References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC948
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
TCMC948
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
TCMC948
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
TCMC948
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
TCMC948
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
TCMC948
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
TCMC948
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
TCMC948
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
TCMC948
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
TCMC948
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
TCMC948
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
TCMC948
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
TCMC1871
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
TCMC1871
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
TCMC1871
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
TCMC1871
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
TCMC1871
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
TCMC1429
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
TCMC1429
|
TCMT65 |
Estradiol 17-beta-dehydrogenase 1 |
Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
TCMC1429
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
TCMC1429
|
TCMT187 |
Androgen Receptor |
Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
TCMC1429
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
TCMC1429
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
TCMC1429
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
TCMC1429
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
TCMC1429
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
TCMC1429
|
TCMT591 |
Estrogen-related receptor alpha |
Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
TCMC1429
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
TCMC1429
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
TCMC1429
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
TCMC1429
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
TCMC1429
|
TCMT159 |
Tyrosinase |
Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
TCMC1985
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 6367.7 (nM), Ref: 26498393 |
TCMC1985
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 67.3 (nM), Ref: 26498393 |
TCMC1985
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 3.9 (nM), Ref: 26498393 |
TCMC1985
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 43.5 (nM), Ref: 26498393 |
TCMC737
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 168 (nM), Ref: 26498393 |
TCMC737
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 5591.2 (nM), Ref: 26498393 |
TCMC737
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 423.7 (nM), Ref: 26498393 |
TCMC737
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4.9 (nM), Ref: 26498393 |
TCMC1430
|
TCMT131 |
Acetylcholinesterase |
Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1986
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 150 (nM), Ref: 18165015 IC50: 2000 (nM), Ref: 22261024 |
TCMC1102
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
TCMC1102
|
TCMT752 |
Casein kinase II alpha |
Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
TCMC1102
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
TCMC1102
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
TCMC1102
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC1102
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
TCMC1102
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
TCMC1102
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
TCMC1102
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
TCMC1102
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
TCMC1102
|
TCMT753 |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
IC50: 142 (nM), Ref: |
TCMC1102
|
TCMT721 |
Heat shock 70 kDa protein 1 |
Homo sapiens |
IC50: 760 (nM), Ref: |
TCMC1102
|
TCMT189 |
Dual specificity protein phosphatase 3 |
Homo sapiens |
IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
TCMC1102
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
TCMC1102
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
TCMC1102
|
TCMT354 |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
TCMC1102
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
TCMC1102
|
TCMT626 |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
TCMC1102
|
TCMT423 |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
TCMC1102
|
TCMT418 |
Ephrin type-B receptor 4 |
Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
TCMC1102
|
TCMT704 |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
TCMC1102
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
TCMC1102
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
TCMC1102
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
TCMC1102
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
TCMC1102
|
TCMT457 |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
TCMC1102
|
TCMT377 |
Insulin receptor |
Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
TCMC1102
|
TCMT536 |
Platelet-derived growth factor receptor beta |
Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
TCMC1102
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT755 |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
TCMC1102
|
TCMT502 |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
TCMC1102
|
TCMT756 |
Mitogen-activated protein kinase kinase kinase 8 |
Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
TCMC1102
|
TCMT739 |
G-protein coupled receptor 35 |
Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
TCMC1102
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
TCMC1102
|
TCMT225 |
Carbonic anhydrase XIII |
Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
TCMC1102
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
TCMC1409
|
TCMT22 |
Intestinal alkaline phosphatase |
Homo sapiens |
IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
TCMC1409
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
TCMC1409
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
TCMC1409
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
TCMC1409
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
TCMC1409
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
TCMC1982
|
TCMT239 |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
TCMC1982
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
TCMC1982
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
TCMC1982
|
TCMT44 |
Glyoxalase I |
Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
TCMC1982
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
TCMC1982
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
TCMC1982
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
TCMC1982
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
TCMC1982
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
TCMC1982
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
TCMC1982
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
TCMC1982
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
TCMC1982
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
TCMC1982
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
TCMC1982
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
TCMC1982
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
TCMC1982
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
TCMC1982
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
TCMC1982
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
TCMC1982
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
TCMC1982
|
TCMT320 |
Matrix metalloproteinase 3 |
Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
TCMC1982
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
TCMC1982
|
TCMT322 |
Matrix metalloproteinase 13 |
Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
TCMC1982
|
TCMT422 |
CaM kinase II beta |
Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
TCMC1982
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1982
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
TCMC1982
|
TCMT784 |
Vasopressin V2 receptor |
Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
TCMC1982
|
TCMT785 |
Interleukin-8 receptor A |
Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
TCMC1982
|
TCMT786 |
C-C chemokine receptor type 4 |
Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
TCMC1982
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
TCMC1982
|
TCMT601 |
Thrombin |
Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
TCMC1982
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
TCMC1982
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
TCMC1982
|
TCMT791 |
Protein kinase N1 |
Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
TCMC1982
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
TCMC1982
|
TCMT462 |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
TCMC1982
|
TCMT445 |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
TCMC1982
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
TCMC1982
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
TCMC1982
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
TCMC1982
|
TCMT388 |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
TCMC1982
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
TCMC1982
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
TCMC1982
|
TCMT402 |
ALK tyrosine kinase receptor |
Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
TCMC1982
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
TCMC1982
|
TCMT592 |
Xanthine dehydrogenase |
Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
TCMC1982
|
TCMT793 |
Liver glycogen phosphorylase |
Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
TCMC1982
|
TCMT33 |
Cytochrome P450 3A4 |
Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
TCMC1982
|
TCMT217 |
Cytochrome P450 2C8 |
Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
TCMC1982
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
TCMC880
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 9910 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 20185318 Ki: 9900 (nM), Ref: 22245047 Ki: 9900 (nM), Ref: 26073005 Ki: 9900 (nM), Ref: 26520662 |
TCMC880
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 4200 (nM), Ref: 18579385 Ki: 4200 (nM), Ref: 20185318 |
TCMC880
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8900 (nM), Ref: 18579385 Ki: 8900 (nM), Ref: 20185318 |
TCMC1202
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
TCMC1202
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1202
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
TCMC1202
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
TCMC1202
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
TCMC1202
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
TCMC1202
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1202
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
TCMC1202
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
TCMC1202
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
TCMC1202
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
TCMC1202
|
TCMT822 |
Alpha-(1,3)-fucosyltransferase 7 |
Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
TCMC1839
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
TCMC1839
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
TCMC1839
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
TCMC1839
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
TCMC1839
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
TCMC1839
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1839
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
TCMC1839
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
TCMC1839
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1839
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
TCMC1839
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
TCMC2002
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 7700 (nM), Ref: 18501600 Ki: 7700 (nM), Ref: 18579385 Ki: 7700 (nM), Ref: 26073005 |
TCMC2002
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 7500 (nM), Ref: 18579385 |
TCMC2002
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7100 (nM), Ref: 18579385 |
TCMC2002
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 8700 (nM), Ref: 18579385 |
TCMC1356
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 3000 (nM), Ref: 22261024 |
TCMC847
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
TCMC847
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
TCMC847
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
TCMC847
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
TCMC847
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
TCMC847
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC847
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
TCMC847
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
TCMC847
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
TCMC847
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
TCMC847
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
TCMC847
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
TCMC847
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
TCMC847
|
TCMT295 |
Matrix metalloproteinase-1 |
Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
TCMC847
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
TCMC897
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
TCMC897
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |