Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
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Ingredient ID & Structure	Target ID	Target Name	Target Organism	Activity Records & Reference
TCMC1881	TCMT151	Protein kinase C alpha	Homo sapiens	Ki: 2.5 (nM), Ref: 11327599 Ki: 6.4 (nM), Ref: 21596562
TCMC1881	TCMT152	Protein kinase C beta	Homo sapiens	Ki: 1.8 (nM), Ref: 11327599
TCMC1881	TCMT153	Protein kinase C gamma	Homo sapiens	Ki: 4.9 (nM), Ref: 11327599
TCMC1881	TCMT154	Protein kinase C delta	Homo sapiens	Ki: 0.8 (nM), Ref: 11327599
TCMC1881	TCMT155	Protein kinase C epsilon	Homo sapiens	Ki: 0.45 (nM), Ref: 11327599
TCMC1173	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394
TCMC1173	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394
TCMC1173	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9870 (nM), Ref: 20185318
TCMC1173	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7410 (nM), Ref: 20185318
TCMC1173	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 8450 (nM), Ref: 20185318
TCMC1173	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7040 (nM), Ref: 20185318
TCMC1173	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2400 (nM), Ref: 20185318
TCMC1173	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2890 (nM), Ref: 20185318
TCMC943	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 810 (nM), Ref: 20100662
TCMC943	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC61	TCMT193	Nuclear factor NF-kappa-B p65 subunit	Homo sapiens	IC50: 250 (nM), Ref: 21513293
TCMC61	TCMT194	Mitogen-activated protein kinase kinase kinase 7	Homo sapiens	IC50: 80 (nM), Ref: 25529738 IC50: 11 (nM), Ref: 26481152 IC50: 8.1 (nM), Ref: 26481152 IC50: 9 (nM), Ref: 27448772
TCMC61	TCMT80	MAP kinase ERK2	Homo sapiens	IC50: 6800 (nM), Ref: 25529738
TCMC61	TCMT195	Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens	IC50: 80 (nM), Ref: 25529738
TCMC61	TCMT196	Dual specificity mitogen-activated protein kinase kinase 7	Homo sapiens	IC50: 1300 (nM), Ref: 25529738
TCMC2051	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 8710 (nM), Ref: 22892213
TCMC2051	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4050 (nM), Ref: 22892213
TCMC2051	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 960 (nM), Ref: 22892213
TCMC957	TCMT191	Signal transducer and activator of transcription 3	Homo sapiens	IC50: 4600 (nM), Ref: 22650325
TCMC957	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 6410 (nM), Ref: 23286284
TCMC957	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 290 (nM), Ref: 23286284 Ki: 141 (nM), Ref: 23286284
TCMC957	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 544 (nM), Ref: 23286284
TCMC761	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 3920 (nM), Ref: 15658857
TCMC948	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394
TCMC948	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394
TCMC948	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5330 (nM), Ref: 20185318
TCMC948	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 5230 (nM), Ref: 20185318
TCMC948	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6720 (nM), Ref: 20185318
TCMC948	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7760 (nM), Ref: 20185318
TCMC948	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 5960 (nM), Ref: 20185318
TCMC948	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9600 (nM), Ref: 20185318
TCMC948	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7570 (nM), Ref: 20185318
TCMC948	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 980 (nM), Ref: 20185318
TCMC948	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1070 (nM), Ref: 20185318
TCMC948	TCMT223	Aldose reductase	Homo sapiens	IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1372	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 2330 (nM), Ref: 22245047
TCMC1372	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 3630 (nM), Ref: 22245047
TCMC1537	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 5930 (nM), Ref: 19846303
TCMC1537	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 630 (nM), Ref: 21561086
TCMC1495	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668
TCMC1495	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668
TCMC1495	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1716	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 4630 (nM), Ref: 26425784
TCMC1957	TCMT34	Cytochrome P450 2D6	Homo sapiens	Ki: 78 (nM), Ref: 26125082
TCMC602	TCMT302	HMG-CoA reductase	Homo sapiens	IC50: 5000 (nM), Ref: 10.1021/np50061a020
TCMC244	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 7900 (nM), Ref: 15916432
TCMC244	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 8300 (nM), Ref: 15658857 IC50: 8298.51 (nM), Ref: 19110342
TCMC820	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5900 (nM), Ref: 23768907
TCMC2126	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 1410 (nM), Ref: 23286284
TCMC2126	TCMT171	Protein-tyrosine phosphatase 1C	Homo sapiens	IC50: 1970 (nM), Ref: 23957426
TCMC2126	TCMT233	Protein-tyrosine phosphatase 2C	Homo sapiens	IC50: 2570 (nM), Ref: 23957426
TCMC1180	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5210 (nM), Ref: 22487176 Ki: 5100 (nM), Ref: 22487176
TCMC1180	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9300 (nM), Ref: 22487176 Ki: 9200 (nM), Ref: 22487176
TCMC1180	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5540 (nM), Ref: 22487176 Ki: 5630 (nM), Ref: 22487176
TCMC1180	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 6590 (nM), Ref: 22487176 Ki: 6650 (nM), Ref: 22487176
TCMC1803	TCMT337	Exportin-1	Homo sapiens	IC50: 1600 (nM), Ref: 20493693
TCMC2052	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 9110 (nM), Ref: 22892213
TCMC2052	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8720 (nM), Ref: 22892213
TCMC2052	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 8430 (nM), Ref: 22892213
TCMC2052	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5930 (nM), Ref: 22892213
TCMC2052	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 780 (nM), Ref: 22892213
TCMC1806	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9600 (nM), Ref: 22137345
TCMC1806	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 3660 (nM), Ref: 22137345
TCMC2037	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662
TCMC2037	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662
TCMC2037	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8800 (nM), Ref: 18579385
TCMC619	TCMT293	Muscarinic acetylcholine receptor M2	Homo sapiens	Ki: 158.49 (nM), Ref: 18077164
TCMC619	TCMT291	Muscarinic acetylcholine receptor M3	Homo sapiens	Ki: 7079.46 (nM), Ref: 18077164
TCMC619	TCMT551	Muscarinic acetylcholine receptor M4	Homo sapiens	Ki: 8511.38 (nM), Ref: 18077164
TCMC619	TCMT290	Muscarinic acetylcholine receptor M5	Homo sapiens	Ki: 9772.37 (nM), Ref: 18077164
TCMC1871	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056
TCMC1871	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662
TCMC1871	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455
TCMC1871	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455
TCMC1871	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662
TCMC619	TCMT241	Neuronal acetylcholine receptor protein alpha-7 subunit	Homo sapiens	Ki: 7943.28 (nM), Ref: 21920761
TCMC1851	TCMT560	Coagulation factor X	Homo sapiens	IC50: 170 (nM), Ref: 9834152 Ki: 570 (nM), Ref: 9834152
TCMC1851	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3760 (nM), Ref: 24835197 Ki: 5130 (nM), Ref: 24835197
TCMC1851	TCMT240	Salivary alpha-amylase	Homo sapiens	IC50: 2350 (nM), Ref: 26395057 Ki: 2600 (nM), Ref: 26395057
TCMC487	TCMT561	5'-nucleotidase	Homo sapiens	IC50: 8200 (nM), Ref: 24215819
TCMC962	TCMT45	Beta amyloid A4 protein	Homo sapiens	Ki: 0.208 (nM), Ref: 17004725 IC50: 800 (nM), Ref: 17270435 IC50: 3900 (nM), Ref: 26099993
TCMC962	TCMT566	Nitric oxide synthase, inducible	Homo sapiens	IC50: 6000 (nM), Ref: 18077363
TCMC962	TCMT87	Cytochrome P450 2C9	Homo sapiens	IC50: 4300 (nM), Ref: 18249473
TCMC962	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 8500 (nM), Ref: 19128977
TCMC962	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2410 (nM), Ref: 20674354
TCMC962	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 380 (nM), Ref: 20674354
TCMC962	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4970 (nM), Ref: 20674354
TCMC962	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9460 (nM), Ref: 20674354
TCMC962	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 9940 (nM), Ref: 20674354
TCMC962	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 9300 (nM), Ref: 20674354
TCMC962	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4050 (nM), Ref: 20674354
TCMC962	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 3480 (nM), Ref: 20674354
TCMC962	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 6850 (nM), Ref: 20674354
TCMC962	TCMT44	Glyoxalase I	Homo sapiens	Ki: 10000 (nM), Ref: 21237663
TCMC962	TCMT22	Intestinal alkaline phosphatase	Homo sapiens	IC50: 7410 (nM), Ref:
TCMC962	TCMT46	Coagulation factor III	Homo sapiens	IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5 IC50: 199.63 (nM), Ref: 23199480
TCMC962	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 8600 (nM), Ref: 23245570
TCMC962	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 4501 (nM), Ref: 23800686
TCMC962	TCMT570	Aminopeptidase N	Homo sapiens	IC50: 10000 (nM), Ref: 23860593
TCMC962	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 3900 (nM), Ref: 24920381 IC50: 500 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381
TCMC962	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 8100 (nM), Ref: 24920381
TCMC962	TCMT301	Prostaglandin E synthase	Homo sapiens	IC50: 600 (nM), Ref: 24920381 IC50: 1200 (nM), Ref: 24920381
TCMC962	TCMT3	Arachidonate 15-lipoxygenase	Homo sapiens	IC50: 1200 (nM), Ref: 24920381
TCMC962	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 5300 (nM), Ref: 25088549
TCMC962	TCMT565	Histone acetyltransferase p300	Homo sapiens	IC50: 6500 (nM), Ref: 25730130
TCMC2119	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9140 (nM), Ref: 20185318
TCMC2119	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9010 (nM), Ref: 20185318
TCMC2119	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8200 (nM), Ref: 20185318
TCMC2119	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7810 (nM), Ref: 20185318
TCMC2119	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7550 (nM), Ref: 20185318
TCMC2119	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6340 (nM), Ref: 20185318
TCMC2119	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8580 (nM), Ref: 20185318
TCMC2119	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3190 (nM), Ref: 20185318
TCMC2119	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4150 (nM), Ref: 20185318
TCMC416	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 4500 (nM), Ref: 14592472
TCMC1293	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2940 (nM), Ref: 19231207
TCMC1439	TCMT588	D-amino-acid oxidase	Homo sapiens	IC50: 2000 (nM), Ref: 23683589
TCMC1439	TCMT159	Tyrosinase	Homo sapiens	IC50: 9150 (nM), Ref: 26386819
TCMC1429	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2700 (nM), Ref: 17378609
TCMC1429	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 1050 (nM), Ref: 18533708
TCMC1429	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 360 (nM), Ref: 18533708
TCMC1429	TCMT187	Androgen Receptor	Homo sapiens	IC50: 9700 (nM), Ref: 19592245
TCMC1429	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 716 (nM), Ref: 20696580
TCMC1429	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 632 (nM), Ref: 20696580
TCMC1429	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 47 (nM), Ref: 20696580
TCMC1429	TCMT223	Aldose reductase	Homo sapiens	IC50: 10000 (nM), Ref: 22261024
TCMC1429	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 2320 (nM), Ref: 23411073
TCMC1429	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 9640 (nM), Ref: 23656512
TCMC1429	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 10000 (nM), Ref: 26322379
TCMC1429	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9525.7 (nM), Ref: 26498393
TCMC1429	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 25 (nM), Ref: 26498393
TCMC1429	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 145.9 (nM), Ref: 26498393
TCMC1429	TCMT159	Tyrosinase	Homo sapiens	IC50: 1000 (nM), Ref: 26841168
TCMC1285	TCMT33	Cytochrome P450 3A4	Homo sapiens	Ki: 399 (nM), Ref: 16248836
TCMC2188	TCMT223	Aldose reductase	Homo sapiens	IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1411	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1261 (nM), Ref: 20696580
TCMC1411	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 56 (nM), Ref: 20696580
TCMC1411	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 17 (nM), Ref: 20696580
TCMC1411	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 212.9 (nM), Ref: 26498393
TCMC1411	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.4 (nM), Ref: 26498393
TCMC1411	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 54.9 (nM), Ref: 26498393 Ki: 220 (nM), Ref: 26498393
TCMC1411	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 440 (nM), Ref: 26498393
TCMC895	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 7630 (nM), Ref: 20053563
TCMC895	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 7630 (nM), Ref: 20053563
TCMC895	TCMT318	Putative hexokinase HKDC1	Homo sapiens	IC50: 8990 (nM), Ref:
TCMC895	TCMT599	Ubiquitin-conjugating enzyme E2 N	Homo sapiens	IC50: 3012 (nM), Ref: IC50: 2197 (nM), Ref:
TCMC895	TCMT608	Solute carrier family 22 member 3	Homo sapiens	IC50: 410 (nM), Ref: 23241029
TCMC895	TCMT213	Solute carrier family 22 member 1	Homo sapiens	IC50: 210 (nM), Ref: 23241029
TCMC895	TCMT309	Solute carrier family 22 member 2	Homo sapiens	IC50: 400 (nM), Ref: 23241029
TCMC895	TCMT310	Multidrug and toxin extrusion protein 2	Homo sapiens	IC50: 500 (nM), Ref: 23241029
TCMC895	TCMT311	Multidrug and toxin extrusion protein 1	Homo sapiens	IC50: 700 (nM), Ref: 23241029
TCMC13	TCMT23	Alkaline phosphatase, tissue-nonspecific isozyme	Homo sapiens	IC50: 407 (nM), Ref:
TCMC1424	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 2100 (nM), Ref: 17994701
TCMC42	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 8390 (nM), Ref: 26696252
TCMC42	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2540 (nM), Ref: 26696252
TCMC737	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 168 (nM), Ref: 26498393
TCMC737	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 5591.2 (nM), Ref: 26498393
TCMC737	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 423.7 (nM), Ref: 26498393
TCMC737	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4.9 (nM), Ref: 26498393
TCMC2025	TCMT61	Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens	IC50: 2025.72 (nM), Ref:
TCMC1041	TCMT636	DNA polymerase alpha subunit	Homo sapiens	Ki: 830 (nM), Ref: 1705574
TCMC1041	TCMT17	DNA polymerase beta	Homo sapiens	Ki: 390 (nM), Ref: 1705574
TCMC1480	TCMT107	Glutamate receptor ionotropic kainate 2	Homo sapiens	Ki: 1106 (nM), Ref: 10821708
TCMC1480	TCMT108	Glutamate receptor ionotropic, AMPA 1	Homo sapiens	Ki: 1360 (nM), Ref: 9357531
TCMC1480	TCMT109	Glutamate receptor ionotropic, AMPA 2	Homo sapiens	Ki: 940 (nM), Ref: 9357531
TCMC1480	TCMT110	Glutamate receptor ionotropic, AMPA 4	Homo sapiens	Ki: 868 (nM), Ref: 9357531
TCMC1480	TCMT111	Glutamate receptor ionotropic kainate 5	Homo sapiens	Ki: 701 (nM), Ref: 9357531
TCMC1480	TCMT660	Metabotropic glutamate receptor 8	Homo sapiens	IC50: 5.7 (nM), Ref: 15603952
TCMC1480	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 613 (nM), Ref: 16250647
TCMC1480	TCMT653	Metabotropic glutamate receptor 1	Homo sapiens	Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT654	Metabotropic glutamate receptor 5	Homo sapiens	Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT657	Metabotropic glutamate receptor 4	Homo sapiens	Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT655	Metabotropic glutamate receptor 2	Homo sapiens	Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT664	Excitatory amino acid transporter 3	Homo sapiens	Ki: 51 (nM), Ref: 18578477
TCMC1480	TCMT656	Metabotropic glutamate receptor 3	Homo sapiens	Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H
TCMC694	TCMT230	Estradiol 17-beta-dehydrogenase 3	Homo sapiens	IC50: 758 (nM), Ref: 11086723 IC50: 758 (nM), Ref: 16078844
TCMC694	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 20 (nM), Ref: 8035427 Ki: 35 (nM), Ref: 26469743
TCMC949	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8900 (nM), Ref: 19911821
TCMC949	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 48 (nM), Ref: 19911821
TCMC949	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9100 (nM), Ref: 19911821
TCMC949	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3300 (nM), Ref: 19911821
TCMC949	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 2000 (nM), Ref: 19911821
TCMC949	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 5200 (nM), Ref: 19911821
TCMC949	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9400 (nM), Ref: 19911821
TCMC949	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 6800 (nM), Ref: 19911821
TCMC949	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 5600 (nM), Ref: 19911821
TCMC949	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270
TCMC949	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270
TCMC1786	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900
TCMC1786	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086
TCMC1786	TCMT190	T-cell protein-tyrosine phosphatase	Homo sapiens	IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900
TCMC1786	TCMT563	Dual specificity phosphatase Cdc25B	Homo sapiens	IC50: 980 (nM), Ref: 25497963
TCMC1735	TCMT599	Ubiquitin-conjugating enzyme E2 N	Homo sapiens	IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC1506	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 101.2 (nM), Ref: 26498393
TCMC1506	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 268.3 (nM), Ref: 26498393
TCMC1506	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4.8 (nM), Ref: 26498393
TCMC845	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 630 (nM), Ref: 19231207
TCMC837	TCMT690	Histone deacetylase 3	Homo sapiens	IC50: 9000 (nM), Ref: 21874153
TCMC2124	TCMT39	Phosphodiesterase 5A	Homo sapiens	IC50: 4703 (nM), Ref:
TCMC2124	TCMT289	Thromboxane-A synthase	Homo sapiens	IC50: 325 (nM), Ref:
TCMC1594	TCMT197	Phosphodiesterase 4D	Homo sapiens	IC50: 2900 (nM), Ref: 22483586 IC50: 2910 (nM), Ref: 26473791
TCMC1594	TCMT698	Phosphodiesterase 4B	Homo sapiens	IC50: 4500 (nM), Ref: 22483586
TCMC632	TCMT597	Solute carrier family 28 member 3	Homo sapiens	Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705
TCMC632	TCMT709	Sodium/nucleoside cotransporter 2	Homo sapiens	Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT710	Sodium/nucleoside cotransporter 1	Homo sapiens	Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT296	Adenosine A1 receptor	Homo sapiens	IC50: 2.344 (nM), Ref: 26756468
TCMC632	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 1.148 (nM), Ref: 26756468
TCMC1956	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1080 (nM), Ref: 21282059
TCMC1956	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 470 (nM), Ref: 21282059
TCMC1956	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4450 (nM), Ref: 21282059
TCMC1956	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4090 (nM), Ref: 21282059
TCMC1956	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439
TCMC1956	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 2450 (nM), Ref: 22687439
TCMC1956	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 690 (nM), Ref: 22668600
TCMC1956	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7870 (nM), Ref: 22668600
TCMC1567	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 890 (nM), Ref: 22668600
TCMC1567	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 960 (nM), Ref: 22668600
TCMC1567	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 790 (nM), Ref: 22668600
TCMC1567	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 810 (nM), Ref: 22668600
TCMC1567	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 580 (nM), Ref: 22668600
TCMC1567	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 710 (nM), Ref: 22668600
TCMC2025	TCMT295	Matrix metalloproteinase-1	Homo sapiens	IC50: 5600 (nM), Ref: 23353736
TCMC1113	TCMT47	Apoptosis regulator Bcl-2	Homo sapiens	Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC43	TCMT301	Prostaglandin E synthase	Homo sapiens	IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43	TCMT565	Histone acetyltransferase p300	Homo sapiens	IC50: 6500 (nM), Ref: 26701186
TCMC43	TCMT208	Monoamine oxidase A	Homo sapiens	Ki: 710 (nM), Ref: 26819666
TCMC43	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601
TCMC2142	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 600 (nM), Ref: 6827528
TCMC2142	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 10000 (nM), Ref: 14552748
TCMC2142	TCMT187	Androgen Receptor	Homo sapiens	IC50: 3.9 (nM), Ref: 15456242 IC50: 2.7 (nM), Ref: 16309907 IC50: 4.571 (nM), Ref: 22746350 IC50: 4.17 (nM), Ref: 25646649 IC50: 4.27 (nM), Ref: 25646649
TCMC2142	TCMT99	Testis-specific androgen-binding protein	Homo sapiens	IC50: 14 (nM), Ref: 17149875
TCMC2142	TCMT725	Voltage-gated L-type calcium channel alpha-1C subunit	Homo sapiens	IC50: 34 (nM), Ref: 22761000 IC50: 38.4 (nM), Ref: 22761000
TCMC2003	TCMT82	Estrogen receptor alpha	Homo sapiens	Ki: 785 (nM), Ref: 15634023
TCMC2003	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref:
TCMC2003	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006
TCMC2003	TCMT329	Quinone reductase 2	Homo sapiens	IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376
TCMC2003	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2210 (nM), Ref: 20674354
TCMC2003	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2770 (nM), Ref: 20674354
TCMC2003	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 9090 (nM), Ref: 20674354
TCMC2003	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4470 (nM), Ref: 20674354
TCMC2003	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4750 (nM), Ref: 20674354
TCMC2003	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4640 (nM), Ref: 20674354
TCMC2003	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 8070 (nM), Ref: 20674354
TCMC2003	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4350 (nM), Ref: 20674354
TCMC2003	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 810 (nM), Ref: 20674354
TCMC2003	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 950 (nM), Ref: 20674354
TCMC2003	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4090 (nM), Ref: 20674354
TCMC2003	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 830 (nM), Ref: 20674354
TCMC2003	TCMT729	PI3-kinase p110-alpha subunit	Homo sapiens	IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003	TCMT730	PI3-kinase p110-beta subunit	Homo sapiens	IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601
TCMC156	TCMT327	Vanilloid receptor	Homo sapiens	IC50: 35 (nM), Ref: 16000002
TCMC2070	TCMT327	Vanilloid receptor	Homo sapiens	IC50: 290 (nM), Ref: 22257892
TCMC1741	TCMT161	Hydroxycarboxylic acid receptor 2	Homo sapiens	IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085
TCMC1446	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 6300 (nM), Ref: 21641214
TCMC1568	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 3580 (nM), Ref: 22658537
TCMC1568	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 610 (nM), Ref: 22658537
TCMC1568	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 2750 (nM), Ref: 22658537
TCMC1609	TCMT44	Glyoxalase I	Homo sapiens	IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529
TCMC1609	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18778944
TCMC1609	TCMT737	DNA dC->dU-editing enzyme APOBEC-3G	Homo sapiens	IC50: 2390 (nM), Ref:
TCMC1609	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 2120 (nM), Ref: 24900447
TCMC1609	TCMT558	DNA topoisomerase II alpha	Homo sapiens	IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1690 (nM), Ref: 23411073
TCMC1609	TCMT2	Microtubule-associated protein tau	Homo sapiens	IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT740	PI3-kinase p110-gamma subunit	Homo sapiens	IC50: 4720 (nM), Ref: 25050878
TCMC1609	TCMT13	DNA-(apurinic or apyrimidinic site) lyase	Homo sapiens	IC50: 320 (nM), Ref: 25280182
TCMC1399	TCMT223	Aldose reductase	Homo sapiens	IC50: 320 (nM), Ref: 22261024
TCMC1986	TCMT223	Aldose reductase	Homo sapiens	IC50: 150 (nM), Ref: 18165015 IC50: 2000 (nM), Ref: 22261024
TCMC2025	TCMT359	Tyrosine-protein kinase FYN	Homo sapiens	IC50: 1300 (nM), Ref: 17315853 IC50: 3600 (nM), Ref: 17315853 Ki: 7500 (nM), Ref: 17315853
TCMC2031	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 7500 (nM), Ref: 16610779
TCMC1102	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 40 (nM), Ref: 19414254
TCMC1102	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2320 (nM), Ref: 20185318
TCMC1102	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2180 (nM), Ref: 20185318
TCMC1102	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9080 (nM), Ref: 20185318
TCMC1102	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7590 (nM), Ref: 20185318
TCMC1102	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7060 (nM), Ref: 20185318
TCMC1102	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213
TCMC1102	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9370 (nM), Ref: 20185318
TCMC1102	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 8910 (nM), Ref: 20185318
TCMC1102	TCMT753	Mothers against decapentaplegic homolog 3	Homo sapiens	IC50: 142 (nM), Ref:
TCMC1102	TCMT721	Heat shock 70 kDa protein 1	Homo sapiens	IC50: 760 (nM), Ref:
TCMC1102	TCMT189	Dual specificity protein phosphatase 3	Homo sapiens	IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102	TCMT223	Aldose reductase	Homo sapiens	IC50: 200 (nM), Ref: 22261024
TCMC1102	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 510 (nM), Ref: 22377675
TCMC1102	TCMT354	Serine/threonine-protein kinase Aurora-A	Homo sapiens	IC50: 2480 (nM), Ref: 22377675
TCMC1102	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 2500 (nM), Ref: 22377675
TCMC1102	TCMT626	Serine/threonine-protein kinase B-raf	Homo sapiens	IC50: 1760 (nM), Ref: 22377675
TCMC1102	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 690 (nM), Ref: 22377675
TCMC1102	TCMT418	Ephrin type-B receptor 4	Homo sapiens	IC50: 1830 (nM), Ref: 22377675
TCMC1102	TCMT704	Receptor protein-tyrosine kinase erbB-2	Homo sapiens	IC50: 3540 (nM), Ref: 22377675
TCMC1102	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 3110 (nM), Ref: 22377675
TCMC1102	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 250 (nM), Ref: 22377675
TCMC1102	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 800 (nM), Ref: 22377675
TCMC1102	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 790 (nM), Ref: 22377675
TCMC1102	TCMT457	Vascular endothelial growth factor receptor 3	Homo sapiens	IC50: 1540 (nM), Ref: 22377675
TCMC1102	TCMT377	Insulin receptor	Homo sapiens	IC50: 340 (nM), Ref: 22377675
TCMC1102	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 22377675
TCMC1102	TCMT536	Platelet-derived growth factor receptor beta	Homo sapiens	IC50: 1300 (nM), Ref: 22377675
TCMC1102	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT755	Serine/threonine-protein kinase PLK4	Homo sapiens	IC50: 2970 (nM), Ref: 22377675
TCMC1102	TCMT502	Tyrosine-protein kinase TIE-2	Homo sapiens	IC50: 260 (nM), Ref: 22377675
TCMC1102	TCMT756	Mitogen-activated protein kinase kinase kinase 8	Homo sapiens	IC50: 2370 (nM), Ref: 22377675
TCMC1102	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 100 (nM), Ref: 24900447
TCMC1102	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8150 (nM), Ref: 22892213
TCMC1102	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4240 (nM), Ref: 22892213
TCMC1102	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3900 (nM), Ref: 24835197
TCMC1409	TCMT22	Intestinal alkaline phosphatase	Homo sapiens	IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409	TCMT223	Aldose reductase	Homo sapiens	IC50: 4500 (nM), Ref: 22261024
TCMC1409	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393
TCMC1409	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 75.7 (nM), Ref: 26498393
TCMC1409	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3.8 (nM), Ref: 26498393
TCMC1409	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393
TCMC1964	TCMT726	Bcr/Abl fusion protein	Homo sapiens	IC50: 10000 (nM), Ref: 16686543
TCMC1964	TCMT329	Quinone reductase 2	Homo sapiens	IC50: 5100 (nM), Ref: 23953689
TCMC1964	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 1400 (nM), Ref: 10.1039/C3MD00317E Ki: 900 (nM), Ref: 10.1039/C0MD00242A
TCMC1964	TCMT215	Cytochrome P450 1A1	Homo sapiens	Ki: 570 (nM), Ref: 10.1039/C0MD00242A
TCMC910	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1118 (nM), Ref: 20696580
TCMC910	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 95 (nM), Ref: 20696580
TCMC910	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 20 (nM), Ref: 20696580
TCMC2048	TCMT771	Serine-protein kinase ATR	Homo sapiens	IC50: 7300 (nM), Ref: 22835870
TCMC1982	TCMT239	Serine/threonine-protein kinase PIM1	Homo sapiens	IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302
TCMC1982	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208
TCMC1982	TCMT223	Aldose reductase	Homo sapiens	IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999
TCMC1982	TCMT44	Glyoxalase I	Homo sapiens	IC50: 3200 (nM), Ref: 18258440
TCMC1982	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 1540 (nM), Ref: 18533708
TCMC452	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2370 (nM), Ref: 21282059
TCMC452	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 600 (nM), Ref: 21282059
TCMC452	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4530 (nM), Ref: 21282059
TCMC452	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 3530 (nM), Ref: 21282059
TCMC452	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 3170 (nM), Ref: 21669522
TCMC1982	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7890 (nM), Ref: 20185318
TCMC1982	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8100 (nM), Ref: 20185318
TCMC1982	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2540 (nM), Ref: 20185318
TCMC1982	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2680 (nM), Ref: 20185318
TCMC1982	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6810 (nM), Ref: 20185318
TCMC1982	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6170 (nM), Ref: 20185318
TCMC1982	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4840 (nM), Ref: 20185318
TCMC1982	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 7000 (nM), Ref: 20185318
TCMC1982	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9390 (nM), Ref: 20185318
TCMC1982	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 5410 (nM), Ref: 20185318
TCMC1158	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3100 (nM), Ref: 24835197 Ki: 6840 (nM), Ref: 24835197
TCMC1982	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 12 (nM), Ref: 20413308
TCMC1982	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583
TCMC1982	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1191 (nM), Ref: 20696580
TCMC1982	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 77 (nM), Ref: 20696580
TCMC1982	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 6680 (nM), Ref: 22658537
TCMC1982	TCMT320	Matrix metalloproteinase 3	Homo sapiens	IC50: 5570 (nM), Ref: 22658537
TCMC1982	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 1610 (nM), Ref: 22658537
TCMC1982	TCMT322	Matrix metalloproteinase 13	Homo sapiens	IC50: 8460 (nM), Ref: 22658537
TCMC1982	TCMT422	CaM kinase II beta	Homo sapiens	IC50: 3000 (nM), Ref: 21798748
TCMC2098	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1400 (nM), Ref: 20590092
TCMC2098	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1110 (nM), Ref: 20590092
TCMC2098	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 112 (nM), Ref: 20590092
TCMC2098	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 1220 (nM), Ref: 20590092
TCMC2098	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 1440 (nM), Ref: 20590092
TCMC2098	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 1410 (nM), Ref: 20590092
TCMC2098	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 1230 (nM), Ref: 20590092
TCMC2098	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 1370 (nM), Ref: 20590092
TCMC2098	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 1000 (nM), Ref: 20590092
TCMC1982	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344
TCMC1982	TCMT784	Vasopressin V2 receptor	Homo sapiens	IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772
TCMC1982	TCMT785	Interleukin-8 receptor A	Homo sapiens	IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772
TCMC1982	TCMT786	C-C chemokine receptor type 4	Homo sapiens	IC50: 10000 (nM), Ref: 23437772
TCMC1982	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 590 (nM), Ref: 23411073
TCMC1982	TCMT601	Thrombin	Homo sapiens	IC50: 1500 (nM), Ref: 24610996
TCMC1982	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 280 (nM), Ref: 24328302
TCMC1982	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 120 (nM), Ref: 24328302
TCMC1982	TCMT791	Protein kinase N1	Homo sapiens	IC50: 5800 (nM), Ref: 24328302
TCMC1982	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 5750 (nM), Ref: 24328302
TCMC1982	TCMT462	Serine/threonine-protein kinase NEK6	Homo sapiens	IC50: 4230 (nM), Ref: 24328302
TCMC1982	TCMT445	Serine/threonine-protein kinase NEK2	Homo sapiens	IC50: 5730 (nM), Ref: 24328302
TCMC1982	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 24328302
TCMC1982	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 300 (nM), Ref: 24328302
TCMC1982	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 1200 (nM), Ref: 24328302
TCMC1982	TCMT388	Tyrosine-protein kinase receptor UFO	Homo sapiens	IC50: 960 (nM), Ref: 24328302
TCMC1982	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 910 (nM), Ref: 24328302
TCMC1982	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 5090 (nM), Ref: 24328302
TCMC1982	TCMT402	ALK tyrosine kinase receptor	Homo sapiens	IC50: 3320 (nM), Ref: 24328302
TCMC1982	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 5390 (nM), Ref: 24328302
TCMC1982	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124
TCMC1982	TCMT793	Liver glycogen phosphorylase	Homo sapiens	IC50: 4800 (nM), Ref: 25092521
TCMC1982	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 2110 (nM), Ref: 22328583
TCMC1982	TCMT217	Cytochrome P450 2C8	Homo sapiens	IC50: 1390 (nM), Ref: 22328583
TCMC1982	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 8900 (nM), Ref: 26322379
TCMC880	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9910 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 20185318 Ki: 9900 (nM), Ref: 22245047 Ki: 9900 (nM), Ref: 26073005 Ki: 9900 (nM), Ref: 26520662
TCMC880	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4200 (nM), Ref: 18579385 Ki: 4200 (nM), Ref: 20185318
TCMC880	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8900 (nM), Ref: 18579385 Ki: 8900 (nM), Ref: 20185318
TCMC916	TCMT161	Hydroxycarboxylic acid receptor 2	Homo sapiens	Ki: 4900 (nM), Ref: 21167710
TCMC1268	TCMT278	Solute carrier organic anion transporter family member 1B1	Homo sapiens	IC50: 1400 (nM), Ref: 22587986 IC50: 2200 (nM), Ref: 22587986
TCMC1268	TCMT221	Bile salt export pump	Homo sapiens	IC50: 5300 (nM), Ref: 21965623
TCMC2105	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC22	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 1000 (nM), Ref: 15679319 Ki: 177 (nM), Ref: 16248836
TCMC1886	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 810 (nM), Ref: 26498394
TCMC1886	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 670 (nM), Ref: 26498394
TCMC1886	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 770 (nM), Ref: 26498394
TCMC1886	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 620 (nM), Ref: 26498394
TCMC1886	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 810 (nM), Ref: 26498394
TCMC1886	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8470 (nM), Ref: 26498394
TCMC1886	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 720 (nM), Ref: 26498394
TCMC124	TCMT194	Mitogen-activated protein kinase kinase kinase 7	Homo sapiens	IC50: 1300 (nM), Ref: 26481152
TCMC1830	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 930 (nM), Ref: 15357969
TCMC1830	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 2600 (nM), Ref: 15357969
TCMC1830	TCMT808	Fatty acid binding protein epidermal	Homo sapiens	IC50: 1200 (nM), Ref: 15357969
TCMC1830	TCMT809	Fatty acid binding protein intestinal	Homo sapiens	IC50: 1700 (nM), Ref: 15357969
TCMC1830	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1830	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1202	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 7030 (nM), Ref: 20185318
TCMC1202	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1202	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6990 (nM), Ref: 20185318
TCMC1202	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6070 (nM), Ref: 20185318
TCMC1202	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6130 (nM), Ref: 20185318
TCMC1202	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9970 (nM), Ref: 20185318
TCMC1202	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1202	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9800 (nM), Ref: 20185318
TCMC1202	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7490 (nM), Ref: 20185318
TCMC1202	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2250 (nM), Ref: 20185318
TCMC1202	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3200 (nM), Ref: 20185318
TCMC1202	TCMT822	Alpha-(1,3)-fucosyltransferase 7	Homo sapiens	IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1143	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 860 (nM), Ref: 22668600
TCMC1143	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 830 (nM), Ref: 22668600
TCMC1143	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 780 (nM), Ref: 22668600
TCMC1143	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 750 (nM), Ref: 22668600
TCMC1143	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 610 (nM), Ref: 22668600
TCMC1143	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 650 (nM), Ref: 22668600
TCMC2128	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 3900 (nM), Ref: 23286284
TCMC1757	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 130 (nM), Ref: 17378609 IC50: 110 (nM), Ref: 19848434 IC50: 25 (nM), Ref: 21958737 IC50: 120 (nM), Ref: 21958738
TCMC1757	TCMT3	Arachidonate 15-lipoxygenase	Homo sapiens	IC50: 110 (nM), Ref: 12608855 IC50: 1100 (nM), Ref: 19848434 IC50: 5100 (nM), Ref: 21739938 IC50: 110 (nM), Ref: 24684213
TCMC1757	TCMT81	Arachidonate 12-lipoxygenase	Homo sapiens	IC50: 180 (nM), Ref: 12608855 IC50: 5900 (nM), Ref: 19848434 IC50: 110 (nM), Ref: 21739938
TCMC1757	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 11 (nM), Ref: 20413308
TCMC983	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref:
TCMC983	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 7300 (nM), Ref: 21030469
TCMC983	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 718.7 (nM), Ref: 26498393
TCMC983	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.2 (nM), Ref: 26498393
TCMC983	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 56.4 (nM), Ref: 26498393
TCMC2111	TCMT614	Egl nine homolog 1	Homo sapiens	IC50: 3000 (nM), Ref: 18942826
TCMC1919	TCMT613	Glucocorticoid receptor	Homo sapiens	IC50: 14 (nM), Ref: 19364854
TCMC1587	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 83.7 (nM), Ref: 23286284 Ki: 40 (nM), Ref: 23286284
TCMC1587	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 2530 (nM), Ref: 23286284
TCMC755	TCMT3	Arachidonate 15-lipoxygenase	Homo sapiens	Ki: 600 (nM), Ref: 21739938
TCMC755	TCMT81	Arachidonate 12-lipoxygenase	Homo sapiens	Ki: 1600 (nM), Ref: 21739938
TCMC755	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469
TCMC755	TCMT384	G protein-coupled receptor kinase 6	Homo sapiens	IC50: 8700 (nM), Ref:
TCMC1428	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 509 (nM), Ref: 20696580
TCMC1428	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 88 (nM), Ref: 20696580
TCMC1428	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC1190	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 9280 (nM), Ref: 22892213
TCMC1190	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6580 (nM), Ref: 22892213
TCMC1190	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4240 (nM), Ref: 22892213
TCMC1190	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9.7 (nM), Ref: 22892213
TCMC1774	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3100 (nM), Ref: 20674354 Ki: 3100 (nM), Ref: 21282059 Ki: 3400 (nM), Ref: 22137345
TCMC1774	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9300 (nM), Ref: 22137345
TCMC2204	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270
TCMC2204	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270
TCMC1168	TCMT117	Kappa opioid receptor	Homo sapiens	Ki: 2515 (nM), Ref: 18166466
TCMC1839	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318
TCMC1839	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318
TCMC1839	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318
TCMC1839	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6160 (nM), Ref: 20185318
TCMC1839	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 3730 (nM), Ref: 20185318
TCMC1839	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1839	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 5700 (nM), Ref: 20185318
TCMC1839	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7130 (nM), Ref: 20185318
TCMC1839	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1839	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 6610 (nM), Ref: 20185318
TCMC1839	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 870 (nM), Ref: 20185318
TCMC850	TCMT307	HERG	Homo sapiens	IC50: 4897.79 (nM), Ref: 21185626
TCMC850	TCMT707	Adenosine A2a receptor	Homo sapiens	Ki: 5011.87 (nM), Ref: 21661720 Ki: 9560 (nM), Ref: 23200243 Ki: 2480 (nM), Ref: 23200243
TCMC850	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 7250 (nM), Ref: 23791077
TCMC378	TCMT848	Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens	IC50: 2370 (nM), Ref: IC50: 5750 (nM), Ref:
TCMC1788	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT126	Telomerase reverse transcriptase	Homo sapiens	IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	Ki: 1500 (nM), Ref: 27460668
TCMC732	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 5900 (nM), Ref: 21561086
TCMC1203	TCMT822	Alpha-(1,3)-fucosyltransferase 7	Homo sapiens	IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC804	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 2000 (nM), Ref: 21561086
TCMC1319	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9700 (nM), Ref: 19911821
TCMC1319	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9000 (nM), Ref: 19911821
TCMC1319	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9800 (nM), Ref: 19911821
TCMC1319	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 2400 (nM), Ref: 19911821
TCMC1319	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 5500 (nM), Ref: 19911821
TCMC1319	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 5100 (nM), Ref: 19911821
TCMC1319	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 8300 (nM), Ref: 19911821
TCMC1319	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5900 (nM), Ref: 19911821
TCMC1787	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3500 (nM), Ref: 18798681 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2002	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 7700 (nM), Ref: 18501600 Ki: 7700 (nM), Ref: 18579385 Ki: 7700 (nM), Ref: 26073005
TCMC2002	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7500 (nM), Ref: 18579385
TCMC2002	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7100 (nM), Ref: 18579385
TCMC2002	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 8700 (nM), Ref: 18579385
TCMC20	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 1100 (nM), Ref: 15679319
TCMC1516	TCMT44	Glyoxalase I	Homo sapiens	IC50: 7700 (nM), Ref: 18258440
TCMC1516	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 3370 (nM), Ref: 20696580
TCMC1516	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1249 (nM), Ref: 20696580
TCMC1516	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 79 (nM), Ref: 20696580
TCMC1516	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 8200 (nM), Ref: 21641214
TCMC1516	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 3610 (nM), Ref: 22658537
TCMC1516	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 5620 (nM), Ref: 22658537
TCMC1516	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 980 (nM), Ref: 22658537
TCMC1516	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 830 (nM), Ref: 23411073
TCMC1516	TCMT127	Poly [ADP-ribose] polymerase-1	Homo sapiens	IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272
TCMC1516	TCMT128	Tankyrase-2	Homo sapiens	IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272
TCMC1516	TCMT129	Tankyrase-1	Homo sapiens	IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272
TCMC1516	TCMT223	Aldose reductase	Homo sapiens	IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431
TCMC1516	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 1600 (nM), Ref: 24368208
TCMC1516	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 6400 (nM), Ref: 24878198
TCMC1516	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677
TCMC1516	TCMT100	Transthyretin	Homo sapiens	IC50: 7000 (nM), Ref: 26214366
TCMC1516	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3691.6 (nM), Ref: 26498393
TCMC1516	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.7 (nM), Ref: 26498393
TCMC1516	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 60.3 (nM), Ref: 26498393
TCMC1516	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 293 (nM), Ref: 26498393
TCMC1516	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 9200 (nM), Ref: 26529431
TCMC392	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 2400 (nM), Ref: 15658857 IC50: 2398.83 (nM), Ref: 19110342
TCMC1977	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 7410 (nM), Ref: 21669522
TCMC1977	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 540 (nM), Ref: 21669522
TCMC1977	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 520 (nM), Ref: 21669522
TCMC1356	TCMT223	Aldose reductase	Homo sapiens	IC50: 3000 (nM), Ref: 22261024
TCMC2127	TCMT223	Aldose reductase	Homo sapiens	IC50: 8690 (nM), Ref: 22261024
TCMC2127	TCMT126	Telomerase reverse transcriptase	Homo sapiens	IC50: 5000 (nM), Ref: 22044621 IC50: 500 (nM), Ref: 22044621
TCMC2127	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 69.4 (nM), Ref: 23286284 Ki: 2450 (nM), Ref: 23286284
TCMC2127	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 6890 (nM), Ref: 23286284
TCMC2127	TCMT171	Protein-tyrosine phosphatase 1C	Homo sapiens	IC50: 2140 (nM), Ref: 23957426
TCMC2127	TCMT233	Protein-tyrosine phosphatase 2C	Homo sapiens	IC50: 2590 (nM), Ref: 23957426
TCMC1734	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 3430 (nM), Ref: 19097799
TCMC1734	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 4960 (nM), Ref: 18533708
TCMC1734	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469
TCMC1734	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 3656 (nM), Ref: 20696580
TCMC1734	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 79.5 (nM), Ref: 26498393
TCMC1734	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.3 (nM), Ref: 26498393
TCMC1734	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 44.3 (nM), Ref: 26498393
TCMC4	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 6000 (nM), Ref: 14592472
TCMC341	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 510 (nM), Ref: 19231207
TCMC1551	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 1900 (nM), Ref: 16248836 Ki: 1900 (nM), Ref: 16248836 Ki: 800 (nM), Ref: 16248836 Ki: 250 (nM), Ref: 22696418
TCMC1551	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 760 (nM), Ref: 23746477
TCMC1551	TCMT268	Cytochrome P450 2A13	Homo sapiens	Ki: 40 (nM), Ref: 22696418
TCMC1798	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1480 (nM), Ref: 23411073
TCMC811	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 2030 (nM), Ref: 19097799
TCMC811	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 9900 (nM), Ref: 18533708
TCMC811	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10.2 (nM), Ref: 20413308
TCMC811	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7078.5 (nM), Ref: 26498393
TCMC811	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 371.5 (nM), Ref: 26498393
TCMC811	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 52.5 (nM), Ref: 26498393
TCMC1496	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT164	Cyclooxygenase-1	Homo sapiens	Ki: 4000 (nM), Ref: 24088053
TCMC847	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394
TCMC847	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394
TCMC847	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 7870 (nM), Ref: 20185318
TCMC847	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6420 (nM), Ref: 20185318
TCMC847	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7330 (nM), Ref: 20185318
TCMC847	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9080 (nM), Ref: 20185318
TCMC847	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6490 (nM), Ref: 20185318
TCMC847	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 10000 (nM), Ref: 20185318
TCMC847	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1610 (nM), Ref: 20185318
TCMC847	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2380 (nM), Ref: 20185318
TCMC847	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3060 (nM), Ref: 19476336
TCMC847	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794
TCMC847	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 24.26 (nM), Ref: 23375794
TCMC847	TCMT295	Matrix metalloproteinase-1	Homo sapiens	IC50: 238.91 (nM), Ref: 23375794
TCMC847	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 8500 (nM), Ref: 26197161
TCMC1892	TCMT508	Tyrosine-protein kinase SYK	Homo sapiens	IC50: 10000 (nM), Ref: 23917087
TCMC2201	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8700 (nM), Ref: 21332115
TCMC1873	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 1840 (nM), Ref: 15828829 Ki: 1840 (nM), Ref: 21733699
TCMC1873	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 5270 (nM), Ref: 15828829 Ki: 5270 (nM), Ref: 21733699
TCMC1611	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1611	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897	TCMT223	Aldose reductase	Homo sapiens	IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024
TCMC897	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 7900 (nM), Ref: 22236472
TCMC1320	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 2786 (nM), Ref: 20696580
TCMC1320	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 511 (nM), Ref: 20696580
TCMC1320	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 102.1 (nM), Ref: 26498393
TCMC1320	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3.3 (nM), Ref: 26498393
TCMC1320	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 454.1 (nM), Ref: 26498393
TCMC1148	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 800 (nM), Ref: 22668600
TCMC1148	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 490 (nM), Ref: 22668600
TCMC1148	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 610 (nM), Ref: 22668600
TCMC1148	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 850 (nM), Ref: 22668600
TCMC1148	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 710 (nM), Ref: 22668600
TCMC1148	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 320 (nM), Ref: 22668600
TCMC1832	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC261	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 6950 (nM), Ref: 26900660
TCMC1237	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7300 (nM), Ref: 22668600
TCMC1237	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6600 (nM), Ref: 22668600
TCMC1237	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 4100 (nM), Ref: 22668600
TCMC1237	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4200 (nM), Ref: 22668600
TCMC2041	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9594.4 (nM), Ref: 26498393
TCMC2041	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 66.6 (nM), Ref: 26498393
TCMC2041	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 71.4 (nM), Ref: 26498393
TCMC2041	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 39.8 (nM), Ref: 26498393
TCMC1236	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref:
TCMC1236	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref:
TCMC1236	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 10 (nM), Ref: 17482813
TCMC1236	TCMT910	Estrogen-related receptor beta	Homo sapiens	IC50: 395 (nM), Ref: 17482813
TCMC1236	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 2210 (nM), Ref: 18533708
TCMC1236	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 340 (nM), Ref: 20853847
TCMC1236	TCMT289	Thromboxane-A synthase	Homo sapiens	IC50: 7720 (nM), Ref:
TCMC273	TCMT332	Amine oxidase, copper containing	Homo sapiens	IC50: 4100 (nM), Ref: 23664164
TCMC1183	TCMT247	Alpha-2a adrenergic receptor	Homo sapiens	Ki: 6.31 (nM), Ref: 11262089
TCMC1183	TCMT307	HERG	Homo sapiens	IC50: 1513.56 (nM), Ref: 12873512 IC50: 1513.56 (nM), Ref: 18448342 IC50: 3100 (nM), Ref: 20637635 IC50: 457.09 (nM), Ref: 21185626 IC50: 10 (nM), Ref: 23919353
TCMC1183	TCMT633	Serotonin transporter	Homo sapiens	Ki: 48 (nM), Ref: 16220969 Ki: 0.72 (nM), Ref: 16162005 IC50: 39.4 (nM), Ref: 16854086 IC50: 16 (nM), Ref: 16750363 IC50: 16 (nM), Ref: 16750359 Ki: 2 (nM), Ref: 17107798 Ki: 2.2 (nM), Ref: 17616397 Ki: 2.2 (nM), Ref: 17127059 Ki: 2.2 (nM), Ref: 17307358 IC50: 47 (nM), Ref: 18667309 Ki: 1.1 (nM), Ref: 19014888 IC50: 7 (nM), Ref: 19014888 IC50: 47 (nM), Ref: 18550369 IC50: 9.4 (nM), Ref: 18557608 IC50: 39.4 (nM), Ref: 18834188 IC50: 10 (nM), Ref: 18771916 IC50: 10 (nM), Ref: 19329313 IC50: 9.4 (nM), Ref: 18951020 Ki: 1.1 (nM), Ref: 19256502 IC50: 7.3 (nM), Ref: 19256502 IC50: 9.4 (nM), Ref: 19722525 IC50: 9.4 (nM), Ref: 19713106 IC50: 9.4 (nM), Ref: 19632110 IC50: 2.5 (nM), Ref: 20034793 IC50: 9.4 (nM), Ref: 20131864 IC50: 9.4 (nM), Ref: 20378347 IC50: 9.4 (nM), Ref: 20462211 IC50: 3.1 (nM), Ref: 20724153 IC50: 5.2 (nM), Ref: 21093273 IC50: 5.012 (nM), Ref: 21310612 IC50: 9.4 (nM), Ref: 21916421 Ki: 98 (nM), Ref: 23602445 IC50: 281.84 (nM), Ref: 23602445 Ki: 1.4 (nM), Ref: 23403082 IC50: 8.6 (nM), Ref: 23403082 IC50: 7.2 (nM), Ref: 24012181 IC50: 150 (nM), Ref: 24974340 IC50: 150 (nM), Ref: 25221656 IC50: 4410 (nM), Ref: 25221656
TCMC1183	TCMT634	Norepinephrine transporter	Homo sapiens	Ki: 2000 (nM), Ref: 16220969 Ki: 440 (nM), Ref: 16162005 IC50: 5200 (nM), Ref: 16750363 IC50: 5200 (nM), Ref: 16750359 IC50: 2000 (nM), Ref: 18667309 Ki: 1560 (nM), Ref: 19014888 IC50: 1020 (nM), Ref: 19014888 IC50: 2000 (nM), Ref: 18550369 IC50: 563 (nM), Ref: 18771916 IC50: 563 (nM), Ref: 19329313 Ki: 1560 (nM), Ref: 19256502 IC50: 1020 (nM), Ref: 19256502 Ki: 1394 (nM), Ref: 23602445 IC50: 6309.57 (nM), Ref: 23602445 IC50: 4410 (nM), Ref: 24974340
TCMC1183	TCMT635	Dopamine transporter	Homo sapiens	Ki: 6000 (nM), Ref: 16220969 Ki: 1900 (nM), Ref: 16162005 IC50: 4400 (nM), Ref: 16750363 IC50: 4400 (nM), Ref: 16750359 IC50: 6000 (nM), Ref: 18667309 Ki: 6670 (nM), Ref: 19014888 IC50: 6000 (nM), Ref: 18550369 Ki: 6670 (nM), Ref: 19256502 Ki: 3764 (nM), Ref: 23602445 IC50: 9120.11 (nM), Ref: 23602445
TCMC1183	TCMT242	Histamine H3 receptor	Homo sapiens	Ki: 7300 (nM), Ref: 17107798 Ki: 7300 (nM), Ref: 17616397 Ki: 7300 (nM), Ref: 17127059 Ki: 7300 (nM), Ref: 17307358
TCMC1183	TCMT31	Cytochrome P450 2C19	Homo sapiens	IC50: 40 (nM), Ref: 26355532
TCMC90	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2400 (nM), Ref: 14592472
TCMC1694	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 2020 (nM), Ref: 10879539 Ki: 1760 (nM), Ref: 16872140
TCMC2209	TCMT597	Solute carrier family 28 member 3	Homo sapiens	Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705
TCMC2209	TCMT710	Sodium/nucleoside cotransporter 1	Homo sapiens	Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705
TCMC1691	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 4720 (nM), Ref: 12027740
TCMC1693	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 4580 (nM), Ref: 20438092
TCMC1133	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030
TCMC1133	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030
TCMC1689	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 8680 (nM), Ref: 15332848
TCMC1133	TCMT187	Androgen Receptor	Homo sapiens	IC50: 19.1 (nM), Ref: 16309907
TCMC1133	TCMT99	Testis-specific androgen-binding protein	Homo sapiens	IC50: 50 (nM), Ref: 17149875
TCMC1133	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346
TCMC1133	TCMT910	Estrogen-related receptor beta	Homo sapiens	IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346
TCMC1133	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261
TCMC1133	TCMT974	G-protein coupled estrogen receptor 1	Homo sapiens	Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A
TCMC710	TCMT249	Cyclin-dependent kinase 6	Homo sapiens	IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554
TCMC710	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 710 (nM), Ref: 18533708
TCMC710	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 800 (nM), Ref: 19414254
TCMC710	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5200 (nM), Ref: 19592245
TCMC710	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 795 (nM), Ref: 20696580
TCMC710	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 427 (nM), Ref: 20696580
TCMC710	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC710	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1450 (nM), Ref: 23411073
TCMC710	TCMT128	Tankyrase-2	Homo sapiens	IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272
TCMC710	TCMT129	Tankyrase-1	Homo sapiens	IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272
TCMC710	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844
TCMC710	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431
TCMC1053	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 1950 (nM), Ref: 23286284 IC50: 1000 (nM), Ref: 24900610 Ki: 600 (nM), Ref: 24900610
TCMC1053	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 1830 (nM), Ref: 23286284 Ki: 118 (nM), Ref: 23286284
TCMC1053	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 398 (nM), Ref: 23286284
TCMC1053	TCMT171	Protein-tyrosine phosphatase 1C	Homo sapiens	IC50: 3670 (nM), Ref: 23957426
TCMC1053	TCMT233	Protein-tyrosine phosphatase 2C	Homo sapiens	IC50: 3940 (nM), Ref: 23957426
TCMC1961	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 600 (nM), Ref: 16248836
TCMC1961	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 6480 (nM), Ref: 23746477
TCMC2216	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168
TCMC2216	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 1900 (nM), Ref: 20100662
TCMC2216	TCMT102	Low molecular weight phosphotyrosine protein phosphatase	Homo sapiens	IC50: 7200 (nM), Ref: 21453996
TCMC2216	TCMT103	Receptor-type tyrosine-protein phosphatase F (LAR)	Homo sapiens	IC50: 3800 (nM), Ref: 21453996
TCMC2216	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086
TCMC2216	TCMT190	T-cell protein-tyrosine phosphatase	Homo sapiens	IC50: 2400 (nM), Ref: 23387824
TCMC2216	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616
TCMC1403	TCMT223	Aldose reductase	Homo sapiens	IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC878	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2420 (nM), Ref: 20674354
TCMC878	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1840 (nM), Ref: 20674354
TCMC878	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 3580 (nM), Ref: 20674354
TCMC878	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4900 (nM), Ref: 20674354
TCMC878	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4210 (nM), Ref: 20674354
TCMC878	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4020 (nM), Ref: 20674354
TCMC878	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 4910 (nM), Ref: 20674354
TCMC878	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 450 (nM), Ref: 20674354
TCMC878	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5030 (nM), Ref: 20674354
TCMC878	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4720 (nM), Ref: 20674354
TCMC1834	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9060 (nM), Ref: 21402476
TCMC1834	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8030 (nM), Ref: 21402476
TCMC770	TCMT588	D-amino-acid oxidase	Homo sapiens	Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755
TCMC1343	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385
TCMC1343	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7800 (nM), Ref: 18579385
TCMC1343	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8200 (nM), Ref: 18579385