References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC550
|
TCMT113 |
Delta opioid receptor |
Homo sapiens |
Ki: 3100 (nM), Ref: 26035635 |
TCMC2126
|
TCMT210 |
Carboxylesterase 2 |
Homo sapiens |
Ki: 1410 (nM), Ref: 23286284 |
TCMC2126
|
TCMT171 |
Protein-tyrosine phosphatase 1C |
Homo sapiens |
IC50: 1970 (nM), Ref: 23957426 |
TCMC2126
|
TCMT233 |
Protein-tyrosine phosphatase 2C |
Homo sapiens |
IC50: 2570 (nM), Ref: 23957426 |
TCMC1786
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
TCMC1786
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
TCMC1786
|
TCMT190 |
T-cell protein-tyrosine phosphatase |
Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
TCMC1786
|
TCMT563 |
Dual specificity phosphatase Cdc25B |
Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC1568
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 3580 (nM), Ref: 22658537 |
TCMC1568
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 610 (nM), Ref: 22658537 |
TCMC1568
|
TCMT734 |
Matrix metalloproteinase 12 |
Homo sapiens |
IC50: 2750 (nM), Ref: 22658537 |
TCMC1886
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 810 (nM), Ref: 26498394 |
TCMC1886
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 670 (nM), Ref: 26498394 |
TCMC1886
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 770 (nM), Ref: 26498394 |
TCMC1886
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 620 (nM), Ref: 26498394 |
TCMC1886
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 810 (nM), Ref: 26498394 |
TCMC1886
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8470 (nM), Ref: 26498394 |
TCMC1886
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 720 (nM), Ref: 26498394 |
TCMC804
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
IC50: 2000 (nM), Ref: 21561086 |
TCMC847
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
TCMC847
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
TCMC847
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
TCMC847
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
TCMC847
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
TCMC847
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC847
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
TCMC847
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
TCMC847
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
TCMC847
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
TCMC847
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
TCMC847
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
TCMC847
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
TCMC847
|
TCMT295 |
Matrix metalloproteinase-1 |
Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
TCMC847
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
TCMC1053
|
TCMT131 |
Acetylcholinesterase |
Homo sapiens |
Ki: 1950 (nM), Ref: 23286284 IC50: 1000 (nM), Ref: 24900610 Ki: 600 (nM), Ref: 24900610 |
TCMC1053
|
TCMT210 |
Carboxylesterase 2 |
Homo sapiens |
Ki: 1830 (nM), Ref: 23286284 Ki: 118 (nM), Ref: 23286284 |
TCMC1053
|
TCMT211 |
Acyl coenzyme A:cholesterol acyltransferase |
Homo sapiens |
Ki: 398 (nM), Ref: 23286284 |
TCMC1053
|
TCMT171 |
Protein-tyrosine phosphatase 1C |
Homo sapiens |
IC50: 3670 (nM), Ref: 23957426 |
TCMC1053
|
TCMT233 |
Protein-tyrosine phosphatase 2C |
Homo sapiens |
IC50: 3940 (nM), Ref: 23957426 |
TCMC2216
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168 |
TCMC2216
|
TCMT174 |
11-beta-hydroxysteroid dehydrogenase 1 |
Homo sapiens |
IC50: 1900 (nM), Ref: 20100662 |
TCMC2216
|
TCMT102 |
Low molecular weight phosphotyrosine protein phosphatase |
Homo sapiens |
IC50: 7200 (nM), Ref: 21453996 |
TCMC2216
|
TCMT103 |
Receptor-type tyrosine-protein phosphatase F (LAR) |
Homo sapiens |
IC50: 3800 (nM), Ref: 21453996 |
TCMC2216
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086 |
TCMC2216
|
TCMT190 |
T-cell protein-tyrosine phosphatase |
Homo sapiens |
IC50: 2400 (nM), Ref: 23387824 |
TCMC2216
|
TCMT150 |
Nuclear receptor ROR-gamma |
Homo sapiens |
IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616 |