628 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
15.27 |
umol/ml |
21215628 |
NPT443 |
Individual Protein |
Histone acetyltransferase GCN5 |
Homo sapiens |
Potency |
|
281.8 |
nM |
PubChem BioAssay data set |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
11.2 |
% |
19500993 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
20.2 |
% |
19500993 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
19.1 |
% |
19500993 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
12.9 |
% |
19500993 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
33 |
% |
20663675 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
43 |
% |
20663675 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
14 |
% |
20663675 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
23 |
% |
20663675 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
EC50 |
= |
270 |
nM |
21856048 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
27 |
% |
22123321 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
15.1 |
umol/ml |
22283497 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
6.3 |
|
22459208 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
41.4 |
% |
22459208 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
67.6 |
% |
22459208 |
NPT1540 |
Individual Protein |
Solute carrier family 22 member 2 |
Homo sapiens |
IC50 |
= |
1700000 |
nM |
12240953 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
IC50 |
= |
2010000 |
nM |
12240953 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
33.2 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
5080.7 |
nM |
PubChem BioAssay data set |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
37 |
mg/dl |
22708876 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
0.8 |
% |
22708876 |
NPT622 |
Individual Protein |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
Inhibition |
= |
-4.5 |
% |
22541068 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
19.6 |
% |
22541068 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
-3.3 |
% |
22541068 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
6.2 |
% |
22524508 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
4.2 |
% |
22524508 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
5.9 |
% |
22524508 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.4 |
% |
22524508 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
24.3 |
% |
22524508 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
22.1 |
% |
22524508 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
3.7 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
46.7 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
44.4 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
29.3 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
66 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
10.3 |
% |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
9.62 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
50 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
48.8 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
13.6 |
ug/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
198.3 |
ug/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
0.28 |
umol/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
0.15 |
umol/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
1.99 |
umol/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
89 |
U/L |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
39 |
U/L |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
1.6 |
umol/ml |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
12.8 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.7 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18.1 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
2.2 |
% |
23025244 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
5.2 |
% |
23025244 |
NPT520 |
Cell Line |
3T3-L1 |
Mus musculus |
Activity |
= |
360.8 |
ug/ml |
23025244 |
NPT520 |
Cell Line |
3T3-L1 |
Mus musculus |
Activity |
= |
125.8 |
ug/ml |
23025244 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.00E-05 |
nM |
23067551 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
14.47 |
nM |
23067551 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
20.72 |
nM |
23067551 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
16.98 |
nM |
23067551 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
2.11 |
nM |
23067551 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
19.1 |
% |
22341243 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18.9 |
% |
22341243 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
9.98 |
umol/ml |
10.1007/s00044-011-9765-3 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
25 |
% |
10.1007/s00044-010-9387-1 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
-26.7 |
% |
10.1007/s00044-010-9387-1 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
24.9 |
% |
10.1007/s00044-010-9401-7 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26 |
% |
10.1007/s00044-010-9401-7 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
26.5 |
% |
10.1007/s00044-007-9043-6 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
23.6 |
% |
10.1007/s00044-007-9043-6 |
NPT5334 |
Individual Protein |
Protein-tyrosine phosphatase 1B |
Rattus norvegicus |
Inhibition |
= |
30.2 |
% |
10.1007/s00044-012-0165-0 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
17 |
% |
10.1007/s00044-012-0007-0 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
18 |
% |
10.1007/s00044-012-0007-0 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
13 |
% |
10.1007/s00044-012-0007-0 |
NPT5334 |
Individual Protein |
Protein-tyrosine phosphatase 1B |
Rattus norvegicus |
Inhibition |
= |
30.2 |
% |
10.1007/s00044-012-0007-0 |
NPT5334 |
Individual Protein |
Protein-tyrosine phosphatase 1B |
Rattus norvegicus |
Inhibition |
= |
30.2 |
% |
10.1007/s00044-013-0528-1 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
2.25 |
umol/ml |
10.1007/s00044-012-0215-7 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Ratio |
= |
3.923 |
|
10.1007/s00044-012-0215-7 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
29.9 |
% |
23218712 |
NPT4037 |
Individual Protein |
Multidrug and toxin extrusion protein 1 |
Homo sapiens |
IC50 |
= |
250000 |
nM |
23241029 |
NPT2268 |
Cell Line |
DOK |
Homo sapiens |
IC50 |
= |
4251537.66 |
nM |
10.6019/CHEMBL1201861 |
NPT1899 |
Cell Line |
DSH1 |
Homo sapiens |
IC50 |
= |
32808699.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1184 |
Cell Line |
Daoy |
Homo sapiens |
IC50 |
= |
43984738.48 |
nM |
10.6019/CHEMBL1201861 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
838320.93 |
nM |
10.6019/CHEMBL1201861 |
NPT1900 |
Cell Line |
DU-4475 |
Homo sapiens |
IC50 |
= |
3835948.46 |
nM |
10.6019/CHEMBL1201861 |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
IC50 |
= |
52114369.72 |
nM |
10.6019/CHEMBL1201861 |
NPT1901 |
Cell Line |
EM-2 |
Homo sapiens |
IC50 |
= |
460688321 |
nM |
10.6019/CHEMBL1201861 |
NPT2269 |
Cell Line |
EPLC-272H |
Homo sapiens |
IC50 |
= |
50826746.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1905 |
Cell Line |
ES4 |
Homo sapiens |
IC50 |
= |
82857786.37 |
nM |
10.6019/CHEMBL1201861 |
NPT1903 |
Cell Line |
ES5 |
Homo sapiens |
IC50 |
= |
14689188.12 |
nM |
10.6019/CHEMBL1201861 |
NPT1902 |
Cell Line |
ES1 |
Homo sapiens |
IC50 |
= |
24548376.48 |
nM |
10.6019/CHEMBL1201861 |
NPT1904 |
Cell Line |
ES3 |
Homo sapiens |
IC50 |
= |
16943202.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2270 |
Cell Line |
Detroit562 |
Homo sapiens |
IC50 |
= |
16478569.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2271 |
Cell Line |
DoTc2-4510 |
Homo sapiens |
IC50 |
= |
31722928.66 |
nM |
10.6019/CHEMBL1201861 |
NPT1908 |
Cell Line |
EC-GI-10 |
Homo sapiens |
IC50 |
= |
26424265.11 |
nM |
10.6019/CHEMBL1201861 |
NPT3465 |
Cell Line |
ECC10 |
Homo sapiens |
IC50 |
= |
2283299.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2272 |
Cell Line |
EFM-19 |
Homo sapiens |
IC50 |
= |
169245398 |
nM |
10.6019/CHEMBL1201861 |
NPT2273 |
Cell Line |
EFO-21 |
Homo sapiens |
IC50 |
= |
55230300.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2274 |
Cell Line |
EFO-27 |
Homo sapiens |
IC50 |
= |
27599391.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2275 |
Cell Line |
EGI-1 |
Homo sapiens |
IC50 |
= |
865126484.4 |
nM |
10.6019/CHEMBL1201861 |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
IC50 |
= |
26205877.59 |
nM |
10.6019/CHEMBL1201861 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
4535624.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2276 |
Cell Line |
A673 |
Homo sapiens |
IC50 |
= |
19160918.71 |
nM |
10.6019/CHEMBL1201861 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
84402727.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2277 |
Cell Line |
C-33-A |
Homo sapiens |
IC50 |
= |
9397293.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2278 |
Cell Line |
COLO-741 |
Homo sapiens |
IC50 |
= |
379329310.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2279 |
Cell Line |
COLO-792 |
Homo sapiens |
IC50 |
= |
7513968.24 |
nM |
10.6019/CHEMBL1201861 |
NPT1913 |
Cell Line |
DJM-1 |
Homo sapiens |
IC50 |
= |
10237390.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2280 |
Cell Line |
A704 |
Homo sapiens |
IC50 |
= |
850354839.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2281 |
Cell Line |
ABC-1 |
Homo sapiens |
IC50 |
= |
30969681.85 |
nM |
10.6019/CHEMBL1201861 |
NPT1911 |
Cell Line |
C2BBe1 |
Homo sapiens |
IC50 |
= |
11823223.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2282 |
Cell Line |
C32 |
Homo sapiens |
IC50 |
= |
43579101.89 |
nM |
10.6019/CHEMBL1201861 |
NPT1912 |
Cell Line |
COLO-800 |
Homo sapiens |
IC50 |
= |
121585865 |
nM |
10.6019/CHEMBL1201861 |
NPT1914 |
Cell Line |
COLO-824 |
Homo sapiens |
IC50 |
= |
21550450.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2283 |
Cell Line |
DK-MG |
Homo sapiens |
IC50 |
= |
860035546.1 |
nM |
10.6019/CHEMBL1201861 |
NPT576 |
Cell Line |
DMS-114 |
Homo sapiens |
IC50 |
= |
90056632.37 |
nM |
10.6019/CHEMBL1201861 |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
IC50 |
= |
47613899.31 |
nM |
10.6019/CHEMBL1201861 |
NPT1916 |
Cell Line |
ACN |
Homo sapiens |
IC50 |
= |
122320019.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2284 |
Cell Line |
C3A |
Homo sapiens |
IC50 |
= |
11278460.1 |
nM |
10.6019/CHEMBL1201861 |
NPT1452 |
Cell Line |
C8166 |
Homo sapiens |
IC50 |
= |
177834389.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1915 |
Cell Line |
COLO-829 |
Homo sapiens |
IC50 |
= |
22432206.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2285 |
Cell Line |
COR-L105 |
Homo sapiens |
IC50 |
= |
24804590.11 |
nM |
10.6019/CHEMBL1201861 |
NPT1918 |
Cell Line |
DMS-79 |
Homo sapiens |
IC50 |
= |
5970482.36 |
nM |
10.6019/CHEMBL1201861 |
NPT1919 |
Cell Line |
DOHH-2 |
Homo sapiens |
IC50 |
= |
7643409.1 |
nM |
10.6019/CHEMBL1201861 |
NPT196 |
Cell Line |
AGS |
Homo sapiens |
IC50 |
= |
15736608.05 |
nM |
10.6019/CHEMBL1201861 |
NPT1920 |
Cell Line |
ALL-PO |
Homo sapiens |
IC50 |
= |
2900904.89 |
nM |
10.6019/CHEMBL1201861 |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
IC50 |
= |
34629146.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2286 |
Cell Line |
CAL-120 |
Homo sapiens |
IC50 |
= |
115735303.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2287 |
Cell Line |
COR-L23 |
Homo sapiens |
IC50 |
= |
23550186.06 |
nM |
10.6019/CHEMBL1201861 |
NPT1922 |
Cell Line |
COR-L88 |
Homo sapiens |
IC50 |
= |
6381318.4 |
nM |
10.6019/CHEMBL1201861 |
NPT572 |
Cell Line |
DMS-273 |
Homo sapiens |
IC50 |
= |
13605290.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1924 |
Cell Line |
AM-38 |
Homo sapiens |
IC50 |
= |
58613187.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2288 |
Cell Line |
AN3-CA |
Homo sapiens |
IC50 |
= |
63308760.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2289 |
Cell Line |
CAL-12T |
Homo sapiens |
IC50 |
= |
237110605.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2290 |
Cell Line |
CAL-27 |
Homo sapiens |
IC50 |
= |
46925194.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2291 |
Cell Line |
CP50-MEL-B |
Homo sapiens |
IC50 |
= |
62097934.1 |
nM |
10.6019/CHEMBL1201861 |
NPT1926 |
Cell Line |
CP66-MEL |
Homo sapiens |
IC50 |
= |
115661141.4 |
nM |
10.6019/CHEMBL1201861 |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
17964484.42 |
nM |
10.6019/CHEMBL1201861 |
NPT1928 |
Cell Line |
ATN-1 |
Homo sapiens |
IC50 |
= |
8646673.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2292 |
Cell Line |
CAL-33 |
Homo sapiens |
IC50 |
= |
43138364.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2293 |
Cell Line |
CAL-39 |
Homo sapiens |
IC50 |
= |
35449236.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1930 |
Cell Line |
CTB-1 |
Homo sapiens |
IC50 |
= |
23007280.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2294 |
Cell Line |
23132-87 |
Homo sapiens |
IC50 |
= |
11226765.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2295 |
Cell Line |
5637 |
Homo sapiens |
IC50 |
= |
5299225.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2296 |
Cell Line |
AU565 |
Homo sapiens |
IC50 |
= |
329122401 |
nM |
10.6019/CHEMBL1201861 |
NPT2297 |
Cell Line |
ASPC1 |
Homo sapiens |
IC50 |
= |
5371642.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2298 |
Cell Line |
BALL-1 |
Homo sapiens |
IC50 |
= |
22981021.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2299 |
Cell Line |
CAL-51 |
Homo sapiens |
IC50 |
= |
163822368.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2300 |
Cell Line |
CAL-54 |
Homo sapiens |
IC50 |
= |
3357983.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2301 |
Cell Line |
CAL-62 |
Homo sapiens |
IC50 |
= |
58560694.02 |
nM |
10.6019/CHEMBL1201861 |
NPT1932 |
Cell Line |
CTV-1 |
Homo sapiens |
IC50 |
= |
1970607.2 |
nM |
10.6019/CHEMBL1201861 |
NPT1933 |
Cell Line |
CW-2 |
Homo sapiens |
IC50 |
= |
4116328.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2302 |
Cell Line |
639-V |
Homo sapiens |
IC50 |
= |
65681461.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2303 |
Cell Line |
647-V |
Homo sapiens |
IC50 |
= |
26686870.98 |
nM |
10.6019/CHEMBL1201861 |
NPT1931 |
Cell Line |
BB30-HNC |
Homo sapiens |
IC50 |
= |
10843618.18 |
nM |
10.6019/CHEMBL1201861 |
NPT1934 |
Cell Line |
BB49-HNC |
Homo sapiens |
IC50 |
= |
27410077.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2304 |
Cell Line |
CAL-72 |
Homo sapiens |
IC50 |
= |
6273031.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2305 |
Cell Line |
CAL-85-1 |
Homo sapiens |
IC50 |
= |
555767322 |
nM |
10.6019/CHEMBL1201861 |
NPT2306 |
Cell Line |
Ca-Ski |
Homo sapiens |
IC50 |
= |
93305468.77 |
nM |
10.6019/CHEMBL1201861 |
NPT1031 |
Cell Line |
Ca9-22 |
Homo sapiens |
IC50 |
= |
7952137.19 |
nM |
10.6019/CHEMBL1201861 |
NPT1094 |
Cell Line |
697 |
Homo sapiens |
IC50 |
= |
6503280.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2307 |
Cell Line |
769-P |
Homo sapiens |
IC50 |
= |
6918899.47 |
nM |
10.6019/CHEMBL1201861 |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
IC50 |
= |
48968132.09 |
nM |
10.6019/CHEMBL1201861 |
NPT1935 |
Cell Line |
BB65-RCC |
Homo sapiens |
IC50 |
= |
112300321.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2308 |
Cell Line |
CAMA-1 |
Homo sapiens |
IC50 |
= |
11038936.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2309 |
Cell Line |
CAPAN-1 |
Homo sapiens |
IC50 |
= |
21285917.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2310 |
Cell Line |
CaR-1 |
Homo sapiens |
IC50 |
= |
47892586.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2311 |
Cell Line |
Calu-3 |
Homo sapiens |
IC50 |
= |
21732280.18 |
nM |
10.6019/CHEMBL1201861 |
NPT1939 |
Cell Line |
8-MG-BA |
Homo sapiens |
IC50 |
= |
20232125.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2312 |
Cell Line |
8305C |
Homo sapiens |
IC50 |
= |
201676861.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2313 |
Cell Line |
BCPAP |
Homo sapiens |
IC50 |
= |
28675804.57 |
nM |
10.6019/CHEMBL1201861 |
NPT1937 |
Cell Line |
CAS-1 |
Homo sapiens |
IC50 |
= |
207230297.1 |
nM |
10.6019/CHEMBL1201861 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
2720842.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1938 |
Cell Line |
Calu-6 |
Homo sapiens |
IC50 |
= |
15241953.45 |
nM |
10.6019/CHEMBL1201861 |
NPT1313 |
Cell Line |
Capan-2 |
Homo sapiens |
IC50 |
= |
214350327.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1215 |
Cell Line |
8505C |
Homo sapiens |
IC50 |
= |
15366314.15 |
nM |
10.6019/CHEMBL1201861 |
NPT1941 |
Cell Line |
A101D |
Homo sapiens |
IC50 |
= |
22504959.81 |
nM |
10.6019/CHEMBL1201861 |
NPT1940 |
Cell Line |
BE-13 |
Homo sapiens |
IC50 |
= |
17990569.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2314 |
Cell Line |
BEN |
Homo sapiens |
IC50 |
= |
15408907.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2315 |
Cell Line |
BFTC-905 |
Homo sapiens |
IC50 |
= |
11741736.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2316 |
Cell Line |
CFPAC-1 |
Homo sapiens |
IC50 |
= |
37288378.92 |
nM |
10.6019/CHEMBL1201861 |
NPT1943 |
Cell Line |
CGTH-W-1 |
Homo sapiens |
IC50 |
= |
25819982.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2317 |
Cell Line |
ChaGo-K-1 |
Homo sapiens |
IC50 |
= |
8885739.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1944 |
Cell Line |
D-247MG |
Homo sapiens |
IC50 |
= |
27260035.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2318 |
Cell Line |
A172 |
Homo sapiens |
IC50 |
= |
17472403.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2319 |
Cell Line |
A204 |
Homo sapiens |
IC50 |
= |
101983875.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1383 |
Cell Line |
A2058 |
Homo sapiens |
IC50 |
= |
65867274.25 |
nM |
10.6019/CHEMBL1201861 |
NPT2320 |
Cell Line |
BFTC-909 |
Homo sapiens |
IC50 |
= |
54922039.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2321 |
Cell Line |
BHT-101 |
Homo sapiens |
IC50 |
= |
6423818.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2322 |
Cell Line |
CHL-1 |
Homo sapiens |
IC50 |
= |
19484800.91 |
nM |
10.6019/CHEMBL1201861 |
NPT1946 |
Cell Line |
D-263MG |
Homo sapiens |
IC50 |
= |
24237395.79 |
nM |
10.6019/CHEMBL1201861 |
NPT1947 |
Cell Line |
D283 Med |
|
IC50 |
= |
34651489.82 |
nM |
10.6019/CHEMBL1201861 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
4876699.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2323 |
Cell Line |
BHY |
Homo sapiens |
IC50 |
= |
50666691.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2324 |
Cell Line |
CHP-212 |
Homo sapiens |
IC50 |
= |
9628695.18 |
nM |
10.6019/CHEMBL1201861 |
NPT1953 |
Cell Line |
D-336MG |
Homo sapiens |
IC50 |
= |
277930121.6 |
nM |
10.6019/CHEMBL1201861 |
NPT1954 |
Cell Line |
D-392MG |
Homo sapiens |
IC50 |
= |
41753768.93 |
nM |
10.6019/CHEMBL1201861 |
NPT1955 |
Cell Line |
A3-KAW |
Homo sapiens |
IC50 |
= |
61798168.06 |
nM |
10.6019/CHEMBL1201861 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
IC50 |
= |
379604044.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2325 |
Cell Line |
BPH-1 |
Homo sapiens |
IC50 |
= |
113545168.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2326 |
Cell Line |
BT-20 |
Homo sapiens |
IC50 |
= |
15263185.02 |
nM |
10.6019/CHEMBL1201861 |
NPT1952 |
Cell Line |
COLO-320-HSR |
Homo sapiens |
IC50 |
= |
83624515.19 |
nM |
10.6019/CHEMBL1201861 |
NPT1956 |
Cell Line |
COLO-668 |
Homo sapiens |
IC50 |
= |
60858331.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2327 |
Cell Line |
D-423MG |
Homo sapiens |
IC50 |
= |
3262010.49 |
nM |
10.6019/CHEMBL1201861 |
NPT1957 |
Cell Line |
D-502MG |
Homo sapiens |
IC50 |
= |
39151616.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1958 |
Cell Line |
A388 |
Homo sapiens |
IC50 |
= |
44196947.3 |
nM |
10.6019/CHEMBL1201861 |
NPT1959 |
Cell Line |
A4-Fuk |
Homo sapiens |
IC50 |
= |
39180717.33 |
nM |
10.6019/CHEMBL1201861 |
NPT845 |
Cell Line |
BT-474 |
Homo sapiens |
IC50 |
= |
39920529.72 |
nM |
10.6019/CHEMBL1201861 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
4195072.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2328 |
Cell Line |
COLO-678 |
Homo sapiens |
IC50 |
= |
60479999.34 |
nM |
10.6019/CHEMBL1201861 |
NPT2329 |
Cell Line |
COLO-679 |
Homo sapiens |
IC50 |
= |
62032207.19 |
nM |
10.6019/CHEMBL1201861 |
NPT1961 |
Cell Line |
D-542MG |
Homo sapiens |
IC50 |
= |
1319594433 |
nM |
10.6019/CHEMBL1201861 |
NPT2330 |
Cell Line |
D-566MG |
Homo sapiens |
IC50 |
= |
10796993.56 |
nM |
10.6019/CHEMBL1201861 |
NPT1962 |
Cell Line |
DB |
Homo sapiens |
IC50 |
= |
34036508.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2331 |
Cell Line |
A-427 |
Homo sapiens |
IC50 |
= |
7174454.43 |
nM |
10.6019/CHEMBL1201861 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
24212976.8 |
nM |
10.6019/CHEMBL1201861 |
NPT1960 |
Cell Line |
BV-173 |
Homo sapiens |
IC50 |
= |
3017500.14 |
nM |
10.6019/CHEMBL1201861 |
NPT1963 |
Cell Line |
Becker |
Homo sapiens |
IC50 |
= |
37314452.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2332 |
Cell Line |
COLO-680N |
Homo sapiens |
IC50 |
= |
600391367.1 |
nM |
10.6019/CHEMBL1201861 |
NPT1964 |
Cell Line |
COLO-684 |
Homo sapiens |
IC50 |
= |
22143715.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2333 |
Cell Line |
DBTRG-05MG |
Homo sapiens |
IC50 |
= |
7269007.2 |
nM |
10.6019/CHEMBL1201861 |
NPT1965 |
Cell Line |
DEL |
Homo sapiens |
IC50 |
= |
255356528.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2334 |
Cell Line |
NCI-H1793 |
Homo sapiens |
IC50 |
= |
18472991.03 |
nM |
10.6019/CHEMBL1201861 |
NPT1966 |
Cell Line |
NCI-H1838 |
Homo sapiens |
IC50 |
= |
35793443.03 |
nM |
10.6019/CHEMBL1201861 |
NPT1967 |
Cell Line |
NCI-H526 |
Homo sapiens |
IC50 |
= |
16089384.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2335 |
Cell Line |
NCI-H596 |
|
IC50 |
= |
108414269.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2336 |
Cell Line |
OE19 |
Homo sapiens |
IC50 |
= |
33393381.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
423198239.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1091 |
Cell Line |
RPMI-7951 |
Homo sapiens |
IC50 |
= |
9101722.86 |
nM |
10.6019/CHEMBL1201861 |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
IC50 |
= |
128564113.9 |
nM |
10.6019/CHEMBL1201861 |
NPT311 |
Cell Line |
SK-LU-1 |
Homo sapiens |
IC50 |
= |
33462878.54 |
nM |
10.6019/CHEMBL1201861 |
NPT926 |
Cell Line |
SK-MEL-1 |
Homo sapiens |
IC50 |
= |
11797512.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1312 |
Cell Line |
SW1990 |
Homo sapiens |
IC50 |
= |
846606258.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2338 |
Cell Line |
SW48 |
Homo sapiens |
IC50 |
= |
41073236.16 |
nM |
10.6019/CHEMBL1201861 |
NPT2339 |
Cell Line |
TGBC24TKB |
Homo sapiens |
IC50 |
= |
265423515.3 |
nM |
10.6019/CHEMBL1201861 |
NPT1971 |
Cell Line |
GI-1 |
Homo sapiens |
IC50 |
= |
46620377.04 |
nM |
10.6019/CHEMBL1201861 |
NPT1972 |
Cell Line |
GI-ME-N |
Homo sapiens |
IC50 |
= |
34633995.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2204 |
Cell Line |
HH |
Homo sapiens |
IC50 |
= |
9630486.28 |
nM |
10.6019/CHEMBL1201861 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
95556693.54 |
nM |
10.6019/CHEMBL1201861 |
NPT1973 |
Cell Line |
IST-SL1 |
Homo sapiens |
IC50 |
= |
203852098 |
nM |
10.6019/CHEMBL1201861 |
NPT1975 |
Cell Line |
KS-1 |
Homo sapiens |
IC50 |
= |
54179506.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2340 |
Cell Line |
KU-19-19 |
Homo sapiens |
IC50 |
= |
9612820.93 |
nM |
10.6019/CHEMBL1201861 |
NPT1976 |
Cell Line |
LNCaP-Clone-FGC |
Homo sapiens |
IC50 |
= |
5234926.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2209 |
Cell Line |
MFH-ino |
Homo sapiens |
IC50 |
= |
824331472.1 |
nM |
10.6019/CHEMBL1201861 |
NPT1978 |
Cell Line |
MFM-223 |
Homo sapiens |
IC50 |
= |
77264432.05 |
nM |
10.6019/CHEMBL1201861 |
NPT1979 |
Cell Line |
NB13 |
Homo sapiens |
IC50 |
= |
867743983.3 |
nM |
10.6019/CHEMBL1201861 |
NPT1980 |
Cell Line |
NB14 |
Homo sapiens |
IC50 |
= |
258999393.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2341 |
Cell Line |
NCI-H1975 |
Homo sapiens |
IC50 |
= |
11679261.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2342 |
Cell Line |
NCI-H630 |
Homo sapiens |
IC50 |
= |
33341628.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2343 |
Cell Line |
NCI-H650 |
Homo sapiens |
IC50 |
= |
366269250.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1968 |
Cell Line |
OMC-1 |
Homo sapiens |
IC50 |
= |
16535783.36 |
nM |
10.6019/CHEMBL1201861 |
NPT1984 |
Cell Line |
ONS-76 |
Homo sapiens |
IC50 |
= |
68537615.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1987 |
Cell Line |
RPMI-8866 |
Homo sapiens |
IC50 |
= |
9028477.25 |
nM |
10.6019/CHEMBL1201861 |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
IC50 |
= |
20109588.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2344 |
Cell Line |
SK-MEL-24 |
Homo sapiens |
IC50 |
= |
35414619.71 |
nM |
10.6019/CHEMBL1201861 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
IC50 |
= |
296888521.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2345 |
Cell Line |
SW626 |
Homo sapiens |
IC50 |
= |
57775552.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2346 |
Cell Line |
TI-73 |
Homo sapiens |
IC50 |
= |
13592521.08 |
nM |
10.6019/CHEMBL1201861 |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
IC50 |
= |
28643075.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2347 |
Cell Line |
GMS-10 |
Homo sapiens |
IC50 |
= |
64902083.15 |
nM |
10.6019/CHEMBL1201861 |
NPT1989 |
Cell Line |
GOTO |
Homo sapiens |
IC50 |
= |
34457535.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2348 |
Cell Line |
HLE |
Homo sapiens |
IC50 |
= |
9860666.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2349 |
Cell Line |
HMV-2 cell line |
|
IC50 |
= |
191793010.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2350 |
Cell Line |
HN |
Homo sapiens |
IC50 |
= |
69206287.69 |
nM |
10.6019/CHEMBL1201861 |
NPT1990 |
Cell Line |
J-RT3-T3-5 |
Homo sapiens |
IC50 |
= |
28901506.48 |
nM |
10.6019/CHEMBL1201861 |
NPT1505 |
Cell Line |
J82 |
Homo sapiens |
IC50 |
= |
12903501.66 |
nM |
10.6019/CHEMBL1201861 |
NPT1991 |
Cell Line |
KU812 cell line |
|
IC50 |
= |
1056639.64 |
nM |
10.6019/CHEMBL1201861 |
NPT1992 |
Cell Line |
KURAMOCHI |
Homo sapiens |
IC50 |
= |
33958857.59 |
nM |
10.6019/CHEMBL1201861 |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
IC50 |
= |
10715301.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2351 |
Cell Line |
MG-63 |
Homo sapiens |
IC50 |
= |
14005914.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2352 |
Cell Line |
MHH-ES-1 |
Homo sapiens |
IC50 |
= |
75350210.67 |
nM |
10.6019/CHEMBL1201861 |
NPT1995 |
Cell Line |
NB17 |
Homo sapiens |
IC50 |
= |
38259761.14 |
nM |
10.6019/CHEMBL1201861 |
NPT1996 |
Cell Line |
NB5 |
Homo sapiens |
IC50 |
= |
28526050.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2353 |
Cell Line |
NCI-H1993 |
Homo sapiens |
IC50 |
= |
906328407.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2354 |
Cell Line |
NCI-H2009 |
Homo sapiens |
IC50 |
= |
442184723.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2355 |
Cell Line |
NCI-H2029 |
Homo sapiens |
IC50 |
= |
14762330.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2356 |
Cell Line |
NCI-H661 |
Homo sapiens |
IC50 |
= |
4558454.87 |
nM |
10.6019/CHEMBL1201861 |
NPT1396 |
Cell Line |
NCI-H69 |
Homo sapiens |
IC50 |
= |
8559722.07 |
nM |
10.6019/CHEMBL1201861 |
NPT1997 |
Cell Line |
OS-RC-2 |
Homo sapiens |
IC50 |
= |
12980467.41 |
nM |
10.6019/CHEMBL1201861 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
IC50 |
= |
17646628.07 |
nM |
10.6019/CHEMBL1201861 |
NPT1998 |
Cell Line |
RS4-11 |
Homo sapiens |
IC50 |
= |
48198153.97 |
nM |
10.6019/CHEMBL1201861 |
NPT2357 |
Cell Line |
RT-112 |
Homo sapiens |
IC50 |
= |
66554803.5 |
nM |
10.6019/CHEMBL1201861 |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
IC50 |
= |
136771372.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2358 |
Cell Line |
SK-MEL3 |
Homo sapiens |
IC50 |
= |
116470464.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2359 |
Cell Line |
SK-MEL-30 |
Homo sapiens |
IC50 |
= |
90805578.51 |
nM |
10.6019/CHEMBL1201861 |
NPT1988 |
Cell Line |
SW684 |
Homo sapiens |
IC50 |
= |
102887763.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2360 |
Cell Line |
SW756 |
Homo sapiens |
IC50 |
= |
63637551.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2361 |
Cell Line |
SW780 |
Homo sapiens |
IC50 |
= |
12398329.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2362 |
Cell Line |
TYK-nu |
Homo sapiens |
IC50 |
= |
16532856.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2363 |
Cell Line |
U-118-MG |
Homo sapiens |
IC50 |
= |
161578116.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2364 |
Cell Line |
GP5d |
Homo sapiens |
IC50 |
= |
59764074.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2000 |
Cell Line |
GR-ST |
Homo sapiens |
IC50 |
= |
22313719.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2365 |
Cell Line |
HO-1-N-1 |
Homo sapiens |
IC50 |
= |
13189416.41 |
nM |
10.6019/CHEMBL1201861 |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
IC50 |
= |
416130004 |
nM |
10.6019/CHEMBL1201861 |
NPT2001 |
Cell Line |
JAR |
Homo sapiens |
IC50 |
= |
9025525.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2366 |
Cell Line |
JEG-3 |
Homo sapiens |
IC50 |
= |
283498185 |
nM |
10.6019/CHEMBL1201861 |
NPT2002 |
Cell Line |
KY821 |
Homo sapiens |
IC50 |
= |
1531549.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2367 |
Cell Line |
KYSE-140 |
Homo sapiens |
IC50 |
= |
95851461.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2003 |
Cell Line |
LS-1034 |
Homo sapiens |
IC50 |
= |
52016486.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2004 |
Cell Line |
LS-123 |
Homo sapiens |
IC50 |
= |
17276059.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2005 |
Cell Line |
MHH-NB-11 |
Homo sapiens |
IC50 |
= |
320681917.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2007 |
Cell Line |
NB6 |
Homo sapiens |
IC50 |
= |
431889479.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2368 |
Cell Line |
NCI-H2030 |
Homo sapiens |
IC50 |
= |
704486184.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2369 |
Cell Line |
NCI-H2052 |
Homo sapiens |
IC50 |
= |
374419086.1 |
nM |
10.6019/CHEMBL1201861 |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
IC50 |
= |
4431821.71 |
nM |
10.6019/CHEMBL1201861 |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
IC50 |
= |
31560859.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2370 |
Cell Line |
RVH-421 |
Homo sapiens |
IC50 |
= |
115930482.3 |
nM |
10.6019/CHEMBL1201861 |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
IC50 |
= |
54145275.49 |
nM |
10.6019/CHEMBL1201861 |
NPT1506 |
Cell Line |
SK-MES-1 |
Homo sapiens |
IC50 |
= |
64080090.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2371 |
Cell Line |
SW837 |
Homo sapiens |
IC50 |
= |
37546933.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2014 |
Cell Line |
SW872 |
Homo sapiens |
IC50 |
= |
149857331.9 |
nM |
10.6019/CHEMBL1201861 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
IC50 |
= |
28782734.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2015 |
Cell Line |
U-266 |
Homo sapiens |
IC50 |
= |
25912972.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2016 |
Cell Line |
ES6 |
Homo sapiens |
IC50 |
= |
34430325.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2017 |
Cell Line |
ES7 |
Homo sapiens |
IC50 |
= |
20627615.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2018 |
Cell Line |
GT3TKB |
Homo sapiens |
IC50 |
= |
56191062.89 |
nM |
10.6019/CHEMBL1201861 |
NPT2372 |
Cell Line |
H-EMC-SS |
Homo sapiens |
IC50 |
= |
25518552.1 |
nM |
10.6019/CHEMBL1201861 |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
IC50 |
= |
863790032.2 |
nM |
10.6019/CHEMBL1201861 |
NPT307 |
Cell Line |
HOS |
Homo sapiens |
IC50 |
= |
20485037.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2019 |
Cell Line |
JVM-2 |
Homo sapiens |
IC50 |
= |
26418610.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2020 |
Cell Line |
JVM-3 |
Homo sapiens |
IC50 |
= |
67784104.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2373 |
Cell Line |
KYSE-150 cell line |
|
IC50 |
= |
157179383.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2374 |
Cell Line |
KYSE-180 |
Homo sapiens |
IC50 |
= |
9061862.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2021 |
Cell Line |
LS-411N |
Homo sapiens |
IC50 |
= |
10383320.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2006 |
Cell Line |
MHH-PREB-1 |
Homo sapiens |
IC50 |
= |
11563917.86 |
nM |
10.6019/CHEMBL1201861 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
22263191.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2375 |
Cell Line |
MKN-1 |
Homo sapiens |
IC50 |
= |
226317916.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2008 |
Cell Line |
NB69 |
Homo sapiens |
IC50 |
= |
30799785.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2023 |
Cell Line |
NB7 |
Homo sapiens |
IC50 |
= |
345740232.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2376 |
Cell Line |
NBsusSR |
Homo sapiens |
IC50 |
= |
9193233.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2377 |
Cell Line |
NCI-H2087 |
Homo sapiens |
IC50 |
= |
47060768.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2024 |
Cell Line |
NCI-H209 |
Homo sapiens |
IC50 |
= |
925298.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2012 |
Cell Line |
NCI-H720 |
Homo sapiens |
IC50 |
= |
533963.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2378 |
Cell Line |
NCI-H727 |
Homo sapiens |
IC50 |
= |
26634029.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2025 |
Cell Line |
NCI-H747 |
Homo sapiens |
IC50 |
= |
39420410.73 |
nM |
10.6019/CHEMBL1201861 |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
IC50 |
= |
54406504.84 |
nM |
10.6019/CHEMBL1201861 |
NPT2379 |
Cell Line |
P12-Ichikawa |
Homo sapiens |
IC50 |
= |
12383348.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2026 |
Cell Line |
Ramos-2G6-4C10 |
Homo sapiens |
IC50 |
= |
83029728.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2380 |
Cell Line |
SK-N-AS |
Homo sapiens |
IC50 |
= |
292697520.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2027 |
Cell Line |
SK-N-DZ |
Homo sapiens |
IC50 |
= |
13296764.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2381 |
Cell Line |
SW900 |
Homo sapiens |
IC50 |
= |
19285388.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2382 |
Cell Line |
SW948 |
Homo sapiens |
IC50 |
= |
52262271.32 |
nM |
10.6019/CHEMBL1201861 |
NPT1535 |
Cell Line |
U-87 MG |
Homo sapiens |
IC50 |
= |
26812085.06 |
nM |
10.6019/CHEMBL1201861 |
NPT2031 |
Cell Line |
ES8 |
Homo sapiens |
IC50 |
= |
17069371.57 |
nM |
10.6019/CHEMBL1201861 |
NPT2383 |
Cell Line |
ESS-1 |
Homo sapiens |
IC50 |
= |
41417012.28 |
nM |
10.6019/CHEMBL1201861 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
IC50 |
= |
56071615.45 |
nM |
10.6019/CHEMBL1201861 |
NPT759 |
Cell Line |
H9 |
Homo sapiens |
IC50 |
= |
7136123.64 |
nM |
10.6019/CHEMBL1201861 |
NPT2032 |
Cell Line |
HAL-01 |
Homo sapiens |
IC50 |
= |
38789311.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2384 |
Cell Line |
HPAF-II |
Homo sapiens |
IC50 |
= |
7743499.53 |
nM |
10.6019/CHEMBL1201861 |
NPT924 |
Cell Line |
HSC-2 |
Homo sapiens |
IC50 |
= |
12116155.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2385 |
Cell Line |
HSC-3 |
Homo sapiens |
IC50 |
= |
36507171.51 |
nM |
10.6019/CHEMBL1201861 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
120774808 |
nM |
10.6019/CHEMBL1201861 |
NPT2386 |
Cell Line |
KYSE-270 |
Homo sapiens |
IC50 |
= |
39394953.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2387 |
Cell Line |
KYSE-410 |
Homo sapiens |
IC50 |
= |
47506508.42 |
nM |
10.6019/CHEMBL1201861 |
NPT2022 |
Cell Line |
LS-513 |
Homo sapiens |
IC50 |
= |
31758922.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2034 |
Cell Line |
LU-134-A |
Homo sapiens |
IC50 |
= |
12994039.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2388 |
Cell Line |
LU-135 |
Homo sapiens |
IC50 |
= |
102281592.6 |
nM |
10.6019/CHEMBL1201861 |
NPT1179 |
Cell Line |
MKN-28 |
Homo sapiens |
IC50 |
= |
86098735.16 |
nM |
10.6019/CHEMBL1201861 |
NPT1097 |
Cell Line |
MKN-45 |
Homo sapiens |
IC50 |
= |
20211337.74 |
nM |
10.6019/CHEMBL1201861 |
NPT2389 |
Cell Line |
NCI-H1048 |
Homo sapiens |
IC50 |
= |
24278925.75 |
nM |
10.6019/CHEMBL1201861 |
NPT2036 |
Cell Line |
NCI-H1092 |
Homo sapiens |
IC50 |
= |
442232924.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2390 |
Cell Line |
NCI-H2122 |
Homo sapiens |
IC50 |
= |
31356253.5 |
nM |
10.6019/CHEMBL1201861 |
NPT1082 |
Cell Line |
NCI-H2126 |
Homo sapiens |
IC50 |
= |
28545740.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2391 |
Cell Line |
NCI-H810 |
Homo sapiens |
IC50 |
= |
67469910.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2040 |
Cell Line |
P30-OHK |
Homo sapiens |
IC50 |
= |
2756329 |
nM |
10.6019/CHEMBL1201861 |
NPT2392 |
Cell Line |
S-117 |
Homo sapiens |
IC50 |
= |
263216456.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2393 |
Cell Line |
SAS |
Homo sapiens |
IC50 |
= |
11279486.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
32669003.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2043 |
Cell Line |
SK-NEP-1 |
Homo sapiens |
IC50 |
= |
15006729.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2029 |
Cell Line |
SW 954 |
Homo sapiens |
IC50 |
= |
53378055.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2044 |
Cell Line |
SW 962 |
Homo sapiens |
IC50 |
= |
115399234.6 |
nM |
10.6019/CHEMBL1201861 |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
IC50 |
= |
61577941.94 |
nM |
10.6019/CHEMBL1201861 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
9900870.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2045 |
Cell Line |
ETK-1 |
Homo sapiens |
IC50 |
= |
14053053.75 |
nM |
10.6019/CHEMBL1201861 |
NPT2047 |
Cell Line |
HC-1 |
Homo sapiens |
IC50 |
= |
4197443.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2394 |
Cell Line |
HSC-4 |
Homo sapiens |
IC50 |
= |
5482656.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2049 |
Cell Line |
HT |
Homo sapiens |
IC50 |
= |
11865614.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2051 |
Cell Line |
K5 |
Homo sapiens |
IC50 |
= |
73727342.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2395 |
Cell Line |
KYSE-450 |
Homo sapiens |
IC50 |
= |
28862458.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2396 |
Cell Line |
KYSE-510 |
Homo sapiens |
IC50 |
= |
45152096.87 |
nM |
10.6019/CHEMBL1201861 |
NPT2397 |
Cell Line |
KYSE-520 cell line |
|
IC50 |
= |
334115493.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2053 |
Cell Line |
LU-139 |
Homo sapiens |
IC50 |
= |
20574238.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2398 |
Cell Line |
MKN-7 |
Homo sapiens |
IC50 |
= |
202097392.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2055 |
Cell Line |
ML-2 |
Homo sapiens |
IC50 |
= |
1486904.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2057 |
Cell Line |
NCI-H1155 |
Homo sapiens |
IC50 |
= |
17718330.43 |
nM |
10.6019/CHEMBL1201861 |
NPT2399 |
Cell Line |
NCI-H2170 |
Homo sapiens |
IC50 |
= |
281979880 |
nM |
10.6019/CHEMBL1201861 |
NPT2039 |
Cell Line |
NCI-H82 |
Homo sapiens |
IC50 |
= |
136989423.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2400 |
Cell Line |
PA-1 |
Homo sapiens |
IC50 |
= |
14188328.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2401 |
Cell Line |
PANC-03-27 |
Homo sapiens |
IC50 |
= |
150520264.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2402 |
Cell Line |
PANC-08-13 |
Homo sapiens |
IC50 |
= |
40546550.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2042 |
Cell Line |
SBC-1 |
Homo sapiens |
IC50 |
= |
6932952.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2403 |
Cell Line |
SBC-5 |
Homo sapiens |
IC50 |
= |
17071146.87 |
nM |
10.6019/CHEMBL1201861 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
1855711985 |
nM |
10.6019/CHEMBL1201861 |
NPT2063 |
Cell Line |
SK-PN-DW |
Homo sapiens |
IC50 |
= |
1149093582 |
nM |
10.6019/CHEMBL1201861 |
NPT2404 |
Cell Line |
SW982 |
Homo sapiens |
IC50 |
= |
35372678.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2405 |
Cell Line |
SAOS-2 |
Homo sapiens |
IC50 |
= |
121614805.9 |
nM |
10.6019/CHEMBL1201861 |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
IC50 |
= |
13920112.28 |
nM |
10.6019/CHEMBL1201861 |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
IC50 |
= |
330080881.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2065 |
Cell Line |
EW-1 |
Homo sapiens |
IC50 |
= |
215035842 |
nM |
10.6019/CHEMBL1201861 |
NPT2048 |
Cell Line |
HCC1187 |
Homo sapiens |
IC50 |
= |
14193210.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2406 |
Cell Line |
HCC1395 |
Homo sapiens |
IC50 |
= |
46239653.05 |
nM |
10.6019/CHEMBL1201861 |
NPT2407 |
Cell Line |
HCC1419 |
Homo sapiens |
IC50 |
= |
20360438.34 |
nM |
10.6019/CHEMBL1201861 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
IC50 |
= |
35496131.58 |
nM |
10.6019/CHEMBL1201861 |
NPT658 |
Cell Line |
HT1197 |
Homo sapiens |
IC50 |
= |
63713324.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2052 |
Cell Line |
KALS-1 |
Homo sapiens |
IC50 |
= |
741326924 |
nM |
10.6019/CHEMBL1201861 |
NPT2067 |
Cell Line |
KARPAS-299 |
Homo sapiens |
IC50 |
= |
29593647.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2408 |
Cell Line |
KYSE-70 cell line |
|
IC50 |
= |
324696441.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2068 |
Cell Line |
L-363 |
Homo sapiens |
IC50 |
= |
6735450.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2069 |
Cell Line |
Lu-65 |
Homo sapiens |
IC50 |
= |
510564.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2409 |
Cell Line |
LU-99A |
Homo sapiens |
IC50 |
= |
530105329.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2056 |
Cell Line |
MLMA |
Homo sapiens |
IC50 |
= |
20800576.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2071 |
Cell Line |
MMAC-SF |
Homo sapiens |
IC50 |
= |
107629494.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2410 |
Cell Line |
NCI-H1299 |
Homo sapiens |
IC50 |
= |
10109066.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2073 |
Cell Line |
NCI-H1304 |
Homo sapiens |
IC50 |
= |
15643910.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2411 |
Cell Line |
NCI-H2228 |
Homo sapiens |
IC50 |
= |
27995834.21 |
nM |
10.6019/CHEMBL1201861 |
NPT465 |
Cell Line |
NCI-N87 |
Homo sapiens |
IC50 |
= |
24094840.27 |
nM |
10.6019/CHEMBL1201861 |
NPT788 |
Cell Line |
SNU1 |
Homo sapiens |
IC50 |
= |
8471450.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2412 |
Cell Line |
Panc1005 |
Homo sapiens |
IC50 |
= |
749154113.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2413 |
Cell Line |
PC-14 |
Homo sapiens |
IC50 |
= |
17586080.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2062 |
Cell Line |
SCC-15 |
Homo sapiens |
IC50 |
= |
52716511.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2414 |
Cell Line |
SCC-25 |
Homo sapiens |
IC50 |
= |
12161372.27 |
nM |
10.6019/CHEMBL1201861 |
NPT2078 |
Cell Line |
SK-UT-1 |
Homo sapiens |
IC50 |
= |
40570764.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2415 |
Cell Line |
SKG-IIIa |
Homo sapiens |
IC50 |
= |
20823032.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2245 |
Cell Line |
SiHa |
Homo sapiens |
IC50 |
= |
37715974.1 |
nM |
10.6019/CHEMBL1201861 |
NPT550 |
Cell Line |
T-24 |
Homo sapiens |
IC50 |
= |
1843576513 |
nM |
10.6019/CHEMBL1201861 |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
IC50 |
= |
19940158.65 |
nM |
10.6019/CHEMBL1201861 |
NPT2416 |
Cell Line |
UACC-893 |
Homo sapiens |
IC50 |
= |
9966372.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2417 |
Cell Line |
UMUC3 |
Homo sapiens |
IC50 |
= |
12815196.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2066 |
Cell Line |
EW-11 |
Homo sapiens |
IC50 |
= |
22190532.21 |
nM |
10.6019/CHEMBL1201861 |
NPT2080 |
Cell Line |
EW-13 |
Homo sapiens |
IC50 |
= |
493323783.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2418 |
Cell Line |
HCC1569 |
Homo sapiens |
IC50 |
= |
1074135812 |
nM |
10.6019/CHEMBL1201861 |
NPT2419 |
Cell Line |
HT-1376 |
Homo sapiens |
IC50 |
= |
10407240.03 |
nM |
10.6019/CHEMBL1201861 |
NPT2082 |
Cell Line |
HT-144 |
Homo sapiens |
IC50 |
= |
31158177.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2084 |
Cell Line |
KARPAS-45 |
Homo sapiens |
IC50 |
= |
3045587.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2086 |
Cell Line |
L-428 |
Homo sapiens |
IC50 |
= |
7764318.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2070 |
Cell Line |
LXF-289 cell line |
|
IC50 |
= |
12032925.94 |
nM |
10.6019/CHEMBL1201861 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
26668143.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2072 |
Cell Line |
MN-60 |
Homo sapiens |
IC50 |
= |
24344470.05 |
nM |
10.6019/CHEMBL1201861 |
NPT3466 |
Cell Line |
MOLT-13 |
Homo sapiens |
IC50 |
= |
556027.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2074 |
Cell Line |
NCI-H1355 |
Homo sapiens |
IC50 |
= |
24747580.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2089 |
Cell Line |
NCI-H1395 |
Homo sapiens |
IC50 |
= |
21920444.08 |
nM |
10.6019/CHEMBL1201861 |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
IC50 |
= |
220985639.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2420 |
Cell Line |
NCI-H2291 |
Homo sapiens |
IC50 |
= |
99154845.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2091 |
Cell Line |
SNU-5 |
Homo sapiens |
IC50 |
= |
3697151.73 |
nM |
10.6019/CHEMBL1201861 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
81483269.83 |
nM |
10.6019/CHEMBL1201861 |
NPT2421 |
Cell Line |
PFSK-1 |
Homo sapiens |
IC50 |
= |
30868699.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2422 |
Cell Line |
SCC-4 |
Homo sapiens |
IC50 |
= |
24417173.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2423 |
Cell Line |
SCC-9 |
Homo sapiens |
IC50 |
= |
10150132.11 |
nM |
10.6019/CHEMBL1201861 |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
IC50 |
= |
306076699 |
nM |
10.6019/CHEMBL1201861 |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
IC50 |
= |
27329855.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2424 |
Cell Line |
T84 |
Homo sapiens |
IC50 |
= |
114457516.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
35620870.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2425 |
Cell Line |
UMC-11 |
Homo sapiens |
IC50 |
= |
52254014.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2096 |
Cell Line |
VA-ES-BJ |
Homo sapiens |
IC50 |
= |
13293573.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2097 |
Cell Line |
EW-16 |
Homo sapiens |
IC50 |
= |
6778804.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2098 |
Cell Line |
EW-18 |
Homo sapiens |
IC50 |
= |
5852920.23 |
nM |
10.6019/CHEMBL1201861 |
NPT2426 |
Cell Line |
HCC1806 |
Homo sapiens |
IC50 |
= |
27568497.37 |
nM |
10.6019/CHEMBL1201861 |
NPT1884 |
Cell Line |
HCC1937 |
Homo sapiens |
IC50 |
= |
34934773.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2427 |
Cell Line |
HCC1954 |
Homo sapiens |
IC50 |
= |
201135079.8 |
nM |
10.6019/CHEMBL1201861 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
39439021.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2428 |
Cell Line |
HT-3 |
Homo sapiens |
IC50 |
= |
8155273.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2429 |
Cell Line |
HT55 |
Homo sapiens |
IC50 |
= |
31769309.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2085 |
Cell Line |
Kasumi 1 |
|
IC50 |
= |
378252.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2099 |
Cell Line |
KE-37 |
Homo sapiens |
IC50 |
= |
7489909.55 |
nM |
10.6019/CHEMBL1201861 |
NPT1358 |
Cell Line |
LAMA-84 |
Homo sapiens |
IC50 |
= |
23557322.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2101 |
Cell Line |
LAN-6 |
Homo sapiens |
IC50 |
= |
355516876.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2430 |
Cell Line |
M059J |
Homo sapiens |
IC50 |
= |
34464221.26 |
nM |
10.6019/CHEMBL1201861 |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
IC50 |
= |
25185230.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2088 |
Cell Line |
MOLT-16 |
Homo sapiens |
IC50 |
= |
21118210.41 |
nM |
10.6019/CHEMBL1201861 |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
IC50 |
= |
54624512.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2431 |
Cell Line |
NCI-H1437 |
Homo sapiens |
IC50 |
= |
27957282.52 |
nM |
10.6019/CHEMBL1201861 |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
IC50 |
= |
17064985.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2432 |
Cell Line |
NCI-H2342 |
Homo sapiens |
IC50 |
= |
8624635.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2092 |
Cell Line |
NEC8 |
Homo sapiens |
IC50 |
= |
16026309.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2106 |
Cell Line |
NH-12 |
Homo sapiens |
IC50 |
= |
112006479.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2107 |
Cell Line |
PSN1 |
Homo sapiens |
IC50 |
= |
25407228.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2109 |
Cell Line |
SCH |
Homo sapiens |
IC50 |
= |
65009845.07 |
nM |
10.6019/CHEMBL1201861 |
NPT890 |
Cell Line |
SNU-387 |
Homo sapiens |
IC50 |
= |
34307387.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2433 |
Cell Line |
SNU-423 |
Homo sapiens |
IC50 |
= |
23686416.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2434 |
Cell Line |
TCC-SUP |
Homo sapiens |
IC50 |
= |
4008406.26 |
nM |
10.6019/CHEMBL1201861 |
NPT2435 |
Cell Line |
VM-CUB-1 |
Homo sapiens |
IC50 |
= |
216257477 |
nM |
10.6019/CHEMBL1201861 |
NPT2436 |
Cell Line |
VMRC-RCZ |
Homo sapiens |
IC50 |
= |
138528034.6 |
nM |
10.6019/CHEMBL1201861 |
NPT1653 |
Cell Line |
WM-115 |
Homo sapiens |
IC50 |
= |
56525378.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2437 |
Cell Line |
EW-22 |
Homo sapiens |
IC50 |
= |
109506370 |
nM |
10.6019/CHEMBL1201861 |
NPT2113 |
Cell Line |
EW-24 |
Homo sapiens |
IC50 |
= |
9448846.98 |
nM |
10.6019/CHEMBL1201861 |
NPT2116 |
Cell Line |
HCC2218 |
Homo sapiens |
IC50 |
= |
701244.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2438 |
Cell Line |
HTC-C3 |
Homo sapiens |
IC50 |
= |
29129450.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2117 |
Cell Line |
HuTu80 |
Homo sapiens |
IC50 |
= |
29848175.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2100 |
Cell Line |
KG-1 |
|
IC50 |
= |
16800030.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2118 |
Cell Line |
KGN |
Homo sapiens |
IC50 |
= |
24717925.79 |
nM |
10.6019/CHEMBL1201861 |
NPT2120 |
Cell Line |
LB1047-RCC |
Homo sapiens |
IC50 |
= |
16393611.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2121 |
Cell Line |
LB2241-RCC |
Homo sapiens |
IC50 |
= |
41003881.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2439 |
Cell Line |
MC-IXC |
Homo sapiens |
IC50 |
= |
7890028.29 |
nM |
10.6019/CHEMBL1201861 |
NPT2122 |
Cell Line |
MC116 |
Homo sapiens |
IC50 |
= |
69653553.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2123 |
Cell Line |
MPP-89 |
Homo sapiens |
IC50 |
= |
37133544.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2440 |
Cell Line |
NCI-H1563 |
Homo sapiens |
IC50 |
= |
8611131.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2441 |
Cell Line |
NCI-H2347 |
Homo sapiens |
IC50 |
= |
211906199.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2442 |
Cell Line |
NCI-H2405 |
Homo sapiens |
IC50 |
= |
569579130.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2126 |
Cell Line |
NKM-1 |
Homo sapiens |
IC50 |
= |
9106393.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2127 |
Cell Line |
NMC-G1 |
Homo sapiens |
IC50 |
= |
46326711.69 |
nM |
10.6019/CHEMBL1201861 |
NPT2108 |
Cell Line |
QIMR-WIL |
Homo sapiens |
IC50 |
= |
50754674.45 |
nM |
10.6019/CHEMBL1201861 |
NPT2128 |
Cell Line |
RCC10RGB |
Homo sapiens |
IC50 |
= |
312349490 |
nM |
10.6019/CHEMBL1201861 |
NPT2111 |
Cell Line |
SF-126 |
Homo sapiens |
IC50 |
= |
40265809.97 |
nM |
10.6019/CHEMBL1201861 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
IC50 |
= |
74942092.93 |
nM |
10.6019/CHEMBL1201861 |
NPT2443 |
Cell Line |
SNU-449 |
Homo sapiens |
IC50 |
= |
29036269.5 |
nM |
10.6019/CHEMBL1201861 |
NPT2112 |
Cell Line |
TE-1 |
Homo sapiens |
IC50 |
= |
23635828.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2130 |
Cell Line |
TE-10 |
Homo sapiens |
IC50 |
= |
41118852.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2444 |
Cell Line |
YAPC |
Homo sapiens |
IC50 |
= |
86555231.19 |
nM |
10.6019/CHEMBL1201861 |
NPT2445 |
Cell Line |
YH-13 |
Homo sapiens |
IC50 |
= |
28266114.54 |
nM |
10.6019/CHEMBL1201861 |
NPT2114 |
Cell Line |
EW-3 |
Homo sapiens |
IC50 |
= |
12151391.88 |
nM |
10.6019/CHEMBL1201861 |
NPT2132 |
Cell Line |
EOL1 |
Homo sapiens |
IC50 |
= |
1816073.44 |
nM |
10.6019/CHEMBL1201861 |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
IC50 |
= |
21339967.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2446 |
Cell Line |
HCC38 |
Homo sapiens |
IC50 |
= |
165320947.5 |
nM |
10.6019/CHEMBL1201861 |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
IC50 |
= |
42952623.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2447 |
Cell Line |
HuCCT-1 |
Homo sapiens |
IC50 |
= |
62409326.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2119 |
Cell Line |
KINGS-1 |
Homo sapiens |
IC50 |
= |
88163118.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2448 |
Cell Line |
KLE |
Homo sapiens |
IC50 |
= |
34253944.33 |
nM |
10.6019/CHEMBL1201861 |
NPT2134 |
Cell Line |
LB2518-MEL |
Homo sapiens |
IC50 |
= |
28878972.09 |
nM |
10.6019/CHEMBL1201861 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
160487285.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2137 |
Cell Line |
MS-1 |
Homo sapiens |
IC50 |
= |
50051211.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2138 |
Cell Line |
MSTO-211H |
Homo sapiens |
IC50 |
= |
31195183.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2449 |
Cell Line |
NCI-H1573 |
Homo sapiens |
IC50 |
= |
16860333.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2139 |
Cell Line |
NCI-H1581 |
Homo sapiens |
IC50 |
= |
14928493.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2450 |
Cell Line |
NCI-H2452 |
Homo sapiens |
IC50 |
= |
122982211.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2451 |
Cell Line |
NCI-H28 |
Homo sapiens |
IC50 |
= |
12044314.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2452 |
Cell Line |
NCI-H292 |
|
IC50 |
= |
5870176.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2140 |
Cell Line |
NOMO-1 |
Homo sapiens |
IC50 |
= |
29009684.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2453 |
Cell Line |
RCM-1 |
Homo sapiens |
IC50 |
= |
30241063.55 |
nM |
10.6019/CHEMBL1201861 |
NPT2454 |
Cell Line |
RD |
Homo sapiens |
IC50 |
= |
44407115.74 |
nM |
10.6019/CHEMBL1201861 |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
IC50 |
= |
6167389.92 |
nM |
10.6019/CHEMBL1201861 |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
IC50 |
= |
31248229.58 |
nM |
10.6019/CHEMBL1201861 |
NPT2455 |
Cell Line |
SNU-C2B |
Homo sapiens |
IC50 |
= |
32795841.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2456 |
Cell Line |
TE-11 |
Homo sapiens |
IC50 |
= |
20523441.51 |
nM |
10.6019/CHEMBL1201861 |
NPT2144 |
Cell Line |
TE-12 |
Homo sapiens |
IC50 |
= |
34356276.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2457 |
Cell Line |
YKG-1 |
Homo sapiens |
IC50 |
= |
277966810.8 |
nM |
10.6019/CHEMBL1201861 |
NPT994 |
Cell Line |
ZR-75-30 |
Homo sapiens |
IC50 |
= |
14885933.71 |
nM |
10.6019/CHEMBL1201861 |
NPT1216 |
Cell Line |
FaDu |
Homo sapiens |
IC50 |
= |
11208951.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2458 |
Cell Line |
FTC-133 |
Homo sapiens |
IC50 |
= |
24793703.28 |
nM |
10.6019/CHEMBL1201861 |
NPT2459 |
Cell Line |
HCC70 |
Homo sapiens |
IC50 |
= |
30423846.37 |
nM |
10.6019/CHEMBL1201861 |
NPT2460 |
Cell Line |
HCE-4 |
Homo sapiens |
IC50 |
= |
11041751.97 |
nM |
10.6019/CHEMBL1201861 |
NPT1229 |
Cell Line |
Huh-7 |
Homo sapiens |
IC50 |
= |
15501157.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2461 |
Cell Line |
HuO-3N1 |
Homo sapiens |
IC50 |
= |
7797566.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2462 |
Cell Line |
HuO9 |
Homo sapiens |
IC50 |
= |
144319085.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2133 |
Cell Line |
KM-H2 |
Homo sapiens |
IC50 |
= |
18689590.69 |
nM |
10.6019/CHEMBL1201861 |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
IC50 |
= |
35184960.09 |
nM |
10.6019/CHEMBL1201861 |
NPT2135 |
Cell Line |
LB373-MEL-D |
Homo sapiens |
IC50 |
= |
432787013.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2148 |
Cell Line |
LB771-HNC |
Homo sapiens |
IC50 |
= |
37926903.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2463 |
Cell Line |
MDA-MB-157 |
Homo sapiens |
IC50 |
= |
759851273.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2464 |
Cell Line |
MDA-MB-175-VII |
Homo sapiens |
IC50 |
= |
24734096.6 |
nM |
10.6019/CHEMBL1201861 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
801348329.7 |
nM |
10.6019/CHEMBL1201861 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
IC50 |
= |
8432368.73 |
nM |
10.6019/CHEMBL1201861 |
NPT2465 |
Cell Line |
NCI-H1623 |
Homo sapiens |
IC50 |
= |
103736053 |
nM |
10.6019/CHEMBL1201861 |
NPT2150 |
Cell Line |
NCI-H1648 |
Homo sapiens |
IC50 |
= |
29765580.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2466 |
Cell Line |
NCI-H358 |
Homo sapiens |
IC50 |
= |
160881283.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2141 |
Cell Line |
NOS-1 |
Homo sapiens |
IC50 |
= |
32232837.18 |
nM |
10.6019/CHEMBL1201861 |
NPT2152 |
Cell Line |
NTERA-2-cl-D1 |
Homo sapiens |
IC50 |
= |
19474262.48 |
nM |
10.6019/CHEMBL1201861 |
NPT2467 |
Cell Line |
RERF-LC-MS |
Homo sapiens |
IC50 |
= |
14379200.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2153 |
Cell Line |
RH-1 |
Homo sapiens |
IC50 |
= |
107647039.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2154 |
Cell Line |
SH-4 |
Homo sapiens |
IC50 |
= |
26196602.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2155 |
Cell Line |
SHP77 |
Homo sapiens |
IC50 |
= |
26563171.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2159 |
Cell Line |
TE-5 |
Homo sapiens |
IC50 |
= |
32242315.02 |
nM |
10.6019/CHEMBL1201861 |
NPT2160 |
Cell Line |
no-10 |
Homo sapiens |
IC50 |
= |
249667422.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2468 |
Cell Line |
G-361 |
Homo sapiens |
IC50 |
= |
2664934400 |
nM |
10.6019/CHEMBL1201861 |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
IC50 |
= |
1591689.01 |
nM |
10.6019/CHEMBL1201861 |
NPT2470 |
Cell Line |
G-402 |
Homo sapiens |
IC50 |
= |
11349193.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2162 |
Cell Line |
HCE-T |
Homo sapiens |
IC50 |
= |
126009678.9 |
nM |
10.6019/CHEMBL1201861 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
65735605.61 |
nM |
10.6019/CHEMBL1201861 |
NPT2471 |
Cell Line |
HuP-T3 |
Homo sapiens |
IC50 |
= |
798533340.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2472 |
Cell Line |
HuP-T4 |
Homo sapiens |
IC50 |
= |
305199518.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2163 |
Cell Line |
KMOE-2 |
Homo sapiens |
IC50 |
= |
89724307.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2166 |
Cell Line |
LB831-BLC |
Homo sapiens |
IC50 |
= |
41603808.81 |
nM |
10.6019/CHEMBL1201861 |
NPT2473 |
Cell Line |
MDA-MB-361 |
Homo sapiens |
IC50 |
= |
41383767.77 |
nM |
10.6019/CHEMBL1201861 |
NPT2474 |
Cell Line |
MDA-MB-415 |
Homo sapiens |
IC50 |
= |
16831610.92 |
nM |
10.6019/CHEMBL1201861 |
NPT2149 |
Cell Line |
MZ1-PC |
Homo sapiens |
IC50 |
= |
178511624.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2168 |
Cell Line |
MZ2-MEL |
Homo sapiens |
IC50 |
= |
26993894.78 |
nM |
10.6019/CHEMBL1201861 |
NPT1820 |
Cell Line |
NCI-H1650 |
Homo sapiens |
IC50 |
= |
289867151.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2475 |
Cell Line |
NCI-H1651 |
Homo sapiens |
IC50 |
= |
18529178.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2476 |
Cell Line |
NCI-H441 |
Homo sapiens |
IC50 |
= |
77587762.97 |
nM |
10.6019/CHEMBL1201861 |
NPT937 |
Cell Line |
NCI-H446 |
Homo sapiens |
IC50 |
= |
120571956.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2477 |
Cell Line |
NUGC-3 |
Homo sapiens |
IC50 |
= |
256839845.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2478 |
Cell Line |
NY |
Homo sapiens |
IC50 |
= |
14121715.53 |
nM |
10.6019/CHEMBL1201861 |
NPT2479 |
Cell Line |
OAW-28 |
Homo sapiens |
IC50 |
= |
36267924.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2480 |
Cell Line |
RH-18 |
Homo sapiens |
IC50 |
= |
140985735.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2170 |
Cell Line |
RKO |
Homo sapiens |
IC50 |
= |
27107751.52 |
nM |
10.6019/CHEMBL1201861 |
NPT2481 |
Cell Line |
SW1088 |
Homo sapiens |
IC50 |
= |
40140938.39 |
nM |
10.6019/CHEMBL1201861 |
NPT2482 |
Cell Line |
SW 1116 |
Homo sapiens |
IC50 |
= |
45059900.24 |
nM |
10.6019/CHEMBL1201861 |
NPT2483 |
Cell Line |
SW13 |
Homo sapiens |
IC50 |
= |
10008099.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2173 |
Cell Line |
TE-6 |
Homo sapiens |
IC50 |
= |
14245495.07 |
nM |
10.6019/CHEMBL1201861 |
NPT2161 |
Cell Line |
no-11 |
Homo sapiens |
IC50 |
= |
31082834.49 |
nM |
10.6019/CHEMBL1201861 |
NPT2175 |
Cell Line |
GAK |
Homo sapiens |
IC50 |
= |
24482748.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2484 |
Cell Line |
GAMG |
Homo sapiens |
IC50 |
= |
21121124.93 |
nM |
10.6019/CHEMBL1201861 |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
IC50 |
= |
8894959.08 |
nM |
10.6019/CHEMBL1201861 |
NPT2176 |
Cell Line |
HD-MY-Z |
Homo sapiens |
IC50 |
= |
29015806.15 |
nM |
10.6019/CHEMBL1201861 |
NPT2485 |
Cell Line |
IA-LM |
Homo sapiens |
IC50 |
= |
51795471.41 |
nM |
10.6019/CHEMBL1201861 |
NPT2486 |
Cell Line |
IGR-1 |
Homo sapiens |
IC50 |
= |
858815162.3 |
nM |
10.6019/CHEMBL1201861 |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
IC50 |
= |
97770385.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2165 |
Cell Line |
KNS-42 |
Homo sapiens |
IC50 |
= |
148495509.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2487 |
Cell Line |
KNS-62 |
Homo sapiens |
IC50 |
= |
22201141.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2180 |
Cell Line |
LC-2-ad |
Homo sapiens |
IC50 |
= |
442037500.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2488 |
Cell Line |
MDA-MB-453 |
Homo sapiens |
IC50 |
= |
12856592.58 |
nM |
10.6019/CHEMBL1201861 |
NPT1773 |
Cell Line |
ME-180 |
Homo sapiens |
IC50 |
= |
86147566.99 |
nM |
10.6019/CHEMBL1201861 |
NPT2169 |
Cell Line |
MZ7-mel |
Homo sapiens |
IC50 |
= |
1540093982 |
nM |
10.6019/CHEMBL1201861 |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
74953859.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2490 |
Cell Line |
NCI-H1666 |
Homo sapiens |
IC50 |
= |
253887110.4 |
nM |
10.6019/CHEMBL1201861 |
NPT2491 |
Cell Line |
NCI-H1693 |
Homo sapiens |
IC50 |
= |
43033751.27 |
nM |
10.6019/CHEMBL1201861 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
23567454.67 |
nM |
10.6019/CHEMBL1201861 |
NPT2184 |
Cell Line |
NCI-H510A |
Homo sapiens |
IC50 |
= |
1313483.44 |
nM |
10.6019/CHEMBL1201861 |
NPT2492 |
Cell Line |
OAW-42 |
Homo sapiens |
IC50 |
= |
18125335.68 |
nM |
10.6019/CHEMBL1201861 |
NPT2493 |
Cell Line |
OC-314 |
Homo sapiens |
IC50 |
= |
26330177.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2494 |
Cell Line |
RMG-I |
Homo sapiens |
IC50 |
= |
73376720.14 |
nM |
10.6019/CHEMBL1201861 |
NPT2188 |
Cell Line |
SJSA-1 |
Homo sapiens |
IC50 |
= |
33067625.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2495 |
Cell Line |
SW1417 |
Homo sapiens |
IC50 |
= |
110297550.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2496 |
Cell Line |
SW1463 |
Homo sapiens |
IC50 |
= |
77942760.77 |
nM |
10.6019/CHEMBL1201861 |
NPT1577 |
Cell Line |
SW1573 |
Homo sapiens |
IC50 |
= |
50285145.78 |
nM |
10.6019/CHEMBL1201861 |
NPT2174 |
Cell Line |
TE-8 |
Homo sapiens |
IC50 |
= |
46779670.66 |
nM |
10.6019/CHEMBL1201861 |
NPT2189 |
Cell Line |
TE-9 |
Homo sapiens |
IC50 |
= |
10467997.24 |
nM |
10.6019/CHEMBL1201861 |
NPT1354 |
Cell Line |
TGBC11TKB |
Homo sapiens |
IC50 |
= |
72091108.94 |
nM |
10.6019/CHEMBL1201861 |
NPT2190 |
Cell Line |
GB-1 |
Homo sapiens |
IC50 |
= |
29779663.3 |
nM |
10.6019/CHEMBL1201861 |
NPT2177 |
Cell Line |
HDLM-2 |
Homo sapiens |
IC50 |
= |
18438847.59 |
nM |
10.6019/CHEMBL1201861 |
NPT2497 |
Cell Line |
HEC-1 |
Homo sapiens |
IC50 |
= |
16218453.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2178 |
Cell Line |
KNS-81-FD |
Homo sapiens |
IC50 |
= |
8876769.72 |
nM |
10.6019/CHEMBL1201861 |
NPT2498 |
Cell Line |
KOSC-2 |
Homo sapiens |
IC50 |
= |
3398019.36 |
nM |
10.6019/CHEMBL1201861 |
NPT2499 |
Cell Line |
KP-4 |
Homo sapiens |
IC50 |
= |
7049605.95 |
nM |
10.6019/CHEMBL1201861 |
NPT2500 |
Cell Line |
LCLC-103H cell line |
|
IC50 |
= |
84133070.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2181 |
Cell Line |
MEG-01 |
Homo sapiens |
IC50 |
= |
8615584.56 |
nM |
10.6019/CHEMBL1201861 |
NPT2501 |
Cell Line |
MEL-HO |
Homo sapiens |
IC50 |
= |
8840007.46 |
nM |
10.6019/CHEMBL1201861 |
NPT2502 |
Cell Line |
MEL-JUSO |
Homo sapiens |
IC50 |
= |
15984087.9 |
nM |
10.6019/CHEMBL1201861 |
NPT2182 |
Cell Line |
Mo |
Homo sapiens |
IC50 |
= |
33960725.38 |
nM |
10.6019/CHEMBL1201861 |
NPT2503 |
Cell Line |
NCI-H1703 |
Homo sapiens |
IC50 |
= |
17289626.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2504 |
Cell Line |
NCI-H1755 |
Homo sapiens |
IC50 |
= |
99305575.85 |
nM |
10.6019/CHEMBL1201861 |
NPT2505 |
Cell Line |
NCI-H520 |
|
IC50 |
= |
101730760.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2185 |
Cell Line |
OCI-AML2 |
Homo sapiens |
IC50 |
= |
25074157.17 |
nM |
10.6019/CHEMBL1201861 |
NPT2199 |
Cell Line |
OCUB-M |
Homo sapiens |
IC50 |
= |
11395650.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2506 |
Cell Line |
RO82-W-1 |
Homo sapiens |
IC50 |
= |
52997445.86 |
nM |
10.6019/CHEMBL1201861 |
NPT2507 |
Cell Line |
RPMI-2650 |
Homo sapiens |
IC50 |
= |
87321239.02 |
nM |
10.6019/CHEMBL1201861 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
26907168.04 |
nM |
10.6019/CHEMBL1201861 |
NPT2201 |
Cell Line |
SK-LMS-1 |
Homo sapiens |
IC50 |
= |
1088494384 |
nM |
10.6019/CHEMBL1201861 |
NPT2508 |
Cell Line |
SW1710 |
Homo sapiens |
IC50 |
= |
95351848.76 |
nM |
10.6019/CHEMBL1201861 |
NPT2509 |
Cell Line |
SW1783 |
Homo sapiens |
IC50 |
= |
24951394.71 |
nM |
10.6019/CHEMBL1201861 |
NPT2202 |
Cell Line |
TGBC1TKB |
Homo sapiens |
IC50 |
= |
32956539.91 |
nM |
10.6019/CHEMBL1201861 |
NPT2191 |
Cell Line |
GCIY |
Homo sapiens |
IC50 |
= |
57213948.35 |
nM |
10.6019/CHEMBL1201861 |
NPT2510 |
Cell Line |
GCT |
Homo sapiens |
IC50 |
= |
854120872.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
IC50 |
= |
332483994.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2511 |
Cell Line |
HGC-27 |
Homo sapiens |
IC50 |
= |
22095671.31 |
nM |
10.6019/CHEMBL1201861 |
NPT2205 |
Cell Line |
IST-MEL1 |
Homo sapiens |
IC50 |
= |
34373733.82 |
nM |
10.6019/CHEMBL1201861 |
NPT2206 |
Cell Line |
IST-MES1 |
Homo sapiens |
IC50 |
= |
23024934.12 |
nM |
10.6019/CHEMBL1201861 |
NPT2207 |
Cell Line |
KP-N-YN |
Homo sapiens |
IC50 |
= |
1441347503 |
nM |
10.6019/CHEMBL1201861 |
NPT2208 |
Cell Line |
KP-N-YS |
Homo sapiens |
IC50 |
= |
879000723.7 |
nM |
10.6019/CHEMBL1201861 |
NPT2512 |
Cell Line |
LCLC-97TM1 |
Homo sapiens |
IC50 |
= |
3174749.47 |
nM |
10.6019/CHEMBL1201861 |
NPT2513 |
Cell Line |
LK-2 |
Homo sapiens |
IC50 |
= |
9238594.11 |
nM |
10.6019/CHEMBL1201861 |
NPT2514 |
Cell Line |
LN-405 |
Homo sapiens |
IC50 |
= |
277557389.6 |
nM |
10.6019/CHEMBL1201861 |
NPT2515 |
Cell Line |
MFE-280 |
Homo sapiens |
IC50 |
= |
214772799.1 |
nM |
10.6019/CHEMBL1201861 |
NPT2210 |
Cell Line |
NB10 |
Homo sapiens |
IC50 |
= |
125084026.2 |
nM |
10.6019/CHEMBL1201861 |
NPT2211 |
Cell Line |
NB12 |
Homo sapiens |
IC50 |
= |
165138368.8 |
nM |
10.6019/CHEMBL1201861 |
NPT2197 |
Cell Line |
NCI-H1770 |
Homo sapiens |
IC50 |
= |
4099720.17 |
nM |
10.6019/CHEMBL1201861 |
NPT1669 |
Cell Line |
NCI-H1792 |
Homo sapiens |
IC50 |
= |
40540347.83 |
nM |
10.6019/CHEMBL1201861 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
37 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.8 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
14.6 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
12.1 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
29.7 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
29.1 |
% |
23567949 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
23.7 |
% |
23567949 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
-24 |
% |
23478147 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
-24 |
mg/dl |
23478147 |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
Activity |
= |
-0.6 |
% |
23478147 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.5 |
nM |
24900695 |
NPT1540 |
Individual Protein |
Solute carrier family 22 member 2 |
Homo sapiens |
FC |
> |
15 |
|
23984907 |
NPT613 |
Individual Protein |
Solute carrier family 22 member 1 |
Homo sapiens |
FC |
> |
1.7 |
|
23984907 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
57.1 |
% |
10.1007/s00044-013-0784-0 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
GI |
= |
32 |
% |
24256410 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1882.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
77.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
149.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
3346.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
30637.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
68589.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
2.7 |
nM |
PubChem BioAssay data set |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
21 |
% |
10.1039/C3MD00138E |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
23.3 |
% |
10.1039/C3MD00138E |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
29.9 |
% |
24588963 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
14.1 |
% |
24813740 |
NPT1135 |
Cell Line |
Hepatocyte |
Rattus norvegicus |
Inhibition |
= |
75 |
% |
24946215 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
24 |
% |
25299458 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
22.94 |
% |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
23.2 |
% |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
19.08 |
% |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
5.32 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
8.1 |
mU |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
21.67 |
U/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
110 |
U/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.92 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.12 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.82 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
21.56 |
ng/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.93 |
|
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
10.73 |
% |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.4 |
% |
25208139 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
83 |
% |
25208139 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
7.57 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
5.48 |
mU |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
46.29 |
U/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
172 |
U/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.07 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.17 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.38 |
nM |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
26.05 |
ng/L |
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.73 |
|
25299682 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
60 |
% |
25122135 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
51 |
% |
25724827 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
3.03 |
nM |
25724827 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
14.1 |
% |
25937008 |
NPT4296 |
Individual Protein |
Equilibrative nucleoside transporter 4 |
Homo sapiens |
Activity |
= |
-2.02 |
nanoampere |
22396231 |
NPT4296 |
Individual Protein |
Equilibrative nucleoside transporter 4 |
Homo sapiens |
Activity |
= |
-38 |
nanoampere |
22396231 |
NPT163 |
Individual Protein |
Nuclear factor NF-kappa-B p105 subunit |
Homo sapiens |
Potency |
|
61644.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5.9 |
nM |
PubChem BioAssay data set |
NPT984 |
Cell Line |
Hepatocyte |
|
Inhibition |
= |
25 |
% |
26562611 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
7.86 |
% |
26920798 |