Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT277 | Solute carrier organic anion transporter family member 1B3 | Homo sapiens |
Ki: 1430 (nM), Ref: 23396419 Ki: 4550 (nM), Ref: 23396419 Ki: 8290 (nM), Ref: 23396419 Ki: 1030 (nM), Ref: 23396419 |
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TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5900 (nM), Ref: 19592245 IC50: 5900 (nM), Ref: 19592245 |
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TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 8 (nM), Ref: 20413308 IC50: 10000 (nM), Ref: 24345481 IC50: 8000 (nM), Ref: 26301554 |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1890 (nM), Ref: 22487176 Ki: 1880 (nM), Ref: 22487176 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8710 (nM), Ref: 22487176 Ki: 8800 (nM), Ref: 22487176 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4130 (nM), Ref: 22487176 Ki: 4220 (nM), Ref: 22487176 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7220 (nM), Ref: 22487176 Ki: 7330 (nM), Ref: 22487176 |
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TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 1380.38 (nM), Ref: 23574272 IC50: 1400 (nM), Ref: 23574272 |
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TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 147.91 (nM), Ref: 23574272 IC50: 140 (nM), Ref: 23574272 |
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TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 323.59 (nM), Ref: 23574272 IC50: 320 (nM), Ref: 23574272 IC50: 323.59 (nM), Ref: 24116873 IC50: 330 (nM), Ref: 24116873 |
Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT1181 | Mycobacterium tuberculosis H37Ra | Mycobacterium tuberculosis H37Ra |
MIC: 50 (ug/ml), Ref: 20691508 |
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TCMT1251 | Candida albicans | Candida albicans |
MIC: 1.56 (ug/ml), Ref: 3373231 MIC: 3.12 (ug/ml), Ref: 3373231 MIC: 6.25 (ug/ml), Ref: 3373231 MIC: 2 (ug/ml), Ref: 15921418 |
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TCMT1458 | Filobasidiella neoformans | Cryptococcus neoformans |
MIC: 25 (ug/ml), Ref: 3373231 MIC: 1 (ug/ml), Ref: 15921418 |
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TCMT1243 | Aspergillus flavus | Aspergillus flavus |
MIC: 100 (ug/ml), Ref: 3373231 |
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TCMT1176 | Streptococcus pneumoniae | Streptococcus pneumoniae |
MIC: 32 (ug/ml), Ref: 15921418 |
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TCMT1218 | Staphylococcus aureus | Staphylococcus aureus |
MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4 |
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TCMT1251 | Candida albicans | Candida albicans |
IC50: 2.82 (ug/ml), Ref: 11958988 |
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TCMT1455 | Mycobacterium tuberculosis H37Rv | Mycobacterium tuberculosis H37Rv |
MIC: 8 (ug/ml), Ref: 24641242 |
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TCMT1438 | Plasmodium falciparum | Plasmodium falciparum |
IC50: 2 (nM), Ref: 19097788 |
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TCMT1455 | Mycobacterium tuberculosis H37Rv | Mycobacterium tuberculosis H37Rv |
MIC: 64 (ug/ml), Ref: 24641242 |