TCM Putative Target References: TCMH2710


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1211
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 270 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 270 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 750 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 2200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC486
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9500 (nM), Ref: 18579385
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC609
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 10000 (nM), Ref: 18501600
Ki: 10000 (nM), Ref: 18579385
Ki: 10000 (nM), Ref: 26520662
TCMC609
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6200 (nM), Ref: 18501600
Ki: 6200 (nM), Ref: 18579385
Ki: 6200 (nM), Ref: 26520662
TCMC609
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4100 (nM), Ref: 18579385
TCMC609
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9100 (nM), Ref: 18579385
TCMC609
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7100 (nM), Ref: 18579385
TCMC609
TCMT216 Myoglobin Homo sapiens IC50: 2300 (nM), Ref: 24482730
TCMC337
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9670 (nM), Ref: 21282059
TCMC337
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1020 (nM), Ref: 21282059
TCMC337
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9070 (nM), Ref: 21282059
TCMC337
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8230 (nM), Ref: 21282059
TCMC337
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 550 (nM), Ref: 22668600
TCMC337
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3220 (nM), Ref: 22668600
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC678
TCMT269 Prostanoid IP receptor Homo sapiens IC50: 1400 (nM), Ref: 10.1016/0960-894X(95)00168-S
Ki: 150 (nM), Ref: 11454474
TCMC903
TCMT175 G-protein coupled bile acid receptor 1 Homo sapiens IC50: 6000 (nM), Ref: 20801037
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC364
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 480 (nM), Ref: 21675776
Ki: 470 (nM), Ref: 22044209
TCMC364
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 1300 (nM), Ref: 21675776
Ki: 1400 (nM), Ref: 22044209
Ki: 1400 (nM), Ref: 23865723
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC37
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC715
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC555
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 15 (nM), Ref: 16392816
TCMC555
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens Ki: 52 (nM), Ref: 16392816
TCMC555
TCMT314 Serotonin 2c (5-HT2c) receptor Homo sapiens Ki: 42 (nM), Ref: 16392816
TCMC555
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 13 (nM), Ref: 16945532
Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
TCMC555
TCMT316 Melatonin receptor 1A Homo sapiens Ki: 210 (nM), Ref: 26023814
TCMC555
TCMT317 Melatonin receptor 1B Homo sapiens Ki: 16 (nM), Ref: 26023814
TCMC820
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 23768907
TCMC2099
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 10 (nM), Ref: 20590092
TCMC2099
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 840 (nM), Ref: 20590092
TCMC2099
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 830 (nM), Ref: 20590092
TCMC2099
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 990 (nM), Ref: 20590092
TCMC2099
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 710 (nM), Ref: 20590092
TCMC2099
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 860 (nM), Ref: 20590092
TCMC2195
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
TCMC2195
TCMT335 Myeloperoxidase Homo sapiens IC50: 770 (nM), Ref: 23581551
TCMC2195
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1700 (nM), Ref: 22696418
TCMC693
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 210 (nM), Ref: 16309907
IC50: 180 (nM), Ref: 17890084
TCMC693
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 16309907
IC50: 9.9 (nM), Ref: 17890084
TCMC693
TCMT187 Androgen Receptor Homo sapiens IC50: 212 (nM), Ref: 16309907
TCMC424
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 550 (nM), Ref: 21282059
TCMC424
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 21282059
TCMC424
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4410 (nM), Ref: 21282059
TCMC424
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3670 (nM), Ref: 21282059
TCMC424
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 650 (nM), Ref: 22668600
TCMC424
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7170 (nM), Ref: 22668600
TCMC1139
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 2 (nM), Ref: 16722623
TCMC1139
TCMT236 Estrogen receptor beta Homo sapiens IC50: 8.1 (nM), Ref: 16722623
TCMC1139
TCMT344 Aldehyde oxidase Homo sapiens IC50: 570 (nM), Ref: 20853847
Ki: 3600 (nM), Ref: 22996261
Ki: 430 (nM), Ref: 22996261
TCMC1139
TCMT218 Cytochrome P450 2B6 Homo sapiens Ki: 800 (nM), Ref: 16248836
Ki: 900 (nM), Ref: 16248836
TCMC1139
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 2200 (nM), Ref: 23241029
TCMC1139
TCMT348 Sulfotransferase 1A1 Homo sapiens IC50: 20 (nM), Ref: 22593037
Ki: 19 (nM), Ref: 22593037
Ki: 8.9 (nM), Ref: 22593037
Ki: 14.9 (nM), Ref: 22593037
TCMC1139
TCMT349 Nuclear receptor subfamily 1 group I member 3 Homo sapiens IC50: 3000 (nM), Ref: 26717202
TCMC505
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 4880 (nM), Ref: 15658857
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC619
TCMT293 Muscarinic acetylcholine receptor M2 Homo sapiens Ki: 158.49 (nM), Ref: 18077164
TCMC619
TCMT291 Muscarinic acetylcholine receptor M3 Homo sapiens Ki: 7079.46 (nM), Ref: 18077164
TCMC619
TCMT551 Muscarinic acetylcholine receptor M4 Homo sapiens Ki: 8511.38 (nM), Ref: 18077164
TCMC619
TCMT290 Muscarinic acetylcholine receptor M5 Homo sapiens Ki: 9772.37 (nM), Ref: 18077164
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC743
TCMT302 HMG-CoA reductase Homo sapiens IC50: 6 (nM), Ref: 15686906
IC50: 12.9 (nM), Ref: 23570542
TCMC743
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 5100 (nM), Ref: 21256005
TCMC743
TCMT278 Solute carrier organic anion transporter family member 1B1 Homo sapiens IC50: 600 (nM), Ref: 22587986
IC50: 800 (nM), Ref: 22587986
IC50: 1600 (nM), Ref: 22587986
TCMC619
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens Ki: 7943.28 (nM), Ref: 21920761
TCMC351
TCMT150 Nuclear receptor ROR-gamma Homo sapiens Ki: 10 (nM), Ref: 10.1039/C3MD00005B
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1731
TCMT167 Aldo-keto-reductase family 1 member C3 Homo sapiens IC50: 480 (nM), Ref: 16183274
IC50: 1100 (nM), Ref: 22877157
TCMC1731
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 211 (nM), Ref:
TCMC1330
TCMT246 Histamine H4 receptor Homo sapiens Ki: 14.45 (nM), Ref: 14640553
Ki: 7.943 (nM), Ref: 15454206
Ki: 12.02 (nM), Ref: 18357976
Ki: 13.4 (nM), Ref: 18459760
Ki: 12.02 (nM), Ref: 20192225
Ki: 60 (nM), Ref: 20452213
Ki: 7.943 (nM), Ref: 21044842
Ki: 12.59 (nM), Ref: 21044842
Ki: 12.02 (nM), Ref: 21348462
Ki: 15.85 (nM), Ref: 22003888
Ki: 9 (nM), Ref: 22153663
Ki: 19.95 (nM), Ref: 10.1039/C2MD20212C
Ki: 4.8 (nM), Ref: 25993395
Ki: 8 (nM), Ref: 25993395
Ki: 15.85 (nM), Ref: 10.1039/C5MD00022J
TCMC1330
TCMT242 Histamine H3 receptor Homo sapiens Ki: 5.2 (nM), Ref: 20384344
Ki: 10 (nM), Ref: 21044842
Ki: 11.75 (nM), Ref: 21348462
Ki: 6.31 (nM), Ref: 22003888
Ki: 16 (nM), Ref: 25993395
TCMC1330
TCMT245 Histamine H2 receptor Homo sapiens Ki: 5000 (nM), Ref: 25993395
TCMC1330
TCMT244 Histamine H1 receptor Homo sapiens Ki: 6000 (nM), Ref: 25993395
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1061
TCMT582 Prostanoid EP1 receptor Homo sapiens Ki: 9.1 (nM), Ref: 17531488
Ki: 9.1 (nM), Ref: 18039575
Ki: 18 (nM), Ref: 24279689
TCMC1061
TCMT583 Prostanoid EP2 receptor Homo sapiens Ki: 4.9 (nM), Ref: 17531488
Ki: 4.9 (nM), Ref: 17931866
Ki: 4.9 (nM), Ref: 18039575
IC50: 2.2 (nM), Ref: 23582449
Ki: 1.7 (nM), Ref: 23466604
IC50: 3.3 (nM), Ref: 23466604
Ki: 38 (nM), Ref: 24279689
IC50: 2.6 (nM), Ref: 26988801
TCMC1061
TCMT584 Prostanoid EP3 receptor Homo sapiens Ki: 0.33 (nM), Ref: 17531488
Ki: 0.33 (nM), Ref: 18039575
Ki: 5 (nM), Ref: 24279689
TCMC1061
TCMT585 Prostanoid EP4 receptor Homo sapiens Ki: 0.79 (nM), Ref: 17531488
Ki: 0.79 (nM), Ref: 17931866
Ki: 0.79 (nM), Ref: 18039575
Ki: 1.9 (nM), Ref: 18983139
IC50: 3.8 (nM), Ref: 18983139
Ki: 0.45 (nM), Ref: 23403082
IC50: 1.1 (nM), Ref: 23403082
Ki: 0.17 (nM), Ref: 23466604
IC50: 0.45 (nM), Ref: 23466604
Ki: 3.1 (nM), Ref: 24279689
TCMC1061
TCMT269 Prostanoid IP receptor Homo sapiens IC50: 260 (nM), Ref: 24279689
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1364
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 4000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC1411
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1261 (nM), Ref: 20696580
TCMC1411
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 56 (nM), Ref: 20696580
TCMC1411
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 17 (nM), Ref: 20696580
TCMC1411
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 212.9 (nM), Ref: 26498393
TCMC1411
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.4 (nM), Ref: 26498393
TCMC1411
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 54.9 (nM), Ref: 26498393
Ki: 220 (nM), Ref: 26498393
TCMC1411
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 440 (nM), Ref: 26498393
TCMC895
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 8990 (nM), Ref:
TCMC895
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 3012 (nM), Ref: IC50: 2197 (nM), Ref:
TCMC895
TCMT608 Solute carrier family 22 member 3 Homo sapiens IC50: 410 (nM), Ref: 23241029
TCMC895
TCMT213 Solute carrier family 22 member 1 Homo sapiens IC50: 210 (nM), Ref: 23241029
TCMC895
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 400 (nM), Ref: 23241029
TCMC895
TCMT310 Multidrug and toxin extrusion protein 2 Homo sapiens IC50: 500 (nM), Ref: 23241029
TCMC895
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 700 (nM), Ref: 23241029
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC2148
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 3200 (nM), Ref: 24920381
TCMC633
TCMT620 Heat shock cognate 71 kDa protein Homo sapiens IC50: 280 (nM), Ref:
TCMC1582
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1582
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 820 (nM), Ref: 22668600
TCMC1582
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5500 (nM), Ref: 22668600
TCMC1582
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 780 (nM), Ref: 22668600
TCMC1582
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3400 (nM), Ref: 22668600
TCMC1582
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2600 (nM), Ref: 22668600
TCMC1112
TCMT203 Glucose-6-phosphate 1-dehydrogenase Homo sapiens Ki: 3400 (nM), Ref: 19231202
Ki: 3000 (nM), Ref: 19231202
IC50: 9400 (nM), Ref: 22506561
TCMC1470
TCMT630 Cysteinyl leukotriene receptor 1 Homo sapiens IC50: 7 (nM), Ref: 20875743
Ki: 0.29 (nM), Ref: 23403082
IC50: 0.7 (nM), Ref: 23403082
TCMC2025
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2025.72 (nM), Ref:
TCMC1584
TCMT571 Adenosine A2b receptor Homo sapiens Ki: 8200 (nM), Ref: 15084123
TCMC1584
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 680 (nM), Ref: 15084123
TCMC1480
TCMT107 Glutamate receptor ionotropic kainate 2 Homo sapiens Ki: 1106 (nM), Ref: 10821708
TCMC1480
TCMT108 Glutamate receptor ionotropic, AMPA 1 Homo sapiens Ki: 1360 (nM), Ref: 9357531
TCMC1480
TCMT109 Glutamate receptor ionotropic, AMPA 2 Homo sapiens Ki: 940 (nM), Ref: 9357531
TCMC1480
TCMT110 Glutamate receptor ionotropic, AMPA 4 Homo sapiens Ki: 868 (nM), Ref: 9357531
TCMC1480
TCMT111 Glutamate receptor ionotropic kainate 5 Homo sapiens Ki: 701 (nM), Ref: 9357531
TCMC1480
TCMT660 Metabotropic glutamate receptor 8 Homo sapiens IC50: 5.7 (nM), Ref: 15603952
TCMC1480
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 613 (nM), Ref: 16250647
TCMC1480
TCMT653 Metabotropic glutamate receptor 1 Homo sapiens Ki: 250 (nM), Ref: 17725337
Ki: 570 (nM), Ref: 19042134
Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT654 Metabotropic glutamate receptor 5 Homo sapiens Ki: 390 (nM), Ref: 17725337
Ki: 1160 (nM), Ref: 19042134
Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT657 Metabotropic glutamate receptor 4 Homo sapiens Ki: 2400 (nM), Ref: 17725337
Ki: 1400 (nM), Ref: 19042134
Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT655 Metabotropic glutamate receptor 2 Homo sapiens Ki: 6400 (nM), Ref: 19042134
Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT664 Excitatory amino acid transporter 3 Homo sapiens Ki: 51 (nM), Ref: 18578477
TCMC1480
TCMT656 Metabotropic glutamate receptor 3 Homo sapiens Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H
TCMC694
TCMT230 Estradiol 17-beta-dehydrogenase 3 Homo sapiens IC50: 758 (nM), Ref: 11086723
IC50: 758 (nM), Ref: 16078844
TCMC694
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 20 (nM), Ref: 8035427
Ki: 35 (nM), Ref: 26469743
TCMC949
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 19911821
TCMC949
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 48 (nM), Ref: 19911821
TCMC949
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9100 (nM), Ref: 19911821
TCMC949
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3300 (nM), Ref: 19911821
TCMC949
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 2000 (nM), Ref: 19911821
TCMC949
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 5200 (nM), Ref: 19911821
TCMC949
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9400 (nM), Ref: 19911821
TCMC949
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 6800 (nM), Ref: 19911821
TCMC949
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 5600 (nM), Ref: 19911821
TCMC949
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3100 (nM), Ref: 19911821
Ki: 3100 (nM), Ref: 21067924
Ki: 3100 (nM), Ref: 22137345
Ki: 3100 (nM), Ref: 22077347
Ki: 3100 (nM), Ref: 22365761
Ki: 3100 (nM), Ref: 22377674
Ki: 3100 (nM), Ref: 23241068
Ki: 3100 (nM), Ref: 22892213
Ki: 3100 (nM), Ref: 26688270
TCMC949
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9200 (nM), Ref: 21067924
Ki: 9200 (nM), Ref: 22137345
Ki: 9200 (nM), Ref: 22077347
Ki: 9200 (nM), Ref: 22365761
Ki: 9200 (nM), Ref: 22377674
Ki: 9200 (nM), Ref: 23241068
Ki: 9200 (nM), Ref: 22892213
Ki: 9200 (nM), Ref: 26688270
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC845
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 630 (nM), Ref: 19231207
TCMC662
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 250 (nM), Ref: 25743213
IC50: 1100 (nM), Ref: 25743213
TCMC1083
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 1.89 (nM), Ref: 10465538
Ki: 759 (nM), Ref: 10465538
Ki: 572 (nM), Ref: 8893836
Ki: 20 (nM), Ref: 10691700
Ki: 17 (nM), Ref: 10691700
Ki: 450 (nM), Ref: 18834111
Ki: 360 (nM), Ref: 18834111
Ki: 2100 (nM), Ref: 20155917
Ki: 2.9 (nM), Ref: 20155917
Ki: 2100 (nM), Ref: 22846798
Ki: 422 (nM), Ref: 23134120
Ki: 110 (nM), Ref: 23428965
Ki: 190 (nM), Ref: 23428965
Ki: 2100 (nM), Ref: 23727194
Ki: 8 (nM), Ref: 24138311
Ki: 8.73 (nM), Ref: 27035329
Ki: 3690 (nM), Ref: 27035329
Ki: 48 (nM), Ref: 27132867
TCMC1083
TCMT651 Dopamine D3 receptor Homo sapiens Ki: 13.2 (nM), Ref: 8893836
Ki: 50 (nM), Ref: 10691700
Ki: 240 (nM), Ref: 18834111
Ki: 72 (nM), Ref: 18834111
Ki: 15 (nM), Ref: 22846798
Ki: 20 (nM), Ref: 23134120
Ki: 21 (nM), Ref: 23428965
Ki: 15 (nM), Ref: 23727194
Ki: 7.58 (nM), Ref: 27035329
Ki: 293 (nM), Ref: 27035329
TCMC1083
TCMT635 Dopamine transporter Homo sapiens Ki: 6400 (nM), Ref: 14592523
IC50: 460 (nM), Ref: 14592523
TCMC1083
TCMT634 Norepinephrine transporter Homo sapiens IC50: 6.63 (nM), Ref: 14592523
TCMC1083
TCMT648 Dopamine D4 receptor Homo sapiens Ki: 1.2 (nM), Ref: 10691700
Ki: 6.2 (nM), Ref: 18834111
Ki: 8.9 (nM), Ref: 23428965
TCMC1083
TCMT316 Melatonin receptor 1A Homo sapiens Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083
TCMT317 Melatonin receptor 1B Homo sapiens Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 4470 (nM), Ref: 23134120
TCMC1083
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC837
TCMT690 Histone deacetylase 3 Homo sapiens IC50: 9000 (nM), Ref: 21874153
TCMC256
TCMT203 Glucose-6-phosphate 1-dehydrogenase Homo sapiens IC50: 4300 (nM), Ref: 22506561
TCMC1930
TCMT203 Glucose-6-phosphate 1-dehydrogenase Homo sapiens Ki: 8900 (nM), Ref: 19231202
Ki: 6200 (nM), Ref: 19231202
TCMC1044
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1400 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 4300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 2400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC287
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3200 (nM), Ref: 15916432
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC2025
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 5600 (nM), Ref: 23353736
TCMC43
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 220 (nM), Ref: 26588603
IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 26701186
TCMC43
TCMT208 Monoamine oxidase A Homo sapiens Ki: 710 (nM), Ref: 26819666
TCMC43
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3100 (nM), Ref: 27190601
IC50: 1500 (nM), Ref: 27190601
TCMC2142
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 600 (nM), Ref: 6827528
TCMC2142
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 10000 (nM), Ref: 14552748
TCMC2142
TCMT187 Androgen Receptor Homo sapiens IC50: 3.9 (nM), Ref: 15456242
IC50: 2.7 (nM), Ref: 16309907
IC50: 4.571 (nM), Ref: 22746350
IC50: 4.17 (nM), Ref: 25646649
IC50: 4.27 (nM), Ref: 25646649
TCMC2142
TCMT99 Testis-specific androgen-binding protein Homo sapiens IC50: 14 (nM), Ref: 17149875
TCMC2142
TCMT725 Voltage-gated L-type calcium channel alpha-1C subunit Homo sapiens IC50: 34 (nM), Ref: 22761000
IC50: 38.4 (nM), Ref: 22761000
TCMC963
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 500 (nM), Ref: 15357993
Ki: 500 (nM), Ref: 15454240
Ki: 500 (nM), Ref: 15501038
Ki: 500 (nM), Ref: 21208801
Ki: 500 (nM), Ref: 26525863
Ki: 500 (nM), Ref: 26853167
Ki: 500 (nM), Ref: 27283786
TCMC963
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4000 (nM), Ref: 15501038
TCMC1499
TCMT131 Acetylcholinesterase Homo sapiens IC50: 1 (nM), Ref: 18181565
TCMC1499
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 0 (nM), Ref: 17976864
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1401
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 15 (nM), Ref: 21561086
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1758
TCMT247 Alpha-2a adrenergic receptor Homo sapiens Ki: 66 (nM), Ref: 8632424
TCMC1758
TCMT243 Alpha-2c adrenergic receptor Homo sapiens Ki: 63 (nM), Ref: 8632424
TCMC1758
TCMT559 Beta-2 adrenergic receptor Homo sapiens Ki: 3300 (nM), Ref: 27132867
TCMC1758
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 1300 (nM), Ref: 27132867
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC1043
TCMT191 Signal transducer and activator of transcription 3 Homo sapiens IC50: 1862 (nM), Ref:
TCMC1043
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 2000 (nM), Ref: 24040486
IC50: 4000 (nM), Ref: 10.1039/C3MD00005B
IC50: 4100 (nM), Ref: 24502334
IC50: 1980 (nM), Ref: 24502334
TCMC1043
TCMT744 Sodium/potassium-transporting ATPase alpha-1 chain Homo sapiens IC50: 290 (nM), Ref: 26122772
TCMC635
TCMT460 MAP kinase-activated protein kinase 2 Homo sapiens IC50: 2800 (nM), Ref: 19919896
IC50: 6300 (nM), Ref: 19919896
TCMC635
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 3370 (nM), Ref:
TCMC2025
TCMT359 Tyrosine-protein kinase FYN Homo sapiens IC50: 1300 (nM), Ref: 17315853
IC50: 3600 (nM), Ref: 17315853
Ki: 7500 (nM), Ref: 17315853
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1743
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 4400 (nM), Ref: 15634016
TCMC1743
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens Ki: 7200 (nM), Ref: 15686879
Ki: 6300 (nM), Ref: 15908213
Ki: 630 (nM), Ref: 16171993
Ki: 10000 (nM), Ref: 17722904
Ki: 1000 (nM), Ref: 19331415
Ki: 1023.29 (nM), Ref: 20828128
Ki: 1000 (nM), Ref: 21920761
Ki: 1000 (nM), Ref: 22243960
Ki: 3000 (nM), Ref: 22793665
Ki: 3000 (nM), Ref: 23126648
Ki: 3800 (nM), Ref: 23561269
IC50: 7600 (nM), Ref: 23561269
Ki: 3000 (nM), Ref: 23692872
TCMC1743
TCMT552 Neuronal acetylcholine receptor subunit alpha-3 Homo sapiens IC50: 45 (nM), Ref: 11312774
TCMC634
TCMT284 Fructose-1,6-bisphosphatase Homo sapiens IC50: 1000 (nM), Ref: 19348494
IC50: 440 (nM), Ref: 19969452
IC50: 140 (nM), Ref: 19969452
IC50: 9800 (nM), Ref: 20116906
IC50: 3200 (nM), Ref: 24530031
IC50: 1000 (nM), Ref: 10.1039/C0MD00269K
IC50: 3200 (nM), Ref: 25461330
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC452
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2370 (nM), Ref: 21282059
TCMC452
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 600 (nM), Ref: 21282059
TCMC452
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4530 (nM), Ref: 21282059
TCMC452
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3530 (nM), Ref: 21282059
TCMC452
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3170 (nM), Ref: 21669522
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1136
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 330 (nM), Ref: 16480268
IC50: 218 (nM), Ref: 18035543
IC50: 109 (nM), Ref: 19836949
Ki: 9500 (nM), Ref: 21413808
TCMC1136
TCMT236 Estrogen receptor beta Homo sapiens IC50: 31 (nM), Ref: 16610787
TCMC1136
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 29 (nM), Ref: 16610787
IC50: 96 (nM), Ref: 19836949
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1136
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2500 (nM), Ref: 26469743
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1744
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 10000 (nM), Ref: 14552748
IC50: 5620 (nM), Ref: 23033255
TCMC1744
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 8290 (nM), Ref: 8917655
TCMC1744
TCMT778 Voltage-gated potassium channel subunit Kv1.5 Homo sapiens IC50: 6100 (nM), Ref: 19004630
TCMC1744
TCMT780 Voltage-gated L-type calcium channel alpha-1D subunit Homo sapiens IC50: 1350 (nM), Ref: 24754640
TCMC1744
TCMT725 Voltage-gated L-type calcium channel alpha-1C subunit Homo sapiens IC50: 22 (nM), Ref: 22761000
IC50: 55 (nM), Ref: 22761000
TCMC1744
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 2300 (nM), Ref: 23033255
TCMC1744
TCMT31 Cytochrome P450 2C19 Homo sapiens IC50: 5420 (nM), Ref: 23033255
TCMC1744
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 4080 (nM), Ref: 23033255
TCMC1744
TCMT220 Cytochrome P450 2J2 Homo sapiens IC50: 3060 (nM), Ref: 23033255
TCMC1744
TCMT407 Myosin light chain kinase, smooth muscle Homo sapiens IC50: 2020 (nM), Ref: 26385444
TCMC649
TCMT783 Mineralocorticoid receptor Homo sapiens IC50: 9.268 (nM), Ref: 20812681
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC2098
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1400 (nM), Ref: 20590092
TCMC2098
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1110 (nM), Ref: 20590092
TCMC2098
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 112 (nM), Ref: 20590092
TCMC2098
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 1220 (nM), Ref: 20590092
TCMC2098
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 1440 (nM), Ref: 20590092
TCMC2098
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 1410 (nM), Ref: 20590092
TCMC2098
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 1230 (nM), Ref: 20590092
TCMC2098
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 1370 (nM), Ref: 20590092
TCMC2098
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 1000 (nM), Ref: 20590092
TCMC339
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 10000 (nM), Ref: 15658857
IC50: 10000 (nM), Ref: 19110342
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC2183
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens IC50: 7000 (nM), Ref: 23713606
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1477
TCMT273 Bile acid receptor FXR Homo sapiens IC50: 7860 (nM), Ref: 23688559
TCMC1477
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 5600 (nM), Ref: 21030469
IC50: 4900 (nM), Ref: 21030469
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC880
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9910 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 20185318
Ki: 9900 (nM), Ref: 22245047
Ki: 9900 (nM), Ref: 26073005
Ki: 9900 (nM), Ref: 26520662
TCMC880
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4200 (nM), Ref: 18579385
Ki: 4200 (nM), Ref: 20185318
TCMC880
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 18579385
Ki: 8900 (nM), Ref: 20185318
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC1824
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 2596 (nM), Ref: 23332369
IC50: 2600 (nM), Ref: 23895532
TCMC1824
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 9.2 (nM), Ref: 23332369
IC50: 7.7 (nM), Ref: 23895532
TCMC1824
TCMT277 Solute carrier organic anion transporter family member 1B3 Homo sapiens Ki: 1800 (nM), Ref: 25618019
IC50: 260 (nM), Ref: 25618019
TCMC1824
TCMT278 Solute carrier organic anion transporter family member 1B1 Homo sapiens Ki: 840 (nM), Ref: 25618019
IC50: 280 (nM), Ref: 25618019
TCMC1824
TCMT393 Proto-oncogene tyrosine-protein kinase MER Homo sapiens IC50: 4900 (nM), Ref: 27238842
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC952
TCMT803 Hypoxanthine-guanine phosphoribosyltransferase Homo sapiens Ki: 5800 (nM), Ref: 19527031
Ki: 5800 (nM), Ref: 25915781
TCMC1155
TCMT230 Estradiol 17-beta-dehydrogenase 3 Homo sapiens IC50: 330 (nM), Ref: 11086723
IC50: 330 (nM), Ref: 16078844
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2063
TCMT646 Serotonin 5a (5-HT5a) receptor Homo sapiens Ki: 126 (nM), Ref: 12825922
IC50: 180 (nM), Ref: 18983139
Ki: 110 (nM), Ref: 18983139
IC50: 184 (nM), Ref: 18588282
Ki: 170 (nM), Ref: 21726069
IC50: 280 (nM), Ref: 23582449
Ki: 82 (nM), Ref: 23466604
IC50: 160 (nM), Ref: 23466604
IC50: 180 (nM), Ref: 26988801
TCMC2063
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 65 (nM), Ref: 12825922
Ki: 100 (nM), Ref: 15357994
IC50: 200 (nM), Ref: 18983139
Ki: 93 (nM), Ref: 18983139
IC50: 262 (nM), Ref: 18588282
IC50: 27.5 (nM), Ref: 20170099
Ki: 84 (nM), Ref: 21726069
Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
IC50: 180 (nM), Ref: 23582449
Ki: 50 (nM), Ref: 23466604
IC50: 100 (nM), Ref: 23466604
Ki: 33 (nM), Ref: 24805037
Ki: 33 (nM), Ref: 25557493
IC50: 120 (nM), Ref: 26988801
Ki: 100 (nM), Ref: 26996373
TCMC2063
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 8.1 (nM), Ref: 12825922
IC50: 0.61 (nM), Ref: 18983139
Ki: 0.22 (nM), Ref: 18983139
IC50: 2.55 (nM), Ref: 12713409
IC50: 1.5 (nM), Ref: 18588282
Ki: 0.13 (nM), Ref: 21726069
IC50: 0.49 (nM), Ref: 23582449
Ki: 0.11 (nM), Ref: 23466604
IC50: 0.29 (nM), Ref: 23466604
Ki: 1.4 (nM), Ref: 24763360
Ki: 0.8 (nM), Ref: 24805037
Ki: 0.8 (nM), Ref: 25557493
IC50: 0.25 (nM), Ref: 26988801
TCMC2063
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 14 (nM), Ref: 15081042
Ki: 8.2 (nM), Ref: 16392816
Ki: 14 (nM), Ref: 16257207
Ki: 120 (nM), Ref: 18468904
Ki: 160 (nM), Ref: 18468904
Ki: 130 (nM), Ref: 18468904
Ki: 150 (nM), Ref: 18468904
Ki: 320 (nM), Ref: 11975483
Ki: 690 (nM), Ref: 17067154
Ki: 323.59 (nM), Ref: 23301527
Ki: 320 (nM), Ref: 23301527
TCMC2063
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens Ki: 12 (nM), Ref: 15081042
Ki: 13 (nM), Ref: 12954071
Ki: 13 (nM), Ref: 16392816
Ki: 12 (nM), Ref: 16257207
Ki: 13.49 (nM), Ref: 24582985
TCMC2063
TCMT314 Serotonin 2c (5-HT2c) receptor Homo sapiens Ki: 6.9 (nM), Ref: 15081042
Ki: 8.3 (nM), Ref: 12954071
Ki: 8.3 (nM), Ref: 16392816
Ki: 6.9 (nM), Ref: 16257207
Ki: 130 (nM), Ref: 11975483
Ki: 20 (nM), Ref: 17067154
Ki: 79.43 (nM), Ref: 23301527
Ki: 79 (nM), Ref: 23301527
TCMC2063
TCMT815 Serotonin 1d (5-HT1d) receptor Homo sapiens Ki: 5.5 (nM), Ref: 8071931
Ki: 0.5 (nM), Ref: 18507369
TCMC2063
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 2.5 (nM), Ref: 7658447
IC50: 1.2 (nM), Ref: 12954071
Ki: 1.259 (nM), Ref: 18433113
Ki: 10000 (nM), Ref: 18433113
Ki: 0.62 (nM), Ref: 22748706
Ki: 0.9 (nM), Ref: 23332346
Ki: 9.5 (nM), Ref: 24161678
Ki: 2.08 (nM), Ref: 25128671
TCMC2063
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 79 (nM), Ref: 16250647
TCMC2063
TCMT816 Serotonin 1b (5-HT1b) receptor Homo sapiens Ki: 1.1 (nM), Ref: 18507369
IC50: 29 (nM), Ref: 18983139
Ki: 18 (nM), Ref: 18983139
Ki: 14 (nM), Ref: 21726069
IC50: 12 (nM), Ref: 23582449
Ki: 4 (nM), Ref: 23466604
IC50: 6.5 (nM), Ref: 23466604
TCMC2063
TCMT817 Serotonin 4 (5-HT4) receptor Homo sapiens Ki: 1049 (nM), Ref: 19334715
Ki: 500 (nM), Ref: 17067154
Ki: 29.51 (nM), Ref: 19223092
Ki: 109.65 (nM), Ref: 19223092
TCMC2063
TCMT645 Serotonin 1e (5-HT1e) receptor Homo sapiens Ki: 10.72 (nM), Ref: 24365159
Ki: 11 (nM), Ref: 24365159
TCMC336
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6500 (nM), Ref: 22668600
TCMC336
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7200 (nM), Ref: 22668600
TCMC336
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5900 (nM), Ref: 22668600
TCMC336
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC336
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5200 (nM), Ref: 22668600
TCMC336
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5700 (nM), Ref: 22668600
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1869
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 4410 (nM), Ref: 15658857
TCMC1111
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 11.78 (nM), Ref: 18242087
IC50: 13 (nM), Ref: 18653260
IC50: 778 (nM), Ref: 20851614
IC50: 778 (nM), Ref: 21376605
IC50: 8.6 (nM), Ref: 21873057
IC50: 29.1 (nM), Ref: 23747808
IC50: 29.1 (nM), Ref: 25590374
TCMC1111
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 257 (nM), Ref: 20851614
IC50: 257 (nM), Ref: 21376605
IC50: 1.22 (nM), Ref: 23747808
IC50: 1.2 (nM), Ref: 25590374
TCMC1111
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4900 (nM), Ref: 21561086
TCMC983
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2800 (nM), Ref: 15887952
IC50: 2800 (nM), Ref: 15887952
IC50: 1200 (nM), Ref: 12502307
IC50: 2800 (nM), Ref:
TCMC983
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 7300 (nM), Ref: 21030469
TCMC983
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 718.7 (nM), Ref: 26498393
TCMC983
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.2 (nM), Ref: 26498393
TCMC983
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 56.4 (nM), Ref: 26498393
TCMC1119
TCMT559 Beta-2 adrenergic receptor Homo sapiens Ki: 360 (nM), Ref: 27132867
TCMC1119
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 910 (nM), Ref: 27132867
TCMC1119
TCMT247 Alpha-2a adrenergic receptor Homo sapiens Ki: 160 (nM), Ref: 27265687
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC1878
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 300 (nM), Ref: 24200808
TCMC689
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 50 (nM), Ref: 16078824
Ki: 72 (nM), Ref: 16213718
Ki: 70 (nM), Ref: 16570929
Ki: 70 (nM), Ref: 16682198
Ki: 72 (nM), Ref: 16279794
Ki: 72 (nM), Ref: 17561406
Ki: 70 (nM), Ref: 19161308
Ki: 72 (nM), Ref: 19331413
Ki: 11 (nM), Ref: 19361197
Ki: 70 (nM), Ref: 22044209
Ki: 89 (nM), Ref: 23865723
Ki: 72 (nM), Ref: 25065940
TCMC689
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 180 (nM), Ref: 16213718
Ki: 180 (nM), Ref: 16570929
Ki: 180 (nM), Ref: 16682198
Ki: 180 (nM), Ref: 19161308
Ki: 168 (nM), Ref: 19361197
Ki: 371 (nM), Ref: 23865723
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC381
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 207 (nM), Ref: 19836949
TCMC2157
TCMT296 Adenosine A1 receptor Homo sapiens Ki: 6200 (nM), Ref: 15214785
Ki: 0.6 (nM), Ref: 15664822
Ki: 6200 (nM), Ref: 16335918
Ki: 6920 (nM), Ref: 16759111
Ki: 6200 (nM), Ref: 16789747
Ki: 6200 (nM), Ref: 17665891
Ki: 6200 (nM), Ref: 19301821
Ki: 6200 (nM), Ref: 18468446
Ki: 6200 (nM), Ref: 19569717
Ki: 6770 (nM), Ref: 20188574
Ki: 6770 (nM), Ref: 24139167
Ki: 6770 (nM), Ref: 10.1039/C5MD00573F
TCMC2157
TCMT571 Adenosine A2b receptor Homo sapiens Ki: 7059 (nM), Ref: 15664822
Ki: 9070 (nM), Ref: 16250640
Ki: 9070 (nM), Ref: 16759111
Ki: 7850 (nM), Ref: 19569717
Ki: 9070 (nM), Ref: 20188574
Ki: 2700 (nM), Ref: 20202853
Ki: 9070 (nM), Ref: 20537438
Ki: 9070 (nM), Ref: 24139167
Ki: 9070 (nM), Ref: 26824742
TCMC2157
TCMT707 Adenosine A2a receptor Homo sapiens Ki: 0.6 (nM), Ref: 15664822
Ki: 7900 (nM), Ref: 16335918
Ki: 6700 (nM), Ref: 16759111
Ki: 7900 (nM), Ref: 16789747
Ki: 7900 (nM), Ref: 17665891
Ki: 7900 (nM), Ref: 19301821
Ki: 7900 (nM), Ref: 18468446
Ki: 4200 (nM), Ref: 19569717
Ki: 6700 (nM), Ref: 20188574
Ki: 1700 (nM), Ref: 23200243
Ki: 2030 (nM), Ref: 23200243
Ki: 6700 (nM), Ref: 24139167
Ki: 1710 (nM), Ref: 10.1039/C5MD00573F
TCMC2157
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 14 (nM), Ref: 15664822
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1377
TCMT186 Monoamine oxidase B Homo sapiens Ki: 3000 (nM), Ref: 16137882
Ki: 3000 (nM), Ref: 19342233
IC50: 7943.28 (nM), Ref: 20934874
Ki: 5340 (nM), Ref: 21134756
Ki: 3000 (nM), Ref: 21778064
Ki: 2000 (nM), Ref: 24140951
TCMC1377
TCMT208 Monoamine oxidase A Homo sapiens Ki: 8380 (nM), Ref: 21134756
TCMC850
TCMT307 HERG Homo sapiens IC50: 4897.79 (nM), Ref: 21185626
TCMC850
TCMT707 Adenosine A2a receptor Homo sapiens Ki: 5011.87 (nM), Ref: 21661720
Ki: 9560 (nM), Ref: 23200243
Ki: 2480 (nM), Ref: 23200243
TCMC850
TCMT131 Acetylcholinesterase Homo sapiens IC50: 7250 (nM), Ref: 23791077
TCMC317
TCMT223 Aldose reductase Homo sapiens IC50: 10 (nM), Ref: 18087047
TCMC204
TCMT803 Hypoxanthine-guanine phosphoribosyltransferase Homo sapiens Ki: 5400 (nM), Ref: 25915781
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC1078
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC588
TCMT855 Nuclear receptor ROR-alpha Homo sapiens Ki: 12 (nM), Ref: 10.1039/C3MD00005B
TCMC1359
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 3000 (nM), Ref: 9544212
IC50: 6900 (nM), Ref: 17517512
IC50: 212 (nM), Ref: IC50: 290 (nM), Ref: 23651359
IC50: 1860 (nM), Ref: 23651359
TCMC1359
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 6200 (nM), Ref: 17517512
IC50: 1100 (nM), Ref: 19884005
IC50: 1100 (nM), Ref: 19500994
IC50: 1100 (nM), Ref: 20097072
IC50: 1100 (nM), Ref: 20202839
IC50: 1100 (nM), Ref: 20576432
IC50: 1400 (nM), Ref: 21280601
IC50: 1100 (nM), Ref: 21641217
IC50: 1100 (nM), Ref: 22148253
IC50: 1350 (nM), Ref: 22091869
IC50: 1100 (nM), Ref: 23200247
IC50: 4300 (nM), Ref: 25221653
IC50: 1100 (nM), Ref: 26487917
IC50: 1100 (nM), Ref: 26691756
TCMC1504
TCMT273 Bile acid receptor FXR Homo sapiens IC50: 18.3 (nM), Ref: 24775917
TCMC1977
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7410 (nM), Ref: 21669522
TCMC1977
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 540 (nM), Ref: 21669522
TCMC1977
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 520 (nM), Ref: 21669522
TCMC1498
TCMT864 Thyroid hormone receptor alpha Homo sapiens IC50: 0.24 (nM), Ref: 16099653
IC50: 0.24 (nM), Ref: 17543524
Ki: 0.33 (nM), Ref: 18975928
Ki: 2.33 (nM), Ref: 22542282
Ki: 2.33 (nM), Ref: 23276448
IC50: 3.2 (nM), Ref: 24290064
TCMC1498
TCMT69 Thyroid hormone receptor beta-1 Homo sapiens IC50: 0.26 (nM), Ref: 16099653
IC50: 0.26 (nM), Ref: 17543524
IC50: 0.257 (nM), Ref: 17524652
Ki: 0.68 (nM), Ref: 18975928
Ki: 2.29 (nM), Ref: 22542282
Ki: 2.29 (nM), Ref: 23276448
IC50: 2.9 (nM), Ref: 24290064
TCMC1498
TCMT796 Proliferating cell nuclear antigen Homo sapiens IC50: 3600 (nM), Ref: 23395113
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC2212
TCMT868 UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit Homo sapiens IC50: 1800 (nM), Ref: 21273069
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC2238
TCMT131 Acetylcholinesterase Homo sapiens IC50: 9000 (nM), Ref: 23791077
TCMC2113
TCMT883 Lysine-specific demethylase 5C Homo sapiens IC50: 4500 (nM), Ref: 22724510
TCMC2113
TCMT884 Histone lysine demethylase PHF8 Homo sapiens IC50: 2300 (nM), Ref: 22724510
TCMC2113
TCMT885 Lysine-specific demethylase 2A Homo sapiens IC50: 570 (nM), Ref: 22724510
TCMC341
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 19231207
TCMC2114
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 2200 (nM), Ref: 25743213
TCMC2114
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 9000 (nM), Ref: 27135370
TCMC811
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 2030 (nM), Ref: 19097799
TCMC811
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 9900 (nM), Ref: 18533708
TCMC811
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10.2 (nM), Ref: 20413308
TCMC811
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7078.5 (nM), Ref: 26498393
TCMC811
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 371.5 (nM), Ref: 26498393
TCMC811
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.5 (nM), Ref: 26498393
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1494
TCMT267 GABA receptor rho-1 subunit Homo sapiens IC50: 91 (nM), Ref: 10.1584/jpestics.R07-07
TCMC1494
TCMT891 GABA receptor beta-3 subunit Homo sapiens IC50: 0.9 (nM), Ref: 10.1584/jpestics.R07-07
TCMC560
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 50 (nM), Ref: 15771424
TCMC560
TCMT817 Serotonin 4 (5-HT4) receptor Homo sapiens Ki: 26.92 (nM), Ref: 19223092
Ki: 245.47 (nM), Ref: 19223092
TCMC2201
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8700 (nM), Ref: 21332115
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2039
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 5400 (nM), Ref: 10.1016/S0960-894X(97)00194-7
TCMC1200
TCMT897 Voltage-gated calcium channel alpha2/delta subunit 1 Homo sapiens IC50: 27 (nM), Ref: 15050626
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC772
TCMT131 Acetylcholinesterase Homo sapiens Ki: 955 (nM), Ref: 15828829
TCMC772
TCMT132 Butyrylcholinesterase Homo sapiens Ki: 2050 (nM), Ref: 15828829
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1856
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 500 (nM), Ref: 20590092
TCMC1856
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 52 (nM), Ref: 20590092
TCMC1856
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 44 (nM), Ref: 20590092
TCMC1856
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 540 (nM), Ref: 20590092
TCMC1856
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 740 (nM), Ref: 20590092
TCMC1856
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 420 (nM), Ref: 20590092
TCMC1856
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 380 (nM), Ref: 20590092
TCMC1856
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 450 (nM), Ref: 20590092
TCMC1856
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 500 (nM), Ref: 20590092
TCMC1742
TCMT637 NAD-dependent deacetylase sirtuin 3 Homo sapiens IC50: 6200 (nM), Ref: 25275824
TCMC1742
TCMT638 NAD-dependent deacetylase sirtuin 2 Homo sapiens IC50: 6300 (nM), Ref: 25549554
IC50: 1200 (nM), Ref: 26696402
TCMC740
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.77 (nM), Ref: 16250647
TCMC740
TCMT675 Beta-1 adrenergic receptor Homo sapiens IC50: 600 (nM), Ref: 18983139
Ki: 430 (nM), Ref: 18983139
IC50: 1740 (nM), Ref: 18588282
IC50: 1640 (nM), Ref: 20875743
Ki: 170 (nM), Ref: 21726069
Ki: 150 (nM), Ref: 23466604
IC50: 260 (nM), Ref: 23466604
IC50: 210 (nM), Ref: 26988801
TCMC2082
TCMT302 HMG-CoA reductase Homo sapiens Ki: 2.6 (nM), Ref: 15686898
IC50: 11.2 (nM), Ref: 15686898
IC50: 11 (nM), Ref: 15686906
IC50: 6110 (nM), Ref: 25311563
IC50: 39.81 (nM), Ref: 25311563
TCMC1940
TCMT187 Androgen Receptor Homo sapiens Ki: 8.5 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12781197
IC50: 37 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 9873735
IC50: 37 (nM), Ref: 9784110
Ki: 35 (nM), Ref: 20510622
TCMC1940
TCMT613 Glucocorticoid receptor Homo sapiens Ki: 30.5 (nM), Ref: 12954062
Ki: 30.5 (nM), Ref: 9873735
Ki: 30.5 (nM), Ref: 9784110
TCMC1940
TCMT783 Mineralocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 12954062
IC50: 14 (nM), Ref: 12781197
IC50: 14 (nM), Ref: 9784110
IC50: 30 (nM), Ref: 8709117
TCMC1940
TCMT904 Progesterone receptor Homo sapiens Ki: 3.5 (nM), Ref: 10212133
IC50: 3.5 (nM), Ref: 11859003
Ki: 3.5 (nM), Ref: 9464361
IC50: 5 (nM), Ref: 8523399
Ki: 3.8 (nM), Ref: 9667968
Ki: 3.467 (nM), Ref: 16821785
Ki: 3.4 (nM), Ref: 18553958
Ki: 5.1 (nM), Ref: 20510622
TCMC1541
TCMT317 Melatonin receptor 1B Homo sapiens Ki: 0.3 (nM), Ref: 15203165
Ki: 0.41 (nM), Ref: 12646022
Ki: 0.29 (nM), Ref: 10.1016/S0960-894X(97)00444-7
Ki: 0.195 (nM), Ref: 12213063
Ki: 0.31 (nM), Ref: 11960497
Ki: 0.7 (nM), Ref: 15713384
Ki: 0.7 (nM), Ref: 15380218
Ki: 0.2818 (nM), Ref: 15293992
Ki: 0.2818 (nM), Ref: 15943478
Ki: 0.35 (nM), Ref: 16759094
Ki: 0.257 (nM), Ref: 17149869
Ki: 0.3 (nM), Ref: 17481904
Ki: 0.3548 (nM), Ref: 17346859
Ki: 0.3388 (nM), Ref: 17459711
Ki: 0.2399 (nM), Ref: 18052314
IC50: 0.53 (nM), Ref: 18372181
Ki: 0.41 (nM), Ref: 18778943
Ki: 0.955 (nM), Ref: 19193160
Ki: 0.741 (nM), Ref: 18657980
Ki: 0.429 (nM), Ref: 20227878
Ki: 0.6166 (nM), Ref: 20674373
Ki: 0.34 (nM), Ref: 21420861
IC50: 0.53 (nM), Ref: 21377769
Ki: 0.21 (nM), Ref: 21473625
Ki: 0.35 (nM), Ref: 21392858
Ki: 0.21 (nM), Ref: 21568291
Ki: 0.3388 (nM), Ref: 21775151
Ki: 0.34 (nM), Ref: 21764185
Ki: 0.5 (nM), Ref: 23265885
Ki: 0.429 (nM), Ref: 23228808
Ki: 0.955 (nM), Ref: 10.1039/C1MD00149C
Ki: 0.41 (nM), Ref: 25232966
Ki: 0.15 (nM), Ref: 26023814
Ki: 0.15 (nM), Ref: 26367450
Ki: 0.955 (nM), Ref: 10.1039/C5MD00190K
Ki: 0.52 (nM), Ref: 26820449
Ki: 0.34 (nM), Ref: 26785296
TCMC1541
TCMT316 Melatonin receptor 1A Homo sapiens Ki: 0.14 (nM), Ref: 12646022
Ki: 0.2 (nM), Ref: 10.1016/S0960-894X(97)00444-7
Ki: 0.0823 (nM), Ref: 12213063
Ki: 0.12 (nM), Ref: 11960497
Ki: 0.3 (nM), Ref: 15713384
Ki: 0.3 (nM), Ref: 15380218
Ki: 0.2884 (nM), Ref: 15293992
Ki: 0.2884 (nM), Ref: 15943478
Ki: 0.39 (nM), Ref: 16759094
Ki: 0.3236 (nM), Ref: 17149869
Ki: 0.2 (nM), Ref: 17481904
Ki: 0.389 (nM), Ref: 17346859
Ki: 0.263 (nM), Ref: 17459711
Ki: 0.1413 (nM), Ref: 18052314
IC50: 0.2 (nM), Ref: 18372181
IC50: 0.18 (nM), Ref: 18983139
Ki: 0.11 (nM), Ref: 18983139
Ki: 0.14 (nM), Ref: 18778943
Ki: 0.4571 (nM), Ref: 19193160
Ki: 0.525 (nM), Ref: 18657980
Ki: 0.296 (nM), Ref: 20227878
Ki: 0.3311 (nM), Ref: 20674373
Ki: 0.25 (nM), Ref: 21420861
IC50: 0.2 (nM), Ref: 21377769
Ki: 0.24 (nM), Ref: 21473625
Ki: 0.22 (nM), Ref: 21392858
Ki: 0.24 (nM), Ref: 21568291
Ki: 0.37 (nM), Ref: 21726069
Ki: 0.263 (nM), Ref: 21775151
Ki: 0.25 (nM), Ref: 21764185
Ki: 0.2 (nM), Ref: 23265885
Ki: 0.296 (nM), Ref: 23228808
IC50: 0.53 (nM), Ref: 23582449
Ki: 0.35 (nM), Ref: 23466604
IC50: 0.44 (nM), Ref: 23466604
Ki: 0.4571 (nM), Ref: 10.1039/C1MD00149C
Ki: 0.14 (nM), Ref: 25232966
Ki: 0.091 (nM), Ref: 26023814
Ki: 0.091 (nM), Ref: 26367450
Ki: 0.4571 (nM), Ref: 10.1039/C5MD00190K
Ki: 0.23 (nM), Ref: 26820449
Ki: 0.25 (nM), Ref: 26785296
IC50: 0.11 (nM), Ref: 26988801
TCMC1541
TCMT329 Quinone reductase 2 Homo sapiens IC50: 64.6 (nM), Ref: 21377769
TCMC307
TCMT333 C-terminal-binding protein 2 Homo sapiens IC50: 7340 (nM), Ref: 27156192
TCMC1540
TCMT302 HMG-CoA reductase Homo sapiens Ki: 23.5 (nM), Ref: 15686898
IC50: 4000 (nM), Ref: 15686898
TCMC736
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 2400 (nM), Ref: 19884005
IC50: 2400 (nM), Ref: 19500994
IC50: 2400 (nM), Ref: 20097072
IC50: 2400 (nM), Ref: 20576432
IC50: 2400 (nM), Ref: 22361134
IC50: 2400 (nM), Ref: 22148253
IC50: 2400 (nM), Ref: 23200247
TCMC736
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 4192 (nM), Ref:
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC2082
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 3700 (nM), Ref: 22328583
TCMC2082
TCMT278 Solute carrier organic anion transporter family member 1B1 Homo sapiens IC50: 4400 (nM), Ref: 22587986
IC50: 6000 (nM), Ref: 22587986
TCMC1974
TCMT905 P2X purinoceptor 1 Homo sapiens IC50: 10000 (nM), Ref: 23510563
TCMC1836
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 2800 (nM), Ref: 23241029
IC50: 2800 (nM), Ref: 23241029
TCMC1836
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 1500 (nM), Ref: 23241029
TCMC1836
TCMT60 Fatty acid synthase Homo sapiens Ki: 4100 (nM), Ref: 25513712
TCMC1067
TCMT307 HERG Homo sapiens IC50: 2570.4 (nM), Ref: 21185626
TCMC1067
TCMT244 Histamine H1 receptor Homo sapiens Ki: 14.79 (nM), Ref: 21944853
TCMC827
TCMT307 HERG Homo sapiens IC50: 891.25 (nM), Ref: 21185626
TCMC1130
TCMT633 Serotonin transporter Homo sapiens Ki: 1 (nM), Ref: 19720528
Ki: 1 (nM), Ref: 20347298
IC50: 4600 (nM), Ref: 24237160
Ki: 7.4 (nM), Ref: 24944746
Ki: 2.2 (nM), Ref: 26153715
TCMC1509
TCMT116 Mu opioid receptor Homo sapiens Ki: 0.53 (nM), Ref: 15454210
TCMC1236
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 15341953
IC50: 10 (nM), Ref: 15456246
IC50: 98.7 (nM), Ref: 15887952
IC50: 98.7 (nM), Ref: 15887952
IC50: 9.7 (nM), Ref: 15943471
IC50: 10 (nM), Ref: 16098741
IC50: 1.3 (nM), Ref: 16219463
IC50: 61 (nM), Ref: 16610787
IC50: 25 (nM), Ref: 17149865
IC50: 395 (nM), Ref: 17049855
IC50: 9.7 (nM), Ref: 17188490
IC50: 6.8 (nM), Ref: 17574424
IC50: 18 (nM), Ref: 12502307
IC50: 98.7 (nM), Ref:
TCMC1236
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 395 (nM), Ref: 15341953
IC50: 395 (nM), Ref: 15456246
IC50: 4660 (nM), Ref: 15887952
IC50: 4660 (nM), Ref: 15887952
IC50: 395 (nM), Ref: 15943471
IC50: 395 (nM), Ref: 16098741
IC50: 29.4 (nM), Ref: 16219463
IC50: 1973 (nM), Ref: 16610787
IC50: 1145 (nM), Ref: 17149865
IC50: 2150 (nM), Ref: 17696335
IC50: 9.7 (nM), Ref: 17049855
IC50: 395 (nM), Ref: 17188490
IC50: 580 (nM), Ref: 17574424
IC50: 300 (nM), Ref: 12502307
IC50: 4680 (nM), Ref:
TCMC883
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 1880 (nM), Ref: 11844666
IC50: 6300 (nM), Ref: 10197970
IC50: 1689 (nM), Ref: 15454242
IC50: 2600 (nM), Ref: 15615524
IC50: 1689 (nM), Ref: 19520573
IC50: 2600 (nM), Ref: 19791801
IC50: 7000 (nM), Ref: 21570308
IC50: 723 (nM), Ref: IC50: 6650 (nM), Ref: 23473947
IC50: 2600 (nM), Ref: 24440378
TCMC883
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 230 (nM), Ref: 11906292
IC50: 1000 (nM), Ref: 10465547
IC50: 1000 (nM), Ref: 10406640
IC50: 68 (nM), Ref: 15454242
IC50: 1200 (nM), Ref: 15546727
IC50: 1200 (nM), Ref: 15916445
IC50: 6 (nM), Ref: 16250658
IC50: 6.8 (nM), Ref: 16250658
IC50: 330 (nM), Ref: 16814546
IC50: 2.2 (nM), Ref: 16806914
IC50: 1300 (nM), Ref: 17335184
IC50: 350 (nM), Ref: 15615524
IC50: 35 (nM), Ref: 17604631
IC50: 540 (nM), Ref: 17915854
IC50: 1200 (nM), Ref: 17994684
IC50: 300 (nM), Ref: 18063374
IC50: 300 (nM), Ref: 17532544
IC50: 1000 (nM), Ref: 17976864
IC50: 2900 (nM), Ref: 19059783
IC50: 80 (nM), Ref: 16252917
IC50: 540 (nM), Ref: 18752957
IC50: 800 (nM), Ref: 19097798
IC50: 120 (nM), Ref: 19136259
IC50: 120 (nM), Ref: 19296694
IC50: 63 (nM), Ref: 19520573
IC50: 68 (nM), Ref: 19520573
IC50: 336 (nM), Ref: 19520573
IC50: 120 (nM), Ref: 19500994
IC50: 120 (nM), Ref: 20097072
IC50: 540 (nM), Ref: 19957931
IC50: 350 (nM), Ref: 19791801
IC50: 800 (nM), Ref: 20451397
IC50: 65 (nM), Ref: 20576432
IC50: 65 (nM), Ref: 20655211
IC50: 300 (nM), Ref: 20970223
IC50: 40 (nM), Ref: 21215625
IC50: 30 (nM), Ref: 21316237
IC50: 10 (nM), Ref: 21434686
IC50: 70 (nM), Ref: 21641217
IC50: 190 (nM), Ref: 21570308
IC50: 100 (nM), Ref: 22119153
IC50: 540 (nM), Ref: 21992176
IC50: 40 (nM), Ref: 22386983
IC50: 70 (nM), Ref: 22361134
IC50: 60 (nM), Ref: 22341941
IC50: 60 (nM), Ref: 22560838
IC50: 140 (nM), Ref: 22749420
IC50: 40 (nM), Ref: 22263894
IC50: 54 (nM), Ref: 22263894
IC50: 42 (nM), Ref: 23010270
IC50: 57 (nM), Ref: 10.1007/s00044-012-0174-z
IC50: 70 (nM), Ref: 23200247
IC50: 100 (nM), Ref: 23353741
IC50: 870 (nM), Ref: 23473947
IC50: 20 (nM), Ref: 23706267
IC50: 320 (nM), Ref: 24211633
IC50: 40 (nM), Ref: 24332492
IC50: 57 (nM), Ref: 24295787
IC50: 540 (nM), Ref: 24373735
IC50: 350 (nM), Ref: 24440378
IC50: 40 (nM), Ref: 24602792
IC50: 280 (nM), Ref: 24607877
IC50: 72 (nM), Ref: 24656662
IC50: 70 (nM), Ref: 24650702
IC50: 2660 (nM), Ref: 24661847
IC50: 40 (nM), Ref: 24745964
IC50: 270 (nM), Ref: 24836072
IC50: 280 (nM), Ref: 24780593
IC50: 290 (nM), Ref: 24900871
IC50: 40 (nM), Ref: 24631898
IC50: 40 (nM), Ref: 24934992
IC50: 50 (nM), Ref: 25221653
IC50: 19 (nM), Ref: 25819096
IC50: 52 (nM), Ref: 25866240
IC50: 16 (nM), Ref: 25980909
IC50: 40 (nM), Ref: 25956953
IC50: 130 (nM), Ref: 26081289
IC50: 19 (nM), Ref: 26316467
IC50: 900 (nM), Ref: 26546221
IC50: 260 (nM), Ref: 26638042
IC50: 870 (nM), Ref: 26691756
IC50: 40 (nM), Ref: 10.1039/C5MD00278H
IC50: 40 (nM), Ref: 26898334
IC50: 40 (nM), Ref: 26898334
IC50: 40 (nM), Ref: 27019010
IC50: 310 (nM), Ref: 27349331
TCMC883
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 880 (nM), Ref: 15686931
Ki: 880 (nM), Ref: 20605094
Ki: 880 (nM), Ref: 23067387
TCMC883
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 21 (nM), Ref: 15686931
Ki: 21 (nM), Ref: 16134940
IC50: 21 (nM), Ref: 16220969
Ki: 21 (nM), Ref: 16290146
Ki: 21 (nM), Ref: 19317447
Ki: 21 (nM), Ref: 19124253
Ki: 21 (nM), Ref: 19193158
Ki: 21 (nM), Ref: 19338333
Ki: 21 (nM), Ref: 19520577
Ki: 21 (nM), Ref: 19846301
Ki: 21 (nM), Ref: 20605094
Ki: 21 (nM), Ref: 20624682
Ki: 21 (nM), Ref: 21208801
Ki: 21 (nM), Ref: 21251841
Ki: 21 (nM), Ref: 21757360
Ki: 21 (nM), Ref: 21852133
IC50: 181 (nM), Ref: Ki: 21 (nM), Ref: 22285172
Ki: 21 (nM), Ref: 22424239
Ki: 21 (nM), Ref: 23067387
Ki: 21 (nM), Ref: 23181552
Ki: 21 (nM), Ref: 23391336
Ki: 21 (nM), Ref: 22883029
Ki: 21 (nM), Ref: 23867389
Ki: 21 (nM), Ref: 23965175
Ki: 21 (nM), Ref: 24314394
Ki: 21 (nM), Ref: 24513184
Ki: 21 (nM), Ref: 24792813
Ki: 21 (nM), Ref: 25129169
Ki: 21 (nM), Ref: 25533402
Ki: 21 (nM), Ref: 25773015
Ki: 21 (nM), Ref: 25882523
Ki: 21 (nM), Ref: 25766630
Ki: 21 (nM), Ref: 26174556
Ki: 21 (nM), Ref: 26525863
Ki: 21 (nM), Ref: 26691758
Ki: 21 (nM), Ref: 26850377
Ki: 21 (nM), Ref: 26832216
Ki: 21 (nM), Ref: 26920803
TCMC883
TCMT507 MAP kinase p38 alpha Homo sapiens IC50: 810 (nM), Ref: 15990304
TCMC883
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 16 (nM), Ref: 16134940
IC50: 16 (nM), Ref: 16220969
Ki: 16 (nM), Ref: 16290146
Ki: 16 (nM), Ref: 19193158
Ki: 16 (nM), Ref: 20605094
Ki: 16 (nM), Ref: 21852133
Ki: 16 (nM), Ref: 23067387
Ki: 16 (nM), Ref: 23965175
Ki: 16 (nM), Ref: 24513184
Ki: 16 (nM), Ref: 25766630
TCMC883
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 18 (nM), Ref: 16290146
Ki: 18 (nM), Ref: 20605094
Ki: 18 (nM), Ref: 21852133
Ki: 18 (nM), Ref: 23067387
Ki: 18 (nM), Ref: 23965175
Ki: 18 (nM), Ref: 24513184
Ki: 18 (nM), Ref: 25766630
TCMC883
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 94 (nM), Ref: 19193158
Ki: 94 (nM), Ref: 20605094
Ki: 94 (nM), Ref: 23067387
TCMC883
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 794 (nM), Ref: 20605094
Ki: 794 (nM), Ref: 23067387
TCMC883
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 93 (nM), Ref: 20605094
Ki: 93 (nM), Ref: 23067387
TCMC883
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 2170 (nM), Ref: 20605094
Ki: 2170 (nM), Ref: 23067387
Ki: 2170 (nM), Ref: 23867389
Ki: 2170 (nM), Ref: 23965175
Ki: 2170 (nM), Ref: 24287559
Ki: 2170 (nM), Ref: 25766630
TCMC883
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 98 (nM), Ref: 20605094
Ki: 98 (nM), Ref: 23067387
TCMC883
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 689 (nM), Ref: 20605094
Ki: 689 (nM), Ref: 23067387
TCMC1236
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 10 (nM), Ref: 17482813
TCMC1236
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 395 (nM), Ref: 17482813
TCMC883
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7400 (nM), Ref: 23067387
TCMC883
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 540 (nM), Ref: 26653180
IC50: 425 (nM), Ref: 26653180
TCMC1236
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 2210 (nM), Ref: 18533708
TCMC2184
TCMT912 Retinoic acid receptor gamma Homo sapiens Ki: 0.7 (nM), Ref: 11412986
Ki: 0.6 (nM), Ref: 10.1016/S0960-894X(97)00420-4
Ki: 0.04 (nM), Ref: 9435893
Ki: 0.5 (nM), Ref: 10.1016/S0960-894X(01)80113-X
TCMC2184
TCMT833 Retinoic acid receptor alpha Homo sapiens Ki: 0.1 (nM), Ref: 10.1016/S0960-894X(97)00420-4
IC50: 9000 (nM), Ref: 15615521
TCMC2184
TCMT913 Retinoic acid receptor beta Homo sapiens Ki: 4.1 (nM), Ref: 9435893
IC50: 3000 (nM), Ref: 15615521
TCMC2184
TCMT735 Retinoid X receptor alpha Homo sapiens Ki: 330 (nM), Ref: 9435893
TCMC2184
TCMT914 Retinoid X receptor beta Homo sapiens Ki: 54 (nM), Ref: 9435893
TCMC2184
TCMT915 Retinoid X receptor gamma Homo sapiens Ki: 120 (nM), Ref: 9435893
TCMC1236
TCMT344 Aldehyde oxidase Homo sapiens IC50: 340 (nM), Ref: 20853847
TCMC2184
TCMT893 Nuclear receptor ROR-beta Homo sapiens IC50: 0.15 (nM), Ref: 10.1039/C3MD00005B
IC50: 125.89 (nM), Ref: 25305688
TCMC2184
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 199.53 (nM), Ref: 25305688
TCMC2184
TCMT855 Nuclear receptor ROR-alpha Homo sapiens IC50: 199.53 (nM), Ref: 25305688
TCMC1236
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 7720 (nM), Ref:
TCMC1946
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 1900 (nM), Ref: 15993593
IC50: 5011.87 (nM), Ref: 26565745
TCMC1946
TCMT559 Beta-2 adrenergic receptor Homo sapiens Ki: 3.69 (nM), Ref: 24326276
Ki: 0.46 (nM), Ref: 24326276
IC50: 50.12 (nM), Ref: 26565745
TCMC1946
TCMT48 Sodium channel protein type V alpha subunit Homo sapiens IC50: 2100 (nM), Ref: 21300721
TCMC1946
TCMT675 Beta-1 adrenergic receptor Homo sapiens IC50: 251.19 (nM), Ref: 26565745
TCMC1946
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens IC50: 3981.07 (nM), Ref: 26565745
TCMC1746
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 980 (nM), Ref: 19719236
TCMC2179
TCMT331 Plasminogen Homo sapiens IC50: 3100 (nM), Ref: 23521080
IC50: 3100 (nM), Ref: 24900876
TCMC1585
TCMT220 Cytochrome P450 2J2 Homo sapiens IC50: 4870 (nM), Ref: 23033255
TCMC1060
TCMT586 Prostanoid FP receptor Homo sapiens IC50: 7 (nM), Ref: 10715159
IC50: 2.5 (nM), Ref: 10915040
TCMC1060
TCMT582 Prostanoid EP1 receptor Homo sapiens IC50: 380 (nM), Ref: 10715159
TCMC1060
TCMT584 Prostanoid EP3 receptor Homo sapiens IC50: 322 (nM), Ref: 10715159
TCMC1060
TCMT585 Prostanoid EP4 receptor Homo sapiens IC50: 4200 (nM), Ref: 10715159
TCMC1060
TCMT921 Prostanoid DP receptor Homo sapiens IC50: 4500 (nM), Ref: 10715159
TCMC2064
TCMT633 Serotonin transporter Homo sapiens IC50: 3 (nM), Ref: 16314097
IC50: 3 (nM), Ref: 21093273
TCMC2064
TCMT635 Dopamine transporter Homo sapiens IC50: 310 (nM), Ref: 16314097
IC50: 310 (nM), Ref: 21093273
TCMC2064
TCMT634 Norepinephrine transporter Homo sapiens IC50: 825 (nM), Ref: 16314097
IC50: 825 (nM), Ref: 21093273
TCMC2064
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 2880 (nM), Ref: 23033255
TCMC151
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 1610 (nM), Ref: 19719236
TCMC1665
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1665
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1338
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 328 (nM), Ref: 21377369
Ki: 328 (nM), Ref: 21757360
Ki: 328 (nM), Ref: 22285172
Ki: 328 (nM), Ref: 23181552
Ki: 328 (nM), Ref: 23391336
Ki: 328 (nM), Ref: 22883029
Ki: 328 (nM), Ref: 24792813
Ki: 328 (nM), Ref: 25129169
Ki: 328 (nM), Ref: 25533402
Ki: 328 (nM), Ref: 25773015
Ki: 328 (nM), Ref: 25882523
Ki: 328 (nM), Ref: 26525863
Ki: 328 (nM), Ref: 26691758
Ki: 328 (nM), Ref: 26850377
Ki: 328 (nM), Ref: 26920803
TCMC1338
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 290 (nM), Ref: 21377369
Ki: 290 (nM), Ref: 21757360
Ki: 290 (nM), Ref: 22285172
Ki: 290 (nM), Ref: 23181552
Ki: 290 (nM), Ref: 23391336
Ki: 290 (nM), Ref: 22883029
Ki: 290 (nM), Ref: 24314394
Ki: 290 (nM), Ref: 24792813
Ki: 290 (nM), Ref: 25129169
Ki: 290 (nM), Ref: 25533402
Ki: 290 (nM), Ref: 25773015
Ki: 290 (nM), Ref: 25882523
Ki: 290 (nM), Ref: 26174556
Ki: 290 (nM), Ref: 26525863
Ki: 290 (nM), Ref: 26691758
Ki: 290 (nM), Ref: 26850377
Ki: 290 (nM), Ref: 26832216
Ki: 290 (nM), Ref: 26920803
TCMC2224
TCMT634 Norepinephrine transporter Homo sapiens Ki: 385 (nM), Ref: 18557608
IC50: 535 (nM), Ref: 18557608
IC50: 535 (nM), Ref: 20378347
IC50: 581 (nM), Ref: 20724153
IC50: 680 (nM), Ref: 24900709
Ki: 1623 (nM), Ref: 23602445
IC50: 7943.28 (nM), Ref: 23602445
IC50: 5722 (nM), Ref: 24974340
TCMC2224
TCMT633 Serotonin transporter Homo sapiens IC50: 31 (nM), Ref: 18557608
IC50: 27 (nM), Ref: 20378347
IC50: 35 (nM), Ref: 20724153
Ki: 11 (nM), Ref: 24900709
Ki: 113 (nM), Ref: 23602445
IC50: 323.59 (nM), Ref: 23602445
IC50: 36.1 (nM), Ref: 24974340
TCMC2224
TCMT635 Dopamine transporter Homo sapiens IC50: 7340 (nM), Ref: 20724153
Ki: 3620 (nM), Ref: 23602445
IC50: 9120.11 (nM), Ref: 23602445
TCMC137
TCMT923 Adenylate cyclase type 10 Homo sapiens IC50: 3000 (nM), Ref: 18630896
TCMC1574
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1989
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 82 (nM), Ref: 11170639
Ki: 63.1 (nM), Ref: 17880057
Ki: 220 (nM), Ref: 18595716
Ki: 101 (nM), Ref: 22268448
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
Ki: 202 (nM), Ref:
TCMC1989
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens Ki: 251.19 (nM), Ref: 17880057
TCMC1989
TCMT651 Dopamine D3 receptor Homo sapiens Ki: 251.19 (nM), Ref: 17880057
Ki: 320 (nM), Ref: 18595716
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 79.43 (nM), Ref: 17880057
Ki: 230 (nM), Ref: 18595716
Ki: 125 (nM), Ref: 22268448
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 63.1 (nM), Ref: 17880057
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT292 Muscarinic acetylcholine receptor M1 Homo sapiens Ki: 398.11 (nM), Ref: 17880057
Ki: 100 (nM), Ref: 18595716
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT551 Muscarinic acetylcholine receptor M4 Homo sapiens Ki: 125.89 (nM), Ref: 17880057
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT244 Histamine H1 receptor Homo sapiens Ki: 8.7 (nM), Ref: 18595716
Ki: 10 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 1300 (nM), Ref: 18595716
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 1400 (nM), Ref: 18595716
TCMC1989
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 180 (nM), Ref: 18595716
Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
Ki: 400 (nM), Ref:
TCMC1989
TCMT648 Dopamine D4 receptor Homo sapiens Ki: 2200 (nM), Ref: 18595716
TCMC1989
TCMT314 Serotonin 2c (5-HT2c) receptor Homo sapiens Ki: 1400 (nM), Ref: 18595716
Ki: 2000 (nM), Ref:
TCMC1989
TCMT307 HERG Homo sapiens IC50: 5754.4 (nM), Ref: 21185626
TCMC1989
TCMT643 Alpha-1a adrenergic receptor Homo sapiens Ki: 100 (nM), Ref: 10.1039/C2MD00311B
Ki: 20 (nM), Ref:
TCMC1989
TCMT650 Alpha-1b adrenergic receptor Homo sapiens Ki: 100 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT647 Alpha-2b adrenergic receptor Homo sapiens Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT243 Alpha-2c adrenergic receptor Homo sapiens Ki: 100 (nM), Ref: 10.1039/C2MD00311B
TCMC1989
TCMT924 Histone H1.0 Homo sapiens Ki: 10 (nM), Ref:
TCMC563
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4690 (nM), Ref: 22137345
TCMC563
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 920 (nM), Ref: 22137345
TCMC660
TCMT592 Xanthine dehydrogenase Homo sapiens IC50: 7820 (nM), Ref: 17379526
Ki: 100 (nM), Ref: 25060641
Ki: 7300 (nM), Ref: 25019478
IC50: 2900 (nM), Ref: 26022844
Ki: 1550 (nM), Ref: 26712096
IC50: 200 (nM), Ref: 26762836
IC50: 950 (nM), Ref: 27162124
TCMC684
TCMT925 Solute carrier family 22 member 6 Homo sapiens Ki: 6020 (nM), Ref: 21571536
TCMC263
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 3000 (nM), Ref: 24924423
TCMC263
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens IC50: 8000 (nM), Ref: 24924423
TCMC683
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9900 (nM), Ref: 15745821
TCMC539
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 225 (nM), Ref: 20926163
IC50: 225 (nM), Ref: 22475216
Ki: 50 (nM), Ref: 22475216
TCMC222
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 3400 (nM), Ref: 10.1016/S0960-894X(97)00194-7
TCMC308
TCMT333 C-terminal-binding protein 2 Homo sapiens IC50: 240 (nM), Ref: 27156192
TCMC1762
TCMT33 Cytochrome P450 3A4 Homo sapiens Ki: 2110 (nM), Ref: 16248836
Ki: 5890 (nM), Ref: 16248836
TCMC1762
TCMT782 Cytochrome P450 3A5 Homo sapiens Ki: 4530 (nM), Ref: 16248836
TCMC2092
TCMT927 Somatostatin receptor 5 Homo sapiens Ki: 120 (nM), Ref: 11266182
Ki: 0.14 (nM), Ref: 11327607
IC50: 10 (nM), Ref: 15658865
Ki: 0.44 (nM), Ref: 15982879
Ki: 0.26 (nM), Ref: 15982879
Ki: 0.71 (nM), Ref: 15982879
Ki: 0.15 (nM), Ref: 15982879
Ki: 1.4 (nM), Ref: 16220980
IC50: 0.2 (nM), Ref: 16220980
IC50: 4.2 (nM), Ref: 21806016
Ki: 0.23 (nM), Ref: 24342240
IC50: 4.2 (nM), Ref: 24378707
Ki: 2 (nM), Ref: 10.1039/C4MD00074A
TCMC2092
TCMT928 Somatostatin receptor 2 Homo sapiens Ki: 0.049 (nM), Ref: 11327607
IC50: 0.7 (nM), Ref: 15658865
Ki: 0.083 (nM), Ref: 15982879
IC50: 0.4 (nM), Ref: 16220980
Ki: 0.23 (nM), Ref: 16220980
IC50: 0.67 (nM), Ref: 21806016
Ki: 0.0016 (nM), Ref: 24342240
IC50: 0.7 (nM), Ref: 24378707
TCMC2092
TCMT929 Somatostatin receptor 1 Homo sapiens Ki: 0.36 (nM), Ref: 11327607
IC50: 1.9 (nM), Ref: 15658865
Ki: 2.3 (nM), Ref: 16220980
IC50: 1.6 (nM), Ref: 21806016
IC50: 0.14 (nM), Ref: 23582449
Ki: 0.43 (nM), Ref: 24342240
IC50: 1.9 (nM), Ref: 24378707
TCMC2092
TCMT930 Somatostatin receptor 3 Homo sapiens Ki: 0.14 (nM), Ref: 11327607
IC50: 3.3 (nM), Ref: 15658865
Ki: 1.17 (nM), Ref: 16220980
IC50: 0.4 (nM), Ref: 16220980
IC50: 3.1 (nM), Ref: 21806016
Ki: 0.53 (nM), Ref: 24342240
IC50: 3.3 (nM), Ref: 24378707
TCMC2092
TCMT931 Somatostatin receptor 4 Homo sapiens Ki: 0.59 (nM), Ref: 11327607
IC50: 1.6 (nM), Ref: 15658865
Ki: 1.7 (nM), Ref: 16220980
IC50: 1.7 (nM), Ref: 21806016
Ki: 0.74 (nM), Ref: 24342240
IC50: 1.6 (nM), Ref: 24378707
Ki: 2 (nM), Ref: 10.1039/C4MD00074A
TCMC1169
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 760 (nM), Ref: 23241029
TCMC2034
TCMT567 DNA (cytosine-5)-methyltransferase 1 Homo sapiens IC50: 2000 (nM), Ref: 19362833
IC50: 800 (nM), Ref: 19364644
IC50: 4000 (nM), Ref: 20006515
IC50: 4000 (nM), Ref: 21958292
IC50: 941 (nM), Ref: 22483584
IC50: 900 (nM), Ref: 22280363
TCMC2034
TCMT568 DNA (cytosine-5)-methyltransferase 3B Homo sapiens IC50: 300 (nM), Ref: 19362833
IC50: 200 (nM), Ref: 19364644
IC50: 250 (nM), Ref: 20006515
TCMC2034
TCMT932 Histone-lysine N-methyltransferase, H3 lysine-79 specific Homo sapiens Ki: 160 (nM), Ref: 22924785
IC50: 600 (nM), Ref: 23433670
IC50: 600 (nM), Ref: 23433670
Ki: 160 (nM), Ref: 23879463
TCMC2034
TCMT757 Histone-arginine methyltransferase CARM1 Homo sapiens Ki: 400 (nM), Ref: 23879463
TCMC2034
TCMT1 Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 Homo sapiens Ki: 570 (nM), Ref: 23879463
IC50: 2000 (nM), Ref: 25746813
TCMC2034
TCMT934 N-lysine methyltransferase SMYD2 Homo sapiens IC50: 180 (nM), Ref: 25746813
TCMC2034
TCMT935 Histone-lysine N-methyltransferase SUV420H2 Homo sapiens IC50: 10000 (nM), Ref: 25746813
TCMC2034
TCMT937 Histone-lysine N-methyltransferase SUV39H1 Homo sapiens IC50: 1200 (nM), Ref: 25746813
TCMC2034
TCMT938 Histone-lysine N-methyltransferase SETDB1 Homo sapiens IC50: 2200 (nM), Ref: 25746813
TCMC2034
TCMT42 Histone-lysine N-methyltransferase MLL Homo sapiens IC50: 2300 (nM), Ref: 25746813
TCMC2034
TCMT940 Histone-lysine N-methyltransferase, H3 lysine-9 specific 5 Homo sapiens IC50: 230 (nM), Ref: 25746813
TCMC2034
TCMT941 Histone-lysine N-methyltransferase EZH1 Homo sapiens IC50: 6400 (nM), Ref: 25746813
TCMC2034
TCMT564 Protein-arginine N-methyltransferase 1 Homo sapiens IC50: 420 (nM), Ref: 25559100
IC50: 500 (nM), Ref: 26428871
TCMC2104
TCMT187 Androgen Receptor Homo sapiens Ki: 2 (nM), Ref: 9871534
IC50: 0 (nM), Ref: 9925725
Ki: 3 (nM), Ref: 9925725
Ki: 0.2 (nM), Ref: 17034117
IC50: 1.82 (nM), Ref: 17149866
Ki: 0.3 (nM), Ref: 17181141
Ki: 0.3 (nM), Ref: 17439112
Ki: 0.2 (nM), Ref: 17257838
Ki: 0.2 (nM), Ref: 17887661
Ki: 0.2 (nM), Ref: 17267219
Ki: 0.9 (nM), Ref: 18400499
Ki: 0.2 (nM), Ref: 18442912
IC50: 0.05 (nM), Ref: 18442912
IC50: 1 (nM), Ref: 19606870
Ki: 4.7 (nM), Ref: 20510622
IC50: 2.1 (nM), Ref: 22094279
IC50: 2.1 (nM), Ref: 23199477
IC50: 11 (nM), Ref: 10.1039/C3MD20341G
IC50: 13.1 (nM), Ref: 26305181
TCMC2104
TCMT99 Testis-specific androgen-binding protein Homo sapiens IC50: 3.8 (nM), Ref: 2296011
TCMC2104
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 1550 (nM), Ref: 2918514
Ki: 220 (nM), Ref: 2918514
TCMC216
TCMT945 Sphingosine 1-phosphate receptor Edg-1 Homo sapiens IC50: 0.16 (nM), Ref: 15149705
IC50: 0.67 (nM), Ref: 15615513
IC50: 0.47 (nM), Ref: 19081720
IC50: 0.78 (nM), Ref: 20304639
TCMC216
TCMT946 Sphingosine 1-phosphate receptor Edg-3 Homo sapiens IC50: 0.04 (nM), Ref: 15149705
IC50: 0.26 (nM), Ref: 15615513
IC50: 0.66 (nM), Ref: 19081720
IC50: 0.92 (nM), Ref: 20304639
TCMC216
TCMT947 Sphingosine 1-phosphate receptor Edg-6 Homo sapiens IC50: 23 (nM), Ref: 15149705
IC50: 34 (nM), Ref: 15615513
IC50: 2.4 (nM), Ref: 19081720
IC50: 1.04 (nM), Ref: 20304639
IC50: 2.9 (nM), Ref: 20446681
TCMC216
TCMT948 Sphingosine 1-phosphate receptor Edg-5 Homo sapiens IC50: 0.23 (nM), Ref: 15149705
IC50: 0.35 (nM), Ref: 15615513
TCMC216
TCMT949 Sphingosine 1-phosphate receptor Edg-8 Homo sapiens IC50: 0.55 (nM), Ref: 15615513
IC50: 1.1 (nM), Ref: 19081720
IC50: 2 (nM), Ref: 20304639
TCMC854
TCMT279 Vitamin D receptor Homo sapiens IC50: 0.7 (nM), Ref: 17149880
IC50: 0.8 (nM), Ref: 17924616
IC50: 9.3 (nM), Ref: 24035340
IC50: 0.08 (nM), Ref: 24742174
IC50: 0.06 (nM), Ref: 26515040
IC50: 0.35 (nM), Ref: 26613420
IC50: 0.1 (nM), Ref: 26613420
IC50: 1.13 (nM), Ref: 26562542
TCMC826
TCMT951 Bradykinin B2 receptor Homo sapiens Ki: 0.11 (nM), Ref: 10882364
Ki: 1.1 (nM), Ref: 23403082
IC50: 1.8 (nM), Ref: 23403082
TCMC1029
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 12 (nM), Ref: 16250647
TCMC129
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens IC50: 1000 (nM), Ref: 24924423
TCMC1822
TCMT760 Oxytocin receptor Homo sapiens Ki: 0.8 (nM), Ref: 12036367
IC50: 2.7 (nM), Ref: 17316912
Ki: 0.79 (nM), Ref: 25642985
Ki: 9.53 (nM), Ref: 25642985
Ki: 6.6 (nM), Ref: 25642985
Ki: 0.79 (nM), Ref: 25642985
Ki: 0.8 (nM), Ref: 26741855
Ki: 0.44 (nM), Ref: 27297999
TCMC1822
TCMT918 Vasopressin V1a receptor Homo sapiens Ki: 120 (nM), Ref: 12036367
Ki: 120 (nM), Ref: 25642985
TCMC1822
TCMT784 Vasopressin V2 receptor Homo sapiens Ki: 3500 (nM), Ref: 12036367
Ki: 1544 (nM), Ref: 25642985
TCMC1822
TCMT672 Vasopressin V1b receptor Homo sapiens Ki: 1782 (nM), Ref: 25642985
TCMC2174
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 500 (nM), Ref: 15771438
Ki: 430 (nM), Ref: 15771438
Ki: 9600 (nM), Ref: 15771438
Ki: 7700 (nM), Ref: 15771438
Ki: 5 (nM), Ref: 15686895
Ki: 5 (nM), Ref: 15686894
Ki: 5 (nM), Ref: 15686931
Ki: 5000 (nM), Ref: 15546717
Ki: 10.3 (nM), Ref: 15837316
Ki: 5 (nM), Ref: 16134940
Ki: 10 (nM), Ref: 16302824
Ki: 10 (nM), Ref: 16539401
Ki: 10 (nM), Ref: 16459077
Ki: 10 (nM), Ref: 17125255
Ki: 10 (nM), Ref: 17228881
Ki: 10 (nM), Ref: 17376683
Ki: 10 (nM), Ref: 17475500
Ki: 450 (nM), Ref: 18363349
Ki: 10 (nM), Ref: 19317447
Ki: 10 (nM), Ref: 19124253
Ki: 10 (nM), Ref: 19193158
Ki: 10 (nM), Ref: 18990571
Ki: 10 (nM), Ref: 19338333
Ki: 10 (nM), Ref: 18640037
Ki: 10 (nM), Ref: 18644716
Ki: 10 (nM), Ref: 19398204
Ki: 10 (nM), Ref: 19520577
Ki: 10 (nM), Ref: 19539481
Ki: 5 (nM), Ref: 19827837
Ki: 10 (nM), Ref: 19846301
Ki: 10 (nM), Ref: 20028100
IC50: 2100 (nM), Ref: 19388676
Ki: 300 (nM), Ref: 19388676
Ki: 5 (nM), Ref: 20201556
Ki: 10 (nM), Ref: 20472429
Ki: 10 (nM), Ref: 20624682
Ki: 10 (nM), Ref: 21208801
Ki: 10 (nM), Ref: 21251841
Ki: 10 (nM), Ref: 21300547
Ki: 5 (nM), Ref: 21314129
Ki: 10 (nM), Ref: 21332115
Ki: 10 (nM), Ref: 19435663
Ki: 10 (nM), Ref: 21506569
Ki: 5 (nM), Ref: 21723123
Ki: 10 (nM), Ref: 21757360
Ki: 10 (nM), Ref: 22285172
Ki: 10 (nM), Ref: 22386980
Ki: 10 (nM), Ref: 22424239
Ki: 10 (nM), Ref: 22443141
Ki: 10 (nM), Ref: 23391336
Ki: 10 (nM), Ref: 22883029
Ki: 10 (nM), Ref: 23867389
Ki: 10 (nM), Ref: 23965175
Ki: 300 (nM), Ref: 24205976
IC50: 500 (nM), Ref: 24205976
Ki: 10 (nM), Ref: 24314394
Ki: 10 (nM), Ref: 24513184
Ki: 10 (nM), Ref: 24792813
Ki: 10 (nM), Ref: 25129169
Ki: 10 (nM), Ref: 25533402
Ki: 10 (nM), Ref: 25773015
Ki: 10 (nM), Ref: 25882523
Ki: 10 (nM), Ref: 26174556
Ki: 10 (nM), Ref: 26525863
Ki: 10 (nM), Ref: 26691758
Ki: 10 (nM), Ref: 26850377
Ki: 10 (nM), Ref: 26832216
Ki: 10 (nM), Ref: 26920803
TCMC2174
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 1590 (nM), Ref: 16039848
Ki: 58 (nM), Ref: 16134940
Ki: 58 (nM), Ref: 17125255
Ki: 1590 (nM), Ref: 17125255
Ki: 1590 (nM), Ref: 17228881
Ki: 58 (nM), Ref: 17228881
Ki: 1590 (nM), Ref: 17376683
Ki: 58 (nM), Ref: 17475500
Ki: 58 (nM), Ref: 19193158
Ki: 58 (nM), Ref: 18640037
Ki: 58 (nM), Ref: 19398204
Ki: 58 (nM), Ref: 19827837
Ki: 58 (nM), Ref: 20028100
Ki: 58 (nM), Ref: 20201556
Ki: 58 (nM), Ref: 20472429
Ki: 58 (nM), Ref: 21314129
Ki: 58 (nM), Ref: 21723123
Ki: 58 (nM), Ref: 22443141
Ki: 58 (nM), Ref: 23965175
Ki: 58 (nM), Ref: 24513184
TCMC2174
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3800 (nM), Ref: 16039848
Ki: 3.8 (nM), Ref: 15686894
Ki: 3.8 (nM), Ref: 17125255
Ki: 3.8 (nM), Ref: 17475500
Ki: 3.8 (nM), Ref: 18640037
Ki: 3800 (nM), Ref: 18406497
Ki: 3.8 (nM), Ref: 19827837
Ki: 3.8 (nM), Ref: 20028100
Ki: 3.8 (nM), Ref: 20201556
Ki: 3.8 (nM), Ref: 20472429
Ki: 3.8 (nM), Ref: 21314129
Ki: 3.8 (nM), Ref: 21723123
Ki: 3.8 (nM), Ref: 23965175
Ki: 3.8 (nM), Ref: 24513184
TCMC2174
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 1460 (nM), Ref: 16039848
Ki: 1460 (nM), Ref: 17125255
Ki: 1460 (nM), Ref: 17376683
Ki: 1460 (nM), Ref: 17475500
Ki: 1460 (nM), Ref: 18640037
Ki: 1460 (nM), Ref: 18406497
Ki: 1460 (nM), Ref: 19398204
Ki: 1460 (nM), Ref: 20028100
Ki: 1460 (nM), Ref: 20472429
Ki: 1460 (nM), Ref: 21506569
Ki: 1460 (nM), Ref: 22443141
TCMC2174
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 250 (nM), Ref: 15686895
Ki: 250 (nM), Ref: 15686894
Ki: 250 (nM), Ref: 15686931
Ki: 250 (nM), Ref: 15546717
Ki: 250 (nM), Ref: 16539401
Ki: 250 (nM), Ref: 16459077
Ki: 250 (nM), Ref: 17125255
Ki: 250 (nM), Ref: 17228881
Ki: 250 (nM), Ref: 17376683
Ki: 250 (nM), Ref: 17475500
Ki: 250 (nM), Ref: 19317447
Ki: 250 (nM), Ref: 19124253
Ki: 250 (nM), Ref: 19193158
Ki: 250 (nM), Ref: 18990571
Ki: 250 (nM), Ref: 19338333
Ki: 250 (nM), Ref: 18640037
Ki: 250 (nM), Ref: 18644716
Ki: 250 (nM), Ref: 19398204
Ki: 250 (nM), Ref: 19450983
Ki: 250 (nM), Ref: 19520577
Ki: 250 (nM), Ref: 19539481
Ki: 250 (nM), Ref: 19827837
Ki: 250 (nM), Ref: 20028100
Ki: 250 (nM), Ref: 20201556
Ki: 250 (nM), Ref: 20472429
Ki: 250 (nM), Ref: 20624682
Ki: 250 (nM), Ref: 21208801
Ki: 250 (nM), Ref: 21251841
Ki: 250 (nM), Ref: 21300547
Ki: 250 (nM), Ref: 21314129
Ki: 250 (nM), Ref: 21332115
Ki: 250 (nM), Ref: 19435663
Ki: 250 (nM), Ref: 21506569
Ki: 250 (nM), Ref: 21723123
Ki: 250 (nM), Ref: 21757360
Ki: 250 (nM), Ref: 22285172
Ki: 250 (nM), Ref: 22443141
Ki: 250 (nM), Ref: 23391336
Ki: 250 (nM), Ref: 22883029
Ki: 250 (nM), Ref: 23867389
Ki: 250 (nM), Ref: 23965175
Ki: 250 (nM), Ref: 24513184
Ki: 250 (nM), Ref: 24792813
Ki: 250 (nM), Ref: 25129169
Ki: 250 (nM), Ref: 25533402
Ki: 250 (nM), Ref: 25773015
Ki: 250 (nM), Ref: 25882523
Ki: 250 (nM), Ref: 26525863
Ki: 250 (nM), Ref: 26691758
Ki: 250 (nM), Ref: 26850377
Ki: 250 (nM), Ref: 26920803
TCMC2174
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 0.87 (nM), Ref: 15686895
Ki: 0.9 (nM), Ref: 17125255
Ki: 0.9 (nM), Ref: 17376683
Ki: 0.9 (nM), Ref: 17475500
Ki: 0.9 (nM), Ref: 18640037
Ki: 0.87 (nM), Ref: 18406497
Ki: 0.9 (nM), Ref: 20028100
Ki: 0.9 (nM), Ref: 20472429
Ki: 0.9 (nM), Ref: 21395315
Ki: 0.9 (nM), Ref: 19435663
Ki: 0.9 (nM), Ref: 21506569
Ki: 0.9 (nM), Ref: 22443141
Ki: 0.9 (nM), Ref: 23867389
Ki: 0.9 (nM), Ref: 23965175
Ki: 0.9 (nM), Ref: 24287559
TCMC2174
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 15686931
Ki: 4900 (nM), Ref: 17125255
Ki: 4900 (nM), Ref: 17376683
Ki: 4900 (nM), Ref: 17475500
Ki: 4900 (nM), Ref: 18990571
Ki: 4900 (nM), Ref: 18640037
Ki: 4900 (nM), Ref: 20028100
Ki: 4900 (nM), Ref: 20472429
TCMC2174
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 63 (nM), Ref: 16302824
Ki: 63 (nM), Ref: 17125255
Ki: 63 (nM), Ref: 17376683
Ki: 63 (nM), Ref: 17475500
Ki: 63 (nM), Ref: 18640037
Ki: 63 (nM), Ref: 18644716
Ki: 63 (nM), Ref: 19539481
Ki: 63 (nM), Ref: 20028100
Ki: 63 (nM), Ref: 20472429
Ki: 63 (nM), Ref: 21300547
TCMC2174
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 30 (nM), Ref: 16302824
Ki: 30 (nM), Ref: 17125255
Ki: 30 (nM), Ref: 17475500
Ki: 30 (nM), Ref: 18640037
Ki: 30 (nM), Ref: 18644716
Ki: 30 (nM), Ref: 19539481
Ki: 30 (nM), Ref: 20028100
Ki: 30 (nM), Ref: 20472429
Ki: 30 (nM), Ref: 21300547
TCMC2174
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 45 (nM), Ref: 17228881
Ki: 45 (nM), Ref: 17475500
Ki: 45 (nM), Ref: 19193158
Ki: 45 (nM), Ref: 18640037
Ki: 45 (nM), Ref: 20028100
Ki: 45 (nM), Ref: 20472429
Ki: 45 (nM), Ref: 21208801
TCMC2174
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 47 (nM), Ref: 20028100
TCMC654
TCMT915 Retinoid X receptor gamma Homo sapiens Ki: 27 (nM), Ref: 10.1016/S0960-894X(97)00420-4
Ki: 14 (nM), Ref: 8765503
Ki: 11 (nM), Ref: 9435893
TCMC654
TCMT735 Retinoid X receptor alpha Homo sapiens Ki: 8 (nM), Ref: 8765503
Ki: 12 (nM), Ref: 9435893
IC50: 29 (nM), Ref: 15317450
TCMC654
TCMT914 Retinoid X receptor beta Homo sapiens Ki: 9 (nM), Ref: 8765503
Ki: 3.8 (nM), Ref: 9435893
TCMC654
TCMT912 Retinoic acid receptor gamma Homo sapiens Ki: 1 (nM), Ref: 9435893
TCMC1820
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 1000 (nM), Ref: 25060641
Ki: 35 (nM), Ref: 25060641
TCMC1472
TCMT105 Solute carrier family 15 member 2 Homo sapiens Ki: 10000 (nM), Ref: 21741846
Ki: 10000 (nM), Ref: 21741846
TCMC950
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 75.7 (nM), Ref: 15887952
IC50: 75.7 (nM), Ref: 15887952
IC50: 75.7 (nM), Ref:
TCMC950
TCMT236 Estrogen receptor beta Homo sapiens IC50: 18.6 (nM), Ref: 15887952
IC50: 18.6 (nM), Ref: 15887952
IC50: 18.6 (nM), Ref:
TCMC806
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8600 (nM), Ref: 15664814
TCMC260
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1160 (nM), Ref: 24074876
TCMC260
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 490 (nM), Ref: 24074876
TCMC2032
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5950 (nM), Ref: 18042384
Ki: 5950 (nM), Ref: 19317447
Ki: 5950 (nM), Ref: 19124253
Ki: 5950 (nM), Ref: 19338333
Ki: 5950 (nM), Ref: 19520577
Ki: 5950 (nM), Ref: 19846301
Ki: 5959 (nM), Ref: 20624682
Ki: 5950 (nM), Ref: 21208801
Ki: 5950 (nM), Ref: 21377369
Ki: 5950 (nM), Ref: 21757360
Ki: 5950 (nM), Ref: 22285172
Ki: 5959 (nM), Ref: 22386980
Ki: 5959 (nM), Ref: 23181552
Ki: 5959 (nM), Ref: 23391336
Ki: 5950 (nM), Ref: 22974493
Ki: 5959 (nM), Ref: 22883029
Ki: 5959 (nM), Ref: 24314394
Ki: 5950 (nM), Ref: 24560739
Ki: 5950 (nM), Ref: 24689792
Ki: 5959 (nM), Ref: 24792813
Ki: 5959 (nM), Ref: 25129169
Ki: 5959 (nM), Ref: 25773015
Ki: 5959 (nM), Ref: 25882523
Ki: 5959 (nM), Ref: 26174556
Ki: 5950 (nM), Ref: 26525863
Ki: 5959 (nM), Ref: 26691758
Ki: 5959 (nM), Ref: 26850377
Ki: 5950 (nM), Ref: 26810710
Ki: 5959 (nM), Ref: 26832216
Ki: 5959 (nM), Ref: 26920803
TCMC2032
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 103 (nM), Ref: 18042384
Ki: 103 (nM), Ref: 22974493
Ki: 103 (nM), Ref: 24560739
Ki: 103 (nM), Ref: 24689792
Ki: 103 (nM), Ref: 26810710
TCMC2032
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 633 (nM), Ref: 18042384
Ki: 633 (nM), Ref: 24560739
Ki: 633 (nM), Ref: 24689792
Ki: 633 (nM), Ref: 26810710
TCMC2032
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 935 (nM), Ref: 21208801
Ki: 935 (nM), Ref: 24689792
TCMC2032
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7920 (nM), Ref: 24689792
TCMC2032
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7210 (nM), Ref: 24689792
TCMC2032
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 10 (nM), Ref: 24689792
TCMC2032
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 773 (nM), Ref: 24689792
TCMC2032
TCMT132 Butyrylcholinesterase Homo sapiens IC50: 3600 (nM), Ref: 25537270
TCMC698
TCMT794 Type-1 angiotensin II receptor Homo sapiens Ki: 0.9 (nM), Ref: 20146480
Ki: 0.24 (nM), Ref: 26824643
IC50: 0.7244 (nM), Ref: 26824643
Ki: 0.16 (nM), Ref: 26824643
TCMC698
TCMT957 Angiotensin II type 2 (AT-2) receptor Homo sapiens Ki: 0.2 (nM), Ref: 26810314
TCMC1789
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 1100 (nM), Ref: 16570929
Ki: 1100 (nM), Ref: 19361197
TCMC566
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 3 (nM), Ref: 21377873
TCMC1437
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 330 (nM), Ref: 18667313
IC50: 14 (nM), Ref:
TCMC1437
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 690 (nM), Ref: 18667313
IC50: 3800 (nM), Ref: 25221653
IC50: 61 (nM), Ref: 26487917
TCMC929
TCMT116 Mu opioid receptor Homo sapiens Ki: 6300 (nM), Ref: 17616524
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC1542
TCMT336 Indoleamine 2,3-dioxygenase Homo sapiens IC50: 1000 (nM), Ref: 18318466
TCMC1542
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 3380 (nM), Ref: 19028102
TCMC1542
TCMT344 Aldehyde oxidase Homo sapiens IC50: 200 (nM), Ref: 20853847
Ki: 1500 (nM), Ref: 22996261
Ki: 470 (nM), Ref: 22996261
TCMC1542
TCMT186 Monoamine oxidase B Homo sapiens Ki: 400 (nM), Ref: 22071524
TCMC1813
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 0.91 (nM), Ref: 25759032
Ki: 1.8 (nM), Ref: 26227779
TCMC1813
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 2.12 (nM), Ref: 25759032
TCMC583
TCMT855 Nuclear receptor ROR-alpha Homo sapiens Ki: 12 (nM), Ref: 10.1039/C3MD00005B
TCMC583
TCMT150 Nuclear receptor ROR-gamma Homo sapiens Ki: 10 (nM), Ref: 10.1039/C3MD00005B
TCMC1133
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 1.3 (nM), Ref: 15203155
IC50: 3 (nM), Ref: 10673099
IC50: 1.3 (nM), Ref: 15203156
Ki: 100 (nM), Ref: 12954056
IC50: 2 (nM), Ref: 12749898
IC50: 5.9 (nM), Ref: 10447957
IC50: 1.3 (nM), Ref: 15745820
IC50: 1.3 (nM), Ref: 15664843
IC50: 1.3 (nM), Ref: 15582421
IC50: 1.3 (nM), Ref: 15225685
IC50: 1.3 (nM), Ref: 15225686
IC50: 3.2 (nM), Ref: 15341953
IC50: 3.2 (nM), Ref: 15456246
IC50: 3.2 (nM), Ref: 15876535
IC50: 3.2 (nM), Ref: 15943471
IC50: 28 (nM), Ref: 15658851
Ki: 1.995 (nM), Ref: 15771467
IC50: 3.2 (nM), Ref: 16098741
IC50: 0.75 (nM), Ref: 16219463
IC50: 1.4 (nM), Ref: 16309907
IC50: 1.35 (nM), Ref: 16412638
IC50: 10 (nM), Ref: 16610787
IC50: 1.3 (nM), Ref: 16632357
IC50: 1.3 (nM), Ref: 16730987
IC50: 46 (nM), Ref: 16942012
IC50: 1.6 (nM), Ref: 16942012
IC50: 1.3 (nM), Ref: 16777408
IC50: 1.2 (nM), Ref: 17149865
IC50: 4.7 (nM), Ref: 17696335
IC50: 3.6 (nM), Ref: 17049855
IC50: 3.2 (nM), Ref: 17188490
IC50: 1 (nM), Ref: 17289385
IC50: 1.4 (nM), Ref: 17448656
IC50: 1.4 (nM), Ref: 17890084
IC50: 4 (nM), Ref: 18760603
Ki: 2 (nM), Ref: 18722117
IC50: 12.5 (nM), Ref: 19836949
IC50: 3.2 (nM), Ref: 19705860
Ki: 0.16 (nM), Ref: 20621492
IC50: 21.04 (nM), Ref: 20812681
IC50: 46 (nM), Ref: 20875743
IC50: 1.3 (nM), Ref: 24315190
IC50: 5.7 (nM), Ref: 25369367
IC50: 0.9 (nM), Ref: 26183544
Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030
TCMC1133
TCMT236 Estrogen receptor beta Homo sapiens IC50: 1.1 (nM), Ref: 15203155
IC50: 4 (nM), Ref: 10673099
IC50: 1.1 (nM), Ref: 15203156
Ki: 100 (nM), Ref: 12954056
IC50: 2 (nM), Ref: 12749898
IC50: 1.1 (nM), Ref: 15745820
IC50: 1.1 (nM), Ref: 15664843
IC50: 1.1 (nM), Ref: 15993065
IC50: 1.1 (nM), Ref: 15582421
IC50: 1.1 (nM), Ref: 15225685
IC50: 1.1 (nM), Ref: 15225686
IC50: 3.6 (nM), Ref: 15341953
IC50: 3.6 (nM), Ref: 15456246
IC50: 3.6 (nM), Ref: 15876535
IC50: 3.6 (nM), Ref: 15943471
IC50: 24 (nM), Ref: 15658851
Ki: 3.162 (nM), Ref: 15771467
IC50: 3.6 (nM), Ref: 16098741
IC50: 1.18 (nM), Ref: 16219463
IC50: 1.2 (nM), Ref: 16309907
IC50: 1.2 (nM), Ref: 16412638
IC50: 11 (nM), Ref: 16610787
IC50: 1.2 (nM), Ref: 16632357
IC50: 1.2 (nM), Ref: 16730987
IC50: 1.4 (nM), Ref: 16942012
IC50: 1.1 (nM), Ref: 16777408
IC50: 1.4 (nM), Ref: 17149865
IC50: 16.7 (nM), Ref: 17696335
IC50: 3.2 (nM), Ref: 17049855
IC50: 3.6 (nM), Ref: 17188490
IC50: 1 (nM), Ref: 17289385
IC50: 1.2 (nM), Ref: 17448656
IC50: 1.2 (nM), Ref: 17890084
IC50: 4 (nM), Ref: 18760603
Ki: 2 (nM), Ref: 18722117
IC50: 2.9 (nM), Ref: 19705860
IC50: 10.74 (nM), Ref: 20812681
IC50: 0.046 (nM), Ref: 24315190
IC50: 5.6 (nM), Ref: 25369367
Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030
TCMC1133
TCMT187 Androgen Receptor Homo sapiens IC50: 19.1 (nM), Ref: 16309907
TCMC1133
TCMT99 Testis-specific androgen-binding protein Homo sapiens IC50: 50 (nM), Ref: 17149875
TCMC1133
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 3.6 (nM), Ref: 17482813
IC50: 6 (nM), Ref: 23448346
TCMC1133
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 3.2 (nM), Ref: 17482813
IC50: 8.7 (nM), Ref: 23448346
TCMC1133
TCMT344 Aldehyde oxidase Homo sapiens IC50: 80 (nM), Ref: 20853847
Ki: 4400 (nM), Ref: 22996261
Ki: 870 (nM), Ref: 22996261
TCMC1133
TCMT974 G-protein coupled estrogen receptor 1 Homo sapiens Ki: 5.7 (nM), Ref: 23672690
Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A
TCMC1471
TCMT976 Leukotriene B4 receptor 1 Homo sapiens IC50: 32 (nM), Ref: 10.1016/S0960-894X(01)80853-2
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC349
TCMT203 Glucose-6-phosphate 1-dehydrogenase Homo sapiens IC50: 5300 (nM), Ref: 22506561
TCMC784
TCMT131 Acetylcholinesterase Homo sapiens IC50: 100 (nM), Ref: 26003344
TCMC784
TCMT132 Butyrylcholinesterase Homo sapiens IC50: 1090 (nM), Ref: 26003344
TCMC2100
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 6425 (nM), Ref: IC50: 6200 (nM), Ref:
TCMC1543
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 840 (nM), Ref: 16248836
Ki: 2500 (nM), Ref: 16248836
TCMC1297
TCMT632 Purine nucleoside phosphorylase Homo sapiens Ki: 5000 (nM), Ref: 31484
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC1343
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 90 (nM), Ref: 18501600
Ki: 90 (nM), Ref: 18579385
TCMC1343
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7800 (nM), Ref: 18579385
TCMC1343
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8200 (nM), Ref: 18579385

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1904
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2268
TCMT1086 Isocitrate lyase Candida albicans IC50: 5.8 (ug/ml), Ref: 18407691
IC50: 4.9 (ug/ml), Ref: 18341287
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC2063
TCMT1086 Isocitrate lyase Candida albicans IC50: 53 (ug/ml), Ref: 21035332
TCMC983
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.43 (ug/ml), Ref: 20116898
TCMC1236
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.84 (ug/ml), Ref: 20116898
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC903
TCMT1251 Candida albicans Candida albicans MIC: 64 (ug/ml), Ref: 18805690
TCMC903
TCMT1246 Escherichia coli Escherichia coli MIC: 64 (ug/ml), Ref: 18805690
MIC: 7.81 (ug/ml), Ref: 20181416
MIC: 4 (ug/ml), Ref: 20038628
MIC: 8 (ug/ml), Ref: 20038628
MIC: 16 (ug/ml), Ref: 20038628
TCMC903
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 15.63 (ug/ml), Ref: 20181416
TCMC903
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 31.25 (ug/ml), Ref: 20181416
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC1352
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 62.5 (ug/ml), Ref: 18823782
TCMC1352
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 18823782
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC895
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.2 (ug/ml), Ref: 6492075
TCMC895
TCMT1246 Escherichia coli Escherichia coli MIC: 0.5 (ug/ml), Ref: 6492075
MIC: 1 (ug/ml), Ref: 6492075
MIC: 2 (ug/ml), Ref: 19770280
MIC: 4 (ug/ml), Ref: 19770280
TCMC895
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 3.9 (ug/ml), Ref: 6492075
TCMC895
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 15.6 (ug/ml), Ref: 6492075
TCMC895
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 15.6 (ug/ml), Ref: 6492075
MIC: 10 (ug/ml), Ref: 18838593
MIC: 2.5 (ug/ml), Ref: 18838593
MIC: 1.25 (ug/ml), Ref: 18838593
MIC: 0.625 (ug/ml), Ref: 18838593
MIC: 5 (ug/ml), Ref: 18838593
MIC: 20 (ug/ml), Ref: 18838593
TCMC895
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 2 (ug/ml), Ref: 17220400
MIC: 0.312 (ug/ml), Ref: 10543897
TCMC895
TCMT1251 Candida albicans Candida albicans MIC: 1.5 (ug/ml), Ref: 19841146
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2148
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 20691508
TCMC2409
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 32 (ug/ml), Ref: 12608857
TCMC2409
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 16 (ug/ml), Ref: 12608857
MIC: 32 (ug/ml), Ref: 12608857
TCMC1582
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 12.5 (ug/ml), Ref: 18539361
TCMC1582
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 25 (ug/ml), Ref: 18539361
TCMC1904
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0541-4
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC845
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 1522419
MIC: 6.25 (ug/ml), Ref: 1522419
TCMC845
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 1522419
MIC: 1.57 (ug/ml), Ref: 1522419
TCMC2134
TCMT1246 Escherichia coli Escherichia coli MIC: 8 (ug/ml), Ref: 20038628
MIC: 4 (ug/ml), Ref: 20038628
MIC: 32 (ug/ml), Ref: 20038628
MIC: 16 (ug/ml), Ref: 20038628
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC887
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 10395496
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC612
TCMT1207 Legionella pneumophila Legionella pneumophila MIC: 0 (ug/ml), Ref: 21244021
TCMC1011
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 MIC: 100 (ug/ml), Ref: 1335077
TCMC1186
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 3430167
TCMC1186
TCMT1284 Penicillium expansum Penicillium expansum MIC: 50 (ug/ml), Ref: 3430167
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC2566
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC915
TCMT1246 Escherichia coli Escherichia coli MIC: 1 (ug/ml), Ref: 25791674
TCMC915
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.5 (ug/ml), Ref: 25791674
TCMC915
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.25 (ug/ml), Ref: 25791674
TCMC2581
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2619
TCMT1462 Streptococcus mutans Streptococcus mutans UA159 MIC: 64 (ug/ml), Ref: 20106564
TCMC2619
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 20106564
TCMC2619
TCMT1251 Candida albicans Candida albicans MIC: 2 (ug/ml), Ref: 20106564
TCMC2619
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 32 (ug/ml), Ref: 20106564
TCMC2634
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC1977
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 19232493
TCMC1977
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 19232493
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2025
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 0.12 (ug/ml), Ref: 18004816
TCMC2025
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MBC: 0.12 (ug/ml), Ref: 18004816
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2025
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC2025
TCMT1246 Escherichia coli Escherichia coli MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC772
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 7714539
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC883
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 22750009
TCMC1236
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (ug/ml), Ref: 19299148
TCMC1970
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 7562923
MIC: 50 (ug/ml), Ref: 1560435
MIC: 100 (ug/ml), Ref: 1560435
MIC: 100 (ug/ml), Ref: 17101678
TCMC1970
TCMT1236 Mycobacterium bovis Mycobacterium bovis MIC: 100 (ug/ml), Ref: 1560435
TCMC1212
TCMT1288 Cytomegalovirus Cytomegalovirus MIC: 0.5 (ug/ml), Ref: 8709116
MIC: 0.9 (ug/ml), Ref: 7932543
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(96)00244-2
IC50: 0.6 (ug/ml), Ref: 11412988
MIC: 6.2 (ug/ml), Ref: 8393114
MIC: 3 (ug/ml), Ref: 8393114
IC50: 0.5 (ug/ml), Ref: 9836626
MIC: 0.6 (ug/ml), Ref: 10691698
MIC: 0.8 (ug/ml), Ref: 10691698
TCMC1212
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 MIC: 0.004 (ug/ml), Ref: 7932543
MIC: 0.08 (ug/ml), Ref: 7932543
MIC: 4.5 (ug/ml), Ref: 7932543
ID50: 0.2 (ug/ml), Ref: 2160539
MIC: 0.0007 (ug/ml), Ref: 10.1016/S0960-894X(96)00244-2
IC50: 0.001 (ug/ml), Ref: 11412988
IC50: 0.48 (ug/ml), Ref: 11412988
MIC: 0.004 (ug/ml), Ref: 8393114
MIC: 0.007 (ug/ml), Ref: 8393114
MIC: 0.001 (ug/ml), Ref: 8393114
MIC: 2 (ug/ml), Ref: 8393114
MIC50: 0.02 (ug/ml), Ref: 8765514
ID50: 0.23 (ug/ml), Ref: 2544723
MIC: 0.2 (ug/ml), Ref: 2329561
MIC: 0.1 (ug/ml), Ref: 2329561
MIC: 20 (ug/ml), Ref: 2329561
MIC: 10 (ug/ml), Ref: 2329561
MIC: 0.006 (ug/ml), Ref: 11708929
MIC: 0.004 (ug/ml), Ref: 11708929
MIC: 0.48 (ug/ml), Ref: 11708929
MIC: 0.07 (ug/ml), Ref: 11708929
MIC50: 0.096 (ug/ml), Ref: 16420056
MIC50: 0.48 (ug/ml), Ref: 16420056
MIC: 0.032 (ug/ml), Ref: 17583388
MIC: 2.4 (ug/ml), Ref: 17583388
MIC50: 0.032 (ug/ml), Ref: 19324473
MIC50: 2.4 (ug/ml), Ref: 19324473
ID50: 0.3 (nM), Ref: 2993615
ID50: 0.04 (nM), Ref: 1849998
TCMC1212
TCMT1228 Human herpesvirus 3 Human herpesvirus 3 MIC: 1.4 (ug/ml), Ref: 7932543
MIC: 1.5 (ug/ml), Ref: 7932543
MIC: 0.072 (ug/ml), Ref: 8393114
MIC: 0.02 (ug/ml), Ref: 8393114
MIC: 0.9 (ug/ml), Ref: 8393114
MIC: 0.1 (ug/ml), Ref: 8393114
MIC: 0.01 (ug/ml), Ref: 10691698
TCMC1212
TCMT1230 Human herpesvirus 5 Human herpesvirus 5 MIC: 1.5 (ug/ml), Ref: 7932543
ID50: 5 (ug/ml), Ref: 2160539
MIC50: 0.7 (ug/ml), Ref: 8765514
ID50: 1.8 (ug/ml), Ref: 2544723
IC50: 0.3 (ug/ml), Ref: 10888336
IC50: 1.2 (ug/ml), Ref: 10197958
IC50: 1.9 (ug/ml), Ref: 10197958
IC50: 0.5 (ug/ml), Ref: 9836626
IC50: 0.3 (ug/ml), Ref: 10447945
IC50: 0.3 (ug/ml), Ref: 12217359
IC50: 0.4 (ug/ml), Ref: 12217359
IC50: 0.1 (ug/ml), Ref: 10.1016/S0960-894X(97)10048-8
ID50: 0.006 (nM), Ref: 2993615
ID50: 0.002 (nM), Ref: 1849998
TCMC1212
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 ID50: 1.6 (ug/ml), Ref: 2160539
IC50: 0.002 (ug/ml), Ref: 11412988
MIC: 0.004 (ug/ml), Ref: 8393114
MIC: 0.02 (ug/ml), Ref: 8393114
MIC50: 0.002 (ug/ml), Ref: 8765514
ID50: 0.94 (ug/ml), Ref: 2544723
MIC: 0.02 (ug/ml), Ref: 2329561
MIC: 0.07 (ug/ml), Ref: 2329561
MIC: 0.1 (ug/ml), Ref: 2329561
MIC: 0.01 (ug/ml), Ref: 11708929
MIC: 0.02 (ug/ml), Ref: 11708929
MIC: 0.04 (ug/ml), Ref: 11708929
MIC50: 0.032 (ug/ml), Ref: 16420056
MIC: 0.032 (ug/ml), Ref: 17583388
MIC50: 0.0064 (ug/ml), Ref: 19324473
ID50: 1.3 (nM), Ref: 2993615
ID50: 0.04 (nM), Ref: 1849998
MIC: 96 (nM), Ref: 17092728
MIC: 6.4 (nM), Ref: 17672445
TCMC1212
TCMT1288 Cytomegalovirus Human herpesvirus 5 MIC: 0.5 (ug/ml), Ref: 8709116
MIC: 0.9 (ug/ml), Ref: 7932543
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(96)00244-2
IC50: 0.6 (ug/ml), Ref: 11412988
MIC: 6.2 (ug/ml), Ref: 8393114
MIC: 3 (ug/ml), Ref: 8393114
IC50: 0.5 (ug/ml), Ref: 9836626
MIC: 0.6 (ug/ml), Ref: 10691698
MIC: 0.8 (ug/ml), Ref: 10691698
TCMC1212
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 45 (ug/ml), Ref: 11412988
TCMC1212
TCMT1293 Vaccinia virus Vaccinia virus MIC: 70 (ug/ml), Ref: 8393114
MIC50: 100 (ug/ml), Ref: 19324473
TCMC1212
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 strain KOS MIC: 0.004 (ug/ml), Ref: 7932543
MIC: 0.08 (ug/ml), Ref: 7932543
MIC: 4.5 (ug/ml), Ref: 7932543
ID50: 0.2 (ug/ml), Ref: 2160539
MIC: 0.0007 (ug/ml), Ref: 10.1016/S0960-894X(96)00244-2
IC50: 0.001 (ug/ml), Ref: 11412988
IC50: 0.48 (ug/ml), Ref: 11412988
MIC: 0.004 (ug/ml), Ref: 8393114
MIC: 0.007 (ug/ml), Ref: 8393114
MIC: 0.001 (ug/ml), Ref: 8393114
MIC: 2 (ug/ml), Ref: 8393114
MIC50: 0.02 (ug/ml), Ref: 8765514
ID50: 0.23 (ug/ml), Ref: 2544723
MIC: 0.2 (ug/ml), Ref: 2329561
MIC: 0.1 (ug/ml), Ref: 2329561
MIC: 20 (ug/ml), Ref: 2329561
MIC: 10 (ug/ml), Ref: 2329561
MIC: 0.006 (ug/ml), Ref: 11708929
MIC: 0.004 (ug/ml), Ref: 11708929
MIC: 0.48 (ug/ml), Ref: 11708929
MIC: 0.07 (ug/ml), Ref: 11708929
MIC50: 0.096 (ug/ml), Ref: 16420056
MIC50: 0.48 (ug/ml), Ref: 16420056
MIC: 0.032 (ug/ml), Ref: 17583388
MIC: 2.4 (ug/ml), Ref: 17583388
MIC50: 0.032 (ug/ml), Ref: 19324473
MIC50: 2.4 (ug/ml), Ref: 19324473
ID50: 0.3 (nM), Ref: 2993615
ID50: 0.04 (nM), Ref: 1849998
TCMC1212
TCMT1231 Human herpesvirus 1 strain KOS Human herpesvirus 1 strain KOS MIC: 12 (ug/ml), Ref: 10.1007/s00044-012-0127-6
MIC: 0.48 (ug/ml), Ref: 10.1007/s00044-012-0127-6
MIC: 96 (nM), Ref: 17092728
MIC: 32 (nM), Ref: 17672445
TCMC1212
TCMT1390 Human herpesvirus 2 strain G Human herpesvirus 2 strain G MIC: 4 (ug/ml), Ref: 10.1007/s00044-012-0127-6
TCMC1789
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 20667727
MIC: 12.5 (ug/ml), Ref: 20667727
TCMC1475
TCMT1246 Escherichia coli Escherichia coli MIC: 0.5 (ug/ml), Ref: 2842501
MIC: 0.016 (ug/ml), Ref: 12824037
MIC: 0.25 (ug/ml), Ref: 12824037
MIC: 0.07 (ug/ml), Ref: 2824776
MIC: 0.04 (ug/ml), Ref: 2824776
MIC: 0.03 (ug/ml), Ref: 7707323
MIC: 0.01 (ug/ml), Ref: 15380226
MIC: 0.06 (ug/ml), Ref: 16078842
MIC: 0.06 (ug/ml), Ref: 17064062
MIC: 0.015 (ug/ml), Ref: 17064062
MIC: 0.008 (ug/ml), Ref: 17064062
MIC: 0.06 (ug/ml), Ref: 17074790
MIC: 0.25 (ug/ml), Ref: 17074790
MIC: 0.5 (ug/ml), Ref: 17074790
MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC: 0.06 (ug/ml), Ref: 17261623
MIC: 8 (ug/ml), Ref: 17220425
MIC: 1.5 (ug/ml), Ref: 17220425
MIC: 0.064 (ug/ml), Ref: 17220425
MIC50: 0.03 (ug/ml), Ref: 17242152
MIC: 0.03 (ug/ml), Ref: 17316916
MIC: 0.016 (ug/ml), Ref: 17157008
MIC: 0.004 (ug/ml), Ref: 17404007
MIC: 0.008 (ug/ml), Ref: 17404007
MIC: 0.125 (ug/ml), Ref: 17404007
MIC: 1 (ug/ml), Ref: 17404007
MIC: 0.03 (ug/ml), Ref: 17404007
MIC: 0.25 (ug/ml), Ref: 17404007
MIC: 2 (ug/ml), Ref: 17404007
MIC: 4 (ug/ml), Ref: 17404007
MIC: 0.06 (ug/ml), Ref: 17404007
MIC: 0.025 (ug/ml), Ref: 18450331
MIC: 0.032 (ug/ml), Ref: 17470656
MIC: 0.016 (ug/ml), Ref: 17470656
MIC: 0.012 (ug/ml), Ref: 17470656
MIC: 0.006 (ug/ml), Ref: 17470656
MIC: 0.002 (ug/ml), Ref: 17470656
MIC: 0.008 (ug/ml), Ref: 17470656
MIC: 0.001 (ug/ml), Ref: 18457383
MIC: 32 (ug/ml), Ref: 17548499
MIC: 0.008 (ug/ml), Ref: 17548499
MIC: 0.016 (ug/ml), Ref: 17548499
MIC: 0.004 (ug/ml), Ref: 17548499
MIC: 0.19 (ug/ml), Ref: 17724159
MIC: 0.38 (ug/ml), Ref: 17724159
MIC: 0.012 (ug/ml), Ref: 17724159
MIC: 0.03 (ug/ml), Ref: 17938184
MIC: 0.5 (ug/ml), Ref: 17938184
MIC: 1 (ug/ml), Ref: 19481308
MIC: 0.015 (ug/ml), Ref: 19939519
MIC: 0.19 (ug/ml), Ref: 19949057
MIC: 0.032 (ug/ml), Ref: 19949057
MIC: 0.125 (ug/ml), Ref: 19949057
MIC: 0.03 (ug/ml), Ref: 20667744
MIC: 25 (ug/ml), Ref: 20667744
MIC: 1 (ug/ml), Ref: 20667731
MIC: 0.5 (ug/ml), Ref: 20591538
MIC: 0.12 (ug/ml), Ref: 20591538
MIC: 1 (ug/ml), Ref: 20038618
MIC: 0.12 (ug/ml), Ref: 20008783
MIC: 0.25 (ug/ml), Ref: 20008783
MIC: 0.0075 (ug/ml), Ref: 20008783
MIC50: 0.5 (ug/ml), Ref: 20065058
MIC90: 1 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 20065058
MIC: 0.06 (ug/ml), Ref: 20065058
MIC: 0.008 (ug/ml), Ref: 18285488
MIC: 0.015 (ug/ml), Ref: 18285488
MIC: 64 (ug/ml), Ref: 18285488
MIC: 0.008 (ug/ml), Ref: 18285488
MIC: 1 (ug/ml), Ref: 18426899
MIC: 0.25 (ug/ml), Ref: 18426899
MIC: 1.5 (ug/ml), Ref: 18426899
MIC: 0.25 (ug/ml), Ref: 18426899
MIC: 0.75 (ug/ml), Ref: 18426899
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 64 (ug/ml), Ref: 20176911
MIC50: 16 (ug/ml), Ref: 20176911
MIC: 4 (ug/ml), Ref: 20176911
MIC90: 0.5 (ug/ml), Ref: 20176911
MIC50: 0.03 (ug/ml), Ref: 20176911
MIC: 0.015 (ug/ml), Ref: 20176911
MIC: 0.03 (ug/ml), Ref: 18644958
MIC: 0.06 (ug/ml), Ref: 18644958
MIC: 0.01 (ug/ml), Ref: 18644958
MIC: 0.008 (ug/ml), Ref: 18644958
MIC: 0.016 (ug/ml), Ref: 18809939
MIC: 0.25 (ug/ml), Ref: 18809939
MIC: 0.5 (ug/ml), Ref: 18809939
MIC: 4 (ug/ml), Ref: 18809939
MIC: 32 (ug/ml), Ref: 19001117
MIC: 0.031 (ug/ml), Ref: 19001117
MIC: 0.004 (ug/ml), Ref: 18644963
MIC: 0.023 (ug/ml), Ref: 18644963
MIC: 0.012 (ug/ml), Ref: 18644963
MIC: 0.006 (ug/ml), Ref: 18644963
MIC: 0.008 (ug/ml), Ref: 18644963
MIC: 0.006 (ug/ml), Ref: 20350950
MIC: 0.5 (ug/ml), Ref: 20421404
MIC: 3 (ug/ml), Ref: 20421404
MIC: 0.023 (ug/ml), Ref: 20421404
MIC: 0.004 (ug/ml), Ref: 20421404
MIC: 0.094 (ug/ml), Ref: 20421404
MIC: 0.002 (ug/ml), Ref: 20421404
MIC90: 1 (ug/ml), Ref: 18591277
MIC50: 16 (ug/ml), Ref: 18299417
MIC90: 16 (ug/ml), Ref: 18299417
MIC90: 32 (ug/ml), Ref: 18299417
MIC50: 0.06 (ug/ml), Ref: 18299417
MIC: 0.023 (ug/ml), Ref: 18519713
MIC: 0.094 (ug/ml), Ref: 18519713
MIC: 0.047 (ug/ml), Ref: 18519713
MIC: 0.012 (ug/ml), Ref: 18519713
MIC50: 0.03 (ug/ml), Ref: 18591277
MIC: 0.015 (ug/ml), Ref: 18591277
MIC: 0.125 (ug/ml), Ref: 20833454
MIC: 16 (ug/ml), Ref: 20833454
MIC: 0.008 (ug/ml), Ref: 18838594
MIC: 0.042 (ug/ml), Ref: 18838594
MIC: 0.023 (ug/ml), Ref: 18838594
MIC: 39 (ug/ml), Ref: 18838594
MIC: 8 (ug/ml), Ref: 18838594
MIC: 0.03 (ug/ml), Ref: 19104025
MIC: 1 (ug/ml), Ref: 19104025
MIC: 0.06 (ug/ml), Ref: 19104025
MIC: 2 (ug/ml), Ref: 19104025
MIC: 0.016 (ug/ml), Ref: 18936192
MIC: 0.25 (ug/ml), Ref: 18936192
MIC: 0.06 (ug/ml), Ref: 18936192
MIC: 16 (ug/ml), Ref: 18936192
MIC: 2 (ug/ml), Ref: 18936192
MIC: 1 (ug/ml), Ref: 18936192
MIC: 0.06 (ug/ml), Ref: 19015359
MIC: 0.5 (ug/ml), Ref: 19015359
MIC: 0.03 (ug/ml), Ref: 19015359
MIC: 16 (ug/ml), Ref: 19015359
MIC: 32 (ug/ml), Ref: 19015359
MIC: 8 (ug/ml), Ref: 19015359
MIC: 4 (ug/ml), Ref: 19015359
MIC: 0.25 (ug/ml), Ref: 19015359
MIC: 2 (ug/ml), Ref: 19015359
MIC: 0.125 (ug/ml), Ref: 19015359
MIC: 0.12 (ug/ml), Ref: 19015360
MIC50: 16 (ug/ml), Ref: 19015360
MIC50: 16 (ug/ml), Ref: 19001109
MIC50: 8 (ug/ml), Ref: 19001109
MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 0.03 (ug/ml), Ref: 19001109
MIC: 3.50E-05 (ug/ml), Ref: 19064900
MIC: 0.015 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC50: 0.25 (ug/ml), Ref: 19114671
MIC90: 0.25 (ug/ml), Ref: 19114671
MIC90: 32 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19364872
MIC90: 4 (ug/ml), Ref: 19364872
MIC50: 1 (ug/ml), Ref: 19364872
MIC: 2 (ug/ml), Ref: 19364872
MIC: 1 (ug/ml), Ref: 19364872
MIC: 0.25 (ug/ml), Ref: 19258263
MIC: 0.023 (ug/ml), Ref: 19258263
MIC: 0.19 (ug/ml), Ref: 19258263
MIC: 0.016 (ug/ml), Ref: 19258263
MIC: 0.006 (ug/ml), Ref: 19258263
MIC: 0.125 (ug/ml), Ref: 19258263
MIC: 0.03 (ug/ml), Ref: 19349512
MBC: 0.06 (ug/ml), Ref: 19349512
MIC: 32 (ug/ml), Ref: 19349512
MIC: 8 (ug/ml), Ref: 19349512
MBC: 32 (ug/ml), Ref: 19349512
MBC: 16 (ug/ml), Ref: 19349512
MIC: 4 (ug/ml), Ref: 19188391
MIC: 8 (ug/ml), Ref: 19188391
MIC: 0.125 (ug/ml), Ref: 19188391
MIC: 0.047 (ug/ml), Ref: 19188391
MIC: 0.03 (ug/ml), Ref: 19188391
MIC: 0.03 (ug/ml), Ref: 19188391
MIC: 0.032 (ug/ml), Ref: 19188391
MIC: 0.006 (ug/ml), Ref: 19451298
MIC: 0.25 (ug/ml), Ref: 19451298
MIC: 0.5 (ug/ml), Ref: 19451298
MIC: 0.015 (ug/ml), Ref: 21232952
MIC: 0.5 (ug/ml), Ref: 21232952
MIC: 0.016 (ug/ml), Ref: 20660686
MIC: 0.004 (ug/ml), Ref: 20660686
MIC: 0.25 (ug/ml), Ref: 20231393
MIC50: 0.03 (ug/ml), Ref: 18625769
MIC90: 16 (ug/ml), Ref: 18625769
MIC: 0.008 (ug/ml), Ref: 21173174
MIC: 0.5 (ug/ml), Ref: 21173174
MIC: 0.125 (ug/ml), Ref: 21173174
MIC: 0.25 (ug/ml), Ref: 21173174
MIC: 1 (ug/ml), Ref: 21173174
MIC: 2 (ug/ml), Ref: 21173174
MIC: 4 (ug/ml), Ref: 21173174
MBC: 0.03 (ug/ml), Ref: 21173174
MBC: 0.5 (ug/ml), Ref: 21173174
MBC: 0.25 (ug/ml), Ref: 21173174
MBC: 2 (ug/ml), Ref: 21173174
MBC: 0.008 (ug/ml), Ref: 21173174
MBC: 4 (ug/ml), Ref: 21173174
MBC: 1 (ug/ml), Ref: 21173174
MIC: 32 (ug/ml), Ref: 19581455
MIC: 0.25 (ug/ml), Ref: 19581455
MIC: 0.03 (ug/ml), Ref: 21458275
MIC: 25 (ug/ml), Ref: 21458275
MIC: 0.03 (ug/ml), Ref: 21515052
MIC: 32 (ug/ml), Ref: 21515052
MIC: 2 (ug/ml), Ref: 21481984
MIC: 16 (ug/ml), Ref: 21481984
MIC: 0.12 (ug/ml), Ref: 21510638
MIC: 2 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 21764484
MIC: 4 (ug/ml), Ref: 21764484
MIC: 0.008 (ug/ml), Ref: 22841282
MIC: 4 (ug/ml), Ref: 22841282
MIC: 0.25 (ug/ml), Ref: 22841282
MIC: 16 (ug/ml), Ref: 22841282
MIC: 8 (ug/ml), Ref: 22841282
MIC: 1 (ug/ml), Ref: 22841282
MIC: 0.12 (ug/ml), Ref: 22939698
MIC: 25 (ug/ml), Ref: 10.1007/s00044-011-9549-9
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.12 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.025 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC50: 0.25 (ug/ml), Ref: 23265890
MIC: 0.012 (ug/ml), Ref: 23409972
MIC: 16 (ug/ml), Ref: 23402878
MIC: 8 (ug/ml), Ref: 23402878
MIC: 0.5 (ug/ml), Ref: 23402878
MIC: 0.015 (ug/ml), Ref: 23402878
MIC50: 0.25 (ug/ml), Ref: 23735742
MIC: 0.25 (ug/ml), Ref: 24447849
MIC: 3.12 (ug/ml), Ref: 24852274
MIC: 0.125 (ug/ml), Ref: 24798098
MIC: 16 (ug/ml), Ref: 25218911
MIC: 32 (ug/ml), Ref: 25218911
MIC90: 16 (ug/ml), Ref: 25155913
MIC: 0.008 (ug/ml), Ref: 25218911
MIC: 0.25 (ug/ml), Ref: 25218911
MIC: 0.13 (ug/ml), Ref: 25646964
MIC: 0.016 (ug/ml), Ref: 26238324
MIC: 8 (ug/ml), Ref: 26238324
MIC: 0.03 (ug/ml), Ref: 26317881
MIC: 0.019 (ug/ml), Ref: 26363871
MIC: 2 (ug/ml), Ref: 26476970
MIC: 8 (ug/ml), Ref: 26476970
MIC: 4 (ug/ml), Ref: 26476970
MIC: 4 (ug/ml), Ref: 26435513
MIC: 8 (ug/ml), Ref: 26435513
MIC: 2 (ug/ml), Ref: 27020299
MIC: 8 (ug/ml), Ref: 27020299
MIC: 4 (ug/ml), Ref: 27020299
MIC: 29 (ug/ml), Ref: 27324976
MIC: 0.5 (ug/ml), Ref: 27293070
MIC: 32 (ug/ml), Ref: 27293070
MIC: 64 (ug/ml), Ref: 27293070
MBC: 0.97 (nM), Ref: 22036229
IC50: 30 (nM), Ref: 24571273
MIC: 63 (nM), Ref: 25818767
MIC: 16 (nM), Ref: 25818767
TCMC1475
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 32 (ug/ml), Ref: 2842501
MIC: 0.5 (ug/ml), Ref: 12824037
MIC: 0.04 (ug/ml), Ref: 2824776
MIC: 0.07 (ug/ml), Ref: 2824776
MIC: 0.5 (ug/ml), Ref: 7707323
MIC: 4 (ug/ml), Ref: 16078842
MIC: 0.5 (ug/ml), Ref: 17064062
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 64 (ug/ml), Ref: 17261623
MIC50: 0.5 (ug/ml), Ref: 17242152
MIC: 4 (ug/ml), Ref: 17316916
MIC: 0.5 (ug/ml), Ref: 17157008
MIC: 0.5 (ug/ml), Ref: 18450331
MIC: 0.5 (ug/ml), Ref: 18457383
MIC: 0.5 (ug/ml), Ref: 17682103
MIC: 64 (ug/ml), Ref: 17682103
MIC: 1 (ug/ml), Ref: 17682103
MIC: 2 (ug/ml), Ref: 17682103
MIC: 0.12 (ug/ml), Ref: 17682103
MIC: 0.06 (ug/ml), Ref: 17682103
MIC: 0.5 (ug/ml), Ref: 19481308
MIC: 0.5 (ug/ml), Ref: 19939519
MIC: 0.064 (ug/ml), Ref: 19917762
MIC: 1 (ug/ml), Ref: 19917762
MIC: 0.125 (ug/ml), Ref: 19917762
MIC50: 8 (ug/ml), Ref: 19917762
MIC50: 32 (ug/ml), Ref: 19917762
MIC50: 16 (ug/ml), Ref: 19917762
MIC50: 4 (ug/ml), Ref: 19917762
MIC90: 64 (ug/ml), Ref: 19917762
MIC: 0.5 (ug/ml), Ref: 19805554
MIC: 1 (ug/ml), Ref: 19805554
MIC: 2 (ug/ml), Ref: 19805554
MIC: 3.5 (ug/ml), Ref: 19805554
MIC50: 4 (ug/ml), Ref: 19805554
MIC: 4 (ug/ml), Ref: 19805554
MIC90: 8 (ug/ml), Ref: 19805554
MIC: 8 (ug/ml), Ref: 19805554
MIC: 16 (ug/ml), Ref: 19805554
MIC: 32 (ug/ml), Ref: 19805554
MIC50: 2 (ug/ml), Ref: 19805554
MIC: 0.3 (ug/ml), Ref: 20667744
MIC: 50 (ug/ml), Ref: 20667744
MIC: 0.25 (ug/ml), Ref: 20667731
MIC: 64 (ug/ml), Ref: 20591538
MIC: 1 (ug/ml), Ref: 20591538
MIC: 1 (ug/ml), Ref: 20038618
MIC50: 8 (ug/ml), Ref: 20065058
MIC: 0.25 (ug/ml), Ref: 20065058
MIC50: 2 (ug/ml), Ref: 18426902
MIC90: 16 (ug/ml), Ref: 18426902
MIC: 0.75 (ug/ml), Ref: 20038614
MIC90: 2 (ug/ml), Ref: 20176911
MIC50: 0.5 (ug/ml), Ref: 20176911
MIC: 0.5 (ug/ml), Ref: 20176911
MIC: 0.12 (ug/ml), Ref: 18591277
MIC50: 4 (ug/ml), Ref: 18591277
MIC90: 64 (ug/ml), Ref: 18591277
MIC: 0.25 (ug/ml), Ref: 18519723
MIC: 0.5 (ug/ml), Ref: 18519723
MIC: 4 (ug/ml), Ref: 18519723
MIC: 2 (ug/ml), Ref: 18519723
MIC: 8 (ug/ml), Ref: 18519723
MIC: 0.5 (ug/ml), Ref: 20833454
MIC: 16 (ug/ml), Ref: 20833454
MIC: 4 (ug/ml), Ref: 20833454
MIC: 2 (ug/ml), Ref: 20833454
MIC: 0.25 (ug/ml), Ref: 20833454
MIC: 2 (ug/ml), Ref: 19104025
MIC: 4 (ug/ml), Ref: 19104025
MIC: 0.5 (ug/ml), Ref: 19104025
MIC: 1 (ug/ml), Ref: 19104025
MIC: 2 (ug/ml), Ref: 19015359
MIC: 16 (ug/ml), Ref: 19015359
MIC50: 1 (ug/ml), Ref: 19001109
MIC: 0.0006 (ug/ml), Ref: 19064900
MIC: 0.25 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19114671
MIC50: 2 (ug/ml), Ref: 19114671
MIC50: 32 (ug/ml), Ref: 19114671
MIC: 0.25 (ug/ml), Ref: 19349512
MBC: 0.5 (ug/ml), Ref: 19349512
MIC: 1 (ug/ml), Ref: 19349512
MIC: 0.5 (ug/ml), Ref: 19349512
MBC: 2 (ug/ml), Ref: 19349512
MBC: 1 (ug/ml), Ref: 19349512
MIC: 0.25 (ug/ml), Ref: 19188391
MIC: 16 (ug/ml), Ref: 19188391
MIC: 0.06 (ug/ml), Ref: 19188391
MIC: 0.06 (ug/ml), Ref: 19506065
MIC: 2 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC50: 16 (ug/ml), Ref: 19506065
MIC90: 1 (ug/ml), Ref: 19506065
MIC90: 64 (ug/ml), Ref: 19506065
MIC: 1 (ug/ml), Ref: 19528273
MIC: 2 (ug/ml), Ref: 19528273
MIC: 4 (ug/ml), Ref: 21232952
MIC: 2 (ug/ml), Ref: 21232952
MIC: 32 (ug/ml), Ref: 19581455
MIC: 0.25 (ug/ml), Ref: 19581455
MIC: 0.3 (ug/ml), Ref: 21458275
MIC: 8 (ug/ml), Ref: 21515052
MIC: 4 (ug/ml), Ref: 21481984
MIC: 16 (ug/ml), Ref: 21481984
MIC: 0.25 (ug/ml), Ref: 21510638
MIC: 4 (ug/ml), Ref: 21764484
MIC: 16 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 21764484
MIC: 1 (ug/ml), Ref: 21764484
MIC: 0.25 (ug/ml), Ref: 22841282
MIC: 0.5 (ug/ml), Ref: 22841282
MIC: 1 (ug/ml), Ref: 22841282
MIC: 0.25 (ug/ml), Ref: 22939698
MIC: 64 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 1 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 3.13 (ug/ml), Ref: 10.1007/s00044-013-0581-9
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC50: 0.25 (ug/ml), Ref: 23265890
MIC: 16 (ug/ml), Ref: 23402878
MIC: 4 (ug/ml), Ref: 23402878
MIC: 1 (ug/ml), Ref: 23402878
MIC50: 0.25 (ug/ml), Ref: 23735742
MIC: 3.12 (ug/ml), Ref: 24852274
MIC: 0.5 (ug/ml), Ref: 25218911
MIC90: 16 (ug/ml), Ref: 25155913
MIC: 16 (ug/ml), Ref: 25218911
MIC: 1 (ug/ml), Ref: 25435146
MIC: 1 (ug/ml), Ref: 25927406
MIC: 1 (ug/ml), Ref: 26238324
MIC: 0.5 (ug/ml), Ref: 26317881
MIC: 2 (ug/ml), Ref: 26476970
MIC: 0.12 (ug/ml), Ref: 26363871
MIC: 1 (ug/ml), Ref: 26476970
MIC: 1 (ug/ml), Ref: 26435513
MIC: 0.5 (ug/ml), Ref: 26435513
MIC: 2 (ug/ml), Ref: 26435513
MIC: 1 (ug/ml), Ref: 27020299
MIC: 2 (ug/ml), Ref: 27020299
MBC: 0.97 (nM), Ref: 22036229
TCMC1475
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 2842501
MIC: 0.12 (ug/ml), Ref: 12824037
MIC: 2 (ug/ml), Ref: 12824037
MIC: 0.15 (ug/ml), Ref: 2824776
MIC: 0.3 (ug/ml), Ref: 2824776
MIC: 0.25 (ug/ml), Ref: 7707323
MIC: 0.2 (ug/ml), Ref: 15380226
MIC: 16 (ug/ml), Ref: 16078842
MIC: 8 (ug/ml), Ref: 16078842
MIC: 32 (ug/ml), Ref: 16078842
MIC: 1 (ug/ml), Ref: 16078842
MIC: 0.25 (ug/ml), Ref: 17064062
MIC: 0.125 (ug/ml), Ref: 17064062
MIC: 0.5 (ug/ml), Ref: 17064062
MIC: 8 (ug/ml), Ref: 17064062
MIC50: 16 (ug/ml), Ref: 17228862
MIC: 16 (ug/ml), Ref: 17228862
MIC: 16 (ug/ml), Ref: 17074796
MIC50: 0.25 (ug/ml), Ref: 17261623
MIC90: 0.25 (ug/ml), Ref: 17261623
MIC50: 8 (ug/ml), Ref: 17261623
MIC90: 8 (ug/ml), Ref: 17261623
MIC50: 32 (ug/ml), Ref: 17261623
MIC90: 64 (ug/ml), Ref: 17261623
MIC: 16 (ug/ml), Ref: 17261623
MIC: 0.125 (ug/ml), Ref: 17261623
MIC: 0.25 (ug/ml), Ref: 17261623
MIC: 8 (ug/ml), Ref: 17261623
MIC: 2 (ug/ml), Ref: 17220419
MIC50: 0.25 (ug/ml), Ref: 17242152
MIC50: 16 (ug/ml), Ref: 17242152
MIC: 0.75 (ug/ml), Ref: 17296740
MIC: 1.5 (ug/ml), Ref: 17296740
MIC: 2 (ug/ml), Ref: 17296740
MIC: 0.125 (ug/ml), Ref: 17303420
MIC: 0.5 (ug/ml), Ref: 17303420
MIC: 0.5 (ug/ml), Ref: 17316916
MIC: 0.25 (ug/ml), Ref: 17316916
MIC: 0.5 (ug/ml), Ref: 17157008
MIC: 4 (ug/ml), Ref: 17157008
MIC: 0.78 (ug/ml), Ref: 17826097
MIC: 0.5 (ug/ml), Ref: 17404009
MIC: 0.25 (ug/ml), Ref: 17404009
MIC: 0.125 (ug/ml), Ref: 17404009
MIC: 0.125 (ug/ml), Ref: 18330977
MIC: 0.25 (ug/ml), Ref: 18450331
MIC: 0.5 (ug/ml), Ref: 18450331
MIC: 0.125 (ug/ml), Ref: 18450331
MIC: 8 (ug/ml), Ref: 18450331
MIC: 16 (ug/ml), Ref: 18450331
MIC: 0.06 (ug/ml), Ref: 17875997
MIC50: 0.25 (ug/ml), Ref: 17875997
MIC90: 4 (ug/ml), Ref: 17875997
MIC: 0.125 (ug/ml), Ref: 17875997
MIC50: 1 (ug/ml), Ref: 17875997
MIC: 0.16 (ug/ml), Ref: 17502404
MBC: 0.32 (ug/ml), Ref: 17502404
MBC: 40 (ug/ml), Ref: 17502404
MIC50: 16 (ug/ml), Ref: 17420210
MIC50: 0.25 (ug/ml), Ref: 17420210
MIC90: 0.5 (ug/ml), Ref: 17420210
MIC: 0.125 (ug/ml), Ref: 18457383
MIC: 0.5 (ug/ml), Ref: 18457383
MIC: 8 (ug/ml), Ref: 18457383
MIC: 32 (ug/ml), Ref: 18457383
MIC: 0.25 (ug/ml), Ref: 17620379
MIC: 1 (ug/ml), Ref: 17620379
MIC: 8 (ug/ml), Ref: 18056272
MIC: 0.25 (ug/ml), Ref: 19481308
MIC: 32 (ug/ml), Ref: 19481308
MIC: 0.4 (ug/ml), Ref: 19552984
MIC: 0.12 (ug/ml), Ref: 19939519
MIC50: 16 (ug/ml), Ref: 19736016
MIC50: 4 (ug/ml), Ref: 19805554
MIC50: 0.125 (ug/ml), Ref: 19805554
MIC90: 0.25 (ug/ml), Ref: 19805554
MIC: 0.07 (ug/ml), Ref: 20667744
MIC: 25 (ug/ml), Ref: 20667744
MIC: 100 (ug/ml), Ref: 20667744
MIC: 0.125 (ug/ml), Ref: 20667731
MIC: 16 (ug/ml), Ref: 20667731
MIC: 0.25 (ug/ml), Ref: 20591538
MIC50: 0.25 (ug/ml), Ref: 20065058
MIC50: 16 (ug/ml), Ref: 20065058
MIC90: 1 (ug/ml), Ref: 20065058
MIC90: 0.25 (ug/ml), Ref: 20065058
MIC90: 16 (ug/ml), Ref: 20065058
MIC: 0.06 (ug/ml), Ref: 20065058
MIC: 0.5 (ug/ml), Ref: 20065058
MIC: 0.025 (ug/ml), Ref: 18316525
MIC: 32 (ug/ml), Ref: 18316525
MIC50: 0.25 (ug/ml), Ref: 18180353
MIC90: 0.5 (ug/ml), Ref: 18180353
MIC: 0.12 (ug/ml), Ref: 18180353
MIC90: 4 (ug/ml), Ref: 20231392
MIC50: 0.5 (ug/ml), Ref: 20385851
MIC90: 0.5 (ug/ml), Ref: 20385851
MIC50: 16 (ug/ml), Ref: 20231392
MIC50: 8 (ug/ml), Ref: 20231392
MIC50: 0.25 (ug/ml), Ref: 20231392
MIC50: 4 (ug/ml), Ref: 20231392
MIC: 16 (ug/ml), Ref: 18838584
MIC: 32 (ug/ml), Ref: 18838584
MIC: 0.125 (ug/ml), Ref: 18838584
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC50: 4 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 0.5 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC90: 4 (ug/ml), Ref: 18591277
MIC: 64 (ug/ml), Ref: 18490505
MIC: 8 (ug/ml), Ref: 18490505
MIC: 4 (ug/ml), Ref: 18490505
MIC: 0.5 (ug/ml), Ref: 18490505
MIC: 0.25 (ug/ml), Ref: 18490505
MIC: 0.25 (ug/ml), Ref: 18411322
MIC: 0.5 (ug/ml), Ref: 18411322
MIC: 8 (ug/ml), Ref: 18411322
MIC: 0.25 (ug/ml), Ref: 18443108
MIC: 1 (ug/ml), Ref: 18443108
MIC: 8 (ug/ml), Ref: 18443108
MIC: 0.06 (ug/ml), Ref: 20833454
MIC: 0.125 (ug/ml), Ref: 20833454
MIC: 0.12 (ug/ml), Ref: 19104025
MIC: 2 (ug/ml), Ref: 19104025
MIC: 0.06 (ug/ml), Ref: 19104025
MIC: 1 (ug/ml), Ref: 19104025
MIC50: 0.25 (ug/ml), Ref: 19001109
MIC: 0.12 (ug/ml), Ref: 19001109
MIC90: 0.5 (ug/ml), Ref: 19001109
MIC50: 4 (ug/ml), Ref: 19001109
MIC: 0.0003 (ug/ml), Ref: 19064900
MIC: 0.16 (ug/ml), Ref: 19075065
MBC: 0.63 (ug/ml), Ref: 19075065
MIC: 0.12 (ug/ml), Ref: 19114671
MIC: 0.25 (ug/ml), Ref: 19114671
MIC: 16 (ug/ml), Ref: 19114671
MIC50: 8 (ug/ml), Ref: 19114671
MIC50: 0.25 (ug/ml), Ref: 19114671
MIC50: 16 (ug/ml), Ref: 19114671
MIC90: 8 (ug/ml), Ref: 19114671
MIC90: 32 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19124664
MIC90: 0.5 (ug/ml), Ref: 19124664
MIC50: 0.5 (ug/ml), Ref: 19124664
MIC: 4 (ug/ml), Ref: 19188391
MIC: 0.06 (ug/ml), Ref: 19188391
MIC90: 0.5 (ug/ml), Ref: 19289528
MIC50: 0.25 (ug/ml), Ref: 19289528
MIC: 0.5 (ug/ml), Ref: 19651906
MIC50: 8 (ug/ml), Ref: 19651906
MIC90: 0.25 (ug/ml), Ref: 19506065
MIC50: 0.12 (ug/ml), Ref: 19506065
MIC: 0.06 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19506065
MIC: 0.125 (ug/ml), Ref: 19651906
MIC50: 0.125 (ug/ml), Ref: 19651906
MIC90: 8 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 16 (ug/ml), Ref: 19651906
MBC: 0.125 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 8 (ug/ml), Ref: 19651906
MIC: 0.25 (ug/ml), Ref: 19546358
MIC: 4 (ug/ml), Ref: 19546358
MIC: 8 (ug/ml), Ref: 19546358
MIC: 16 (ug/ml), Ref: 19546358
MIC: 32 (ug/ml), Ref: 19546358
MIC: 64 (ug/ml), Ref: 19546358
MIC: 0.25 (ug/ml), Ref: 19738006
MIC: 0.5 (ug/ml), Ref: 19738006
MIC: 8 (ug/ml), Ref: 19738006
MIC: 0.125 (ug/ml), Ref: 21232952
MIC: 8 (ug/ml), Ref: 21232952
MIC: 32 (ug/ml), Ref: 21232952
MIC: 1 (ug/ml), Ref: 20660686
MIC: 0.25 (ug/ml), Ref: 20660686
MIC50: 0.12 (ug/ml), Ref: 18625769
MIC50: 8 (ug/ml), Ref: 18625769
MIC90: 16 (ug/ml), Ref: 18625769
MIC90: 8 (ug/ml), Ref: 18625769
MIC90: 16 (ug/ml), Ref: 19738018
MIC: 0.25 (ug/ml), Ref: 20660673
MIC: 0.5 (ug/ml), Ref: 18676888
MBC: 0.015 (ug/ml), Ref: 18676888
MIC: 0.07 (ug/ml), Ref: 21458275
MIC: 25 (ug/ml), Ref: 21458275
MIC: 100 (ug/ml), Ref: 21458275
MIC50: 16 (ug/ml), Ref: 21425851
MIC: 0.06 (ug/ml), Ref: 21515052
MIC: 1 (ug/ml), Ref: 21515052
MIC: 0.25 (ug/ml), Ref: 21481984
MIC: 0.125 (ug/ml), Ref: 21481984
MIC: 0.12 (ug/ml), Ref: 21510638
MIC: 0.25 (ug/ml), Ref: 21764484
MIC: 0.06 (ug/ml), Ref: 21764484
MIC50: 16 (ug/ml), Ref: 22148555
MIC: 0.25 (ug/ml), Ref: 22148555
MIC: 0.25 (ug/ml), Ref: 22841282
MIC: 32 (ug/ml), Ref: 22841282
MIC: 16 (ug/ml), Ref: 22841282
MIC: 0.5 (ug/ml), Ref: 22841282
MIC: 0.12 (ug/ml), Ref: 22939698
MIC: 16 (ug/ml), Ref: 22779424
MIC: 0.125 (ug/ml), Ref: 22779424
MIC: 8 (ug/ml), Ref: 22779424
MIC: 100 (ug/ml), Ref: 10.1007/s00044-011-9549-9
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-011-9549-9
MIC: 0.25 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.39 (ug/ml), Ref: 10.1007/s00044-013-0581-9
MIC50: 16 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC: 16 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC: 8 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC90: 0.5 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC50: 0.5 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC50: 0.25 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MBC: 0.5 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MBC: 0.25 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC: 0.25 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC: 0.125 (ug/ml), Ref: 10.1007/s00044-012-0429-8
MIC50: 0.25 (ug/ml), Ref: 23265890
MIC: 0.1 (ug/ml), Ref: 23409972
MIC: 32 (ug/ml), Ref: 23402878
MIC: 0.125 (ug/ml), Ref: 23402878
MIC: 0.06 (ug/ml), Ref: 23402878
MIC90: 16 (ug/ml), Ref: 23206863
MIC50: 0.25 (ug/ml), Ref: 23735742
MBC: 8 (ug/ml), Ref: 10.1007/s00044-013-0844-5
MIC: 2 (ug/ml), Ref: 10.1007/s00044-013-0844-5
MIC: 0.5 (ug/ml), Ref: 24447849
MIC: 0.13 (ug/ml), Ref: 24098982
MIC: 4 (ug/ml), Ref: 24098982
MIC: 3.12 (ug/ml), Ref: 24852274
MIC: 0.5 (ug/ml), Ref: 24798098
MIC90: 32 (ug/ml), Ref: 24959892
MIC90: 64 (ug/ml), Ref: 24959892
MIC: 0.008 (ug/ml), Ref: 25218911
MIC: 0.125 (ug/ml), Ref: 25218911
MIC: 32 (ug/ml), Ref: 25218911
MIC: 0.13 (ug/ml), Ref: 25286019
MIC: 0.25 (ug/ml), Ref: 25286019
MIC: 0.25 (ug/ml), Ref: 25851938
MIC: 0.25 (ug/ml), Ref: 25911300
MIC: 0.25 (ug/ml), Ref: 25978963
MIC: 0.25 (ug/ml), Ref: 26152426
MIC: 32 (ug/ml), Ref: 26238324
MIC: 0.25 (ug/ml), Ref: 26238324
MIC: 4 (ug/ml), Ref: 26238324
MIC: 0.25 (ug/ml), Ref: 26191374
MIC: 8 (ug/ml), Ref: 26191374
MIC: 0.25 (ug/ml), Ref: 26317881
MIC: 0.125 (ug/ml), Ref: 26476970
MIC: 8 (ug/ml), Ref: 26476970
MIC: 0.25 (ug/ml), Ref: 26476970
MIC: 0.5 (ug/ml), Ref: 26476970
MIC: 64 (ug/ml), Ref: 26476970
MIC: 0.125 (ug/ml), Ref: 26522947
MIC: 4 (ug/ml), Ref: 26522947
MIC: 8 (ug/ml), Ref: 26522947
MIC: 0.25 (ug/ml), Ref: 26435513
MIC: 8 (ug/ml), Ref: 26435513
MIC: 0.125 (ug/ml), Ref: 26435513
MIC: 0.5 (ug/ml), Ref: 26435513
MIC: 64 (ug/ml), Ref: 26435513
MIC: 0.26 (ug/ml), Ref: 10.1039/C5MD00297D
MIC: 0.125 (ug/ml), Ref: 27020299
MIC: 0.25 (ug/ml), Ref: 27020299
MIC: 0.5 (ug/ml), Ref: 27020299
MIC: 64 (ug/ml), Ref: 27020299
MIC: 8 (ug/ml), Ref: 27020299
MIC: 28 (ug/ml), Ref: 27324976
MIC: 16 (ug/ml), Ref: 27293070
MIC: 0.5 (ug/ml), Ref: 27293070
MIC: 32 (ug/ml), Ref: 27293070
MBC: 0.97 (nM), Ref: 22036229
TCMC1475
TCMT1340 Staphylococcus faecalis Staphylococcus faecalis MIC: 16 (ug/ml), Ref: 2842501
TCMC1475
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 2842501
MIC: 16 (ug/ml), Ref: 15149694
MIC: 0.25 (ug/ml), Ref: 12824037
MIC: 0.5 (ug/ml), Ref: 12824037
MIC: 0.78 (ug/ml), Ref: 15380226
MIC: 1 (ug/ml), Ref: 16078842
MIC: 2 (ug/ml), Ref: 16078842
MIC: 16 (ug/ml), Ref: 15911248
MIC: 0.5 (ug/ml), Ref: 17064062
MIC: 16 (ug/ml), Ref: 17064062
MIC50: 16 (ug/ml), Ref: 17101672
MIC: 1 (ug/ml), Ref: 17116668
MIC: 1 (ug/ml), Ref: 17116666
MIC: 2 (ug/ml), Ref: 17116668
MIC: 3 (ug/ml), Ref: 17116668
MIC: 16 (ug/ml), Ref: 17116666
MIC: 32 (ug/ml), Ref: 17116666
MIC: 0.5 (ug/ml), Ref: 17116666
MIC: 2 (ug/ml), Ref: 17116666
MIC: 4 (ug/ml), Ref: 17116666
MIC: 64 (ug/ml), Ref: 17116666
MIC50: 0.5 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 17261623
MIC50: 16 (ug/ml), Ref: 17261623
MIC90: 16 (ug/ml), Ref: 17261623
MIC: 0.5 (ug/ml), Ref: 17261623
MIC: 32 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 17220419
MIC: 2 (ug/ml), Ref: 17220419
MIC: 4 (ug/ml), Ref: 17220419
MIC: 64 (ug/ml), Ref: 17220419
MIC: 16 (ug/ml), Ref: 17220419
MIC: 8 (ug/ml), Ref: 17220419
MIC: 0.5 (ug/ml), Ref: 17220419
MIC: 32 (ug/ml), Ref: 17220419
MIC50: 1 (ug/ml), Ref: 17242152
MIC90: 1 (ug/ml), Ref: 17242152
MIC50: 1 (ug/ml), Ref: 17210772
MIC90: 1 (ug/ml), Ref: 17210772
MIC: 0.025 (ug/ml), Ref: 17296740
MIC: 0.5 (ug/ml), Ref: 17303420
MIC: 16 (ug/ml), Ref: 17303420
MIC: 1 (ug/ml), Ref: 17157008
MIC: 0.195 (ug/ml), Ref: 17826097
MIC: 1 (ug/ml), Ref: 17371817
MIC: 0.5 (ug/ml), Ref: 18330977
MIC: 8 (ug/ml), Ref: 18330977
MIC50: 1 (ug/ml), Ref: 17502407
MIC90: 2 (ug/ml), Ref: 17502407
MIC: 0.032 (ug/ml), Ref: 17502407
MIC: 0.008 (ug/ml), Ref: 17502407
MIC: 0.064 (ug/ml), Ref: 17502407
MIC: 0.004 (ug/ml), Ref: 17502407
MIC: 0.5 (ug/ml), Ref: 18457383
MIC: 32 (ug/ml), Ref: 18457383
MIC50: 1 (ug/ml), Ref: 17606677
MIC90: 1 (ug/ml), Ref: 17606677
MIC: 0.25 (ug/ml), Ref: 17606689
MIC: 0.5 (ug/ml), Ref: 17606689
MIC50: 0.5 (ug/ml), Ref: 17606689
MIC90: 1 (ug/ml), Ref: 17606689
MIC90: 4 (ug/ml), Ref: 17606689
MIC: 0.5 (ug/ml), Ref: 17664329
MIC: 16 (ug/ml), Ref: 17664329
MIC: 8 (ug/ml), Ref: 17664329
MIC: 2 (ug/ml), Ref: 17548487
MIC: 16 (ug/ml), Ref: 17548487
MIC: 8 (ug/ml), Ref: 17548487
MIC: 1 (ug/ml), Ref: 17548487
MIC: 0.5 (ug/ml), Ref: 17548487
MIC: 1 (ug/ml), Ref: 17876003
MIC: 4 (ug/ml), Ref: 17876003
MIC: 16 (ug/ml), Ref: 17876003
MIC: 0.5 (ug/ml), Ref: 17876003
MIC: 8 (ug/ml), Ref: 17876003
MIC: 32 (ug/ml), Ref: 17876003
MIC: 2 (ug/ml), Ref: 17876003
MIC50: 1 (ug/ml), Ref: 17908940
MIC90: 1 (ug/ml), Ref: 17908940
MIC: 1 (ug/ml), Ref: 17938189
MIC: 2 (ug/ml), Ref: 17938189
MIC: 0.5 (ug/ml), Ref: 17938189
MIC: 16 (ug/ml), Ref: 17938189
MIC: 8 (ug/ml), Ref: 17938189
MIC: 32 (ug/ml), Ref: 17938189
MIC: 4 (ug/ml), Ref: 17938189
MIC90: 16 (ug/ml), Ref: 17938189
MIC50: 16 (ug/ml), Ref: 17938189
MIC90: 1 (ug/ml), Ref: 17938189
MIC50: 1 (ug/ml), Ref: 17938189
MIC90: 2 (ug/ml), Ref: 17938189
MIC90: 8 (ug/ml), Ref: 17938189
MIC90: 4 (ug/ml), Ref: 17938189
MIC: 64 (ug/ml), Ref: 17938189
MIC: 1 (ug/ml), Ref: 17664314
MIC: 0.5 (ug/ml), Ref: 17664314
MIC: 2 (ug/ml), Ref: 17664314
MIC: 8 (ug/ml), Ref: 17664314
MIC: 1 (ug/ml), Ref: 17846144
MBC: 1 (ug/ml), Ref: 17846144
MIC: 2 (ug/ml), Ref: 17846144
MIC: 32 (ug/ml), Ref: 19481308
MIC: 16 (ug/ml), Ref: 20008781
MIC: 4 (ug/ml), Ref: 20008781
MIC: 8 (ug/ml), Ref: 20008781
MIC: 2 (ug/ml), Ref: 20008781
MIC: 32 (ug/ml), Ref: 20008781
MIC90: 32 (ug/ml), Ref: 20008781
MIC50: 2 (ug/ml), Ref: 20008781
MIC: 2 (ug/ml), Ref: 20667731
MIC50: 1 (ug/ml), Ref: 19884376
MIC90: 2 (ug/ml), Ref: 19884376
MIC90: 16 (ug/ml), Ref: 19884376
MIC: 1 (ug/ml), Ref: 19884376
MIC: 0.06 (ug/ml), Ref: 19884376
MIC50: 16 (ug/ml), Ref: 19884376
MIC50: 1 (ug/ml), Ref: 20065058
MIC50: 16 (ug/ml), Ref: 20065058
MIC: 0.5 (ug/ml), Ref: 20065058
MIC: 8 (ug/ml), Ref: 20065058
MIC90: 2 (ug/ml), Ref: 20065058
MIC: 0.5 (ug/ml), Ref: 18316525
MIC: 1 (ug/ml), Ref: 18316525
MIC: 2 (ug/ml), Ref: 18316525
MIC: 8 (ug/ml), Ref: 18316525
MIC90: 1 (ug/ml), Ref: 18362188
MIC50: 1 (ug/ml), Ref: 18362188
MIC: 0.5 (ug/ml), Ref: 18362188
MIC: 1 (ug/ml), Ref: 18362188
MIC: 0.25 (ug/ml), Ref: 18362188
MIC50: 1 (ug/ml), Ref: 18362189
MIC90: 1 (ug/ml), Ref: 18362189
MIC90: 2 (ug/ml), Ref: 18362189
MIC90: 4 (ug/ml), Ref: 18362189
MIC90: 8 (ug/ml), Ref: 18362189
MIC50: 16 (ug/ml), Ref: 18362189
MIC90: 16 (ug/ml), Ref: 18362189
MIC: 0.5 (ug/ml), Ref: 18362189
MIC: 4 (ug/ml), Ref: 18362189
MIC50: 1 (ug/ml), Ref: 18413298
MIC90: 1 (ug/ml), Ref: 18413298
MIC50: 1 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC: 0.5 (ug/ml), Ref: 18443115
MIC90: 64 (ug/ml), Ref: 20176911
MIC50: 16 (ug/ml), Ref: 20176911
MIC: 8 (ug/ml), Ref: 20176911
MIC: 0.5 (ug/ml), Ref: 18180346
MIC50: 1 (ug/ml), Ref: 18180346
MIC: 2 (ug/ml), Ref: 18160515
MIC: 16 (ug/ml), Ref: 18160515
MIC: 32 (ug/ml), Ref: 18160515
MIC: 8 (ug/ml), Ref: 18160515
MIC90: 1 (ug/ml), Ref: 20231392
MIC50: 1 (ug/ml), Ref: 20231392
MIC: 0.25 (ug/ml), Ref: 20231392
MIC: 0.5 (ug/ml), Ref: 20231392
MIC90: 0.25 (ug/ml), Ref: 20439616
MIC50: 0.125 (ug/ml), Ref: 20439616
MIC90: 1 (ug/ml), Ref: 18725443
MIC90: 16 (ug/ml), Ref: 18725443
MIC50: 16 (ug/ml), Ref: 18725443
MIC50: 1 (ug/ml), Ref: 18725443
MIC90: 1 (ug/ml), Ref: 18725443
MIC50: 1 (ug/ml), Ref: 18725443
MIC90: 1 (ug/ml), Ref: 18443117
MIC90: 2 (ug/ml), Ref: 18443117
MIC90: 0 (ug/ml), Ref: 18443117
MIC90: 100 (ug/ml), Ref: 18443117
MIC90: 97 (ug/ml), Ref: 18443117
MIC: 0.12 (ug/ml), Ref: 18443122
MIC50: 0.5 (ug/ml), Ref: 18443122
MIC90: 1 (ug/ml), Ref: 18443122
MIC: 0.25 (ug/ml), Ref: 18443122
MIC: 4 (ug/ml), Ref: 20833454
MIC: 2 (ug/ml), Ref: 20833454
MIC: 4 (ug/ml), Ref: 18725440
MIC: 2 (ug/ml), Ref: 18725440
MIC: 1 (ug/ml), Ref: 18725440
MIC50: 1 (ug/ml), Ref: 19001109
MIC: 0.5 (ug/ml), Ref: 19001109
MIC90: 1 (ug/ml), Ref: 19001109
MIC50: 0.5 (ug/ml), Ref: 19001109
MIC: 0.25 (ug/ml), Ref: 19001109
MIC: 32 (ug/ml), Ref: 18725440
MIC: 16 (ug/ml), Ref: 18725440
MIC: 8 (ug/ml), Ref: 18725440
MIC: 4 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19114671
MIC50: 16 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 1 (ug/ml), Ref: 19114671
MIC90: 2 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19307366
MIC: 0.5 (ug/ml), Ref: 19307366
MIC: 16 (ug/ml), Ref: 19307366
MIC: 2 (ug/ml), Ref: 19307366
MIC: 32 (ug/ml), Ref: 19307366
MIC50: 1 (ug/ml), Ref: 19307366
MIC90: 16 (ug/ml), Ref: 19307366
MIC90: 2 (ug/ml), Ref: 19307366
MIC90: 4 (ug/ml), Ref: 19307366
MIC50: 2 (ug/ml), Ref: 19307366
MIC: 8 (ug/ml), Ref: 19307366
MIC: 0.5 (ug/ml), Ref: 19451290
MIC: 0.25 (ug/ml), Ref: 19451290
MIC: 1 (ug/ml), Ref: 19451290
MIC: 16 (ug/ml), Ref: 19451290
MIC: 0.25 (ug/ml), Ref: 19506065
MIC: 4 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC50: 16 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
MIC90: 16 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19487444
MIC90: 1 (ug/ml), Ref: 19487444
MIC: 0.06 (ug/ml), Ref: 19487444
MIC90: 1 (ug/ml), Ref: 19738026
MIC: 0.015 (ug/ml), Ref: 21232952
MIC50: 1 (ug/ml), Ref: 20308374
MIC90: 1 (ug/ml), Ref: 20308374
MIC90: 2 (ug/ml), Ref: 20308374
MIC: 0.25 (ug/ml), Ref: 20308374
MIC: 0.5 (ug/ml), Ref: 20308374
MIC50: 0.5 (ug/ml), Ref: 18625769
MIC90: 1 (ug/ml), Ref: 18625769
MIC: 0.25 (ug/ml), Ref: 18625769
MIC: 0.12 (ug/ml), Ref: 18625769
MIC: 0.5 (ug/ml), Ref: 20065057
MIC50: 1 (ug/ml), Ref: 20065057
MIC90: 1 (ug/ml), Ref: 20065057
MIC: 2 (ug/ml), Ref: 21515052
MIC: 0.5 (ug/ml), Ref: 21515052
MIC: 2 (ug/ml), Ref: 21481984
MIC: 16 (ug/ml), Ref: 21764484
MIC: 4 (ug/ml), Ref: 21764484
MIC50: 1 (ug/ml), Ref: 22148555
MIC90: 1 (ug/ml), Ref: 22148555
MIC: 0.5 (ug/ml), Ref: 22148555
MIC: 16 (ug/ml), Ref: 22841282
MIC: 32 (ug/ml), Ref: 22841282
MIC90: 16 (ug/ml), Ref: 23409972
MIC80: 16 (ug/ml), Ref: 23409972
MIC50: 8 (ug/ml), Ref: 23409972
MIC: 0.78 (ug/ml), Ref: 23409972
MIC: 0.125 (ug/ml), Ref: 23402878
MIC: 2 (ug/ml), Ref: 23206863
MIC: 1 (ug/ml), Ref: 24098982
MIC: 1 (ug/ml), Ref: 25286019
MIC: 16 (ug/ml), Ref: 25286019
MIC: 0.125 (ug/ml), Ref: 25218911
MIC: 2 (ug/ml), Ref: 25218911
MIC: 0.5 (ug/ml), Ref: 26238324
MIC: 0.25 (ug/ml), Ref: 26238324
MIC: 0.5 (ug/ml), Ref: 26476970
MIC: 0.5 (ug/ml), Ref: 26435513
MIC: 0.5 (ug/ml), Ref: 27020299
TCMC1475
TCMT1177 Haemophilus influenzae Haemophilus influenzae MIC: 0.015 (ug/ml), Ref: 15149694
MIC: 0.015 (ug/ml), Ref: 15911248
MIC: 0.008 (ug/ml), Ref: 17064062
MIC50: 0.016 (ug/ml), Ref: 17116681
MIC90: 0.32 (ug/ml), Ref: 17116681
MIC50: 0.023 (ug/ml), Ref: 17116681
MIC90: 1 (ug/ml), Ref: 17116681
MIC90: 0.032 (ug/ml), Ref: 17116681
MIC90: 0.047 (ug/ml), Ref: 17116681
MIC: 0.03 (ug/ml), Ref: 17283196
MIC: 0.25 (ug/ml), Ref: 17283196
MIC: 0.5 (ug/ml), Ref: 17283196
MIC: 4 (ug/ml), Ref: 17283196
MIC: 0.12 (ug/ml), Ref: 17283196
MIC: 2 (ug/ml), Ref: 17283196
MIC: 8 (ug/ml), Ref: 17283196
MIC50: 0.015 (ug/ml), Ref: 17261623
MIC90: 0.03 (ug/ml), Ref: 17261623
MIC50: 0.008 (ug/ml), Ref: 17261623
MIC90: 0.015 (ug/ml), Ref: 17261623
MIC50: 0.015 (ug/ml), Ref: 17242152
MIC90: 0.03 (ug/ml), Ref: 17242152
MIC: 0.015 (ug/ml), Ref: 17303420
MIC: 0.008 (ug/ml), Ref: 17157008
MIC: 0.032 (ug/ml), Ref: 18330977
MIC: 0.008 (ug/ml), Ref: 18457383
MIC: 0.06 (ug/ml), Ref: 17606681
MIC: 1 (ug/ml), Ref: 17606681
MIC: 0.016 (ug/ml), Ref: 17606681
MIC50: 0.06 (ug/ml), Ref: 17698631
MIC90: 0.06 (ug/ml), Ref: 17698631
MIC50: 0.06 (ug/ml), Ref: 17908940
MIC90: 0.06 (ug/ml), Ref: 17908940
MIC50: 0.016 (ug/ml), Ref: 19884366
MIC90: 0.031 (ug/ml), Ref: 19884366
MIC90: 0.016 (ug/ml), Ref: 19884366
MIC: 0.15 (ug/ml), Ref: 20667744
MIC: 0.06 (ug/ml), Ref: 20065058
MIC50: 0.25 (ug/ml), Ref: 20065058
MIC90: 8 (ug/ml), Ref: 20065058
MIC: 0.008 (ug/ml), Ref: 18316525
MIC: 0.016 (ug/ml), Ref: 18316525
MIC: 0.004 (ug/ml), Ref: 18426902
MIC50: 0.015 (ug/ml), Ref: 18426902
MIC90: 0.25 (ug/ml), Ref: 18426902
MIC50: 0.12 (ug/ml), Ref: 20231392
MIC90: 0.12 (ug/ml), Ref: 20231392
MIC: 0.12 (ug/ml), Ref: 20231392
MIC50: 0.015 (ug/ml), Ref: 20439616
MIC90: 0.015 (ug/ml), Ref: 20439616
MIC90: 0.015 (ug/ml), Ref: 19001109
MIC50: 0.015 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
MIC: 7.00E-05 (ug/ml), Ref: 19064900
MIC: 0.015 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.06 (ug/ml), Ref: 19114671
MIC: 0.008 (ug/ml), Ref: 19506065
MIC: 1 (ug/ml), Ref: 19506065
MIC50: 0.015 (ug/ml), Ref: 19506065
MIC50: 8 (ug/ml), Ref: 19506065
MIC90: 0.015 (ug/ml), Ref: 19506065
MIC90: 16 (ug/ml), Ref: 19506065
MIC50: 0.015 (ug/ml), Ref: 18625769
MIC90: 0.03 (ug/ml), Ref: 18625769
MIC: 0.004 (ug/ml), Ref: 18625769
MIC: 0.08 (ug/ml), Ref: 20625154
MIC90: 0.06 (ug/ml), Ref: 20625154
MIC50: 0.015 (ug/ml), Ref: 20625154
MIC: 0.15 (ug/ml), Ref: 21458275
MIC50: 0.016 (ug/ml), Ref: 22148555
MIC90: 0.031 (ug/ml), Ref: 22148555
MIC: 0.016 (ug/ml), Ref: 22148555
MIC90: 0.03 (ug/ml), Ref: 23092194
MIC: 0.012 (ug/ml), Ref: 23409972
MIC90: 0.015 (ug/ml), Ref: 24959892
TCMC1475
TCMT1244 Staphylococcus saprophyticus Staphylococcus saprophyticus MIC: 0.12 (ug/ml), Ref: 12824037
MIC: 0.5 (ug/ml), Ref: 16078842
MIC50: 0.25 (ug/ml), Ref: 17261623
MIC90: 0.5 (ug/ml), Ref: 17261623
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 19506065
MIC50: 0.25 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
TCMC1475
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 2 (ug/ml), Ref: 12824037
MIC: 0.3 (ug/ml), Ref: 2824776
MIC: 0.12 (ug/ml), Ref: 7707323
MIC: 0.39 (ug/ml), Ref: 15380226
MIC: 0.25 (ug/ml), Ref: 17261623
MIC50: 8 (ug/ml), Ref: 17261623
MIC90: 64 (ug/ml), Ref: 17261623
MIC: 0.5 (ug/ml), Ref: 17316916
MIC: 0.25 (ug/ml), Ref: 17316916
MIC: 0.78 (ug/ml), Ref: 17826097
MIC: 0.25 (ug/ml), Ref: 18330977
MIC: 32 (ug/ml), Ref: 19481308
MIC: 0.25 (ug/ml), Ref: 20667731
MIC: 0.125 (ug/ml), Ref: 20667731
MIC50: 0.5 (ug/ml), Ref: 20065058
MIC90: 8 (ug/ml), Ref: 20065058
MIC: 0.12 (ug/ml), Ref: 20065058
MIC90: 16 (ug/ml), Ref: 20176911
MIC50: 16 (ug/ml), Ref: 20176911
MIC: 4 (ug/ml), Ref: 20176911
MIC50: 8 (ug/ml), Ref: 20176911
MIC: 0.12 (ug/ml), Ref: 20176911
MIC90: 0.25 (ug/ml), Ref: 20176911
MIC50: 0.12 (ug/ml), Ref: 20176911
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC: 0.25 (ug/ml), Ref: 20833454
MIC: 0.125 (ug/ml), Ref: 20833454
MIC: 2 (ug/ml), Ref: 20833454
MIC50: 0.12 (ug/ml), Ref: 19001109
MIC: 0.06 (ug/ml), Ref: 19001109
MIC90: 0.25 (ug/ml), Ref: 19001109
MIC50: 2 (ug/ml), Ref: 19001109
MIC: 8 (ug/ml), Ref: 19188391
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 0.12 (ug/ml), Ref: 19506065
MIC: 2 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19651906
MIC50: 0.25 (ug/ml), Ref: 19651906
MIC90: 4 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 4 (ug/ml), Ref: 19651906
MBC90: 16 (ug/ml), Ref: 19651906
MIC50: 8 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 4 (ug/ml), Ref: 19651906
MIC: 2 (ug/ml), Ref: 21232952
MIC: 8 (ug/ml), Ref: 21232952
MIC: 0.15 (ug/ml), Ref: 21458275
MIC: 0.125 (ug/ml), Ref: 21515052
MIC: 1 (ug/ml), Ref: 21515052
MIC: 4 (ug/ml), Ref: 21481984
MIC: 0.25 (ug/ml), Ref: 21481984
MIC: 0.5 (ug/ml), Ref: 21764484
MIC: 0.06 (ug/ml), Ref: 21764484
MIC: 2 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 22841282
MIC: 4 (ug/ml), Ref: 22841282
MIC: 0.39 (ug/ml), Ref: 23409972
MIC: 8 (ug/ml), Ref: 23402878
MIC: 0.25 (ug/ml), Ref: 23402878
MIC: 0.125 (ug/ml), Ref: 23402878
MIC: 0.125 (ug/ml), Ref: 25218911
MIC: 0.5 (ug/ml), Ref: 25218911
MIC: 4 (ug/ml), Ref: 25218911
MIC: 32 (ug/ml), Ref: 25218911
MIC: 8 (ug/ml), Ref: 26238324
MIC: 0.5 (ug/ml), Ref: 26317881
MIC: 8 (ug/ml), Ref: 26317881
MIC: 64 (ug/ml), Ref: 26476970
MIC: 32 (ug/ml), Ref: 26476970
MIC: 64 (ug/ml), Ref: 26435513
MIC: 32 (ug/ml), Ref: 26435513
MIC: 1 (ug/ml), Ref: 27020299
MIC: 2 (ug/ml), Ref: 27020299
MIC: 32 (ug/ml), Ref: 27020299
MIC: 64 (ug/ml), Ref: 27020299
MIC: 16 (ug/ml), Ref: 27293070
MIC: 0.5 (ug/ml), Ref: 27293070
TCMC1475
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 0.25 (ug/ml), Ref: 12824037
MIC: 1 (ug/ml), Ref: 12824037
MIC: 0.46 (ug/ml), Ref: 2824776
MIC: 64 (ug/ml), Ref: 17064062
MIC50: 32 (ug/ml), Ref: 17261623
MIC90: 64 (ug/ml), Ref: 17261623
MIC50: 64 (ug/ml), Ref: 17261623
MIC: 4 (ug/ml), Ref: 17261623
MIC: 4 (ug/ml), Ref: 18330977
MIC: 64 (ug/ml), Ref: 18330977
MIC: 2 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 18316525
MIC: 4 (ug/ml), Ref: 18316525
MIC50: 4 (ug/ml), Ref: 20231392
MIC50: 4 (ug/ml), Ref: 18591277
MIC: 1 (ug/ml), Ref: 18591277
MIC: 8 (ug/ml), Ref: 20833454
MIC: 2 (ug/ml), Ref: 20833454
MIC50: 4 (ug/ml), Ref: 19001109
MIC: 1 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19114671
MIC50: 2 (ug/ml), Ref: 19114671
MIC50: 32 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19506065
MIC: 4 (ug/ml), Ref: 21481984
MIC: 16 (ug/ml), Ref: 21481984
MIC: 4 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 21764484
MIC: 32 (ug/ml), Ref: 22841282
MIC: 32 (ug/ml), Ref: 26317881
MIC: 64 (ug/ml), Ref: 26317881
MIC: 16 (ug/ml), Ref: 26476970
MIC: 32 (ug/ml), Ref: 26476970
MIC: 64 (ug/ml), Ref: 26476970
MIC: 32 (ug/ml), Ref: 26435513
MIC: 64 (ug/ml), Ref: 26435513
MIC: 1 (ug/ml), Ref: 27020299
TCMC1475
TCMT1314 Streptococcus viridans Streptococcus viridans MIC: 0.25 (ug/ml), Ref: 12824037
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 17242152
MIC90: 1 (ug/ml), Ref: 17242152
MIC: 0.25 (ug/ml), Ref: 17606689
MIC50: 0.5 (ug/ml), Ref: 17606689
MIC90: 1 (ug/ml), Ref: 17606689
MIC: 2 (ug/ml), Ref: 17548487
MIC: 1 (ug/ml), Ref: 17548487
MIC: 16 (ug/ml), Ref: 17548487
MIC50: 1 (ug/ml), Ref: 20065058
MIC: 0.25 (ug/ml), Ref: 20065058
MIC90: 2 (ug/ml), Ref: 20065058
MIC50: 1 (ug/ml), Ref: 20231392
MIC90: 2 (ug/ml), Ref: 20231392
MIC: 0.25 (ug/ml), Ref: 20231392
MIC: 0.12 (ug/ml), Ref: 18443122
MIC: 0.12 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 2 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 18625769
MIC90: 1 (ug/ml), Ref: 18625769
MIC: 0.015 (ug/ml), Ref: 18625769
MIC90: 2 (ug/ml), Ref: 18625769
TCMC1475
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0.008 (ug/ml), Ref: 12824037
MIC: 0.03 (ug/ml), Ref: 7707323
MIC50: 0.06 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC: 0.125 (ug/ml), Ref: 19481308
MIC: 0.125 (ug/ml), Ref: 20667731
MIC50: 2 (ug/ml), Ref: 20065058
MIC90: 16 (ug/ml), Ref: 20065058
MIC: 0.12 (ug/ml), Ref: 20065058
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 0.12 (ug/ml), Ref: 20176911
MIC50: 0.06 (ug/ml), Ref: 20176911
MIC: 0.008 (ug/ml), Ref: 20176911
MIC: 0.25 (ug/ml), Ref: 18809939
MIC: 0.5 (ug/ml), Ref: 18809939
MIC: 1 (ug/ml), Ref: 18809939
MIC: 2 (ug/ml), Ref: 18809939
MIC: 8 (ug/ml), Ref: 18809939
MIC: 32 (ug/ml), Ref: 18809939
MIC: 2 (ug/ml), Ref: 18852270
MIC90: 4 (ug/ml), Ref: 18591277
MIC: 0.38 (ug/ml), Ref: 18519713
MIC: 0.5 (ug/ml), Ref: 18519713
MIC: 0.094 (ug/ml), Ref: 18519713
MIC: 0.75 (ug/ml), Ref: 18519713
MIC: 0.19 (ug/ml), Ref: 18519713
MIC: 1 (ug/ml), Ref: 18519713
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC: 0.03 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 19015359
MIC: 16 (ug/ml), Ref: 19015359
MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 0.12 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
MIC50: 0.06 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.06 (ug/ml), Ref: 19114671
MIC: 0.25 (ug/ml), Ref: 19364872
MIC: 2 (ug/ml), Ref: 19364872
MIC: 0.03 (ug/ml), Ref: 19349512
MBC: 0.03 (ug/ml), Ref: 19349512
MIC: 0.06 (ug/ml), Ref: 19349512
MBC: 0.06 (ug/ml), Ref: 19349512
MIC: 0.008 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 19506065
MIC90: 0.25 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 18625769
MIC50: 0.12 (ug/ml), Ref: 18625769
MIC90: 0.5 (ug/ml), Ref: 18625769
MIC: 0.03 (ug/ml), Ref: 18625769
MIC90: 1 (ug/ml), Ref: 18625769
MIC: 0.06 (ug/ml), Ref: 21515052
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 0.004 (ug/ml), Ref: 12824037
MIC: 4 (ug/ml), Ref: 12824037
MIC: 0.04 (ug/ml), Ref: 2824776
MIC: 0.03 (ug/ml), Ref: 7707323
MIC: 0.05 (ug/ml), Ref: 15380226
MIC: 0.008 (ug/ml), Ref: 16078842
MIC: 0.03 (ug/ml), Ref: 17064062
MIC: 8 (ug/ml), Ref: 17064062
MIC: 4 (ug/ml), Ref: 17074790
MIC: 8 (ug/ml), Ref: 17074790
MIC: 16 (ug/ml), Ref: 17074790
MIC50: 0.06 (ug/ml), Ref: 17261623
MIC90: 0.5 (ug/ml), Ref: 17261623
MIC50: 0.5 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC: 0.25 (ug/ml), Ref: 17316916
MIC: 0.098 (ug/ml), Ref: 17826097
MIC50: 2 (ug/ml), Ref: 17387156
MIC: 2 (ug/ml), Ref: 17404007
MIC: 16 (ug/ml), Ref: 17404007
MIC: 0.5 (ug/ml), Ref: 17404007
MIC: 8 (ug/ml), Ref: 17404007
MIC: 64 (ug/ml), Ref: 17404007
MIC: 4 (ug/ml), Ref: 17404007
MIC: 0.25 (ug/ml), Ref: 17404007
MIC: 0.016 (ug/ml), Ref: 18457383
MIC: 4 (ug/ml), Ref: 17938184
MIC: 1 (ug/ml), Ref: 19481308
MIC: 0.09 (ug/ml), Ref: 19858254
MIC: 0.006 (ug/ml), Ref: 19858254
MIC: 0.19 (ug/ml), Ref: 19858254
MIC: 1 (ug/ml), Ref: 20667731
MIC: 1 (ug/ml), Ref: 20591538
MIC: 0.12 (ug/ml), Ref: 20591538
MIC50: 2 (ug/ml), Ref: 20065058
MIC: 0.06 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 18426899
MIC: 0.75 (ug/ml), Ref: 18426899
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 0.12 (ug/ml), Ref: 20176911
MIC50: 0.06 (ug/ml), Ref: 20176911
MIC: 0.015 (ug/ml), Ref: 20176911
MIC: 0.25 (ug/ml), Ref: 18809939
MIC: 0.5 (ug/ml), Ref: 18809939
MIC: 8 (ug/ml), Ref: 18809939
MIC: 32 (ug/ml), Ref: 18809939
MIC: 0.5 (ug/ml), Ref: 20350950
MIC: 0.12 (ug/ml), Ref: 20350950
MIC: 0.25 (ug/ml), Ref: 20350950
MIC: 0.25 (ug/ml), Ref: 20350950
MIC90: 4 (ug/ml), Ref: 18591277
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC: 0.03 (ug/ml), Ref: 18591277
MIC: 8 (ug/ml), Ref: 20833454
MIC: 16 (ug/ml), Ref: 20833454
MIC: 16 (ug/ml), Ref: 18936192
MIC: 1 (ug/ml), Ref: 18936192
MIC: 0.25 (ug/ml), Ref: 19015359
MIC: 16 (ug/ml), Ref: 19015359
MIC: 0.5 (ug/ml), Ref: 19015359
MIC: 0.125 (ug/ml), Ref: 19015359
MIC: 0.06 (ug/ml), Ref: 19015359
MIC: 2 (ug/ml), Ref: 19015359
MIC: 8 (ug/ml), Ref: 19015359
MIC: 64 (ug/ml), Ref: 19015359
MIC: 32 (ug/ml), Ref: 19015359
MIC: 1 (ug/ml), Ref: 19015359
MIC: 4 (ug/ml), Ref: 19015359
MIC: 0.12 (ug/ml), Ref: 19015360
MIC: 2 (ug/ml), Ref: 19015360
MIC: 1 (ug/ml), Ref: 19015360
MIC50: 2 (ug/ml), Ref: 19015360
MIC50: 0.5 (ug/ml), Ref: 19015360
MIC90: 16 (ug/ml), Ref: 19015360
MIC50: 4 (ug/ml), Ref: 19015360
MIC50: 2 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 0.5 (ug/ml), Ref: 19001109
MIC90: 0.5 (ug/ml), Ref: 19001109
MIC50: 0.06 (ug/ml), Ref: 19001109
MIC: 0.00015 (ug/ml), Ref: 19064900
MIC: 0.015 (ug/ml), Ref: 19114671
MIC: 0.03 (ug/ml), Ref: 19114671
MIC50: 0.06 (ug/ml), Ref: 19114671
MIC50: 0.5 (ug/ml), Ref: 19114671
MIC90: 0.5 (ug/ml), Ref: 19114671
MIC90: 8 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19364872
MIC: 2 (ug/ml), Ref: 19364872
MIC: 0.25 (ug/ml), Ref: 19349512
MIC: 4 (ug/ml), Ref: 19349512
MBC: 2 (ug/ml), Ref: 19349512
MBC: 4 (ug/ml), Ref: 19349512
MIC: 0.004 (ug/ml), Ref: 19506065
MIC50: 0.06 (ug/ml), Ref: 19506065
MIC90: 2 (ug/ml), Ref: 19506065
MIC: 32 (ug/ml), Ref: 21232952
MIC50: 0.06 (ug/ml), Ref: 18625769
MIC50: 8 (ug/ml), Ref: 18625769
MIC90: 0.25 (ug/ml), Ref: 18625769
MIC: 0.03 (ug/ml), Ref: 20679507
MIC: 1 (ug/ml), Ref: 20679507
MIC: 0.06 (ug/ml), Ref: 20679507
MIC: 0.5 (ug/ml), Ref: 20679507
MIC: 0.015 (ug/ml), Ref: 20679507
MIC: 0.125 (ug/ml), Ref: 20679507
MIC: 2 (ug/ml), Ref: 19581455
MIC: 0.5 (ug/ml), Ref: 21515052
MIC: 16 (ug/ml), Ref: 21481984
MIC: 16 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 22841282
MIC: 32 (ug/ml), Ref: 22841282
MIC: 1 (ug/ml), Ref: 22841282
MIC: 1 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.12 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.39 (ug/ml), Ref: 10.1007/s00044-013-0581-9
MIC: 0.05 (ug/ml), Ref: 23409972
MIC: 8 (ug/ml), Ref: 23402878
MIC: 4 (ug/ml), Ref: 23402878
MIC: 1 (ug/ml), Ref: 23402878
MIC: 0.25 (ug/ml), Ref: 23402878
MIC: 0.06 (ug/ml), Ref: 23402878
MIC: 0.06 (ug/ml), Ref: 25218911
MIC: 0.008 (ug/ml), Ref: 25218911
MIC: 16 (ug/ml), Ref: 25218911
MIC: 8 (ug/ml), Ref: 25218911
MIC: 0.5 (ug/ml), Ref: 25218911
MIC90: 64 (ug/ml), Ref: 25155913
MIC: 1 (ug/ml), Ref: 25435146
MIC: 1 (ug/ml), Ref: 26317881
MIC: 0.12 (ug/ml), Ref: 26363871
MIC: 4 (ug/ml), Ref: 26476970
MIC: 1 (ug/ml), Ref: 26476970
MIC: 64 (ug/ml), Ref: 26476970
MIC: 16 (ug/ml), Ref: 26476970
MIC: 8 (ug/ml), Ref: 26476970
MIC: 0.5 (ug/ml), Ref: 26435513
MIC: 64 (ug/ml), Ref: 26435513
MIC: 16 (ug/ml), Ref: 26435513
MIC: 8 (ug/ml), Ref: 26435513
MIC: 32 (ug/ml), Ref: 26435513
MIC: 4 (ug/ml), Ref: 27020299
MIC: 1 (ug/ml), Ref: 27020299
MIC: 64 (ug/ml), Ref: 27020299
MIC: 16 (ug/ml), Ref: 27020299
MIC: 8 (ug/ml), Ref: 27020299
MIC: 30 (nM), Ref: 26214729
TCMC1475
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 0.06 (ug/ml), Ref: 12824037
MIC50: 0.125 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 20591538
MIC: 0.12 (ug/ml), Ref: 20591538
MIC50: 2 (ug/ml), Ref: 20065058
MIC: 0.06 (ug/ml), Ref: 20065058
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC: 0.03 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 19015360
MIC: 2 (ug/ml), Ref: 19015360
MIC: 4 (ug/ml), Ref: 19015360
MIC50: 8 (ug/ml), Ref: 19015360
MIC90: 16 (ug/ml), Ref: 19001109
MIC50: 0.5 (ug/ml), Ref: 19001109
MIC: 0.03 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.25 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19258263
MIC: 0.015 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 19506065
MIC90: 8 (ug/ml), Ref: 19506065
MIC50: 0.06 (ug/ml), Ref: 18625769
MIC90: 16 (ug/ml), Ref: 18625769
MIC: 32 (ug/ml), Ref: 19581455
MIC: 0.25 (ug/ml), Ref: 19581455
MIC90: 0.06 (ug/ml), Ref: 23092194
MIC: 1 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.12 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 1.21 (ug/ml), Ref: 2824776
MIC: 1 (ug/ml), Ref: 16078842
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 20065058
MIC: 0.5 (ug/ml), Ref: 20065058
MIC90: 2 (ug/ml), Ref: 20065058
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18591277
MIC50: 0.5 (ug/ml), Ref: 18591277
MIC: 0.5 (ug/ml), Ref: 18591277
MIC90: 1 (ug/ml), Ref: 18443122
MIC50: 0.5 (ug/ml), Ref: 18443122
MIC: 0.12 (ug/ml), Ref: 18443122
MIC90: 1 (ug/ml), Ref: 19001109
MIC: 0.5 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
MIC: 0.5 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 1 (ug/ml), Ref: 19114671
MIC50: 2 (ug/ml), Ref: 19332682
MIC: 0.5 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
MIC90: 1 (ug/ml), Ref: 19738026
MIC50: 0.5 (ug/ml), Ref: 18625769
MIC50: 1 (ug/ml), Ref: 18625769
MIC90: 1 (ug/ml), Ref: 18625769
MIC: 0.12 (ug/ml), Ref: 18625769
TCMC1475
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 0.07 (ug/ml), Ref: 2824776
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 0.06 (ug/ml), Ref: 20176911
MIC50: 0.06 (ug/ml), Ref: 20176911
MIC: 0.03 (ug/ml), Ref: 20176911
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC90: 0.5 (ug/ml), Ref: 19001109
MIC50: 0.06 (ug/ml), Ref: 19001109
MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 0.12 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
MIC: 0.03 (ug/ml), Ref: 19114671
MIC50: 0.06 (ug/ml), Ref: 19114671
MIC90: 0.5 (ug/ml), Ref: 19114671
MIC: 0.03 (ug/ml), Ref: 19506065
MIC50: 0.06 (ug/ml), Ref: 19506065
MIC90: 16 (ug/ml), Ref: 19506065
MIC: 0.03 (ug/ml), Ref: 21515052
MIC: 0.78 (ug/ml), Ref: 24852274
TCMC1475
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.03 (ug/ml), Ref: 7707323
MIC: 0.5 (ug/ml), Ref: 17316916
MIC: 0.03 (ug/ml), Ref: 20667744
MIC: 0.03 (ug/ml), Ref: 21458275
MIC: 0.12 (ug/ml), Ref: 21510638
MIC: 0.12 (ug/ml), Ref: 22939698
MIC: 0.78 (ug/ml), Ref: 10.1007/s00044-013-0581-9
MIC: 1.56 (ug/ml), Ref: 23409972
MIC50: 0.25 (ug/ml), Ref: 23735742
MIC: 1 (ug/ml), Ref: 24447849
MIC: 0.25 (ug/ml), Ref: 24798098
MIC: 29 (ug/ml), Ref: 27324976
TCMC1475
TCMT1286 Bacillus cereus Bacillus cereus MIC: 0.25 (ug/ml), Ref: 7707323
MIC: 0.15 (ug/ml), Ref: 21458275
TCMC1475
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0.25 (ug/ml), Ref: 7707323
MIC: 0.78 (ug/ml), Ref: 15380226
MIC: 1 (ug/ml), Ref: 16078842
MIC: 1 (ug/ml), Ref: 17064062
MIC: 32 (ug/ml), Ref: 17064062
MIC50: 16 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC: 16 (ug/ml), Ref: 17261623
MIC: 0.5 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 17261623
MIC50: 16 (ug/ml), Ref: 17242152
MIC: 1 (ug/ml), Ref: 17316916
MIC: 2 (ug/ml), Ref: 17157008
MIC: 0.5 (ug/ml), Ref: 18330977
MIC: 1 (ug/ml), Ref: 18457383
MIC: 64 (ug/ml), Ref: 18457383
MIC: 32 (ug/ml), Ref: 18457383
MIC: 8 (ug/ml), Ref: 18056272
MIC: 1 (ug/ml), Ref: 19481308
MIC: 0.5 (ug/ml), Ref: 20667731
MIC: 32 (ug/ml), Ref: 20591538
MIC: 0.5 (ug/ml), Ref: 20591538
MIC50: 2 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 18316525
MIC: 2 (ug/ml), Ref: 18316525
MIC: 32 (ug/ml), Ref: 18316525
MIC: 0.5 (ug/ml), Ref: 18316525
MIC50: 1 (ug/ml), Ref: 20231392
MIC90: 2 (ug/ml), Ref: 18591277
MIC50: 1 (ug/ml), Ref: 18591277
MIC: 0.25 (ug/ml), Ref: 18591277
MIC: 8 (ug/ml), Ref: 20833454
MIC: 4 (ug/ml), Ref: 20833454
MIC50: 2 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
MIC: 0.5 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 32 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19188391
MIC50: 1 (ug/ml), Ref: 19289528
MIC90: 64 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 18625769
MIC: 16 (ug/ml), Ref: 19581455
MIC: 0.25 (ug/ml), Ref: 21515052
MIC: 2 (ug/ml), Ref: 21515052
MIC: 8 (ug/ml), Ref: 21481984
MIC: 0.5 (ug/ml), Ref: 21510638
MIC: 8 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 22841282
MIC: 64 (ug/ml), Ref: 22841282
MIC: 16 (ug/ml), Ref: 22841282
MIC: 0.5 (ug/ml), Ref: 22939698
MIC: 32 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.78 (ug/ml), Ref: 23409972
MIC90: 32 (ug/ml), Ref: 24959892
MIC90: 64 (ug/ml), Ref: 24959892
MIC: 0.5 (ug/ml), Ref: 26317881
MIC: 1 (ug/ml), Ref: 26476970
MIC: 1 (ug/ml), Ref: 26435513
MIC: 16 (ug/ml), Ref: 27020299
MIC: 32 (ug/ml), Ref: 27020299
MIC: 64 (ug/ml), Ref: 27020299
MIC: 2 (ug/ml), Ref: 27293070
MIC: 4 (ug/ml), Ref: 27293070
TCMC1475
TCMT1299 Morganella morganii Morganella morganii MIC: 0.03 (ug/ml), Ref: 7707323
MIC50: 0.125 (ug/ml), Ref: 17261623
MIC90: 16 (ug/ml), Ref: 17261623
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 64 (ug/ml), Ref: 18591277
MIC50: 1 (ug/ml), Ref: 18591277
MIC50: 0.03 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19114671
MIC50: 0.06 (ug/ml), Ref: 19114671
MIC90: 8 (ug/ml), Ref: 19114671
MIC: 0.015 (ug/ml), Ref: 19506065
MIC50: 0.06 (ug/ml), Ref: 19506065
MIC90: 8 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 18625769
MIC90: 8 (ug/ml), Ref: 18625769
MIC: 0.03 (ug/ml), Ref: 21515052
MIC: 16 (ug/ml), Ref: 21510638
MIC: 16 (ug/ml), Ref: 22939698
MIC: 0.78 (ug/ml), Ref: 24852274
MIC: 0.06 (ug/ml), Ref: 26317881
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 0.39 (ug/ml), Ref: 15380226
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 17548487
MIC: 0.25 (ug/ml), Ref: 17548487
MIC: 0.5 (ug/ml), Ref: 17548487
MIC: 2 (ug/ml), Ref: 17548487
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.03 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 18443122
MIC90: 0.12 (ug/ml), Ref: 18591277
MIC50: 0.03 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 2 (ug/ml), Ref: 16078842
MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1358 Bacteroides vulgatus Bacteroides vulgatus MIC: 1 (ug/ml), Ref: 16078842
MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 8 (ug/ml), Ref: 18625771
TCMC1475
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 0.12 (ug/ml), Ref: 16078842
MIC50: 0.25 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 8 (ug/ml), Ref: 19001109
MIC90: 16 (ug/ml), Ref: 19001109
MIC: 0.06 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19651906
MIC50: 0.25 (ug/ml), Ref: 19651906
MIC90: 4 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 4 (ug/ml), Ref: 19651906
MIC50: 4 (ug/ml), Ref: 19506065
MBC90: 16 (ug/ml), Ref: 19651906
MIC90: 0.5 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 4 (ug/ml), Ref: 19651906
TCMC1475
TCMT1207 Legionella pneumophila Legionella pneumophila MIC50: 0.12 (ug/ml), Ref: 17101672
MIC90: 0.5 (ug/ml), Ref: 17101672
MIC50: 0.008 (ug/ml), Ref: 17261623
MIC90: 0.015 (ug/ml), Ref: 17261623
MIC: 0.015 (ug/ml), Ref: 17242152
MIC: 0.002 (ug/ml), Ref: 18426902
MIC50: 0.004 (ug/ml), Ref: 18426902
MIC90: 0.015 (ug/ml), Ref: 18426902
MIC: 0.015 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 19506065
MIC90: 0.03 (ug/ml), Ref: 19506065
TCMC1475
TCMT1203 Mycoplasma pneumoniae Mycoplasma pneumoniae MIC50: 0.5 (ug/ml), Ref: 17101672
MIC90: 1 (ug/ml), Ref: 17101672
MIC: 0.5 (ug/ml), Ref: 17242152
MIC: 0.5 (ug/ml), Ref: 17387152
MIC: 0.25 (ug/ml), Ref: 17387152
MIC: 0.125 (ug/ml), Ref: 18330977
MIC: 0.063 (ug/ml), Ref: 18330977
MIC50: 0.5 (ug/ml), Ref: 17954691
MIC50: 1 (ug/ml), Ref: 17954691
MIC90: 1 (ug/ml), Ref: 17954691
MIC: 0.125 (ug/ml), Ref: 17954691
MIC: 0.5 (ug/ml), Ref: 17954691
MIC: 0.25 (ug/ml), Ref: 18663020
MIC50: 0.5 (ug/ml), Ref: 18663020
MIC90: 1 (ug/ml), Ref: 18663020
MIC: 0.125 (ug/ml), Ref: 19258276
MIC50: 0.5 (ug/ml), Ref: 19258276
MIC90: 0.5 (ug/ml), Ref: 19258276
MIC: 0.015 (ug/ml), Ref: 19273684
MIC: 0.25 (ug/ml), Ref: 19273684
MIC50: 0.25 (ug/ml), Ref: 19273684
MIC90: 0.5 (ug/ml), Ref: 19273684
MIC: 0.012 (ug/ml), Ref: 19738013
MIC50: 1 (ug/ml), Ref: 19738013
MIC90: 1 (ug/ml), Ref: 19738013
MIC: 1 (ug/ml), Ref: 23409972
MIC: 2 (ug/ml), Ref: 23409972
TCMC1475
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 0.03 (ug/ml), Ref: 17043131
MIC: 0.015 (ug/ml), Ref: 17043131
MIC: 0.5 (ug/ml), Ref: 17043131
MIC: 0.06 (ug/ml), Ref: 17043131
MIC: 1 (ug/ml), Ref: 17043131
MIC: 0.25 (ug/ml), Ref: 17043131
MIC: 0.12 (ug/ml), Ref: 17043131
MIC: 2 (ug/ml), Ref: 17043131
MIC: 8 (ug/ml), Ref: 17043131
MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 0.06 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 19596880
MIC: 0.78 (ug/ml), Ref: 24852274
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC50: 0.008 (ug/ml), Ref: 17261623
MIC90: 0.008 (ug/ml), Ref: 17261623
MIC: 2 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 20065058
MIC: 0.5 (ug/ml), Ref: 20065058
MIC90: 0.5 (ug/ml), Ref: 23092194
TCMC1475
TCMT1401 Staphylococcus warneri Staphylococcus warneri MIC: 0.125 (ug/ml), Ref: 17261623
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 19506065
MIC50: 0.12 (ug/ml), Ref: 19506065
TCMC1475
TCMT1380 Enterococcus gallinarum Enterococcus gallinarum MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
TCMC1475
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC50: 0.5 (ug/ml), Ref: 18227183
MIC90: 1 (ug/ml), Ref: 18227183
MIC: 0.5 (ug/ml), Ref: 18426902
MIC50: 1 (ug/ml), Ref: 18426902
MIC90: 1 (ug/ml), Ref: 18426902
MIC: 0.125 (ug/ml), Ref: 18227183
MIC50: 1 (ug/ml), Ref: 20231392
MIC90: 1 (ug/ml), Ref: 20231392
MIC: 1 (ug/ml), Ref: 20231392
MIC: 1 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 1 (ug/ml), Ref: 19114671
MIC90: 1 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19506065
TCMC1475
TCMT1397 Corynebacterium jeikeium Corynebacterium jeikeium MIC50: 0.25 (ug/ml), Ref: 17261623
MIC90: 0.5 (ug/ml), Ref: 17261623
MIC: 0.06 (ug/ml), Ref: 18227183
MIC50: 4 (ug/ml), Ref: 18227183
MIC: 0.5 (ug/ml), Ref: 19114671
TCMC1475
TCMT1436 Corynebacterium sp. Corynebacterium sp. MIC50: 0.5 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC: 0.25 (ug/ml), Ref: 18426902
MIC50: 0.5 (ug/ml), Ref: 18426902
MIC90: 32 (ug/ml), Ref: 18426902
TCMC1475
TCMT1389 Klebsiella oxytoca Klebsiella oxytoca MIC50: 0.06 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC90: 0.25 (ug/ml), Ref: 19001109
MIC50: 0.03 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
MIC: 0.25 (ug/ml), Ref: 19364872
MIC: 4 (ug/ml), Ref: 19364872
MIC: 0.5 (ug/ml), Ref: 19364872
MIC: 0.015 (ug/ml), Ref: 19506065
MIC50: 0.03 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
TCMC1475
TCMT1289 Shigella dysenteriae Shigella dysenteriae MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 0.06 (ug/ml), Ref: 17261623
TCMC1475
TCMT1271 Shigella flexneri Shigella flexneri MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 0.06 (ug/ml), Ref: 17261623
MIC: 0.03 (ug/ml), Ref: 17316916
TCMC1475
TCMT1194 Shigella sonnei Shigella sonnei MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 0.06 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 19481308
MIC: 1 (ug/ml), Ref: 20667731
MIC: 0.03 (ug/ml), Ref: 21515052
MIC: 3.12 (ug/ml), Ref: 24852274
TCMC1475
TCMT1198 Serratia marcescens Serratia marcescens MIC50: 0.125 (ug/ml), Ref: 17261623
MIC90: 4 (ug/ml), Ref: 17261623
MIC: 0.5 (ug/ml), Ref: 17316916
MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.06 (ug/ml), Ref: 18591277
MIC90: 4 (ug/ml), Ref: 19001109
MIC50: 0.12 (ug/ml), Ref: 19001109
MIC: 0.06 (ug/ml), Ref: 19001109
MIC90: 8 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
MIC: 0.06 (ug/ml), Ref: 19114671
MIC50: 0.12 (ug/ml), Ref: 19114671
MIC90: 0.25 (ug/ml), Ref: 19114671
MIC: 0.19 (ug/ml), Ref: 19188391
MIC: 0.03 (ug/ml), Ref: 19506065
MIC50: 0.12 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
MIC50: 0.12 (ug/ml), Ref: 18625769
MIC90: 1 (ug/ml), Ref: 18625769
MIC: 0.03 (ug/ml), Ref: 18625769
MIC: 0.25 (ug/ml), Ref: 21515052
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1331 Acinetobacter sp. Acinetobacter sp. MIC50: 0.125 (ug/ml), Ref: 17261623
MIC90: 16 (ug/ml), Ref: 17261623
MIC: 2 (ug/ml), Ref: 17470660
MIC: 4 (ug/ml), Ref: 17470660
MIC50: 2 (ug/ml), Ref: 18426902
MIC90: 16 (ug/ml), Ref: 18426902
TCMC1475
TCMT1360 Bacteroides ovatus Bacteroides ovatus MIC50: 8 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
TCMC1475
TCMT1281 Clostridium difficile Clostridium difficile MIC50: 0.5 (ug/ml), Ref: 17261623
MIC90: 0.5 (ug/ml), Ref: 17261623
MIC: 8 (ug/ml), Ref: 17562807
MIC50: 4 (ug/ml), Ref: 17517836
MIC90: 32 (ug/ml), Ref: 17517836
MIC: 2 (ug/ml), Ref: 19364867
MIC: 1 (ug/ml), Ref: 19364867
MIC: 64 (ug/ml), Ref: 19364867
MIC: 8 (ug/ml), Ref: 19364867
MIC: 16 (ug/ml), Ref: 19364867
MIC: 4 (ug/ml), Ref: 19364867
TCMC1475
TCMT1204 Clostridium perfringens Clostridium perfringens MIC50: 0.5 (ug/ml), Ref: 17261623
MIC90: 0.5 (ug/ml), Ref: 17261623
MIC: 0.25 (ug/ml), Ref: 18330977
MIC: 0.25 (ug/ml), Ref: 18625771
MIC50: 0.5 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 0.03 (ug/ml), Ref: 17261623
MIC: 0.12 (ug/ml), Ref: 18625771
MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1369 Fusobacterium necrophorum Fusobacterium necrophorum MIC: 0.03 (ug/ml), Ref: 17261623
MIC: 0.12 (ug/ml), Ref: 18625771
MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1386 Fusobacterium sp. Fusobacterium sp. MIC: 0.03 (ug/ml), Ref: 17261623
TCMC1475
TCMT1363 Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC: 0.125 (ug/ml), Ref: 17261623
MIC: 0.125 (ug/ml), Ref: 18330977
MIC50: 0.5 (ug/ml), Ref: 18625771
MIC90: 32 (ug/ml), Ref: 18625771
TCMC1475
TCMT1366 Prevotella bivia Prevotella bivia MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 18625771
MIC90: 16 (ug/ml), Ref: 18625771
TCMC1475
TCMT1365 Prevotella buccae Prevotella buccae MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 18625771
MIC90: 16 (ug/ml), Ref: 18625771
TCMC1475
TCMT1387 Prevotella corporis Prevotella corporis MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
TCMC1475
TCMT1370 Prevotella melaninogenica Prevotella melaninogenica MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
MIC50: 1 (ug/ml), Ref: 18625771
MIC90: 16 (ug/ml), Ref: 18625771
TCMC1475
TCMT1364 Prevotella oralis Prevotella oralis MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 2 (ug/ml), Ref: 17261623
TCMC1475
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC50: 0.008 (ug/ml), Ref: 17261623
MIC90: 0.008 (ug/ml), Ref: 17261623
MIC50: 0.12 (ug/ml), Ref: 17242152
MIC90: 0.12 (ug/ml), Ref: 17242152
MIC50: 0.008 (ug/ml), Ref: 20625152
MIC90: 0.008 (ug/ml), Ref: 20625152
MIC: 0.008 (ug/ml), Ref: 20625152
MIC: 0.004 (ug/ml), Ref: 19506065
MIC50: 0.008 (ug/ml), Ref: 19506065
MIC90: 0.015 (ug/ml), Ref: 19506065
MIC90: 0.008 (ug/ml), Ref: 23092194
TCMC1475
TCMT1342 Streptococcus salivarius Streptococcus salivarius MIC50: 1 (ug/ml), Ref: 17261623
MIC90: 1 (ug/ml), Ref: 17261623
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1440 Actinomyces sp. Actinomyces sp. MIC: 0.25 (ug/ml), Ref: 17261623
TCMC1475
TCMT1219 Enterococcus Enterococcus MIC: 16 (ug/ml), Ref: 17220419
TCMC1475
TCMT1305 Salmonella enteritidis Salmonella enterica subsp. enterica serovar Enteritidis MIC50: 0.03 (ug/ml), Ref: 17261623
MIC90: 0.06 (ug/ml), Ref: 17261623
TCMC1475
TCMT1274 Shigella boydii Shigella boydii MIC: 0.098 (ug/ml), Ref: 17826097
TCMC1475
TCMT1196 Salmonella Salmonella MIC: 0.098 (ug/ml), Ref: 17826097
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.06 (ug/ml), Ref: 18591277
TCMC1475
TCMT1406 Mycobacterium leprae Mycobacterium leprae IC50: 7 (ug/ml), Ref: 17325221
TCMC1475
TCMT1404 Streptococcus intermedius Streptococcus intermedius MIC: 0.5 (ug/ml), Ref: 18330977
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.12 (ug/ml), Ref: 18443122
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1395 Staphylococcus sp. Staphylococcus sp. MIC50: 4 (ug/ml), Ref: 17420210
MIC90: 32 (ug/ml), Ref: 17420210
MIC50: 0.25 (ug/ml), Ref: 17420210
MIC90: 0.25 (ug/ml), Ref: 17420210
MIC90: 1 (ug/ml), Ref: 20231392
MIC90: 0.5 (ug/ml), Ref: 20231392
MIC50: 1 (ug/ml), Ref: 20231392
MIC50: 0.25 (ug/ml), Ref: 20231392
MIC50: 8 (ug/ml), Ref: 20231392
MIC50: 0.5 (ug/ml), Ref: 20231392
MIC: 0.06 (ug/ml), Ref: 20231392
MIC: 0.25 (ug/ml), Ref: 20231392
TCMC1475
TCMT1199 Streptococcus sp. 'group A' Streptococcus sp. 'group A' MIC: 0.12 (ug/ml), Ref: 17606689
MIC50: 0.5 (ug/ml), Ref: 17606689
MIC90: 0.5 (ug/ml), Ref: 17606689
MIC50: 0.5 (ug/ml), Ref: 18362189
MIC90: 1 (ug/ml), Ref: 18362189
MIC90: 2 (ug/ml), Ref: 18362189
MIC: 0.25 (ug/ml), Ref: 18362189
MIC: 0.5 (ug/ml), Ref: 18362189
MIC: 0.25 (ug/ml), Ref: 19289528
MIC90: 1 (ug/ml), Ref: 19289528
MIC50: 0.5 (ug/ml), Ref: 19289528
TCMC1475
TCMT1341 Streptococcus oralis Streptococcus oralis MIC: 1 (ug/ml), Ref: 17548487
MIC: 2 (ug/ml), Ref: 17548487
MIC: 32 (ug/ml), Ref: 17548487
MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.12 (ug/ml), Ref: 18443122
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 0.5 (ug/ml), Ref: 17682103
MIC: 0.06 (ug/ml), Ref: 17682103
MIC: 0.5 (ug/ml), Ref: 18519723
MIC: 0.5 (ug/ml), Ref: 19364849
MIC: 2 (ug/ml), Ref: 20696867
MIC: 0.5 (ug/ml), Ref: 20696867
MIC: 1 (ug/ml), Ref: 20696867
MIC: 0.25 (ug/ml), Ref: 20696867
MIC: 0.39 (ug/ml), Ref: 23409972
TCMC1475
TCMT1460 Mycobacterium intracellulare Mycobacterium intracellulare MIC: 4 (ug/ml), Ref: 17709469
MIC50: 8 (ug/ml), Ref: 20368403
MIC90: 32 (ug/ml), Ref: 20368403
MIC: 2 (ug/ml), Ref: 20368403
TCMC1475
TCMT1328 Enterococcus avium Enterococcus avium MIC: 8 (ug/ml), Ref: 18056272
MIC50: 2 (ug/ml), Ref: 19001109
MIC90: 2 (ug/ml), Ref: 19001109
TCMC1475
TCMT1201 Staphylococcus epidermidis ATCC 12228 Staphylococcus epidermidis ATCC 12228 MIC: 0.5 (ug/ml), Ref: 19481308
MIC: 0.15 (ug/ml), Ref: 20667744
MIC: 0.39 (ug/ml), Ref: 10.1007/s00044-013-0581-9
MIC: 0.125 (ug/ml), Ref: 26238324
MIC: 0.25 (ug/ml), Ref: 26317881
TCMC1475
TCMT1193 Staphylococcus Staphylococcus MIC50: 0.5 (ug/ml), Ref: 20065058
MIC90: 8 (ug/ml), Ref: 20065058
MIC: 0.12 (ug/ml), Ref: 20065058
MIC: 0.125 (ug/ml), Ref: 18316525
MIC: 0.025 (ug/ml), Ref: 18316525
MIC: 4 (ug/ml), Ref: 18316525
MIC: 0.06 (ug/ml), Ref: 18426902
MIC50: 0.25 (ug/ml), Ref: 18426902
MIC90: 32 (ug/ml), Ref: 18426902
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 0.25 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 19114671
MIC: 0.06 (ug/ml), Ref: 19114671
MIC50: 8 (ug/ml), Ref: 19114671
MIC50: 0.25 (ug/ml), Ref: 19114671
MIC90: 16 (ug/ml), Ref: 19114671
MIC: 0.5 (ug/ml), Ref: 19124664
MIC50: 4 (ug/ml), Ref: 19124664
MIC90: 4 (ug/ml), Ref: 19124664
MIC50: 0.5 (ug/ml), Ref: 19124664
TCMC1475
TCMT1355 Rhodococcus equi Rhodococcus equi MIC50: 1 (ug/ml), Ref: 18227183
MIC90: 2 (ug/ml), Ref: 18227183
MIC: 0.125 (ug/ml), Ref: 18227183
TCMC1475
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC90: 4 (ug/ml), Ref: 18227183
MIC: 0.06 (ug/ml), Ref: 18227183
MIC50: 0.25 (ug/ml), Ref: 18227183
TCMC1475
TCMT1280 Salmonella sp. Salmonella sp. MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC: 0.03 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.06 (ug/ml), Ref: 19114671
TCMC1475
TCMT1197 Shigella sp. Shigella sp. MIC: 0.008 (ug/ml), Ref: 18426902
MIC50: 0.06 (ug/ml), Ref: 18426902
MIC90: 8 (ug/ml), Ref: 18426902
MIC: 0.015 (ug/ml), Ref: 19114671
MIC50: 0.03 (ug/ml), Ref: 19114671
MIC90: 0.06 (ug/ml), Ref: 19114671
TCMC1475
TCMT1441 Streptococcus dysgalactiae subsp. equisimilis Streptococcus dysgalactiae subsp. equisimilis MIC: 12 (ug/ml), Ref: 20145082
MIC: 8 (ug/ml), Ref: 20145082
MIC: 4 (ug/ml), Ref: 20145082
MIC: 3 (ug/ml), Ref: 20145082
MIC: 1.5 (ug/ml), Ref: 20145082
MIC: 2 (ug/ml), Ref: 20145082
MIC: 1 (ug/ml), Ref: 20145082
MIC: 0.75 (ug/ml), Ref: 20145082
MIC: 0.19 (ug/ml), Ref: 20145082
MIC: 0.5 (ug/ml), Ref: 20145082
MIC: 0.38 (ug/ml), Ref: 20145082
TCMC1475
TCMT1315 Streptococcus sp. Streptococcus sp. MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 0.5 (ug/ml), Ref: 18443115
MIC: 0.12 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19506065
TCMC1475
TCMT1403 Streptococcus constellatus Streptococcus constellatus MIC50: 0.5 (ug/ml), Ref: 18443115
MIC90: 1 (ug/ml), Ref: 18443115
MIC: 0.25 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 18443122
MIC90: 1 (ug/ml), Ref: 18591277
MIC50: 0.25 (ug/ml), Ref: 18591277
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC90: 4 (ug/ml), Ref: 19506065
TCMC1475
TCMT1220 Streptococcus pneumoniae R6 Streptococcus pneumoniae R6 MIC: 0.25 (ug/ml), Ref: 18160515
MIC: 2 (ug/ml), Ref: 18725440
MIC: 1 (ug/ml), Ref: 18725440
MIC: 16 (ug/ml), Ref: 18725440
TCMC1475
TCMT1398 Corynebacterium amycolatum Corynebacterium amycolatum MIC: 0.06 (ug/ml), Ref: 18227183
TCMC1475
TCMT1320 Corynebacterium minutissimum Corynebacterium minutissimum MIC: 0.03 (ug/ml), Ref: 18227183
MIC50: 0.06 (ug/ml), Ref: 18227183
TCMC1475
TCMT1379 Corynebacterium striatum Corynebacterium striatum MIC: 0.03 (ug/ml), Ref: 18227183
TCMC1475
TCMT1419 Corynebacterium urealyticum Corynebacterium urealyticum MIC: 0.03 (ug/ml), Ref: 18227183
TCMC1475
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 0.125 (ug/ml), Ref: 18227183
MIC50: 32 (ug/ml), Ref: 18227183
TCMC1475
TCMT1266 Mycobacterium abscessus Mycobacterium abscessus MIC: 16 (ug/ml), Ref: 20368403
MIC50: 64 (ug/ml), Ref: 20368403
MIC50: 16 (ug/ml), Ref: 18725441
MIC90: 32 (ug/ml), Ref: 18725441
TCMC1475
TCMT1418 Enterobacteriaceae Enterobacteriaceae MIC90: 64 (ug/ml), Ref: 20211892
MIC50: 16 (ug/ml), Ref: 20211892
MIC90: 32 (ug/ml), Ref: 20211892
MIC50: 8 (ug/ml), Ref: 20211892
MIC90: 8 (ug/ml), Ref: 20211892
MIC50: 0.03 (ug/ml), Ref: 20211892
MIC50: 0.06 (ug/ml), Ref: 18625769
MIC50: 8 (ug/ml), Ref: 18625769
MIC90: 4 (ug/ml), Ref: 18625769
MIC90: 0.06 (ug/ml), Ref: 19738018
TCMC1475
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50: 0.5 (ug/ml), Ref: 20368403
MIC50: 8 (ug/ml), Ref: 20368403
MIC90: 0.5 (ug/ml), Ref: 20368403
MIC90: 16 (ug/ml), Ref: 20368403
MIC: 0.25 (ug/ml), Ref: 20368403
MIC: 2 (ug/ml), Ref: 20368403
MIC: 0.5 (ug/ml), Ref: 18070980
MIC90: 1 (ug/ml), Ref: 10.1007/s00044-012-0101-3
MIC: 0.125 (ug/ml), Ref: 25218911
TCMC1475
TCMT1237 Mycobacterium kansasii Mycobacterium kansasii MIC50: 0.25 (ug/ml), Ref: 20368403
MIC90: 1 (ug/ml), Ref: 20368403
MIC: 0.25 (ug/ml), Ref: 20368403
TCMC1475
TCMT1184 Mycobacterium fortuitum Mycobacterium fortuitum MIC50: 0.25 (ug/ml), Ref: 20368403
MIC90: 0.5 (ug/ml), Ref: 20368403
MIC: 0.06 (ug/ml), Ref: 20368403
MIC50: 0.06 (ug/ml), Ref: 18725441
MIC90: 0.25 (ug/ml), Ref: 18725441
TCMC1475
TCMT1267 Mycobacterium chelonae Mycobacterium chelonae MIC50: 32 (ug/ml), Ref: 20368403
MIC90: 64 (ug/ml), Ref: 20368403
MIC: 4 (ug/ml), Ref: 20368403
MIC50: 0.5 (ug/ml), Ref: 18725441
MIC90: 8 (ug/ml), Ref: 18725441
TCMC1475
TCMT1202 Mycoplasma hominis Mycoplasma hominis MIC: 0.125 (ug/ml), Ref: 18663020
MIC50: 0.25 (ug/ml), Ref: 18663020
MIC90: 0.5 (ug/ml), Ref: 18663020
MIC: 0.125 (ug/ml), Ref: 19258276
MIC50: 0.25 (ug/ml), Ref: 19258276
MIC90: 0.5 (ug/ml), Ref: 19258276
MIC: 0.1 (ug/ml), Ref: 19738013
MIC50: 0.25 (ug/ml), Ref: 19738013
MIC90: 0.5 (ug/ml), Ref: 19738013
TCMC1475
TCMT1273 Pseudomonas putida Pseudomonas putida MIC: 0.25 (ug/ml), Ref: 18809945
TCMC1475
TCMT1172 Staphylococcus aureus subsp. aureus RN4220 Staphylococcus aureus subsp. aureus RN4220 MIC: 0.125 (ug/ml), Ref: 18838584
TCMC1475
TCMT1400 Mycobacterium mageritense Mycobacterium mageritense MIC: 0.03 (ug/ml), Ref: 18725441
TCMC1475
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 0.03 (ug/ml), Ref: 18725441
MIC99: 0.58 (nM), Ref: 10.1039/C3MD00387F
TCMC1475
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 19651906
MIC50: 0.25 (ug/ml), Ref: 19651906
MIC90: 4 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 4 (ug/ml), Ref: 19651906
MBC90: 16 (ug/ml), Ref: 19651906
MIC50: 8 (ug/ml), Ref: 19506065
MIC90: 0.5 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 4 (ug/ml), Ref: 19651906
TCMC1475
TCMT1377 Staphylococcus lugdunensis Staphylococcus lugdunensis MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.25 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 19506065
MIC50: 0.25 (ug/ml), Ref: 19506065
TCMC1475
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
MIC: 0.25 (ug/ml), Ref: 19651906
MIC50: 0.25 (ug/ml), Ref: 19651906
MIC90: 4 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 4 (ug/ml), Ref: 19651906
MBC90: 16 (ug/ml), Ref: 19651906
MIC90: 0.5 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 4 (ug/ml), Ref: 19651906
TCMC1475
TCMT1402 Staphylococcus cohnii Staphylococcus cohnii MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
TCMC1475
TCMT1304 Staphylococcus capitis Staphylococcus capitis MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC50: 0.12 (ug/ml), Ref: 18591277
TCMC1475
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC50: 4 (ug/ml), Ref: 18591277
MIC90: 8 (ug/ml), Ref: 18591277
MIC: 0.06 (ug/ml), Ref: 18591277
TCMC1475
TCMT1303 Bacillus Bacillus MIC: 0.06 (ug/ml), Ref: 18591277
MIC90: 4 (ug/ml), Ref: 18591277
MIC50: 0.5 (ug/ml), Ref: 18591277
TCMC1475
TCMT1376 Staphylococcus intermedius Staphylococcus intermedius MIC: 0.03 (ug/ml), Ref: 18591277
MIC90: 0.12 (ug/ml), Ref: 18591277
MIC50: 0.03 (ug/ml), Ref: 18591277
TCMC1475
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 50 (ug/ml), Ref: 18838592
MIC: 10 (ug/ml), Ref: 18838592
MIC: 2 (ug/ml), Ref: 18838592
MIC: 30 (ug/ml), Ref: 18838592
MIC: 20 (ug/ml), Ref: 18838592
MIC: 8 (ug/ml), Ref: 18838592
MIC: 0.034 (ug/ml), Ref: 18838592
MIC: 0.168 (ug/ml), Ref: 18838592
MIC: 0.016 (ug/ml), Ref: 18838592
MIC: 0.25 (ug/ml), Ref: 20231393
MIC: 1 (ug/ml), Ref: 18936189
MIC: 0.06 (ug/ml), Ref: 18936189
MIC: 0.2 (ug/ml), Ref: 20855738
TCMC1475
TCMT1291 Haemophilus parainfluenzae Haemophilus parainfluenzae MIC90: 0.06 (ug/ml), Ref: 19001109
MIC50: 0.015 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19001109
TCMC1475
TCMT1378 Acinetobacter haemolyticus Acinetobacter haemolyticus MIC90: 2 (ug/ml), Ref: 19001109
MIC50: 0.12 (ug/ml), Ref: 19001109
MIC: 0.03 (ug/ml), Ref: 19001109
TCMC1475
TCMT1290 Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC90: 16 (ug/ml), Ref: 19001109
MIC50: 8 (ug/ml), Ref: 19001109
MIC: 0.06 (ug/ml), Ref: 19001109
MIC: 0.015 (ug/ml), Ref: 19506065
MIC50: 0.5 (ug/ml), Ref: 19506065
MIC90: 8 (ug/ml), Ref: 19506065
MIC: 0.25 (ug/ml), Ref: 21515052
MIC: 0.5 (ug/ml), Ref: 26317881
MIC: 0.12 (ug/ml), Ref: 26363871
TCMC1475
TCMT1312 Enterococcus durans Enterococcus durans MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
TCMC1475
TCMT1310 Enterococcus hirae Enterococcus hirae MIC90: 8 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
MBC: 1.9 (nM), Ref: 22036229
TCMC1475
TCMT1227 Streptococcus Streptococcus MIC90: 1 (ug/ml), Ref: 19124664
MIC50: 0.5 (ug/ml), Ref: 19124664
MIC: 0.5 (ug/ml), Ref: 19124664
MIC50: 1 (ug/ml), Ref: 19124664
MIC90: 2 (ug/ml), Ref: 19124664
MIC: 0.03 (ug/ml), Ref: 19738026
MIC: 0.25 (ug/ml), Ref: 19738026
MIC90: 0.5 (ug/ml), Ref: 19738026
TCMC1475
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 4 (ug/ml), Ref: 19380599
MIC: 2 (ug/ml), Ref: 19380599
MIC: 0.12 (ug/ml), Ref: 19380599
MIC50: 8 (ug/ml), Ref: 19380599
MIC50: 4 (ug/ml), Ref: 19380599
MIC50: 0.25 (ug/ml), Ref: 19380599
MIC90: 16 (ug/ml), Ref: 19380599
MIC90: 8 (ug/ml), Ref: 19380599
MIC90: 0.25 (ug/ml), Ref: 19380599
MIC90: 1 (ug/ml), Ref: 24775303
TCMC1475
TCMT1362 Bordetella pertussis Bordetella pertussis MIC: 0.016 (ug/ml), Ref: 19414571
MIC: 0.008 (ug/ml), Ref: 19414571
MIC: 0.004 (ug/ml), Ref: 19414571
MIC: 0.064 (ug/ml), Ref: 19414571
TCMC1475
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 0.25 (ug/ml), Ref: 19651906
MIC50: 0.25 (ug/ml), Ref: 19651906
MIC90: 4 (ug/ml), Ref: 19651906
MBC: 0.5 (ug/ml), Ref: 19651906
MBC50: 4 (ug/ml), Ref: 19651906
MBC90: 16 (ug/ml), Ref: 19651906
MIC90: 0.5 (ug/ml), Ref: 19651906
MBC50: 1 (ug/ml), Ref: 19651906
MBC90: 4 (ug/ml), Ref: 19651906
TCMC1475
TCMT1334 Chlamydia trachomatis Chlamydia trachomatis MIC: 0.5 (ug/ml), Ref: 20855744
MIC: 0.25 (ug/ml), Ref: 20855744
MBC: 0.5 (ug/ml), Ref: 20855744
MBC: 0.25 (ug/ml), Ref: 20855744
TCMC1475
TCMT1357 Bacteroides uniformis Bacteroides uniformis MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 8 (ug/ml), Ref: 18625771
TCMC1475
TCMT1359 Bacteroides caccae Bacteroides caccae MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 8 (ug/ml), Ref: 18625771
TCMC1475
TCMT1368 Fusobacterium varium Fusobacterium varium MIC: 0.12 (ug/ml), Ref: 18625771
MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1367 Fusobacterium mortiferum Fusobacterium mortiferum MIC: 0.12 (ug/ml), Ref: 18625771
MIC50: 2 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1371 Veillonella parvula Veillonella parvula MIC: 0.06 (ug/ml), Ref: 18625771
TCMC1475
TCMT1372 Clostridium paraputrificum Clostridium paraputrificum MIC: 0.25 (ug/ml), Ref: 18625771
MIC50: 0.5 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1373 Clostridium septicum Clostridium septicum MIC: 0.25 (ug/ml), Ref: 18625771
MIC50: 0.5 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1374 Clostridium tertium Clostridium tertium MIC: 0.25 (ug/ml), Ref: 18625771
MIC50: 0.5 (ug/ml), Ref: 18625771
MIC90: 4 (ug/ml), Ref: 18625771
TCMC1475
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 0.03 (ug/ml), Ref: 21458275
TCMC1475
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 0.5 (ug/ml), Ref: 21510638
MIC: 0.5 (ug/ml), Ref: 22939698
MIC: 0.25 (ug/ml), Ref: 25218911
MIC: 0.25 (ug/ml), Ref: 27020299
MIC99: 0.78 (nM), Ref: 10.1039/C4MD00303A
TCMC1475
TCMT1411 Vibrio parahaemolyticus Vibrio parahaemolyticus MIC: 0.156 (ug/ml), Ref: 21744790
TCMC1475
TCMT1229 Enterococcus faecalis Enterococcus faecalis ATCC 29212 MIC: 0.25 (ug/ml), Ref: 7707323
MIC: 0.78 (ug/ml), Ref: 15380226
MIC: 1 (ug/ml), Ref: 16078842
MIC: 1 (ug/ml), Ref: 17064062
MIC: 32 (ug/ml), Ref: 17064062
MIC50: 16 (ug/ml), Ref: 17261623
MIC90: 32 (ug/ml), Ref: 17261623
MIC: 16 (ug/ml), Ref: 17261623
MIC: 0.5 (ug/ml), Ref: 17261623
MIC: 1 (ug/ml), Ref: 17261623
MIC50: 16 (ug/ml), Ref: 17242152
MIC: 1 (ug/ml), Ref: 17316916
MIC: 2 (ug/ml), Ref: 17157008
MIC: 0.5 (ug/ml), Ref: 18330977
MIC: 1 (ug/ml), Ref: 18457383
MIC: 64 (ug/ml), Ref: 18457383
MIC: 32 (ug/ml), Ref: 18457383
MIC: 8 (ug/ml), Ref: 18056272
MIC: 1 (ug/ml), Ref: 19481308
MIC: 0.5 (ug/ml), Ref: 20667731
MIC: 32 (ug/ml), Ref: 20591538
MIC: 0.5 (ug/ml), Ref: 20591538
MIC50: 2 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 20065058
MIC: 1 (ug/ml), Ref: 18316525
MIC: 2 (ug/ml), Ref: 18316525
MIC: 32 (ug/ml), Ref: 18316525
MIC: 0.5 (ug/ml), Ref: 18316525
MIC50: 1 (ug/ml), Ref: 20231392
MIC90: 2 (ug/ml), Ref: 18591277
MIC50: 1 (ug/ml), Ref: 18591277
MIC: 0.25 (ug/ml), Ref: 18591277
MIC: 8 (ug/ml), Ref: 20833454
MIC: 4 (ug/ml), Ref: 20833454
MIC50: 2 (ug/ml), Ref: 19001109
MIC50: 1 (ug/ml), Ref: 19001109
MIC: 0.5 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19114671
MIC50: 1 (ug/ml), Ref: 19114671
MIC90: 32 (ug/ml), Ref: 19114671
MIC: 1 (ug/ml), Ref: 19188391
MIC50: 1 (ug/ml), Ref: 19289528
MIC90: 64 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 19506065
MIC: 0.12 (ug/ml), Ref: 19506065
MIC50: 1 (ug/ml), Ref: 18625769
MIC: 16 (ug/ml), Ref: 19581455
MIC: 0.25 (ug/ml), Ref: 21515052
MIC: 2 (ug/ml), Ref: 21515052
MIC: 8 (ug/ml), Ref: 21481984
MIC: 0.5 (ug/ml), Ref: 21510638
MIC: 8 (ug/ml), Ref: 21764484
MIC: 8 (ug/ml), Ref: 22841282
MIC: 64 (ug/ml), Ref: 22841282
MIC: 16 (ug/ml), Ref: 22841282
MIC: 0.5 (ug/ml), Ref: 22939698
MIC: 32 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-010-9338-x
MIC: 0.78 (ug/ml), Ref: 23409972
MIC90: 32 (ug/ml), Ref: 24959892
MIC90: 64 (ug/ml), Ref: 24959892
MIC: 0.5 (ug/ml), Ref: 26317881
MIC: 1 (ug/ml), Ref: 26476970
MIC: 1 (ug/ml), Ref: 26435513
MIC: 16 (ug/ml), Ref: 27020299
MIC: 32 (ug/ml), Ref: 27020299
MIC: 64 (ug/ml), Ref: 27020299
MIC: 2 (ug/ml), Ref: 27293070
MIC: 4 (ug/ml), Ref: 27293070
TCMC1475
TCMT1399 Chlamydophila pneumoniae Chlamydophila pneumoniae MIC: 0.5 (ug/ml), Ref: 23409972
TCMC1475
TCMT1287 Bacillus subtilis subsp. spizizenii ATCC 6633 Bacillus subtilis subsp. spizizenii ATCC 6633 MIC: 3.12 (ug/ml), Ref: 24852274
TCMC1475
TCMT1426 Enterococcus sp. Enterococcus sp. MIC: 0.78 (ug/ml), Ref: 24852274
TCMC1475
TCMT1187 Enterococcus faecalis ATCC 29212 Enterococcus faecalis ATCC 29212 MIC: 0.5 (ug/ml), Ref: 26317881
TCMC1542
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 5 (ug/ml), Ref: 17888665
TCMC1542
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 15.6 (ug/ml), Ref: 24913712
TCMC1542
TCMT1251 Candida albicans Candida albicans MIC: 15.6 (ug/ml), Ref: 24913712
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC784
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2100
TCMT1251 Candida albicans Candida albicans MIC: 6 (ug/ml), Ref: 18778047
TCMC2100
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 18778047
MIC: 4 (ug/ml), Ref: 18778047
TCMC2100
TCMT1246 Escherichia coli Escherichia coli MIC: 42 (ug/ml), Ref: 18778047
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC1012
TCMT1246 Escherichia coli Escherichia coli MIC: 0.25 (ug/ml), Ref: 19770280
MIC: 5 (ug/ml), Ref: 19770280
TCMC1850
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 24360560
TCMC1850
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.78 (ug/ml), Ref: 24360560
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1059
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 0.3 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC1059
TCMT1251 Candida albicans Candida albicans MIC: 0.4 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC1059
TCMT1246 Escherichia coli Escherichia coli MIC: 0.3 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC1059
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 0.4 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC1059
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.3 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC1059
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-007-9047-2
TCMC634
TCMT1158 Human immunodeficiency virus type 1 protease Human immunodeficiency virus 1 Kd: 1.13 (nM), Ref: 12459011
Ki: 0.23 (nM), Ref: 12459011
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC812
TCMT1095 Streptavidin Streptomyces avidinii Kd: 1.00E-05 (nM), Ref: 24913411
TCMC883
TCMT1088 Carbonic anhydrase Helicobacter pylori Ki: 21 (nM), Ref: 19450983
TCMC2033
TCMT1159 Met repressor Escherichia coli Kd: 4 (nM), Ref: 22137339
TCMC2174
TCMT1088 Carbonic anhydrase Helicobacter pylori Ki: 10 (nM), Ref: 19450983
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1824
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.09 (nM), Ref: 19734910
IC50: 0.15 (nM), Ref: 19734910
IC50: 1.78 (nM), Ref: 19734910
IC50: 0.07 (nM), Ref: 19734910
IC50: 79.43 (nM), Ref: 19734910
IC50: 63.1 (nM), Ref: 19734910
TCMC1824
TCMT1316 Leishmania sp. Leishmania sp. IC50: 35 (nM), Ref: 18070965
TCMC1836
TCMT1168 Trichomonas vaginalis Trichomonas vaginalis IC50: 75.6 (nM), Ref: 22047694
TCMC1836
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 2.6 (nM), Ref: 22047694
TCMC2184
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 15.4 (nM), Ref: 17503850
TCMC1762
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC99: 0.0042 (nM), Ref: 24894561
MIC99: 0.5 (nM), Ref: 24894561
TCMC1475
TCMT1174 Mycobacterium bovis BCG Mycobacterium bovis BCG MIC99: 0.39 (nM), Ref: 10.1039/C4MD00303A