Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
160 |
nM |
11814804 |
NPT4168 |
Individual Protein |
Serine-threonine protein phosphatase 2A regulatory subunit |
Gallus gallus |
IC50 |
= |
1700 |
nM |
11814804 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
11881984 |
NPT4168 |
Individual Protein |
Serine-threonine protein phosphatase 2A regulatory subunit |
Gallus gallus |
IC50 |
= |
200 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
1000000 |
nM |
11881984 |
NPT4167 |
Individual Protein |
Serine/threonine protein phosphatase PP1-gamma catalytic subunit |
Homo sapiens |
IC50 |
= |
1780 |
nM |
11881984 |
NPT4168 |
Individual Protein |
Serine-threonine protein phosphatase 2A regulatory subunit |
Gallus gallus |
IC50 |
= |
260 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
10000 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
11000 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
9000 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
6400 |
nM |
11881984 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
10800 |
nM |
10.1016/S0960-894X(97)10005-1 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
65 |
nM |
10.1016/S0960-894X(97)10005-1 |
NPT178 |
Individual Protein |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50 |
= |
3600 |
nM |
11677131 |
NPT4168 |
Individual Protein |
Serine-threonine protein phosphatase 2A regulatory subunit |
Gallus gallus |
IC50 |
= |
360 |
nM |
11677131 |
NPT4366 |
Individual Protein |
Protein phosphatase 2C beta |
Homo sapiens |
IC50 |
= |
1780 |
nM |
10937725 |
NPT4168 |
Individual Protein |
Serine-threonine protein phosphatase 2A regulatory subunit |
Gallus gallus |
IC50 |
= |
260 |
nM |
10937725 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
10937725 |
NPT4368 |
Cell Line |
ADDP cell line |
|
IC50 |
= |
11000 |
nM |
10937725 |
NPT3792 |
Cell Line |
143B |
Homo sapiens |
IC50 |
= |
10000 |
nM |
10937725 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
10937725 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
6400 |
nM |
10937725 |
NPT4366 |
Individual Protein |
Protein phosphatase 2C beta |
Homo sapiens |
IC50 |
= |
430 |
nM |
15050639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600 |
nM |
15050639 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
10000 |
nM |
15050639 |
NPT2469 |
Cell Line |
G-401 |
Homo sapiens |
GI50 |
= |
3500 |
nM |
15050639 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
6400 |
nM |
15050639 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
4300 |
nM |
15050639 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
GI50 |
= |
15000 |
nM |
15050639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11000 |
nM |
17451951 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
17451951 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
3300 |
nM |
17451951 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
GI50 |
= |
4600 |
nM |
17451951 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
7000 |
nM |
17451951 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
5800 |
nM |
17451951 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
4000 |
nM |
17451951 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
3400 |
nM |
17451951 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
2400 |
nM |
17451951 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
4900 |
nM |
17451951 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
3000 |
nM |
17451951 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
GI50 |
= |
4500 |
nM |
17606377 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
3200 |
nM |
17606377 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
7500 |
nM |
17606377 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
4400 |
nM |
17606377 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
3300 |
nM |
17606377 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
2900 |
nM |
17606377 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
2100 |
nM |
17606377 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
3700 |
nM |
17606377 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1700 |
nM |
17606377 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7600 |
nM |
17870547 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
990 |
nM |
17870547 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
0.1 |
nM |
17870547 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
7.7 |
|
17870547 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
0.07 |
|
17870547 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
24.47 |
% |
18024584 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
259.49 |
% |
18024584 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
332.84 |
% |
18024584 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
463.81 |
% |
18024584 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
GI50 |
= |
4400 |
nM |
20153915 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
3300 |
nM |
20153915 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
900 |
nM |
20153915 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
= |
2100 |
nM |
20153915 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6000 |
nM |
20153915 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
3700 |
nM |
20153915 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
1700 |
nM |
20153915 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
7500 |
nM |
20153915 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
GI50 |
= |
4500 |
nM |
20153915 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
GI50 |
= |
2900 |
nM |
20153915 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
= |
3200 |
nM |
20153915 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
20691337 |
NPT1086 |
Cell Line |
SK-HEP1 |
Homo sapiens |
IC50 |
= |
34000 |
nM |
20691337 |
NPT1135 |
Cell Line |
Hepatocyte |
Rattus norvegicus |
IC50 |
= |
21000 |
nM |
20691337 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
5011.87 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3981.07 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3162.28 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
2511.89 |
nM |
19734910 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
9000 |
nM |
20888768 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1800 |
nM |
20888768 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
200 |
nM |
20888768 |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
1122 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT93 |
Individual Protein |
Survival motor neuron protein |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT211 |
Individual Protein |
Hypoxia-inducible factor 1 alpha |
Homo sapiens |
Potency |
= |
2511.9 |
nM |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
5011.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT443 |
Individual Protein |
Histone acetyltransferase GCN5 |
Homo sapiens |
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
15848.93 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
1018.2 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
2031.5 |
nM |
PubChem BioAssay data set |
NPT367 |
Cell Line |
MDA-N |
Homo sapiens |
GI50 |
|
2910.72 |
nM |
PubChem BioAssay data set |
NPT368 |
Cell Line |
SN12C |
Homo sapiens |
GI50 |
|
2009.09 |
nM |
PubChem BioAssay data set |
NPT369 |
Cell Line |
ACHN |
Homo sapiens |
GI50 |
|
1183.04 |
nM |
PubChem BioAssay data set |
NPT370 |
Cell Line |
NCI-H23 |
Homo sapiens |
GI50 |
|
5069.91 |
nM |
PubChem BioAssay data set |
NPT372 |
Cell Line |
HOP-92 |
Homo sapiens |
GI50 |
|
609.54 |
nM |
PubChem BioAssay data set |
NPT371 |
Cell Line |
UO-31 |
Homo sapiens |
GI50 |
|
2636.33 |
nM |
PubChem BioAssay data set |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
GI50 |
|
1020.94 |
nM |
PubChem BioAssay data set |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
GI50 |
|
1633.05 |
nM |
PubChem BioAssay data set |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
GI50 |
|
972.75 |
nM |
PubChem BioAssay data set |
NPT374 |
Cell Line |
SF-539 |
Homo sapiens |
GI50 |
|
2041.74 |
nM |
PubChem BioAssay data set |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
GI50 |
|
2301.44 |
nM |
PubChem BioAssay data set |
NPT375 |
Cell Line |
Malme-3M |
Homo sapiens |
GI50 |
|
1336.6 |
nM |
PubChem BioAssay data set |
NPT376 |
Cell Line |
A498 |
Homo sapiens |
GI50 |
|
1124.6 |
nM |
PubChem BioAssay data set |
NPT112 |
Cell Line |
MOLT-4 |
Homo sapiens |
GI50 |
|
9794.9 |
nM |
PubChem BioAssay data set |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
GI50 |
|
758.58 |
nM |
PubChem BioAssay data set |
NPT378 |
Cell Line |
NCI/ADR-RES |
Homo sapiens |
GI50 |
|
6501.3 |
nM |
PubChem BioAssay data set |
NPT379 |
Cell Line |
HOP-62 |
Homo sapiens |
GI50 |
|
2443.43 |
nM |
PubChem BioAssay data set |
NPT381 |
Cell Line |
OVCAR-8 |
Homo sapiens |
GI50 |
|
5984.12 |
nM |
PubChem BioAssay data set |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
GI50 |
|
1412.54 |
nM |
PubChem BioAssay data set |
NPT383 |
Cell Line |
SNB-19 |
Homo sapiens |
GI50 |
|
1099.01 |
nM |
PubChem BioAssay data set |
NPT382 |
Cell Line |
OVCAR-5 |
Homo sapiens |
GI50 |
|
2454.71 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
3374.7 |
nM |
PubChem BioAssay data set |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
GI50 |
|
1330.45 |
nM |
PubChem BioAssay data set |
NPT384 |
Cell Line |
TK-10 |
Homo sapiens |
GI50 |
|
312.61 |
nM |
PubChem BioAssay data set |
NPT385 |
Cell Line |
SR |
Homo sapiens |
GI50 |
|
2606.15 |
nM |
PubChem BioAssay data set |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
|
3837.07 |
nM |
PubChem BioAssay data set |
NPT386 |
Cell Line |
KM12 |
Homo sapiens |
GI50 |
|
5420.01 |
nM |
PubChem BioAssay data set |
NPT455 |
Cell Line |
NCI-H522 |
Homo sapiens |
GI50 |
|
935.41 |
nM |
PubChem BioAssay data set |
NPT387 |
Cell Line |
M14 |
Homo sapiens |
GI50 |
|
1702.16 |
nM |
PubChem BioAssay data set |
NPT388 |
Cell Line |
NCI-H322M |
Homo sapiens |
GI50 |
|
2018.37 |
nM |
PubChem BioAssay data set |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
615.9 |
nM |
PubChem BioAssay data set |
NPT389 |
Cell Line |
RPMI-8226 |
Homo sapiens |
GI50 |
|
2084.49 |
nM |
PubChem BioAssay data set |
NPT456 |
Cell Line |
OVCAR-4 |
Homo sapiens |
GI50 |
|
2582.26 |
nM |
PubChem BioAssay data set |
NPT390 |
Cell Line |
LOX IMVI |
Homo sapiens |
GI50 |
|
2233.57 |
nM |
PubChem BioAssay data set |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
GI50 |
|
1698.24 |
nM |
PubChem BioAssay data set |
NPT147 |
Cell Line |
SK-MEL-2 |
Homo sapiens |
GI50 |
|
1452.11 |
nM |
PubChem BioAssay data set |
NPT391 |
Cell Line |
HCC 2998 |
Homo sapiens |
GI50 |
|
1531.09 |
nM |
PubChem BioAssay data set |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
|
918.33 |
nM |
PubChem BioAssay data set |
NPT392 |
Cell Line |
SNB-75 |
Homo sapiens |
GI50 |
|
472.06 |
nM |
PubChem BioAssay data set |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
GI50 |
|
1976.97 |
nM |
PubChem BioAssay data set |
NPT148 |
Cell Line |
HCT-15 |
Homo sapiens |
GI50 |
|
4055.09 |
nM |
PubChem BioAssay data set |
NPT394 |
Cell Line |
EKVX |
Homo sapiens |
GI50 |
|
449.78 |
nM |
PubChem BioAssay data set |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
|
1766.04 |
nM |
PubChem BioAssay data set |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
GI50 |
|
279.25 |
nM |
PubChem BioAssay data set |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
|
7762.47 |
nM |
PubChem BioAssay data set |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
GI50 |
|
2167.7 |
nM |
PubChem BioAssay data set |
NPT396 |
Cell Line |
T47D |
Homo sapiens |
GI50 |
|
1682.67 |
nM |
PubChem BioAssay data set |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
|
2722.7 |
nM |
PubChem BioAssay data set |
NPT398 |
Cell Line |
UACC-62 |
Homo sapiens |
GI50 |
|
2118.36 |
nM |
PubChem BioAssay data set |
NPT308 |
Cell Line |
CAKI-1 |
Homo sapiens |
GI50 |
|
790.68 |
nM |
PubChem BioAssay data set |
NPT399 |
Cell Line |
SF-295 |
Homo sapiens |
GI50 |
|
1367.73 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
6911.1 |
nM |
PubChem BioAssay data set |
NPT400 |
Cell Line |
MDA-MB-435 |
Homo sapiens |
GI50 |
|
1892.34 |
nM |
PubChem BioAssay data set |
NPT458 |
Cell Line |
IGROV-1 |
Homo sapiens |
GI50 |
|
2157.74 |
nM |
PubChem BioAssay data set |
NPT402 |
Cell Line |
Hs-578T |
Homo sapiens |
GI50 |
|
1032.76 |
nM |
PubChem BioAssay data set |
NPT401 |
Cell Line |
786-0 |
Homo sapiens |
GI50 |
|
1737.8 |
nM |
PubChem BioAssay data set |
NPT403 |
Cell Line |
UACC-257 |
Homo sapiens |
GI50 |
|
2654.61 |
nM |
PubChem BioAssay data set |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
GI50 |
|
1193.99 |
nM |
PubChem BioAssay data set |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI50 |
|
1655.77 |
nM |
PubChem BioAssay data set |
NPT405 |
Cell Line |
NCI-H226 |
Homo sapiens |
GI50 |
|
1061.7 |
nM |
PubChem BioAssay data set |
NPT406 |
Cell Line |
RXF 393 |
Homo sapiens |
GI50 |
|
484.17 |
nM |
PubChem BioAssay data set |
NPT170 |
Cell Line |
SK-MEL-28 |
Homo sapiens |
GI50 |
|
3483.37 |
nM |
PubChem BioAssay data set |
NPT407 |
Cell Line |
COLO 205 |
Homo sapiens |
GI50 |
|
426.58 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
903.5 |
nM |
PubChem BioAssay data set |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
-7.81 |
% |
23062825 |
NPT67 |
Individual Protein |
Cholinesterase |
Equus caballus |
Inhibition |
= |
-2.13 |
% |
23062825 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
102.45 |
% |
23571415 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
105.74 |
% |
23571415 |