References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1173
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
TCMC1173
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
TCMC1173
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
TCMC1173
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
TCMC1173
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
TCMC1173
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
TCMC1173
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
TCMC1173
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
TCMC948
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
TCMC948
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
TCMC948
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
TCMC948
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
TCMC948
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
TCMC948
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
TCMC948
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
TCMC948
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
TCMC948
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
TCMC948
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
TCMC948
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
TCMC948
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
TCMC1429
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
TCMC1429
|
TCMT65 |
Estradiol 17-beta-dehydrogenase 1 |
Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
TCMC1429
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
TCMC1429
|
TCMT187 |
Androgen Receptor |
Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
TCMC1429
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
TCMC1429
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
TCMC1429
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
TCMC1429
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
TCMC1429
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
TCMC1429
|
TCMT591 |
Estrogen-related receptor alpha |
Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
TCMC1429
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
TCMC1429
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
TCMC1429
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
TCMC1429
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
TCMC1429
|
TCMT159 |
Tyrosinase |
Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
TCMC656
|
TCMT126 |
Telomerase reverse transcriptase |
Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C0MD00241K |
TCMC1480
|
TCMT107 |
Glutamate receptor ionotropic kainate 2 |
Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
TCMC1480
|
TCMT108 |
Glutamate receptor ionotropic, AMPA 1 |
Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
TCMC1480
|
TCMT109 |
Glutamate receptor ionotropic, AMPA 2 |
Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
TCMC1480
|
TCMT110 |
Glutamate receptor ionotropic, AMPA 4 |
Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
TCMC1480
|
TCMT111 |
Glutamate receptor ionotropic kainate 5 |
Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
TCMC1480
|
TCMT660 |
Metabotropic glutamate receptor 8 |
Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
TCMC1480
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
TCMC1480
|
TCMT653 |
Metabotropic glutamate receptor 1 |
Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT654 |
Metabotropic glutamate receptor 5 |
Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT657 |
Metabotropic glutamate receptor 4 |
Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT655 |
Metabotropic glutamate receptor 2 |
Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT664 |
Excitatory amino acid transporter 3 |
Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
TCMC1480
|
TCMT656 |
Metabotropic glutamate receptor 3 |
Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
TCMC632
|
TCMT597 |
Solute carrier family 28 member 3 |
Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
TCMC632
|
TCMT709 |
Sodium/nucleoside cotransporter 2 |
Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT710 |
Sodium/nucleoside cotransporter 1 |
Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT296 |
Adenosine A1 receptor |
Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
TCMC632
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC1982
|
TCMT239 |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
TCMC1982
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
TCMC1982
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
TCMC1982
|
TCMT44 |
Glyoxalase I |
Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
TCMC1982
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
TCMC1982
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
TCMC1982
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
TCMC1982
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
TCMC1982
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
TCMC1982
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
TCMC1982
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
TCMC1982
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
TCMC1982
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
TCMC1982
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
TCMC1982
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
TCMC1982
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
TCMC1982
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
TCMC1982
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
TCMC1982
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
TCMC1982
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
TCMC1982
|
TCMT320 |
Matrix metalloproteinase 3 |
Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
TCMC1982
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
TCMC1982
|
TCMT322 |
Matrix metalloproteinase 13 |
Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
TCMC1982
|
TCMT422 |
CaM kinase II beta |
Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
TCMC1982
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1982
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
TCMC1982
|
TCMT784 |
Vasopressin V2 receptor |
Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
TCMC1982
|
TCMT785 |
Interleukin-8 receptor A |
Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
TCMC1982
|
TCMT786 |
C-C chemokine receptor type 4 |
Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
TCMC1982
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
TCMC1982
|
TCMT601 |
Thrombin |
Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
TCMC1982
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
TCMC1982
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
TCMC1982
|
TCMT791 |
Protein kinase N1 |
Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
TCMC1982
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
TCMC1982
|
TCMT462 |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
TCMC1982
|
TCMT445 |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
TCMC1982
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
TCMC1982
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
TCMC1982
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
TCMC1982
|
TCMT388 |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
TCMC1982
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
TCMC1982
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
TCMC1982
|
TCMT402 |
ALK tyrosine kinase receptor |
Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
TCMC1982
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
TCMC1982
|
TCMT592 |
Xanthine dehydrogenase |
Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
TCMC1982
|
TCMT793 |
Liver glycogen phosphorylase |
Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
TCMC1982
|
TCMT33 |
Cytochrome P450 3A4 |
Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
TCMC1982
|
TCMT217 |
Cytochrome P450 2C8 |
Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
TCMC1982
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
TCMC1839
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
TCMC1839
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
TCMC1839
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
TCMC1839
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
TCMC1839
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
TCMC1839
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1839
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
TCMC1839
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
TCMC1839
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1839
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
TCMC1839
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
TCMC847
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
TCMC847
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
TCMC847
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
TCMC847
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
TCMC847
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
TCMC847
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC847
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
TCMC847
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
TCMC847
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
TCMC847
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
TCMC847
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
TCMC847
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
TCMC847
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
TCMC847
|
TCMT295 |
Matrix metalloproteinase-1 |
Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
TCMC847
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
TCMC1974
|
TCMT905 |
P2X purinoceptor 1 |
Homo sapiens |
IC50: 10000 (nM), Ref: 23510563 |