Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 810 (nM), Ref: 20100662 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 5930 (nM), Ref: 19846303 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 630 (nM), Ref: 21561086 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 1720 (nM), Ref: 8576921 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1118 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 95 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 20 (nM), Ref: 20696580 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 5900 (nM), Ref: 21561086 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 1900 (nM), Ref: 20100662 |
|
TCMT102 | Low molecular weight phosphotyrosine protein phosphatase | Homo sapiens |
IC50: 7200 (nM), Ref: 21453996 |
|
TCMT103 | Receptor-type tyrosine-protein phosphatase F (LAR) | Homo sapiens |
IC50: 3800 (nM), Ref: 21453996 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 2400 (nM), Ref: 23387824 |
|
TCMT150 | Nuclear receptor ROR-gamma | Homo sapiens |
IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616 |
|
TCMT632 | Purine nucleoside phosphorylase | Homo sapiens |
Ki: 5000 (nM), Ref: 31484 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 7400 (nM), Ref: 22940448 |