References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1173
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
TCMC1173
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
TCMC1173
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
TCMC1173
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
TCMC1173
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
TCMC1173
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
TCMC1173
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
TCMC1173
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
TCMC1187
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
IC50: 1900 (nM), Ref: 9834166 |
TCMC1495
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
TCMC1495
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
TCMC1495
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2037
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
TCMC2037
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
TCMC2037
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
TCMC619
|
TCMT293 |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki: 158.49 (nM), Ref: 18077164 |
TCMC619
|
TCMT291 |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
Ki: 7079.46 (nM), Ref: 18077164 |
TCMC619
|
TCMT551 |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki: 8511.38 (nM), Ref: 18077164 |
TCMC619
|
TCMT290 |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
Ki: 9772.37 (nM), Ref: 18077164 |
TCMC619
|
TCMT241 |
Neuronal acetylcholine receptor protein alpha-7 subunit |
Homo sapiens |
Ki: 7943.28 (nM), Ref: 21920761 |
TCMC1330
|
TCMT246 |
Histamine H4 receptor |
Homo sapiens |
Ki: 14.45 (nM), Ref: 14640553 Ki: 7.943 (nM), Ref: 15454206 Ki: 12.02 (nM), Ref: 18357976 Ki: 13.4 (nM), Ref: 18459760 Ki: 12.02 (nM), Ref: 20192225 Ki: 60 (nM), Ref: 20452213 Ki: 7.943 (nM), Ref: 21044842 Ki: 12.59 (nM), Ref: 21044842 Ki: 12.02 (nM), Ref: 21348462 Ki: 15.85 (nM), Ref: 22003888 Ki: 9 (nM), Ref: 22153663 Ki: 19.95 (nM), Ref: 10.1039/C2MD20212C Ki: 4.8 (nM), Ref: 25993395 Ki: 8 (nM), Ref: 25993395 Ki: 15.85 (nM), Ref: 10.1039/C5MD00022J |
TCMC1330
|
TCMT242 |
Histamine H3 receptor |
Homo sapiens |
Ki: 5.2 (nM), Ref: 20384344 Ki: 10 (nM), Ref: 21044842 Ki: 11.75 (nM), Ref: 21348462 Ki: 6.31 (nM), Ref: 22003888 Ki: 16 (nM), Ref: 25993395 |
TCMC1330
|
TCMT245 |
Histamine H2 receptor |
Homo sapiens |
Ki: 5000 (nM), Ref: 25993395 |
TCMC1330
|
TCMT244 |
Histamine H1 receptor |
Homo sapiens |
Ki: 6000 (nM), Ref: 25993395 |
TCMC632
|
TCMT597 |
Solute carrier family 28 member 3 |
Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
TCMC632
|
TCMT709 |
Sodium/nucleoside cotransporter 2 |
Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT710 |
Sodium/nucleoside cotransporter 1 |
Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT296 |
Adenosine A1 receptor |
Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
TCMC632
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC614
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
TCMC916
|
TCMT161 |
Hydroxycarboxylic acid receptor 2 |
Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
TCMC2105
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2105
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1202
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
TCMC1202
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1202
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
TCMC1202
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
TCMC1202
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
TCMC1202
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
TCMC1202
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1202
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
TCMC1202
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
TCMC1202
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
TCMC1202
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
TCMC1202
|
TCMT822 |
Alpha-(1,3)-fucosyltransferase 7 |
Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
TCMC2111
|
TCMT614 |
Egl nine homolog 1 |
Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
TCMC1839
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
TCMC1839
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
TCMC1839
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
TCMC1839
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
TCMC1839
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
TCMC1839
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1839
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
TCMC1839
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
TCMC1839
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1839
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
TCMC1839
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
TCMC1788
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT126 |
Telomerase reverse transcriptase |
Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
TCMC1788
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
TCMC2201
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
TCMC1611
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1611
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2209
|
TCMT597 |
Solute carrier family 28 member 3 |
Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
TCMC2209
|
TCMT710 |
Sodium/nucleoside cotransporter 1 |
Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
TCMC770
|
TCMT588 |
D-amino-acid oxidase |
Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |
TCMC1378
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
TCMC1378
|
TCMT734 |
Matrix metalloproteinase 12 |
Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |