Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
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Ingredient ID & Structure	Target ID	Target Name	Target Organism	Activity Records & Reference
TCMC1211	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 270 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 270 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 750 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 2200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC486	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 9500 (nM), Ref: 18579385
TCMC1173	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394
TCMC1173	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394
TCMC1173	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9870 (nM), Ref: 20185318
TCMC1173	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7410 (nM), Ref: 20185318
TCMC1173	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 8450 (nM), Ref: 20185318
TCMC1173	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7040 (nM), Ref: 20185318
TCMC1173	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2400 (nM), Ref: 20185318
TCMC1173	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2890 (nM), Ref: 20185318
TCMC609	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 10000 (nM), Ref: 18501600 Ki: 10000 (nM), Ref: 18579385 Ki: 10000 (nM), Ref: 26520662
TCMC609	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 6200 (nM), Ref: 18501600 Ki: 6200 (nM), Ref: 18579385 Ki: 6200 (nM), Ref: 26520662
TCMC609	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4100 (nM), Ref: 18579385
TCMC609	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 9100 (nM), Ref: 18579385
TCMC609	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7100 (nM), Ref: 18579385
TCMC609	TCMT216	Myoglobin	Homo sapiens	IC50: 2300 (nM), Ref: 24482730
TCMC337	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9670 (nM), Ref: 21282059
TCMC337	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1020 (nM), Ref: 21282059
TCMC337	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9070 (nM), Ref: 21282059
TCMC337	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8230 (nM), Ref: 21282059
TCMC337	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 550 (nM), Ref: 22668600
TCMC337	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3220 (nM), Ref: 22668600
TCMC2051	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 8710 (nM), Ref: 22892213
TCMC2051	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4050 (nM), Ref: 22892213
TCMC2051	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 960 (nM), Ref: 22892213
TCMC761	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 3920 (nM), Ref: 15658857
TCMC678	TCMT269	Prostanoid IP receptor	Homo sapiens	IC50: 1400 (nM), Ref: 10.1016/0960-894X(95)00168-S Ki: 150 (nM), Ref: 11454474
TCMC903	TCMT175	G-protein coupled bile acid receptor 1	Homo sapiens	IC50: 6000 (nM), Ref: 20801037
TCMC948	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394
TCMC948	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394
TCMC948	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5330 (nM), Ref: 20185318
TCMC948	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 5230 (nM), Ref: 20185318
TCMC948	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6720 (nM), Ref: 20185318
TCMC948	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7760 (nM), Ref: 20185318
TCMC948	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 5960 (nM), Ref: 20185318
TCMC948	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9600 (nM), Ref: 20185318
TCMC948	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7570 (nM), Ref: 20185318
TCMC948	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 980 (nM), Ref: 20185318
TCMC948	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1070 (nM), Ref: 20185318
TCMC948	TCMT223	Aldose reductase	Homo sapiens	IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1447	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 3000 (nM), Ref: 18565755 IC50: 2600 (nM), Ref: 18565755
TCMC364	TCMT115	Cannabinoid CB1 receptor	Homo sapiens	Ki: 480 (nM), Ref: 21675776 Ki: 470 (nM), Ref: 22044209
TCMC364	TCMT114	Cannabinoid CB2 receptor	Homo sapiens	Ki: 1300 (nM), Ref: 21675776 Ki: 1400 (nM), Ref: 22044209 Ki: 1400 (nM), Ref: 23865723
TCMC1495	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668
TCMC1495	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668
TCMC1495	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC37	TCMT308	Oxoeicosanoid receptor 1	Homo sapiens	IC50: 2000 (nM), Ref: 24351031
TCMC715	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC88	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 3400 (nM), Ref: 11678652
TCMC555	TCMT37	Serotonin 2a (5-HT2a) receptor	Homo sapiens	Ki: 15 (nM), Ref: 16392816
TCMC555	TCMT313	Serotonin 2b (5-HT2b) receptor	Homo sapiens	Ki: 52 (nM), Ref: 16392816
TCMC555	TCMT314	Serotonin 2c (5-HT2c) receptor	Homo sapiens	Ki: 42 (nM), Ref: 16392816
TCMC555	TCMT315	Serotonin 6 (5-HT6) receptor	Homo sapiens	Ki: 13 (nM), Ref: 16945532 Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
TCMC555	TCMT316	Melatonin receptor 1A	Homo sapiens	Ki: 210 (nM), Ref: 26023814
TCMC555	TCMT317	Melatonin receptor 1B	Homo sapiens	Ki: 16 (nM), Ref: 26023814
TCMC820	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5900 (nM), Ref: 23768907
TCMC2099	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 10 (nM), Ref: 20590092
TCMC2099	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 840 (nM), Ref: 20590092
TCMC2099	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 830 (nM), Ref: 20590092
TCMC2099	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 990 (nM), Ref: 20590092
TCMC2099	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 710 (nM), Ref: 20590092
TCMC2099	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 860 (nM), Ref: 20590092
TCMC1098	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 240 (nM), Ref: 16412638
TCMC1098	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 12 (nM), Ref: 16412638
TCMC2195	TCMT315	Serotonin 6 (5-HT6) receptor	Homo sapiens	Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
TCMC2195	TCMT335	Myeloperoxidase	Homo sapiens	IC50: 770 (nM), Ref: 23581551
TCMC2195	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 1700 (nM), Ref: 22696418
TCMC693	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 210 (nM), Ref: 16309907 IC50: 180 (nM), Ref: 17890084
TCMC693	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 10 (nM), Ref: 16309907 IC50: 9.9 (nM), Ref: 17890084
TCMC693	TCMT187	Androgen Receptor	Homo sapiens	IC50: 212 (nM), Ref: 16309907
TCMC424	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 550 (nM), Ref: 21282059
TCMC424	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 510 (nM), Ref: 21282059
TCMC424	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4410 (nM), Ref: 21282059
TCMC424	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 3670 (nM), Ref: 21282059
TCMC424	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 650 (nM), Ref: 22668600
TCMC424	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7170 (nM), Ref: 22668600
TCMC1139	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 2 (nM), Ref: 16722623
TCMC1139	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 8.1 (nM), Ref: 16722623
TCMC1139	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 570 (nM), Ref: 20853847 Ki: 3600 (nM), Ref: 22996261 Ki: 430 (nM), Ref: 22996261
TCMC1139	TCMT218	Cytochrome P450 2B6	Homo sapiens	Ki: 800 (nM), Ref: 16248836 Ki: 900 (nM), Ref: 16248836
TCMC1139	TCMT309	Solute carrier family 22 member 2	Homo sapiens	IC50: 2200 (nM), Ref: 23241029
TCMC1139	TCMT348	Sulfotransferase 1A1	Homo sapiens	IC50: 20 (nM), Ref: 22593037 Ki: 19 (nM), Ref: 22593037 Ki: 8.9 (nM), Ref: 22593037 Ki: 14.9 (nM), Ref: 22593037
TCMC1139	TCMT349	Nuclear receptor subfamily 1 group I member 3	Homo sapiens	IC50: 3000 (nM), Ref: 26717202
TCMC505	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 4880 (nM), Ref: 15658857
TCMC2037	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662
TCMC2037	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662
TCMC2037	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8800 (nM), Ref: 18579385
TCMC619	TCMT293	Muscarinic acetylcholine receptor M2	Homo sapiens	Ki: 158.49 (nM), Ref: 18077164
TCMC619	TCMT291	Muscarinic acetylcholine receptor M3	Homo sapiens	Ki: 7079.46 (nM), Ref: 18077164
TCMC619	TCMT551	Muscarinic acetylcholine receptor M4	Homo sapiens	Ki: 8511.38 (nM), Ref: 18077164
TCMC619	TCMT290	Muscarinic acetylcholine receptor M5	Homo sapiens	Ki: 9772.37 (nM), Ref: 18077164
TCMC1871	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056
TCMC1871	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662
TCMC1871	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455
TCMC1871	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455
TCMC1871	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662
TCMC743	TCMT302	HMG-CoA reductase	Homo sapiens	IC50: 6 (nM), Ref: 15686906 IC50: 12.9 (nM), Ref: 23570542
TCMC743	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 5100 (nM), Ref: 21256005
TCMC743	TCMT278	Solute carrier organic anion transporter family member 1B1	Homo sapiens	IC50: 600 (nM), Ref: 22587986 IC50: 800 (nM), Ref: 22587986 IC50: 1600 (nM), Ref: 22587986
TCMC619	TCMT241	Neuronal acetylcholine receptor protein alpha-7 subunit	Homo sapiens	Ki: 7943.28 (nM), Ref: 21920761
TCMC351	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	Ki: 10 (nM), Ref: 10.1039/C3MD00005B
TCMC1464	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 3900 (nM), Ref: 18565755 IC50: 8400 (nM), Ref: 18565755
TCMC2119	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9140 (nM), Ref: 20185318
TCMC2119	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9010 (nM), Ref: 20185318
TCMC2119	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8200 (nM), Ref: 20185318
TCMC2119	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7810 (nM), Ref: 20185318
TCMC2119	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7550 (nM), Ref: 20185318
TCMC2119	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6340 (nM), Ref: 20185318
TCMC2119	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8580 (nM), Ref: 20185318
TCMC2119	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3190 (nM), Ref: 20185318
TCMC2119	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4150 (nM), Ref: 20185318
TCMC1731	TCMT167	Aldo-keto-reductase family 1 member C3	Homo sapiens	IC50: 480 (nM), Ref: 16183274 IC50: 1100 (nM), Ref: 22877157
TCMC1731	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 211 (nM), Ref:
TCMC1330	TCMT246	Histamine H4 receptor	Homo sapiens	Ki: 14.45 (nM), Ref: 14640553 Ki: 7.943 (nM), Ref: 15454206 Ki: 12.02 (nM), Ref: 18357976 Ki: 13.4 (nM), Ref: 18459760 Ki: 12.02 (nM), Ref: 20192225 Ki: 60 (nM), Ref: 20452213 Ki: 7.943 (nM), Ref: 21044842 Ki: 12.59 (nM), Ref: 21044842 Ki: 12.02 (nM), Ref: 21348462 Ki: 15.85 (nM), Ref: 22003888 Ki: 9 (nM), Ref: 22153663 Ki: 19.95 (nM), Ref: 10.1039/C2MD20212C Ki: 4.8 (nM), Ref: 25993395 Ki: 8 (nM), Ref: 25993395 Ki: 15.85 (nM), Ref: 10.1039/C5MD00022J
TCMC1330	TCMT242	Histamine H3 receptor	Homo sapiens	Ki: 5.2 (nM), Ref: 20384344 Ki: 10 (nM), Ref: 21044842 Ki: 11.75 (nM), Ref: 21348462 Ki: 6.31 (nM), Ref: 22003888 Ki: 16 (nM), Ref: 25993395
TCMC1330	TCMT245	Histamine H2 receptor	Homo sapiens	Ki: 5000 (nM), Ref: 25993395
TCMC1330	TCMT244	Histamine H1 receptor	Homo sapiens	Ki: 6000 (nM), Ref: 25993395
TCMC1293	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2940 (nM), Ref: 19231207
TCMC1061	TCMT582	Prostanoid EP1 receptor	Homo sapiens	Ki: 9.1 (nM), Ref: 17531488 Ki: 9.1 (nM), Ref: 18039575 Ki: 18 (nM), Ref: 24279689
TCMC1061	TCMT583	Prostanoid EP2 receptor	Homo sapiens	Ki: 4.9 (nM), Ref: 17531488 Ki: 4.9 (nM), Ref: 17931866 Ki: 4.9 (nM), Ref: 18039575 IC50: 2.2 (nM), Ref: 23582449 Ki: 1.7 (nM), Ref: 23466604 IC50: 3.3 (nM), Ref: 23466604 Ki: 38 (nM), Ref: 24279689 IC50: 2.6 (nM), Ref: 26988801
TCMC1061	TCMT584	Prostanoid EP3 receptor	Homo sapiens	Ki: 0.33 (nM), Ref: 17531488 Ki: 0.33 (nM), Ref: 18039575 Ki: 5 (nM), Ref: 24279689
TCMC1061	TCMT585	Prostanoid EP4 receptor	Homo sapiens	Ki: 0.79 (nM), Ref: 17531488 Ki: 0.79 (nM), Ref: 17931866 Ki: 0.79 (nM), Ref: 18039575 Ki: 1.9 (nM), Ref: 18983139 IC50: 3.8 (nM), Ref: 18983139 Ki: 0.45 (nM), Ref: 23403082 IC50: 1.1 (nM), Ref: 23403082 Ki: 0.17 (nM), Ref: 23466604 IC50: 0.45 (nM), Ref: 23466604 Ki: 3.1 (nM), Ref: 24279689
TCMC1061	TCMT269	Prostanoid IP receptor	Homo sapiens	IC50: 260 (nM), Ref: 24279689
TCMC1429	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2700 (nM), Ref: 17378609
TCMC1429	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 1050 (nM), Ref: 18533708
TCMC1429	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 360 (nM), Ref: 18533708
TCMC1429	TCMT187	Androgen Receptor	Homo sapiens	IC50: 9700 (nM), Ref: 19592245
TCMC1429	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 716 (nM), Ref: 20696580
TCMC1429	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 632 (nM), Ref: 20696580
TCMC1429	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 47 (nM), Ref: 20696580
TCMC1429	TCMT223	Aldose reductase	Homo sapiens	IC50: 10000 (nM), Ref: 22261024
TCMC1429	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 2320 (nM), Ref: 23411073
TCMC1429	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 9640 (nM), Ref: 23656512
TCMC1429	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 10000 (nM), Ref: 26322379
TCMC1429	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9525.7 (nM), Ref: 26498393
TCMC1429	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 25 (nM), Ref: 26498393
TCMC1429	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 145.9 (nM), Ref: 26498393
TCMC1429	TCMT159	Tyrosinase	Homo sapiens	IC50: 1000 (nM), Ref: 26841168
TCMC1364	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 4000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364	TCMT308	Oxoeicosanoid receptor 1	Homo sapiens	IC50: 2000 (nM), Ref: 24351031
TCMC1411	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1261 (nM), Ref: 20696580
TCMC1411	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 56 (nM), Ref: 20696580
TCMC1411	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 17 (nM), Ref: 20696580
TCMC1411	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 212.9 (nM), Ref: 26498393
TCMC1411	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.4 (nM), Ref: 26498393
TCMC1411	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 54.9 (nM), Ref: 26498393 Ki: 220 (nM), Ref: 26498393
TCMC1411	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 440 (nM), Ref: 26498393
TCMC895	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 7630 (nM), Ref: 20053563
TCMC895	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 7630 (nM), Ref: 20053563
TCMC895	TCMT318	Putative hexokinase HKDC1	Homo sapiens	IC50: 8990 (nM), Ref:
TCMC895	TCMT599	Ubiquitin-conjugating enzyme E2 N	Homo sapiens	IC50: 3012 (nM), Ref: IC50: 2197 (nM), Ref:
TCMC895	TCMT608	Solute carrier family 22 member 3	Homo sapiens	IC50: 410 (nM), Ref: 23241029
TCMC895	TCMT213	Solute carrier family 22 member 1	Homo sapiens	IC50: 210 (nM), Ref: 23241029
TCMC895	TCMT309	Solute carrier family 22 member 2	Homo sapiens	IC50: 400 (nM), Ref: 23241029
TCMC895	TCMT310	Multidrug and toxin extrusion protein 2	Homo sapiens	IC50: 500 (nM), Ref: 23241029
TCMC895	TCMT311	Multidrug and toxin extrusion protein 1	Homo sapiens	IC50: 700 (nM), Ref: 23241029
TCMC13	TCMT23	Alkaline phosphatase, tissue-nonspecific isozyme	Homo sapiens	IC50: 407 (nM), Ref:
TCMC2148	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 3200 (nM), Ref: 24920381
TCMC633	TCMT620	Heat shock cognate 71 kDa protein	Homo sapiens	IC50: 280 (nM), Ref:
TCMC1582	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 4100 (nM), Ref: 22668600
TCMC1582	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 820 (nM), Ref: 22668600
TCMC1582	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5500 (nM), Ref: 22668600
TCMC1582	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 780 (nM), Ref: 22668600
TCMC1582	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3400 (nM), Ref: 22668600
TCMC1582	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2600 (nM), Ref: 22668600
TCMC1112	TCMT203	Glucose-6-phosphate 1-dehydrogenase	Homo sapiens	Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561
TCMC1470	TCMT630	Cysteinyl leukotriene receptor 1	Homo sapiens	IC50: 7 (nM), Ref: 20875743 Ki: 0.29 (nM), Ref: 23403082 IC50: 0.7 (nM), Ref: 23403082
TCMC2025	TCMT61	Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens	IC50: 2025.72 (nM), Ref:
TCMC1584	TCMT571	Adenosine A2b receptor	Homo sapiens	Ki: 8200 (nM), Ref: 15084123
TCMC1584	TCMT112	Adenosine A3 receptor	Homo sapiens	Ki: 680 (nM), Ref: 15084123
TCMC1480	TCMT107	Glutamate receptor ionotropic kainate 2	Homo sapiens	Ki: 1106 (nM), Ref: 10821708
TCMC1480	TCMT108	Glutamate receptor ionotropic, AMPA 1	Homo sapiens	Ki: 1360 (nM), Ref: 9357531
TCMC1480	TCMT109	Glutamate receptor ionotropic, AMPA 2	Homo sapiens	Ki: 940 (nM), Ref: 9357531
TCMC1480	TCMT110	Glutamate receptor ionotropic, AMPA 4	Homo sapiens	Ki: 868 (nM), Ref: 9357531
TCMC1480	TCMT111	Glutamate receptor ionotropic kainate 5	Homo sapiens	Ki: 701 (nM), Ref: 9357531
TCMC1480	TCMT660	Metabotropic glutamate receptor 8	Homo sapiens	IC50: 5.7 (nM), Ref: 15603952
TCMC1480	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 613 (nM), Ref: 16250647
TCMC1480	TCMT653	Metabotropic glutamate receptor 1	Homo sapiens	Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT654	Metabotropic glutamate receptor 5	Homo sapiens	Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT657	Metabotropic glutamate receptor 4	Homo sapiens	Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT655	Metabotropic glutamate receptor 2	Homo sapiens	Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H
TCMC1480	TCMT664	Excitatory amino acid transporter 3	Homo sapiens	Ki: 51 (nM), Ref: 18578477
TCMC1480	TCMT656	Metabotropic glutamate receptor 3	Homo sapiens	Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H
TCMC694	TCMT230	Estradiol 17-beta-dehydrogenase 3	Homo sapiens	IC50: 758 (nM), Ref: 11086723 IC50: 758 (nM), Ref: 16078844
TCMC694	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 20 (nM), Ref: 8035427 Ki: 35 (nM), Ref: 26469743
TCMC949	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8900 (nM), Ref: 19911821
TCMC949	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 48 (nM), Ref: 19911821
TCMC949	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9100 (nM), Ref: 19911821
TCMC949	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3300 (nM), Ref: 19911821
TCMC949	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 2000 (nM), Ref: 19911821
TCMC949	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 5200 (nM), Ref: 19911821
TCMC949	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9400 (nM), Ref: 19911821
TCMC949	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 6800 (nM), Ref: 19911821
TCMC949	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 5600 (nM), Ref: 19911821
TCMC949	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270
TCMC949	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270
TCMC1786	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900
TCMC1786	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086
TCMC1786	TCMT190	T-cell protein-tyrosine phosphatase	Homo sapiens	IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900
TCMC1786	TCMT563	Dual specificity phosphatase Cdc25B	Homo sapiens	IC50: 980 (nM), Ref: 25497963
TCMC845	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 630 (nM), Ref: 19231207
TCMC662	TCMT683	Macrophage migration inhibitory factor	Homo sapiens	IC50: 250 (nM), Ref: 25743213 IC50: 1100 (nM), Ref: 25743213
TCMC1083	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867
TCMC1083	TCMT651	Dopamine D3 receptor	Homo sapiens	Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329
TCMC1083	TCMT635	Dopamine transporter	Homo sapiens	Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523
TCMC1083	TCMT634	Norepinephrine transporter	Homo sapiens	IC50: 6.63 (nM), Ref: 14592523
TCMC1083	TCMT648	Dopamine D4 receptor	Homo sapiens	Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965
TCMC1083	TCMT316	Melatonin receptor 1A	Homo sapiens	Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083	TCMT317	Melatonin receptor 1B	Homo sapiens	Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083	TCMT27	Dopamine D1 receptor	Homo sapiens	Ki: 4470 (nM), Ref: 23134120
TCMC1083	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1396	TCMT689	Protein-glutamine gamma-glutamyltransferase	Homo sapiens	IC50: 8000 (nM), Ref: 21215619
TCMC837	TCMT690	Histone deacetylase 3	Homo sapiens	IC50: 9000 (nM), Ref: 21874153
TCMC256	TCMT203	Glucose-6-phosphate 1-dehydrogenase	Homo sapiens	IC50: 4300 (nM), Ref: 22506561
TCMC1930	TCMT203	Glucose-6-phosphate 1-dehydrogenase	Homo sapiens	Ki: 8900 (nM), Ref: 19231202 Ki: 6200 (nM), Ref: 19231202
TCMC1044	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1400 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 4300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 2400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1044	TCMT308	Oxoeicosanoid receptor 1	Homo sapiens	IC50: 2000 (nM), Ref: 24351031
TCMC287	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 3200 (nM), Ref: 15916432
TCMC632	TCMT597	Solute carrier family 28 member 3	Homo sapiens	Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705
TCMC632	TCMT709	Sodium/nucleoside cotransporter 2	Homo sapiens	Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT710	Sodium/nucleoside cotransporter 1	Homo sapiens	Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT296	Adenosine A1 receptor	Homo sapiens	IC50: 2.344 (nM), Ref: 26756468
TCMC632	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 1.148 (nM), Ref: 26756468
TCMC1956	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1080 (nM), Ref: 21282059
TCMC1956	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 470 (nM), Ref: 21282059
TCMC1956	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4450 (nM), Ref: 21282059
TCMC1956	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4090 (nM), Ref: 21282059
TCMC1956	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439
TCMC1956	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 2450 (nM), Ref: 22687439
TCMC1956	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 690 (nM), Ref: 22668600
TCMC1956	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7870 (nM), Ref: 22668600
TCMC2025	TCMT295	Matrix metalloproteinase-1	Homo sapiens	IC50: 5600 (nM), Ref: 23353736
TCMC43	TCMT301	Prostaglandin E synthase	Homo sapiens	IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43	TCMT565	Histone acetyltransferase p300	Homo sapiens	IC50: 6500 (nM), Ref: 26701186
TCMC43	TCMT208	Monoamine oxidase A	Homo sapiens	Ki: 710 (nM), Ref: 26819666
TCMC43	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601
TCMC2142	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 600 (nM), Ref: 6827528
TCMC2142	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 10000 (nM), Ref: 14552748
TCMC2142	TCMT187	Androgen Receptor	Homo sapiens	IC50: 3.9 (nM), Ref: 15456242 IC50: 2.7 (nM), Ref: 16309907 IC50: 4.571 (nM), Ref: 22746350 IC50: 4.17 (nM), Ref: 25646649 IC50: 4.27 (nM), Ref: 25646649
TCMC2142	TCMT99	Testis-specific androgen-binding protein	Homo sapiens	IC50: 14 (nM), Ref: 17149875
TCMC2142	TCMT725	Voltage-gated L-type calcium channel alpha-1C subunit	Homo sapiens	IC50: 34 (nM), Ref: 22761000 IC50: 38.4 (nM), Ref: 22761000
TCMC963	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 500 (nM), Ref: 15357993 Ki: 500 (nM), Ref: 15454240 Ki: 500 (nM), Ref: 15501038 Ki: 500 (nM), Ref: 21208801 Ki: 500 (nM), Ref: 26525863 Ki: 500 (nM), Ref: 26853167 Ki: 500 (nM), Ref: 27283786
TCMC963	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4000 (nM), Ref: 15501038
TCMC1499	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 1 (nM), Ref: 18181565
TCMC1499	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 0 (nM), Ref: 17976864
TCMC1741	TCMT161	Hydroxycarboxylic acid receptor 2	Homo sapiens	IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085
TCMC1401	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 15 (nM), Ref: 21561086
TCMC1446	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 6300 (nM), Ref: 21641214
TCMC1758	TCMT247	Alpha-2a adrenergic receptor	Homo sapiens	Ki: 66 (nM), Ref: 8632424
TCMC1758	TCMT243	Alpha-2c adrenergic receptor	Homo sapiens	Ki: 63 (nM), Ref: 8632424
TCMC1758	TCMT559	Beta-2 adrenergic receptor	Homo sapiens	Ki: 3300 (nM), Ref: 27132867
TCMC1758	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 1300 (nM), Ref: 27132867
TCMC1609	TCMT44	Glyoxalase I	Homo sapiens	IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529
TCMC1609	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18778944
TCMC1609	TCMT737	DNA dC->dU-editing enzyme APOBEC-3G	Homo sapiens	IC50: 2390 (nM), Ref:
TCMC1609	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 2120 (nM), Ref: 24900447
TCMC1609	TCMT558	DNA topoisomerase II alpha	Homo sapiens	IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1690 (nM), Ref: 23411073
TCMC1609	TCMT2	Microtubule-associated protein tau	Homo sapiens	IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT740	PI3-kinase p110-gamma subunit	Homo sapiens	IC50: 4720 (nM), Ref: 25050878
TCMC1609	TCMT13	DNA-(apurinic or apyrimidinic site) lyase	Homo sapiens	IC50: 320 (nM), Ref: 25280182
TCMC1043	TCMT191	Signal transducer and activator of transcription 3	Homo sapiens	IC50: 1862 (nM), Ref:
TCMC1043	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	IC50: 2000 (nM), Ref: 24040486 IC50: 4000 (nM), Ref: 10.1039/C3MD00005B IC50: 4100 (nM), Ref: 24502334 IC50: 1980 (nM), Ref: 24502334
TCMC1043	TCMT744	Sodium/potassium-transporting ATPase alpha-1 chain	Homo sapiens	IC50: 290 (nM), Ref: 26122772
TCMC635	TCMT460	MAP kinase-activated protein kinase 2	Homo sapiens	IC50: 2800 (nM), Ref: 19919896 IC50: 6300 (nM), Ref: 19919896
TCMC635	TCMT721	Heat shock 70 kDa protein 1	Homo sapiens	IC50: 3370 (nM), Ref:
TCMC2025	TCMT359	Tyrosine-protein kinase FYN	Homo sapiens	IC50: 1300 (nM), Ref: 17315853 IC50: 3600 (nM), Ref: 17315853 Ki: 7500 (nM), Ref: 17315853
TCMC2031	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 7500 (nM), Ref: 16610779
TCMC1102	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 40 (nM), Ref: 19414254
TCMC1102	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2320 (nM), Ref: 20185318
TCMC1102	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2180 (nM), Ref: 20185318
TCMC1102	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9080 (nM), Ref: 20185318
TCMC1102	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7590 (nM), Ref: 20185318
TCMC1102	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7060 (nM), Ref: 20185318
TCMC1102	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213
TCMC1102	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9370 (nM), Ref: 20185318
TCMC1102	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 8910 (nM), Ref: 20185318
TCMC1102	TCMT753	Mothers against decapentaplegic homolog 3	Homo sapiens	IC50: 142 (nM), Ref:
TCMC1102	TCMT721	Heat shock 70 kDa protein 1	Homo sapiens	IC50: 760 (nM), Ref:
TCMC1102	TCMT189	Dual specificity protein phosphatase 3	Homo sapiens	IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102	TCMT223	Aldose reductase	Homo sapiens	IC50: 200 (nM), Ref: 22261024
TCMC1102	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 510 (nM), Ref: 22377675
TCMC1102	TCMT354	Serine/threonine-protein kinase Aurora-A	Homo sapiens	IC50: 2480 (nM), Ref: 22377675
TCMC1102	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 2500 (nM), Ref: 22377675
TCMC1102	TCMT626	Serine/threonine-protein kinase B-raf	Homo sapiens	IC50: 1760 (nM), Ref: 22377675
TCMC1102	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 690 (nM), Ref: 22377675
TCMC1102	TCMT418	Ephrin type-B receptor 4	Homo sapiens	IC50: 1830 (nM), Ref: 22377675
TCMC1102	TCMT704	Receptor protein-tyrosine kinase erbB-2	Homo sapiens	IC50: 3540 (nM), Ref: 22377675
TCMC1102	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 3110 (nM), Ref: 22377675
TCMC1102	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 250 (nM), Ref: 22377675
TCMC1102	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 800 (nM), Ref: 22377675
TCMC1102	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 790 (nM), Ref: 22377675
TCMC1102	TCMT457	Vascular endothelial growth factor receptor 3	Homo sapiens	IC50: 1540 (nM), Ref: 22377675
TCMC1102	TCMT377	Insulin receptor	Homo sapiens	IC50: 340 (nM), Ref: 22377675
TCMC1102	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 22377675
TCMC1102	TCMT536	Platelet-derived growth factor receptor beta	Homo sapiens	IC50: 1300 (nM), Ref: 22377675
TCMC1102	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT755	Serine/threonine-protein kinase PLK4	Homo sapiens	IC50: 2970 (nM), Ref: 22377675
TCMC1102	TCMT502	Tyrosine-protein kinase TIE-2	Homo sapiens	IC50: 260 (nM), Ref: 22377675
TCMC1102	TCMT756	Mitogen-activated protein kinase kinase kinase 8	Homo sapiens	IC50: 2370 (nM), Ref: 22377675
TCMC1102	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 100 (nM), Ref: 24900447
TCMC1102	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8150 (nM), Ref: 22892213
TCMC1102	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4240 (nM), Ref: 22892213
TCMC1102	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3900 (nM), Ref: 24835197
TCMC1743	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 4400 (nM), Ref: 15634016
TCMC1743	TCMT241	Neuronal acetylcholine receptor protein alpha-7 subunit	Homo sapiens	Ki: 7200 (nM), Ref: 15686879 Ki: 6300 (nM), Ref: 15908213 Ki: 630 (nM), Ref: 16171993 Ki: 10000 (nM), Ref: 17722904 Ki: 1000 (nM), Ref: 19331415 Ki: 1023.29 (nM), Ref: 20828128 Ki: 1000 (nM), Ref: 21920761 Ki: 1000 (nM), Ref: 22243960 Ki: 3000 (nM), Ref: 22793665 Ki: 3000 (nM), Ref: 23126648 Ki: 3800 (nM), Ref: 23561269 IC50: 7600 (nM), Ref: 23561269 Ki: 3000 (nM), Ref: 23692872
TCMC1743	TCMT552	Neuronal acetylcholine receptor subunit alpha-3	Homo sapiens	IC50: 45 (nM), Ref: 11312774
TCMC634	TCMT284	Fructose-1,6-bisphosphatase	Homo sapiens	IC50: 1000 (nM), Ref: 19348494 IC50: 440 (nM), Ref: 19969452 IC50: 140 (nM), Ref: 19969452 IC50: 9800 (nM), Ref: 20116906 IC50: 3200 (nM), Ref: 24530031 IC50: 1000 (nM), Ref: 10.1039/C0MD00269K IC50: 3200 (nM), Ref: 25461330
TCMC1982	TCMT239	Serine/threonine-protein kinase PIM1	Homo sapiens	IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302
TCMC1982	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208
TCMC1982	TCMT223	Aldose reductase	Homo sapiens	IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999
TCMC1982	TCMT44	Glyoxalase I	Homo sapiens	IC50: 3200 (nM), Ref: 18258440
TCMC1982	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 1540 (nM), Ref: 18533708
TCMC452	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2370 (nM), Ref: 21282059
TCMC452	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 600 (nM), Ref: 21282059
TCMC452	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4530 (nM), Ref: 21282059
TCMC452	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 3530 (nM), Ref: 21282059
TCMC452	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 3170 (nM), Ref: 21669522
TCMC1982	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7890 (nM), Ref: 20185318
TCMC1982	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8100 (nM), Ref: 20185318
TCMC1982	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2540 (nM), Ref: 20185318
TCMC1982	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2680 (nM), Ref: 20185318
TCMC1982	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6810 (nM), Ref: 20185318
TCMC1982	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6170 (nM), Ref: 20185318
TCMC1982	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4840 (nM), Ref: 20185318
TCMC1982	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 7000 (nM), Ref: 20185318
TCMC1982	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9390 (nM), Ref: 20185318
TCMC1982	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 5410 (nM), Ref: 20185318
TCMC1136	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 330 (nM), Ref: 16480268 IC50: 218 (nM), Ref: 18035543 IC50: 109 (nM), Ref: 19836949 Ki: 9500 (nM), Ref: 21413808
TCMC1136	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 31 (nM), Ref: 16610787
TCMC1136	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 29 (nM), Ref: 16610787 IC50: 96 (nM), Ref: 19836949
TCMC1982	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 12 (nM), Ref: 20413308
TCMC1136	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 2500 (nM), Ref: 26469743
TCMC1982	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583
TCMC1982	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1191 (nM), Ref: 20696580
TCMC1982	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 77 (nM), Ref: 20696580
TCMC1744	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 10000 (nM), Ref: 14552748 IC50: 5620 (nM), Ref: 23033255
TCMC1744	TCMT112	Adenosine A3 receptor	Homo sapiens	Ki: 8290 (nM), Ref: 8917655
TCMC1744	TCMT778	Voltage-gated potassium channel subunit Kv1.5	Homo sapiens	IC50: 6100 (nM), Ref: 19004630
TCMC1744	TCMT780	Voltage-gated L-type calcium channel alpha-1D subunit	Homo sapiens	IC50: 1350 (nM), Ref: 24754640
TCMC1744	TCMT725	Voltage-gated L-type calcium channel alpha-1C subunit	Homo sapiens	IC50: 22 (nM), Ref: 22761000 IC50: 55 (nM), Ref: 22761000
TCMC1744	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 2300 (nM), Ref: 23033255
TCMC1744	TCMT31	Cytochrome P450 2C19	Homo sapiens	IC50: 5420 (nM), Ref: 23033255
TCMC1744	TCMT87	Cytochrome P450 2C9	Homo sapiens	IC50: 4080 (nM), Ref: 23033255
TCMC1744	TCMT220	Cytochrome P450 2J2	Homo sapiens	IC50: 3060 (nM), Ref: 23033255
TCMC1744	TCMT407	Myosin light chain kinase, smooth muscle	Homo sapiens	IC50: 2020 (nM), Ref: 26385444
TCMC649	TCMT783	Mineralocorticoid receptor	Homo sapiens	IC50: 9.268 (nM), Ref: 20812681
TCMC1982	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 6680 (nM), Ref: 22658537
TCMC1982	TCMT320	Matrix metalloproteinase 3	Homo sapiens	IC50: 5570 (nM), Ref: 22658537
TCMC1982	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 1610 (nM), Ref: 22658537
TCMC1982	TCMT322	Matrix metalloproteinase 13	Homo sapiens	IC50: 8460 (nM), Ref: 22658537
TCMC1982	TCMT422	CaM kinase II beta	Homo sapiens	IC50: 3000 (nM), Ref: 21798748
TCMC2098	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1400 (nM), Ref: 20590092
TCMC2098	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1110 (nM), Ref: 20590092
TCMC2098	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 112 (nM), Ref: 20590092
TCMC2098	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 1220 (nM), Ref: 20590092
TCMC2098	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 1440 (nM), Ref: 20590092
TCMC2098	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 1410 (nM), Ref: 20590092
TCMC2098	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 1230 (nM), Ref: 20590092
TCMC2098	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 1370 (nM), Ref: 20590092
TCMC2098	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 1000 (nM), Ref: 20590092
TCMC339	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 10000 (nM), Ref: 15658857 IC50: 10000 (nM), Ref: 19110342
TCMC1982	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344
TCMC1982	TCMT784	Vasopressin V2 receptor	Homo sapiens	IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772
TCMC1982	TCMT785	Interleukin-8 receptor A	Homo sapiens	IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772
TCMC1982	TCMT786	C-C chemokine receptor type 4	Homo sapiens	IC50: 10000 (nM), Ref: 23437772
TCMC1982	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 590 (nM), Ref: 23411073
TCMC2183	TCMT241	Neuronal acetylcholine receptor protein alpha-7 subunit	Homo sapiens	IC50: 7000 (nM), Ref: 23713606
TCMC1982	TCMT601	Thrombin	Homo sapiens	IC50: 1500 (nM), Ref: 24610996
TCMC1982	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 280 (nM), Ref: 24328302
TCMC1982	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 120 (nM), Ref: 24328302
TCMC1982	TCMT791	Protein kinase N1	Homo sapiens	IC50: 5800 (nM), Ref: 24328302
TCMC1982	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 5750 (nM), Ref: 24328302
TCMC1982	TCMT462	Serine/threonine-protein kinase NEK6	Homo sapiens	IC50: 4230 (nM), Ref: 24328302
TCMC1982	TCMT445	Serine/threonine-protein kinase NEK2	Homo sapiens	IC50: 5730 (nM), Ref: 24328302
TCMC1982	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 24328302
TCMC1982	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 300 (nM), Ref: 24328302
TCMC1982	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 1200 (nM), Ref: 24328302
TCMC1982	TCMT388	Tyrosine-protein kinase receptor UFO	Homo sapiens	IC50: 960 (nM), Ref: 24328302
TCMC1982	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 910 (nM), Ref: 24328302
TCMC1982	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 5090 (nM), Ref: 24328302
TCMC1982	TCMT402	ALK tyrosine kinase receptor	Homo sapiens	IC50: 3320 (nM), Ref: 24328302
TCMC1982	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 5390 (nM), Ref: 24328302
TCMC1982	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124
TCMC1982	TCMT793	Liver glycogen phosphorylase	Homo sapiens	IC50: 4800 (nM), Ref: 25092521
TCMC1982	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 2110 (nM), Ref: 22328583
TCMC1982	TCMT217	Cytochrome P450 2C8	Homo sapiens	IC50: 1390 (nM), Ref: 22328583
TCMC1477	TCMT273	Bile acid receptor FXR	Homo sapiens	IC50: 7860 (nM), Ref: 23688559
TCMC1477	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 5600 (nM), Ref: 21030469 IC50: 4900 (nM), Ref: 21030469
TCMC1982	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 8900 (nM), Ref: 26322379
TCMC880	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9910 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 20185318 Ki: 9900 (nM), Ref: 22245047 Ki: 9900 (nM), Ref: 26073005 Ki: 9900 (nM), Ref: 26520662
TCMC880	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4200 (nM), Ref: 18579385 Ki: 4200 (nM), Ref: 20185318
TCMC880	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8900 (nM), Ref: 18579385 Ki: 8900 (nM), Ref: 20185318
TCMC916	TCMT161	Hydroxycarboxylic acid receptor 2	Homo sapiens	Ki: 4900 (nM), Ref: 21167710
TCMC2196	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 64 (nM), Ref: 22819942 IC50: 64 (nM), Ref: 23146282
TCMC2196	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 150 (nM), Ref: 22819942
TCMC2196	TCMT336	Indoleamine 2,3-dioxygenase	Homo sapiens	IC50: 53.7 (nM), Ref: 24099220 IC50: 7150 (nM), Ref: 24099220 Ki: 4810 (nM), Ref: 24099220
TCMC1824	TCMT232	P-glycoprotein 1	Homo sapiens	IC50: 2596 (nM), Ref: 23332369 IC50: 2600 (nM), Ref: 23895532
TCMC1824	TCMT801	Tubulin beta-3 chain	Homo sapiens	IC50: 9.2 (nM), Ref: 23332369 IC50: 7.7 (nM), Ref: 23895532
TCMC1824	TCMT277	Solute carrier organic anion transporter family member 1B3	Homo sapiens	Ki: 1800 (nM), Ref: 25618019 IC50: 260 (nM), Ref: 25618019
TCMC1824	TCMT278	Solute carrier organic anion transporter family member 1B1	Homo sapiens	Ki: 840 (nM), Ref: 25618019 IC50: 280 (nM), Ref: 25618019
TCMC1824	TCMT393	Proto-oncogene tyrosine-protein kinase MER	Homo sapiens	IC50: 4900 (nM), Ref: 27238842
TCMC2105	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC952	TCMT803	Hypoxanthine-guanine phosphoribosyltransferase	Homo sapiens	Ki: 5800 (nM), Ref: 19527031 Ki: 5800 (nM), Ref: 25915781
TCMC1155	TCMT230	Estradiol 17-beta-dehydrogenase 3	Homo sapiens	IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844
TCMC1597	TCMT807	Solute carrier family 22 member 12	Homo sapiens	IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024
TCMC1597	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 2927.18 (nM), Ref:
TCMC1597	TCMT61	Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens	IC50: 2988.26 (nM), Ref:
TCMC1597	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 1600 (nM), Ref: 24900447
TCMC1597	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 1600 (nM), Ref: 26322379
TCMC1597	TCMT283	Receptor-type tyrosine-protein phosphatase S	Homo sapiens	IC50: 4300 (nM), Ref: 26602279
TCMC1830	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 930 (nM), Ref: 15357969
TCMC1830	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 2600 (nM), Ref: 15357969
TCMC1830	TCMT808	Fatty acid binding protein epidermal	Homo sapiens	IC50: 1200 (nM), Ref: 15357969
TCMC1830	TCMT809	Fatty acid binding protein intestinal	Homo sapiens	IC50: 1700 (nM), Ref: 15357969
TCMC1830	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1830	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2063	TCMT646	Serotonin 5a (5-HT5a) receptor	Homo sapiens	Ki: 126 (nM), Ref: 12825922 IC50: 180 (nM), Ref: 18983139 Ki: 110 (nM), Ref: 18983139 IC50: 184 (nM), Ref: 18588282 Ki: 170 (nM), Ref: 21726069 IC50: 280 (nM), Ref: 23582449 Ki: 82 (nM), Ref: 23466604 IC50: 160 (nM), Ref: 23466604 IC50: 180 (nM), Ref: 26988801
TCMC2063	TCMT315	Serotonin 6 (5-HT6) receptor	Homo sapiens	Ki: 65 (nM), Ref: 12825922 Ki: 100 (nM), Ref: 15357994 IC50: 200 (nM), Ref: 18983139 Ki: 93 (nM), Ref: 18983139 IC50: 262 (nM), Ref: 18588282 IC50: 27.5 (nM), Ref: 20170099 Ki: 84 (nM), Ref: 21726069 Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8 IC50: 180 (nM), Ref: 23582449 Ki: 50 (nM), Ref: 23466604 IC50: 100 (nM), Ref: 23466604 Ki: 33 (nM), Ref: 24805037 Ki: 33 (nM), Ref: 25557493 IC50: 120 (nM), Ref: 26988801 Ki: 100 (nM), Ref: 26996373
TCMC2063	TCMT160	Serotonin 7 (5-HT7) receptor	Homo sapiens	Ki: 8.1 (nM), Ref: 12825922 IC50: 0.61 (nM), Ref: 18983139 Ki: 0.22 (nM), Ref: 18983139 IC50: 2.55 (nM), Ref: 12713409 IC50: 1.5 (nM), Ref: 18588282 Ki: 0.13 (nM), Ref: 21726069 IC50: 0.49 (nM), Ref: 23582449 Ki: 0.11 (nM), Ref: 23466604 IC50: 0.29 (nM), Ref: 23466604 Ki: 1.4 (nM), Ref: 24763360 Ki: 0.8 (nM), Ref: 24805037 Ki: 0.8 (nM), Ref: 25557493 IC50: 0.25 (nM), Ref: 26988801
TCMC2063	TCMT37	Serotonin 2a (5-HT2a) receptor	Homo sapiens	Ki: 14 (nM), Ref: 15081042 Ki: 8.2 (nM), Ref: 16392816 Ki: 14 (nM), Ref: 16257207 Ki: 120 (nM), Ref: 18468904 Ki: 160 (nM), Ref: 18468904 Ki: 130 (nM), Ref: 18468904 Ki: 150 (nM), Ref: 18468904 Ki: 320 (nM), Ref: 11975483 Ki: 690 (nM), Ref: 17067154 Ki: 323.59 (nM), Ref: 23301527 Ki: 320 (nM), Ref: 23301527
TCMC2063	TCMT313	Serotonin 2b (5-HT2b) receptor	Homo sapiens	Ki: 12 (nM), Ref: 15081042 Ki: 13 (nM), Ref: 12954071 Ki: 13 (nM), Ref: 16392816 Ki: 12 (nM), Ref: 16257207 Ki: 13.49 (nM), Ref: 24582985
TCMC2063	TCMT314	Serotonin 2c (5-HT2c) receptor	Homo sapiens	Ki: 6.9 (nM), Ref: 15081042 Ki: 8.3 (nM), Ref: 12954071 Ki: 8.3 (nM), Ref: 16392816 Ki: 6.9 (nM), Ref: 16257207 Ki: 130 (nM), Ref: 11975483 Ki: 20 (nM), Ref: 17067154 Ki: 79.43 (nM), Ref: 23301527 Ki: 79 (nM), Ref: 23301527
TCMC2063	TCMT815	Serotonin 1d (5-HT1d) receptor	Homo sapiens	Ki: 5.5 (nM), Ref: 8071931 Ki: 0.5 (nM), Ref: 18507369
TCMC2063	TCMT36	Serotonin 1a (5-HT1a) receptor	Homo sapiens	Ki: 2.5 (nM), Ref: 7658447 IC50: 1.2 (nM), Ref: 12954071 Ki: 1.259 (nM), Ref: 18433113 Ki: 10000 (nM), Ref: 18433113 Ki: 0.62 (nM), Ref: 22748706 Ki: 0.9 (nM), Ref: 23332346 Ki: 9.5 (nM), Ref: 24161678 Ki: 2.08 (nM), Ref: 25128671
TCMC2063	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 79 (nM), Ref: 16250647
TCMC2063	TCMT816	Serotonin 1b (5-HT1b) receptor	Homo sapiens	Ki: 1.1 (nM), Ref: 18507369 IC50: 29 (nM), Ref: 18983139 Ki: 18 (nM), Ref: 18983139 Ki: 14 (nM), Ref: 21726069 IC50: 12 (nM), Ref: 23582449 Ki: 4 (nM), Ref: 23466604 IC50: 6.5 (nM), Ref: 23466604
TCMC2063	TCMT817	Serotonin 4 (5-HT4) receptor	Homo sapiens	Ki: 1049 (nM), Ref: 19334715 Ki: 500 (nM), Ref: 17067154 Ki: 29.51 (nM), Ref: 19223092 Ki: 109.65 (nM), Ref: 19223092
TCMC2063	TCMT645	Serotonin 1e (5-HT1e) receptor	Homo sapiens	Ki: 10.72 (nM), Ref: 24365159 Ki: 11 (nM), Ref: 24365159
TCMC336	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6500 (nM), Ref: 22668600
TCMC336	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7200 (nM), Ref: 22668600
TCMC336	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5900 (nM), Ref: 22668600
TCMC336	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6600 (nM), Ref: 22668600
TCMC336	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 5200 (nM), Ref: 22668600
TCMC336	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5700 (nM), Ref: 22668600
TCMC2094	TCMT238	Sodium/glucose cotransporter 2	Homo sapiens	IC50: 4100 (nM), Ref: 17374486
TCMC2094	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 1100 (nM), Ref: 18565755 IC50: 5200 (nM), Ref: 18565755
TCMC1202	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 7030 (nM), Ref: 20185318
TCMC1202	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1202	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6990 (nM), Ref: 20185318
TCMC1202	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6070 (nM), Ref: 20185318
TCMC1202	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6130 (nM), Ref: 20185318
TCMC1202	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9970 (nM), Ref: 20185318
TCMC1202	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1202	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9800 (nM), Ref: 20185318
TCMC1202	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7490 (nM), Ref: 20185318
TCMC1202	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2250 (nM), Ref: 20185318
TCMC1202	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3200 (nM), Ref: 20185318
TCMC1202	TCMT822	Alpha-(1,3)-fucosyltransferase 7	Homo sapiens	IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1869	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 4410 (nM), Ref: 15658857
TCMC1111	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 11.78 (nM), Ref: 18242087 IC50: 13 (nM), Ref: 18653260 IC50: 778 (nM), Ref: 20851614 IC50: 778 (nM), Ref: 21376605 IC50: 8.6 (nM), Ref: 21873057 IC50: 29.1 (nM), Ref: 23747808 IC50: 29.1 (nM), Ref: 25590374
TCMC1111	TCMT209	11-beta-hydroxysteroid dehydrogenase 2	Homo sapiens	IC50: 257 (nM), Ref: 20851614 IC50: 257 (nM), Ref: 21376605 IC50: 1.22 (nM), Ref: 23747808 IC50: 1.2 (nM), Ref: 25590374
TCMC1111	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 4900 (nM), Ref: 21561086
TCMC983	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref:
TCMC983	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 7300 (nM), Ref: 21030469
TCMC983	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 718.7 (nM), Ref: 26498393
TCMC983	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.2 (nM), Ref: 26498393
TCMC983	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 56.4 (nM), Ref: 26498393
TCMC84	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 6700 (nM), Ref: 18565755
TCMC1119	TCMT559	Beta-2 adrenergic receptor	Homo sapiens	Ki: 360 (nM), Ref: 27132867
TCMC1119	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 910 (nM), Ref: 27132867
TCMC1119	TCMT247	Alpha-2a adrenergic receptor	Homo sapiens	Ki: 160 (nM), Ref: 27265687
TCMC2111	TCMT614	Egl nine homolog 1	Homo sapiens	IC50: 3000 (nM), Ref: 18942826
TCMC412	TCMT683	Macrophage migration inhibitory factor	Homo sapiens	Ki: 38 (nM), Ref: 19090668 IC50: 38 (nM), Ref: 27156768
TCMC1878	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 300 (nM), Ref: 24200808
TCMC689	TCMT115	Cannabinoid CB1 receptor	Homo sapiens	Ki: 50 (nM), Ref: 16078824 Ki: 72 (nM), Ref: 16213718 Ki: 70 (nM), Ref: 16570929 Ki: 70 (nM), Ref: 16682198 Ki: 72 (nM), Ref: 16279794 Ki: 72 (nM), Ref: 17561406 Ki: 70 (nM), Ref: 19161308 Ki: 72 (nM), Ref: 19331413 Ki: 11 (nM), Ref: 19361197 Ki: 70 (nM), Ref: 22044209 Ki: 89 (nM), Ref: 23865723 Ki: 72 (nM), Ref: 25065940
TCMC689	TCMT114	Cannabinoid CB2 receptor	Homo sapiens	Ki: 180 (nM), Ref: 16213718 Ki: 180 (nM), Ref: 16570929 Ki: 180 (nM), Ref: 16682198 Ki: 180 (nM), Ref: 19161308 Ki: 168 (nM), Ref: 19361197 Ki: 371 (nM), Ref: 23865723
TCMC1898	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 7906 (nM), Ref: 20696580
TCMC1898	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 1679 (nM), Ref: 20696580
TCMC1898	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1491 (nM), Ref: 20696580
TCMC1898	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 900 (nM), Ref: 10.1039/C3MD00166K
TCMC2204	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270
TCMC2204	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270
TCMC2239	TCMT226	3-phosphoinositide dependent protein kinase-1	Homo sapiens	IC50: 6600 (nM), Ref: 22537682
TCMC2239	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2100 (nM), Ref: 26918635 IC50: 2900 (nM), Ref: 26918635
TCMC381	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 207 (nM), Ref: 19836949
TCMC2157	TCMT296	Adenosine A1 receptor	Homo sapiens	Ki: 6200 (nM), Ref: 15214785 Ki: 0.6 (nM), Ref: 15664822 Ki: 6200 (nM), Ref: 16335918 Ki: 6920 (nM), Ref: 16759111 Ki: 6200 (nM), Ref: 16789747 Ki: 6200 (nM), Ref: 17665891 Ki: 6200 (nM), Ref: 19301821 Ki: 6200 (nM), Ref: 18468446 Ki: 6200 (nM), Ref: 19569717 Ki: 6770 (nM), Ref: 20188574 Ki: 6770 (nM), Ref: 24139167 Ki: 6770 (nM), Ref: 10.1039/C5MD00573F
TCMC2157	TCMT571	Adenosine A2b receptor	Homo sapiens	Ki: 7059 (nM), Ref: 15664822 Ki: 9070 (nM), Ref: 16250640 Ki: 9070 (nM), Ref: 16759111 Ki: 7850 (nM), Ref: 19569717 Ki: 9070 (nM), Ref: 20188574 Ki: 2700 (nM), Ref: 20202853 Ki: 9070 (nM), Ref: 20537438 Ki: 9070 (nM), Ref: 24139167 Ki: 9070 (nM), Ref: 26824742
TCMC2157	TCMT707	Adenosine A2a receptor	Homo sapiens	Ki: 0.6 (nM), Ref: 15664822 Ki: 7900 (nM), Ref: 16335918 Ki: 6700 (nM), Ref: 16759111 Ki: 7900 (nM), Ref: 16789747 Ki: 7900 (nM), Ref: 17665891 Ki: 7900 (nM), Ref: 19301821 Ki: 7900 (nM), Ref: 18468446 Ki: 4200 (nM), Ref: 19569717 Ki: 6700 (nM), Ref: 20188574 Ki: 1700 (nM), Ref: 23200243 Ki: 2030 (nM), Ref: 23200243 Ki: 6700 (nM), Ref: 24139167 Ki: 1710 (nM), Ref: 10.1039/C5MD00573F
TCMC2157	TCMT112	Adenosine A3 receptor	Homo sapiens	Ki: 14 (nM), Ref: 15664822
TCMC1839	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318
TCMC1839	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318
TCMC1839	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318
TCMC1839	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6160 (nM), Ref: 20185318
TCMC1839	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 3730 (nM), Ref: 20185318
TCMC1839	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1839	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 5700 (nM), Ref: 20185318
TCMC1839	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7130 (nM), Ref: 20185318
TCMC1839	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1839	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 6610 (nM), Ref: 20185318
TCMC1839	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 870 (nM), Ref: 20185318
TCMC1377	TCMT186	Monoamine oxidase B	Homo sapiens	Ki: 3000 (nM), Ref: 16137882 Ki: 3000 (nM), Ref: 19342233 IC50: 7943.28 (nM), Ref: 20934874 Ki: 5340 (nM), Ref: 21134756 Ki: 3000 (nM), Ref: 21778064 Ki: 2000 (nM), Ref: 24140951
TCMC1377	TCMT208	Monoamine oxidase A	Homo sapiens	Ki: 8380 (nM), Ref: 21134756
TCMC2250	TCMT334	3-beta-hydroxysteroid-delta(8),delta(7)-isomerase	Homo sapiens	Ki: 2 (nM), Ref: 16033255
TCMC2250	TCMT307	HERG	Homo sapiens	IC50: 181.97 (nM), Ref: 21185626
TCMC850	TCMT307	HERG	Homo sapiens	IC50: 4897.79 (nM), Ref: 21185626
TCMC850	TCMT707	Adenosine A2a receptor	Homo sapiens	Ki: 5011.87 (nM), Ref: 21661720 Ki: 9560 (nM), Ref: 23200243 Ki: 2480 (nM), Ref: 23200243
TCMC850	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 7250 (nM), Ref: 23791077
TCMC317	TCMT223	Aldose reductase	Homo sapiens	IC50: 10 (nM), Ref: 18087047
TCMC204	TCMT803	Hypoxanthine-guanine phosphoribosyltransferase	Homo sapiens	Ki: 5400 (nM), Ref: 25915781
TCMC1788	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT126	Telomerase reverse transcriptase	Homo sapiens	IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	Ki: 1500 (nM), Ref: 27460668
TCMC732	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 5900 (nM), Ref: 21561086
TCMC1078	TCMT308	Oxoeicosanoid receptor 1	Homo sapiens	IC50: 2000 (nM), Ref: 24351031
TCMC588	TCMT855	Nuclear receptor ROR-alpha	Homo sapiens	Ki: 12 (nM), Ref: 10.1039/C3MD00005B
TCMC1359	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 3000 (nM), Ref: 9544212 IC50: 6900 (nM), Ref: 17517512 IC50: 212 (nM), Ref: IC50: 290 (nM), Ref: 23651359 IC50: 1860 (nM), Ref: 23651359
TCMC1359	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 6200 (nM), Ref: 17517512 IC50: 1100 (nM), Ref: 19884005 IC50: 1100 (nM), Ref: 19500994 IC50: 1100 (nM), Ref: 20097072 IC50: 1100 (nM), Ref: 20202839 IC50: 1100 (nM), Ref: 20576432 IC50: 1400 (nM), Ref: 21280601 IC50: 1100 (nM), Ref: 21641217 IC50: 1100 (nM), Ref: 22148253 IC50: 1350 (nM), Ref: 22091869 IC50: 1100 (nM), Ref: 23200247 IC50: 4300 (nM), Ref: 25221653 IC50: 1100 (nM), Ref: 26487917 IC50: 1100 (nM), Ref: 26691756
TCMC1516	TCMT44	Glyoxalase I	Homo sapiens	IC50: 7700 (nM), Ref: 18258440
TCMC1516	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 3370 (nM), Ref: 20696580
TCMC1516	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1249 (nM), Ref: 20696580
TCMC1516	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 79 (nM), Ref: 20696580
TCMC1516	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 8200 (nM), Ref: 21641214
TCMC1516	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 3610 (nM), Ref: 22658537
TCMC1516	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 5620 (nM), Ref: 22658537
TCMC1516	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 980 (nM), Ref: 22658537
TCMC1516	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 830 (nM), Ref: 23411073
TCMC1516	TCMT127	Poly [ADP-ribose] polymerase-1	Homo sapiens	IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272
TCMC1516	TCMT128	Tankyrase-2	Homo sapiens	IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272
TCMC1516	TCMT129	Tankyrase-1	Homo sapiens	IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272
TCMC1516	TCMT223	Aldose reductase	Homo sapiens	IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431
TCMC1516	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 1600 (nM), Ref: 24368208
TCMC1516	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 6400 (nM), Ref: 24878198
TCMC1516	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677
TCMC1516	TCMT100	Transthyretin	Homo sapiens	IC50: 7000 (nM), Ref: 26214366
TCMC1516	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3691.6 (nM), Ref: 26498393
TCMC1516	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.7 (nM), Ref: 26498393
TCMC1516	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 60.3 (nM), Ref: 26498393
TCMC1516	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 293 (nM), Ref: 26498393
TCMC1516	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 9200 (nM), Ref: 26529431
TCMC1504	TCMT273	Bile acid receptor FXR	Homo sapiens	IC50: 18.3 (nM), Ref: 24775917
TCMC1977	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 7410 (nM), Ref: 21669522
TCMC1977	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 540 (nM), Ref: 21669522
TCMC1977	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 520 (nM), Ref: 21669522
TCMC1498	TCMT864	Thyroid hormone receptor alpha	Homo sapiens	IC50: 0.24 (nM), Ref: 16099653 IC50: 0.24 (nM), Ref: 17543524 Ki: 0.33 (nM), Ref: 18975928 Ki: 2.33 (nM), Ref: 22542282 Ki: 2.33 (nM), Ref: 23276448 IC50: 3.2 (nM), Ref: 24290064
TCMC1498	TCMT69	Thyroid hormone receptor beta-1	Homo sapiens	IC50: 0.26 (nM), Ref: 16099653 IC50: 0.26 (nM), Ref: 17543524 IC50: 0.257 (nM), Ref: 17524652 Ki: 0.68 (nM), Ref: 18975928 Ki: 2.29 (nM), Ref: 22542282 Ki: 2.29 (nM), Ref: 23276448 IC50: 2.9 (nM), Ref: 24290064
TCMC1498	TCMT796	Proliferating cell nuclear antigen	Homo sapiens	IC50: 3600 (nM), Ref: 23395113
TCMC1734	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 3430 (nM), Ref: 19097799
TCMC1734	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 4960 (nM), Ref: 18533708
TCMC2212	TCMT868	UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit	Homo sapiens	IC50: 1800 (nM), Ref: 21273069
TCMC1734	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469
TCMC1734	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 3656 (nM), Ref: 20696580
TCMC1734	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 79.5 (nM), Ref: 26498393
TCMC1734	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.3 (nM), Ref: 26498393
TCMC1734	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 44.3 (nM), Ref: 26498393
TCMC2238	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 9000 (nM), Ref: 23791077
TCMC2113	TCMT883	Lysine-specific demethylase 5C	Homo sapiens	IC50: 4500 (nM), Ref: 22724510
TCMC2113	TCMT884	Histone lysine demethylase PHF8	Homo sapiens	IC50: 2300 (nM), Ref: 22724510
TCMC2113	TCMT885	Lysine-specific demethylase 2A	Homo sapiens	IC50: 570 (nM), Ref: 22724510
TCMC341	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 510 (nM), Ref: 19231207
TCMC2114	TCMT683	Macrophage migration inhibitory factor	Homo sapiens	IC50: 2200 (nM), Ref: 25743213
TCMC2114	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 9000 (nM), Ref: 27135370
TCMC811	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 2030 (nM), Ref: 19097799
TCMC811	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 9900 (nM), Ref: 18533708
TCMC811	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10.2 (nM), Ref: 20413308
TCMC811	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7078.5 (nM), Ref: 26498393
TCMC811	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 371.5 (nM), Ref: 26498393
TCMC811	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 52.5 (nM), Ref: 26498393
TCMC1496	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT164	Cyclooxygenase-1	Homo sapiens	Ki: 4000 (nM), Ref: 24088053
TCMC1494	TCMT267	GABA receptor rho-1 subunit	Homo sapiens	IC50: 91 (nM), Ref: 10.1584/jpestics.R07-07
TCMC1494	TCMT891	GABA receptor beta-3 subunit	Homo sapiens	IC50: 0.9 (nM), Ref: 10.1584/jpestics.R07-07
TCMC560	TCMT315	Serotonin 6 (5-HT6) receptor	Homo sapiens	Ki: 50 (nM), Ref: 15771424
TCMC560	TCMT817	Serotonin 4 (5-HT4) receptor	Homo sapiens	Ki: 26.92 (nM), Ref: 19223092 Ki: 245.47 (nM), Ref: 19223092
TCMC2201	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8700 (nM), Ref: 21332115
TCMC1873	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 1840 (nM), Ref: 15828829 Ki: 1840 (nM), Ref: 21733699
TCMC1873	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 5270 (nM), Ref: 15828829 Ki: 5270 (nM), Ref: 21733699
TCMC1611	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1611	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2039	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 5400 (nM), Ref: 10.1016/S0960-894X(97)00194-7
TCMC1200	TCMT897	Voltage-gated calcium channel alpha2/delta subunit 1	Homo sapiens	IC50: 27 (nM), Ref: 15050626
TCMC897	TCMT223	Aldose reductase	Homo sapiens	IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024
TCMC897	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 7900 (nM), Ref: 22236472
TCMC1320	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 2786 (nM), Ref: 20696580
TCMC1320	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 511 (nM), Ref: 20696580
TCMC1320	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 102.1 (nM), Ref: 26498393
TCMC1320	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3.3 (nM), Ref: 26498393
TCMC1320	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 454.1 (nM), Ref: 26498393
TCMC772	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 955 (nM), Ref: 15828829
TCMC772	TCMT132	Butyrylcholinesterase	Homo sapiens	Ki: 2050 (nM), Ref: 15828829
TCMC1832	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1856	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 500 (nM), Ref: 20590092
TCMC1856	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 52 (nM), Ref: 20590092
TCMC1856	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 44 (nM), Ref: 20590092
TCMC1856	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 540 (nM), Ref: 20590092
TCMC1856	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 740 (nM), Ref: 20590092
TCMC1856	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 420 (nM), Ref: 20590092
TCMC1856	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 380 (nM), Ref: 20590092
TCMC1856	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 450 (nM), Ref: 20590092
TCMC1856	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 500 (nM), Ref: 20590092
TCMC1742	TCMT637	NAD-dependent deacetylase sirtuin 3	Homo sapiens	IC50: 6200 (nM), Ref: 25275824
TCMC1742	TCMT638	NAD-dependent deacetylase sirtuin 2	Homo sapiens	IC50: 6300 (nM), Ref: 25549554 IC50: 1200 (nM), Ref: 26696402
TCMC740	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 1.77 (nM), Ref: 16250647
TCMC740	TCMT675	Beta-1 adrenergic receptor	Homo sapiens	IC50: 600 (nM), Ref: 18983139 Ki: 430 (nM), Ref: 18983139 IC50: 1740 (nM), Ref: 18588282 IC50: 1640 (nM), Ref: 20875743 Ki: 170 (nM), Ref: 21726069 Ki: 150 (nM), Ref: 23466604 IC50: 260 (nM), Ref: 23466604 IC50: 210 (nM), Ref: 26988801
TCMC2082	TCMT302	HMG-CoA reductase	Homo sapiens	Ki: 2.6 (nM), Ref: 15686898 IC50: 11.2 (nM), Ref: 15686898 IC50: 11 (nM), Ref: 15686906 IC50: 6110 (nM), Ref: 25311563 IC50: 39.81 (nM), Ref: 25311563
TCMC1940	TCMT187	Androgen Receptor	Homo sapiens	Ki: 8.5 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12781197 IC50: 37 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 9873735 IC50: 37 (nM), Ref: 9784110 Ki: 35 (nM), Ref: 20510622
TCMC1940	TCMT613	Glucocorticoid receptor	Homo sapiens	Ki: 30.5 (nM), Ref: 12954062 Ki: 30.5 (nM), Ref: 9873735 Ki: 30.5 (nM), Ref: 9784110
TCMC1940	TCMT783	Mineralocorticoid receptor	Homo sapiens	IC50: 14 (nM), Ref: 12954062 IC50: 14 (nM), Ref: 12781197 IC50: 14 (nM), Ref: 9784110 IC50: 30 (nM), Ref: 8709117
TCMC1940	TCMT904	Progesterone receptor	Homo sapiens	Ki: 3.5 (nM), Ref: 10212133 IC50: 3.5 (nM), Ref: 11859003 Ki: 3.5 (nM), Ref: 9464361 IC50: 5 (nM), Ref: 8523399 Ki: 3.8 (nM), Ref: 9667968 Ki: 3.467 (nM), Ref: 16821785 Ki: 3.4 (nM), Ref: 18553958 Ki: 5.1 (nM), Ref: 20510622
TCMC1541	TCMT317	Melatonin receptor 1B	Homo sapiens	Ki: 0.3 (nM), Ref: 15203165 Ki: 0.41 (nM), Ref: 12646022 Ki: 0.29 (nM), Ref: 10.1016/S0960-894X(97)00444-7 Ki: 0.195 (nM), Ref: 12213063 Ki: 0.31 (nM), Ref: 11960497 Ki: 0.7 (nM), Ref: 15713384 Ki: 0.7 (nM), Ref: 15380218 Ki: 0.2818 (nM), Ref: 15293992 Ki: 0.2818 (nM), Ref: 15943478 Ki: 0.35 (nM), Ref: 16759094 Ki: 0.257 (nM), Ref: 17149869 Ki: 0.3 (nM), Ref: 17481904 Ki: 0.3548 (nM), Ref: 17346859 Ki: 0.3388 (nM), Ref: 17459711 Ki: 0.2399 (nM), Ref: 18052314 IC50: 0.53 (nM), Ref: 18372181 Ki: 0.41 (nM), Ref: 18778943 Ki: 0.955 (nM), Ref: 19193160 Ki: 0.741 (nM), Ref: 18657980 Ki: 0.429 (nM), Ref: 20227878 Ki: 0.6166 (nM), Ref: 20674373 Ki: 0.34 (nM), Ref: 21420861 IC50: 0.53 (nM), Ref: 21377769 Ki: 0.21 (nM), Ref: 21473625 Ki: 0.35 (nM), Ref: 21392858 Ki: 0.21 (nM), Ref: 21568291 Ki: 0.3388 (nM), Ref: 21775151 Ki: 0.34 (nM), Ref: 21764185 Ki: 0.5 (nM), Ref: 23265885 Ki: 0.429 (nM), Ref: 23228808 Ki: 0.955 (nM), Ref: 10.1039/C1MD00149C Ki: 0.41 (nM), Ref: 25232966 Ki: 0.15 (nM), Ref: 26023814 Ki: 0.15 (nM), Ref: 26367450 Ki: 0.955 (nM), Ref: 10.1039/C5MD00190K Ki: 0.52 (nM), Ref: 26820449 Ki: 0.34 (nM), Ref: 26785296
TCMC1541	TCMT316	Melatonin receptor 1A	Homo sapiens	Ki: 0.14 (nM), Ref: 12646022 Ki: 0.2 (nM), Ref: 10.1016/S0960-894X(97)00444-7 Ki: 0.0823 (nM), Ref: 12213063 Ki: 0.12 (nM), Ref: 11960497 Ki: 0.3 (nM), Ref: 15713384 Ki: 0.3 (nM), Ref: 15380218 Ki: 0.2884 (nM), Ref: 15293992 Ki: 0.2884 (nM), Ref: 15943478 Ki: 0.39 (nM), Ref: 16759094 Ki: 0.3236 (nM), Ref: 17149869 Ki: 0.2 (nM), Ref: 17481904 Ki: 0.389 (nM), Ref: 17346859 Ki: 0.263 (nM), Ref: 17459711 Ki: 0.1413 (nM), Ref: 18052314 IC50: 0.2 (nM), Ref: 18372181 IC50: 0.18 (nM), Ref: 18983139 Ki: 0.11 (nM), Ref: 18983139 Ki: 0.14 (nM), Ref: 18778943 Ki: 0.4571 (nM), Ref: 19193160 Ki: 0.525 (nM), Ref: 18657980 Ki: 0.296 (nM), Ref: 20227878 Ki: 0.3311 (nM), Ref: 20674373 Ki: 0.25 (nM), Ref: 21420861 IC50: 0.2 (nM), Ref: 21377769 Ki: 0.24 (nM), Ref: 21473625 Ki: 0.22 (nM), Ref: 21392858 Ki: 0.24 (nM), Ref: 21568291 Ki: 0.37 (nM), Ref: 21726069 Ki: 0.263 (nM), Ref: 21775151 Ki: 0.25 (nM), Ref: 21764185 Ki: 0.2 (nM), Ref: 23265885 Ki: 0.296 (nM), Ref: 23228808 IC50: 0.53 (nM), Ref: 23582449 Ki: 0.35 (nM), Ref: 23466604 IC50: 0.44 (nM), Ref: 23466604 Ki: 0.4571 (nM), Ref: 10.1039/C1MD00149C Ki: 0.14 (nM), Ref: 25232966 Ki: 0.091 (nM), Ref: 26023814 Ki: 0.091 (nM), Ref: 26367450 Ki: 0.4571 (nM), Ref: 10.1039/C5MD00190K Ki: 0.23 (nM), Ref: 26820449 Ki: 0.25 (nM), Ref: 26785296 IC50: 0.11 (nM), Ref: 26988801
TCMC1541	TCMT329	Quinone reductase 2	Homo sapiens	IC50: 64.6 (nM), Ref: 21377769
TCMC2163	TCMT214	Monoglyceride lipase	Homo sapiens	IC50: 977.24 (nM), Ref: 19883085
TCMC2163	TCMT434	Tyrosine-protein kinase JAK2	Homo sapiens	IC50: 223 (nM), Ref:
TCMC2163	TCMT881	Gamma-butyrobetaine dioxygenase	Homo sapiens	IC50: 5800 (nM), Ref: 25266780 IC50: 7900 (nM), Ref: 25266780
TCMC307	TCMT333	C-terminal-binding protein 2	Homo sapiens	IC50: 7340 (nM), Ref: 27156192
TCMC1540	TCMT302	HMG-CoA reductase	Homo sapiens	Ki: 23.5 (nM), Ref: 15686898 IC50: 4000 (nM), Ref: 15686898
TCMC736	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 2400 (nM), Ref: 19884005 IC50: 2400 (nM), Ref: 19500994 IC50: 2400 (nM), Ref: 20097072 IC50: 2400 (nM), Ref: 20576432 IC50: 2400 (nM), Ref: 22361134 IC50: 2400 (nM), Ref: 22148253 IC50: 2400 (nM), Ref: 23200247
TCMC736	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 4192 (nM), Ref:
TCMC1237	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7300 (nM), Ref: 22668600
TCMC1237	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6600 (nM), Ref: 22668600
TCMC1237	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 4100 (nM), Ref: 22668600
TCMC1237	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4200 (nM), Ref: 22668600
TCMC2082	TCMT217	Cytochrome P450 2C8	Homo sapiens	IC50: 3700 (nM), Ref: 22328583
TCMC2082	TCMT278	Solute carrier organic anion transporter family member 1B1	Homo sapiens	IC50: 4400 (nM), Ref: 22587986 IC50: 6000 (nM), Ref: 22587986
TCMC1974	TCMT905	P2X purinoceptor 1	Homo sapiens	IC50: 10000 (nM), Ref: 23510563
TCMC2018	TCMT907	Farnesyl diphosphate synthase	Homo sapiens	IC50: 452.9 (nM), Ref: 18327899 Ki: 82.2 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18327899 Ki: 0.36 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18434151 IC50: 300 (nM), Ref: 20801032 IC50: 11 (nM), Ref: 22390415 IC50: 860 (nM), Ref: 22390415 IC50: 11 (nM), Ref: 22884353 IC50: 10 (nM), Ref: 21780776 IC50: 5.2 (nM), Ref: 23998921 IC50: 11 (nM), Ref: 23998921 IC50: 6 (nM), Ref: 24911527 IC50: 11 (nM), Ref: 25630225 IC50: 6 (nM), Ref: 25935643 IC50: 0.36 (nM), Ref: 25815158 IC50: 82 (nM), Ref: 25815158
TCMC1836	TCMT311	Multidrug and toxin extrusion protein 1	Homo sapiens	IC50: 2800 (nM), Ref: 23241029 IC50: 2800 (nM), Ref: 23241029
TCMC1836	TCMT309	Solute carrier family 22 member 2	Homo sapiens	IC50: 1500 (nM), Ref: 23241029
TCMC1836	TCMT60	Fatty acid synthase	Homo sapiens	Ki: 4100 (nM), Ref: 25513712
TCMC1067	TCMT307	HERG	Homo sapiens	IC50: 2570.4 (nM), Ref: 21185626
TCMC1067	TCMT244	Histamine H1 receptor	Homo sapiens	Ki: 14.79 (nM), Ref: 21944853
TCMC827	TCMT307	HERG	Homo sapiens	IC50: 891.25 (nM), Ref: 21185626
TCMC1130	TCMT633	Serotonin transporter	Homo sapiens	Ki: 1 (nM), Ref: 19720528 Ki: 1 (nM), Ref: 20347298 IC50: 4600 (nM), Ref: 24237160 Ki: 7.4 (nM), Ref: 24944746 Ki: 2.2 (nM), Ref: 26153715
TCMC1509	TCMT116	Mu opioid receptor	Homo sapiens	Ki: 0.53 (nM), Ref: 15454210
TCMC1236	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref:
TCMC1236	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref:
TCMC883	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 1880 (nM), Ref: 11844666 IC50: 6300 (nM), Ref: 10197970 IC50: 1689 (nM), Ref: 15454242 IC50: 2600 (nM), Ref: 15615524 IC50: 1689 (nM), Ref: 19520573 IC50: 2600 (nM), Ref: 19791801 IC50: 7000 (nM), Ref: 21570308 IC50: 723 (nM), Ref: IC50: 6650 (nM), Ref: 23473947 IC50: 2600 (nM), Ref: 24440378
TCMC883	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 230 (nM), Ref: 11906292 IC50: 1000 (nM), Ref: 10465547 IC50: 1000 (nM), Ref: 10406640 IC50: 68 (nM), Ref: 15454242 IC50: 1200 (nM), Ref: 15546727 IC50: 1200 (nM), Ref: 15916445 IC50: 6 (nM), Ref: 16250658 IC50: 6.8 (nM), Ref: 16250658 IC50: 330 (nM), Ref: 16814546 IC50: 2.2 (nM), Ref: 16806914 IC50: 1300 (nM), Ref: 17335184 IC50: 350 (nM), Ref: 15615524 IC50: 35 (nM), Ref: 17604631 IC50: 540 (nM), Ref: 17915854 IC50: 1200 (nM), Ref: 17994684 IC50: 300 (nM), Ref: 18063374 IC50: 300 (nM), Ref: 17532544 IC50: 1000 (nM), Ref: 17976864 IC50: 2900 (nM), Ref: 19059783 IC50: 80 (nM), Ref: 16252917 IC50: 540 (nM), Ref: 18752957 IC50: 800 (nM), Ref: 19097798 IC50: 120 (nM), Ref: 19136259 IC50: 120 (nM), Ref: 19296694 IC50: 63 (nM), Ref: 19520573 IC50: 68 (nM), Ref: 19520573 IC50: 336 (nM), Ref: 19520573 IC50: 120 (nM), Ref: 19500994 IC50: 120 (nM), Ref: 20097072 IC50: 540 (nM), Ref: 19957931 IC50: 350 (nM), Ref: 19791801 IC50: 800 (nM), Ref: 20451397 IC50: 65 (nM), Ref: 20576432 IC50: 65 (nM), Ref: 20655211 IC50: 300 (nM), Ref: 20970223 IC50: 40 (nM), Ref: 21215625 IC50: 30 (nM), Ref: 21316237 IC50: 10 (nM), Ref: 21434686 IC50: 70 (nM), Ref: 21641217 IC50: 190 (nM), Ref: 21570308 IC50: 100 (nM), Ref: 22119153 IC50: 540 (nM), Ref: 21992176 IC50: 40 (nM), Ref: 22386983 IC50: 70 (nM), Ref: 22361134 IC50: 60 (nM), Ref: 22341941 IC50: 60 (nM), Ref: 22560838 IC50: 140 (nM), Ref: 22749420 IC50: 40 (nM), Ref: 22263894 IC50: 54 (nM), Ref: 22263894 IC50: 42 (nM), Ref: 23010270 IC50: 57 (nM), Ref: 10.1007/s00044-012-0174-z IC50: 70 (nM), Ref: 23200247 IC50: 100 (nM), Ref: 23353741 IC50: 870 (nM), Ref: 23473947 IC50: 20 (nM), Ref: 23706267 IC50: 320 (nM), Ref: 24211633 IC50: 40 (nM), Ref: 24332492 IC50: 57 (nM), Ref: 24295787 IC50: 540 (nM), Ref: 24373735 IC50: 350 (nM), Ref: 24440378 IC50: 40 (nM), Ref: 24602792 IC50: 280 (nM), Ref: 24607877 IC50: 72 (nM), Ref: 24656662 IC50: 70 (nM), Ref: 24650702 IC50: 2660 (nM), Ref: 24661847 IC50: 40 (nM), Ref: 24745964 IC50: 270 (nM), Ref: 24836072 IC50: 280 (nM), Ref: 24780593 IC50: 290 (nM), Ref: 24900871 IC50: 40 (nM), Ref: 24631898 IC50: 40 (nM), Ref: 24934992 IC50: 50 (nM), Ref: 25221653 IC50: 19 (nM), Ref: 25819096 IC50: 52 (nM), Ref: 25866240 IC50: 16 (nM), Ref: 25980909 IC50: 40 (nM), Ref: 25956953 IC50: 130 (nM), Ref: 26081289 IC50: 19 (nM), Ref: 26316467 IC50: 900 (nM), Ref: 26546221 IC50: 260 (nM), Ref: 26638042 IC50: 870 (nM), Ref: 26691756 IC50: 40 (nM), Ref: 10.1039/C5MD00278H IC50: 40 (nM), Ref: 26898334 IC50: 40 (nM), Ref: 26898334 IC50: 40 (nM), Ref: 27019010 IC50: 310 (nM), Ref: 27349331
TCMC883	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 880 (nM), Ref: 15686931 Ki: 880 (nM), Ref: 20605094 Ki: 880 (nM), Ref: 23067387
TCMC883	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 21 (nM), Ref: 15686931 Ki: 21 (nM), Ref: 16134940 IC50: 21 (nM), Ref: 16220969 Ki: 21 (nM), Ref: 16290146 Ki: 21 (nM), Ref: 19317447 Ki: 21 (nM), Ref: 19124253 Ki: 21 (nM), Ref: 19193158 Ki: 21 (nM), Ref: 19338333 Ki: 21 (nM), Ref: 19520577 Ki: 21 (nM), Ref: 19846301 Ki: 21 (nM), Ref: 20605094 Ki: 21 (nM), Ref: 20624682 Ki: 21 (nM), Ref: 21208801 Ki: 21 (nM), Ref: 21251841 Ki: 21 (nM), Ref: 21757360 Ki: 21 (nM), Ref: 21852133 IC50: 181 (nM), Ref: Ki: 21 (nM), Ref: 22285172 Ki: 21 (nM), Ref: 22424239 Ki: 21 (nM), Ref: 23067387 Ki: 21 (nM), Ref: 23181552 Ki: 21 (nM), Ref: 23391336 Ki: 21 (nM), Ref: 22883029 Ki: 21 (nM), Ref: 23867389 Ki: 21 (nM), Ref: 23965175 Ki: 21 (nM), Ref: 24314394 Ki: 21 (nM), Ref: 24513184 Ki: 21 (nM), Ref: 24792813 Ki: 21 (nM), Ref: 25129169 Ki: 21 (nM), Ref: 25533402 Ki: 21 (nM), Ref: 25773015 Ki: 21 (nM), Ref: 25882523 Ki: 21 (nM), Ref: 25766630 Ki: 21 (nM), Ref: 26174556 Ki: 21 (nM), Ref: 26525863 Ki: 21 (nM), Ref: 26691758 Ki: 21 (nM), Ref: 26850377 Ki: 21 (nM), Ref: 26832216 Ki: 21 (nM), Ref: 26920803
TCMC883	TCMT507	MAP kinase p38 alpha	Homo sapiens	IC50: 810 (nM), Ref: 15990304
TCMC883	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 16 (nM), Ref: 16134940 IC50: 16 (nM), Ref: 16220969 Ki: 16 (nM), Ref: 16290146 Ki: 16 (nM), Ref: 19193158 Ki: 16 (nM), Ref: 20605094 Ki: 16 (nM), Ref: 21852133 Ki: 16 (nM), Ref: 23067387 Ki: 16 (nM), Ref: 23965175 Ki: 16 (nM), Ref: 24513184 Ki: 16 (nM), Ref: 25766630
TCMC883	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 18 (nM), Ref: 16290146 Ki: 18 (nM), Ref: 20605094 Ki: 18 (nM), Ref: 21852133 Ki: 18 (nM), Ref: 23067387 Ki: 18 (nM), Ref: 23965175 Ki: 18 (nM), Ref: 24513184 Ki: 18 (nM), Ref: 25766630
TCMC883	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 94 (nM), Ref: 19193158 Ki: 94 (nM), Ref: 20605094 Ki: 94 (nM), Ref: 23067387
TCMC883	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 794 (nM), Ref: 20605094 Ki: 794 (nM), Ref: 23067387
TCMC883	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 93 (nM), Ref: 20605094 Ki: 93 (nM), Ref: 23067387
TCMC883	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 2170 (nM), Ref: 20605094 Ki: 2170 (nM), Ref: 23067387 Ki: 2170 (nM), Ref: 23867389 Ki: 2170 (nM), Ref: 23965175 Ki: 2170 (nM), Ref: 24287559 Ki: 2170 (nM), Ref: 25766630
TCMC883	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 98 (nM), Ref: 20605094 Ki: 98 (nM), Ref: 23067387
TCMC883	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 689 (nM), Ref: 20605094 Ki: 689 (nM), Ref: 23067387
TCMC1236	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 10 (nM), Ref: 17482813
TCMC1236	TCMT910	Estrogen-related receptor beta	Homo sapiens	IC50: 395 (nM), Ref: 17482813
TCMC883	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7400 (nM), Ref: 23067387
TCMC883	TCMT301	Prostaglandin E synthase	Homo sapiens	IC50: 540 (nM), Ref: 26653180 IC50: 425 (nM), Ref: 26653180
TCMC1236	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 2210 (nM), Ref: 18533708
TCMC2184	TCMT912	Retinoic acid receptor gamma	Homo sapiens	Ki: 0.7 (nM), Ref: 11412986 Ki: 0.6 (nM), Ref: 10.1016/S0960-894X(97)00420-4 Ki: 0.04 (nM), Ref: 9435893 Ki: 0.5 (nM), Ref: 10.1016/S0960-894X(01)80113-X
TCMC2184	TCMT833	Retinoic acid receptor alpha	Homo sapiens	Ki: 0.1 (nM), Ref: 10.1016/S0960-894X(97)00420-4 IC50: 9000 (nM), Ref: 15615521
TCMC2184	TCMT913	Retinoic acid receptor beta	Homo sapiens	Ki: 4.1 (nM), Ref: 9435893 IC50: 3000 (nM), Ref: 15615521
TCMC2184	TCMT735	Retinoid X receptor alpha	Homo sapiens	Ki: 330 (nM), Ref: 9435893
TCMC2184	TCMT914	Retinoid X receptor beta	Homo sapiens	Ki: 54 (nM), Ref: 9435893
TCMC2184	TCMT915	Retinoid X receptor gamma	Homo sapiens	Ki: 120 (nM), Ref: 9435893
TCMC1236	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 340 (nM), Ref: 20853847
TCMC2184	TCMT893	Nuclear receptor ROR-beta	Homo sapiens	IC50: 0.15 (nM), Ref: 10.1039/C3MD00005B IC50: 125.89 (nM), Ref: 25305688
TCMC2184	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	IC50: 199.53 (nM), Ref: 25305688
TCMC2184	TCMT855	Nuclear receptor ROR-alpha	Homo sapiens	IC50: 199.53 (nM), Ref: 25305688
TCMC1236	TCMT289	Thromboxane-A synthase	Homo sapiens	IC50: 7720 (nM), Ref:
TCMC1946	TCMT34	Cytochrome P450 2D6	Homo sapiens	IC50: 1900 (nM), Ref: 15993593 IC50: 5011.87 (nM), Ref: 26565745
TCMC1946	TCMT559	Beta-2 adrenergic receptor	Homo sapiens	Ki: 3.69 (nM), Ref: 24326276 Ki: 0.46 (nM), Ref: 24326276 IC50: 50.12 (nM), Ref: 26565745
TCMC1946	TCMT48	Sodium channel protein type V alpha subunit	Homo sapiens	IC50: 2100 (nM), Ref: 21300721
TCMC1946	TCMT675	Beta-1 adrenergic receptor	Homo sapiens	IC50: 251.19 (nM), Ref: 26565745
TCMC1946	TCMT36	Serotonin 1a (5-HT1a) receptor	Homo sapiens	IC50: 3981.07 (nM), Ref: 26565745
TCMC1746	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 980 (nM), Ref: 19719236
TCMC2179	TCMT331	Plasminogen	Homo sapiens	IC50: 3100 (nM), Ref: 23521080 IC50: 3100 (nM), Ref: 24900876
TCMC1585	TCMT220	Cytochrome P450 2J2	Homo sapiens	IC50: 4870 (nM), Ref: 23033255
TCMC1060	TCMT586	Prostanoid FP receptor	Homo sapiens	IC50: 7 (nM), Ref: 10715159 IC50: 2.5 (nM), Ref: 10915040
TCMC1060	TCMT582	Prostanoid EP1 receptor	Homo sapiens	IC50: 380 (nM), Ref: 10715159
TCMC1060	TCMT584	Prostanoid EP3 receptor	Homo sapiens	IC50: 322 (nM), Ref: 10715159
TCMC1060	TCMT585	Prostanoid EP4 receptor	Homo sapiens	IC50: 4200 (nM), Ref: 10715159
TCMC1060	TCMT921	Prostanoid DP receptor	Homo sapiens	IC50: 4500 (nM), Ref: 10715159
TCMC2064	TCMT633	Serotonin transporter	Homo sapiens	IC50: 3 (nM), Ref: 16314097 IC50: 3 (nM), Ref: 21093273
TCMC2064	TCMT635	Dopamine transporter	Homo sapiens	IC50: 310 (nM), Ref: 16314097 IC50: 310 (nM), Ref: 21093273
TCMC2064	TCMT634	Norepinephrine transporter	Homo sapiens	IC50: 825 (nM), Ref: 16314097 IC50: 825 (nM), Ref: 21093273
TCMC2064	TCMT34	Cytochrome P450 2D6	Homo sapiens	IC50: 2880 (nM), Ref: 23033255
TCMC151	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 1610 (nM), Ref: 19719236
TCMC1665	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3000 (nM), Ref: 25086914
TCMC1665	TCMT2	Microtubule-associated protein tau	Homo sapiens	IC50: 3000 (nM), Ref: 25086914
TCMC1338	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 328 (nM), Ref: 21377369 Ki: 328 (nM), Ref: 21757360 Ki: 328 (nM), Ref: 22285172 Ki: 328 (nM), Ref: 23181552 Ki: 328 (nM), Ref: 23391336 Ki: 328 (nM), Ref: 22883029 Ki: 328 (nM), Ref: 24792813 Ki: 328 (nM), Ref: 25129169 Ki: 328 (nM), Ref: 25533402 Ki: 328 (nM), Ref: 25773015 Ki: 328 (nM), Ref: 25882523 Ki: 328 (nM), Ref: 26525863 Ki: 328 (nM), Ref: 26691758 Ki: 328 (nM), Ref: 26850377 Ki: 328 (nM), Ref: 26920803
TCMC1338	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 290 (nM), Ref: 21377369 Ki: 290 (nM), Ref: 21757360 Ki: 290 (nM), Ref: 22285172 Ki: 290 (nM), Ref: 23181552 Ki: 290 (nM), Ref: 23391336 Ki: 290 (nM), Ref: 22883029 Ki: 290 (nM), Ref: 24314394 Ki: 290 (nM), Ref: 24792813 Ki: 290 (nM), Ref: 25129169 Ki: 290 (nM), Ref: 25533402 Ki: 290 (nM), Ref: 25773015 Ki: 290 (nM), Ref: 25882523 Ki: 290 (nM), Ref: 26174556 Ki: 290 (nM), Ref: 26525863 Ki: 290 (nM), Ref: 26691758 Ki: 290 (nM), Ref: 26850377 Ki: 290 (nM), Ref: 26832216 Ki: 290 (nM), Ref: 26920803
TCMC2224	TCMT634	Norepinephrine transporter	Homo sapiens	Ki: 385 (nM), Ref: 18557608 IC50: 535 (nM), Ref: 18557608 IC50: 535 (nM), Ref: 20378347 IC50: 581 (nM), Ref: 20724153 IC50: 680 (nM), Ref: 24900709 Ki: 1623 (nM), Ref: 23602445 IC50: 7943.28 (nM), Ref: 23602445 IC50: 5722 (nM), Ref: 24974340
TCMC2224	TCMT633	Serotonin transporter	Homo sapiens	IC50: 31 (nM), Ref: 18557608 IC50: 27 (nM), Ref: 20378347 IC50: 35 (nM), Ref: 20724153 Ki: 11 (nM), Ref: 24900709 Ki: 113 (nM), Ref: 23602445 IC50: 323.59 (nM), Ref: 23602445 IC50: 36.1 (nM), Ref: 24974340
TCMC2224	TCMT635	Dopamine transporter	Homo sapiens	IC50: 7340 (nM), Ref: 20724153 Ki: 3620 (nM), Ref: 23602445 IC50: 9120.11 (nM), Ref: 23602445
TCMC137	TCMT923	Adenylate cyclase type 10	Homo sapiens	IC50: 3000 (nM), Ref: 18630896
TCMC1574	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1989	TCMT37	Serotonin 2a (5-HT2a) receptor	Homo sapiens	Ki: 82 (nM), Ref: 11170639 Ki: 63.1 (nM), Ref: 17880057 Ki: 220 (nM), Ref: 18595716 Ki: 101 (nM), Ref: 22268448 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B Ki: 202 (nM), Ref:
TCMC1989	TCMT313	Serotonin 2b (5-HT2b) receptor	Homo sapiens	Ki: 251.19 (nM), Ref: 17880057
TCMC1989	TCMT651	Dopamine D3 receptor	Homo sapiens	Ki: 251.19 (nM), Ref: 17880057 Ki: 320 (nM), Ref: 18595716 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT36	Serotonin 1a (5-HT1a) receptor	Homo sapiens	Ki: 79.43 (nM), Ref: 17880057 Ki: 230 (nM), Ref: 18595716 Ki: 125 (nM), Ref: 22268448 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT160	Serotonin 7 (5-HT7) receptor	Homo sapiens	Ki: 63.1 (nM), Ref: 17880057 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT292	Muscarinic acetylcholine receptor M1	Homo sapiens	Ki: 398.11 (nM), Ref: 17880057 Ki: 100 (nM), Ref: 18595716 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT551	Muscarinic acetylcholine receptor M4	Homo sapiens	Ki: 125.89 (nM), Ref: 17880057 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT244	Histamine H1 receptor	Homo sapiens	Ki: 8.7 (nM), Ref: 18595716 Ki: 10 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT27	Dopamine D1 receptor	Homo sapiens	Ki: 1300 (nM), Ref: 18595716 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT315	Serotonin 6 (5-HT6) receptor	Homo sapiens	Ki: 1400 (nM), Ref: 18595716
TCMC1989	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 180 (nM), Ref: 18595716 Ki: 1000 (nM), Ref: 10.1039/C2MD00311B Ki: 400 (nM), Ref:
TCMC1989	TCMT648	Dopamine D4 receptor	Homo sapiens	Ki: 2200 (nM), Ref: 18595716
TCMC1989	TCMT314	Serotonin 2c (5-HT2c) receptor	Homo sapiens	Ki: 1400 (nM), Ref: 18595716 Ki: 2000 (nM), Ref:
TCMC1989	TCMT307	HERG	Homo sapiens	IC50: 5754.4 (nM), Ref: 21185626
TCMC1989	TCMT643	Alpha-1a adrenergic receptor	Homo sapiens	Ki: 100 (nM), Ref: 10.1039/C2MD00311B Ki: 20 (nM), Ref:
TCMC1989	TCMT650	Alpha-1b adrenergic receptor	Homo sapiens	Ki: 100 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT647	Alpha-2b adrenergic receptor	Homo sapiens	Ki: 1000 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT243	Alpha-2c adrenergic receptor	Homo sapiens	Ki: 100 (nM), Ref: 10.1039/C2MD00311B
TCMC1989	TCMT924	Histone H1.0	Homo sapiens	Ki: 10 (nM), Ref:
TCMC563	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4690 (nM), Ref: 22137345
TCMC563	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 920 (nM), Ref: 22137345
TCMC660	TCMT592	Xanthine dehydrogenase	Homo sapiens	IC50: 7820 (nM), Ref: 17379526 Ki: 100 (nM), Ref: 25060641 Ki: 7300 (nM), Ref: 25019478 IC50: 2900 (nM), Ref: 26022844 Ki: 1550 (nM), Ref: 26712096 IC50: 200 (nM), Ref: 26762836 IC50: 950 (nM), Ref: 27162124
TCMC684	TCMT925	Solute carrier family 22 member 6	Homo sapiens	Ki: 6020 (nM), Ref: 21571536
TCMC263	TCMT3	Arachidonate 15-lipoxygenase	Homo sapiens	IC50: 3000 (nM), Ref: 24924423
TCMC263	TCMT81	Arachidonate 12-lipoxygenase	Homo sapiens	IC50: 8000 (nM), Ref: 24924423
TCMC683	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9900 (nM), Ref: 15745821
TCMC539	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 225 (nM), Ref: 20926163 IC50: 225 (nM), Ref: 22475216 Ki: 50 (nM), Ref: 22475216
TCMC222	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 3400 (nM), Ref: 10.1016/S0960-894X(97)00194-7
TCMC308	TCMT333	C-terminal-binding protein 2	Homo sapiens	IC50: 240 (nM), Ref: 27156192
TCMC1762	TCMT33	Cytochrome P450 3A4	Homo sapiens	Ki: 2110 (nM), Ref: 16248836 Ki: 5890 (nM), Ref: 16248836
TCMC1762	TCMT782	Cytochrome P450 3A5	Homo sapiens	Ki: 4530 (nM), Ref: 16248836
TCMC2092	TCMT927	Somatostatin receptor 5	Homo sapiens	Ki: 120 (nM), Ref: 11266182 Ki: 0.14 (nM), Ref: 11327607 IC50: 10 (nM), Ref: 15658865 Ki: 0.44 (nM), Ref: 15982879 Ki: 0.26 (nM), Ref: 15982879 Ki: 0.71 (nM), Ref: 15982879 Ki: 0.15 (nM), Ref: 15982879 Ki: 1.4 (nM), Ref: 16220980 IC50: 0.2 (nM), Ref: 16220980 IC50: 4.2 (nM), Ref: 21806016 Ki: 0.23 (nM), Ref: 24342240 IC50: 4.2 (nM), Ref: 24378707 Ki: 2 (nM), Ref: 10.1039/C4MD00074A
TCMC2092	TCMT928	Somatostatin receptor 2	Homo sapiens	Ki: 0.049 (nM), Ref: 11327607 IC50: 0.7 (nM), Ref: 15658865 Ki: 0.083 (nM), Ref: 15982879 IC50: 0.4 (nM), Ref: 16220980 Ki: 0.23 (nM), Ref: 16220980 IC50: 0.67 (nM), Ref: 21806016 Ki: 0.0016 (nM), Ref: 24342240 IC50: 0.7 (nM), Ref: 24378707
TCMC2092	TCMT929	Somatostatin receptor 1	Homo sapiens	Ki: 0.36 (nM), Ref: 11327607 IC50: 1.9 (nM), Ref: 15658865 Ki: 2.3 (nM), Ref: 16220980 IC50: 1.6 (nM), Ref: 21806016 IC50: 0.14 (nM), Ref: 23582449 Ki: 0.43 (nM), Ref: 24342240 IC50: 1.9 (nM), Ref: 24378707
TCMC2092	TCMT930	Somatostatin receptor 3	Homo sapiens	Ki: 0.14 (nM), Ref: 11327607 IC50: 3.3 (nM), Ref: 15658865 Ki: 1.17 (nM), Ref: 16220980 IC50: 0.4 (nM), Ref: 16220980 IC50: 3.1 (nM), Ref: 21806016 Ki: 0.53 (nM), Ref: 24342240 IC50: 3.3 (nM), Ref: 24378707
TCMC2092	TCMT931	Somatostatin receptor 4	Homo sapiens	Ki: 0.59 (nM), Ref: 11327607 IC50: 1.6 (nM), Ref: 15658865 Ki: 1.7 (nM), Ref: 16220980 IC50: 1.7 (nM), Ref: 21806016 Ki: 0.74 (nM), Ref: 24342240 IC50: 1.6 (nM), Ref: 24378707 Ki: 2 (nM), Ref: 10.1039/C4MD00074A
TCMC1169	TCMT311	Multidrug and toxin extrusion protein 1	Homo sapiens	IC50: 760 (nM), Ref: 23241029
TCMC2034	TCMT567	DNA (cytosine-5)-methyltransferase 1	Homo sapiens	IC50: 2000 (nM), Ref: 19362833 IC50: 800 (nM), Ref: 19364644 IC50: 4000 (nM), Ref: 20006515 IC50: 4000 (nM), Ref: 21958292 IC50: 941 (nM), Ref: 22483584 IC50: 900 (nM), Ref: 22280363
TCMC2034	TCMT568	DNA (cytosine-5)-methyltransferase 3B	Homo sapiens	IC50: 300 (nM), Ref: 19362833 IC50: 200 (nM), Ref: 19364644 IC50: 250 (nM), Ref: 20006515
TCMC2034	TCMT932	Histone-lysine N-methyltransferase, H3 lysine-79 specific	Homo sapiens	Ki: 160 (nM), Ref: 22924785 IC50: 600 (nM), Ref: 23433670 IC50: 600 (nM), Ref: 23433670 Ki: 160 (nM), Ref: 23879463
TCMC2034	TCMT757	Histone-arginine methyltransferase CARM1	Homo sapiens	Ki: 400 (nM), Ref: 23879463
TCMC2034	TCMT1	Histone-lysine N-methyltransferase, H3 lysine-9 specific 3	Homo sapiens	Ki: 570 (nM), Ref: 23879463 IC50: 2000 (nM), Ref: 25746813
TCMC2034	TCMT934	N-lysine methyltransferase SMYD2	Homo sapiens	IC50: 180 (nM), Ref: 25746813
TCMC2034	TCMT935	Histone-lysine N-methyltransferase SUV420H2	Homo sapiens	IC50: 10000 (nM), Ref: 25746813
TCMC2034	TCMT937	Histone-lysine N-methyltransferase SUV39H1	Homo sapiens	IC50: 1200 (nM), Ref: 25746813
TCMC2034	TCMT938	Histone-lysine N-methyltransferase SETDB1	Homo sapiens	IC50: 2200 (nM), Ref: 25746813
TCMC2034	TCMT42	Histone-lysine N-methyltransferase MLL	Homo sapiens	IC50: 2300 (nM), Ref: 25746813
TCMC2034	TCMT940	Histone-lysine N-methyltransferase, H3 lysine-9 specific 5	Homo sapiens	IC50: 230 (nM), Ref: 25746813
TCMC2034	TCMT941	Histone-lysine N-methyltransferase EZH1	Homo sapiens	IC50: 6400 (nM), Ref: 25746813
TCMC2034	TCMT564	Protein-arginine N-methyltransferase 1	Homo sapiens	IC50: 420 (nM), Ref: 25559100 IC50: 500 (nM), Ref: 26428871
TCMC2104	TCMT187	Androgen Receptor	Homo sapiens	Ki: 2 (nM), Ref: 9871534 IC50: 0 (nM), Ref: 9925725 Ki: 3 (nM), Ref: 9925725 Ki: 0.2 (nM), Ref: 17034117 IC50: 1.82 (nM), Ref: 17149866 Ki: 0.3 (nM), Ref: 17181141 Ki: 0.3 (nM), Ref: 17439112 Ki: 0.2 (nM), Ref: 17257838 Ki: 0.2 (nM), Ref: 17887661 Ki: 0.2 (nM), Ref: 17267219 Ki: 0.9 (nM), Ref: 18400499 Ki: 0.2 (nM), Ref: 18442912 IC50: 0.05 (nM), Ref: 18442912 IC50: 1 (nM), Ref: 19606870 Ki: 4.7 (nM), Ref: 20510622 IC50: 2.1 (nM), Ref: 22094279 IC50: 2.1 (nM), Ref: 23199477 IC50: 11 (nM), Ref: 10.1039/C3MD20341G IC50: 13.1 (nM), Ref: 26305181
TCMC2104	TCMT99	Testis-specific androgen-binding protein	Homo sapiens	IC50: 3.8 (nM), Ref: 2296011
TCMC2104	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 1550 (nM), Ref: 2918514 Ki: 220 (nM), Ref: 2918514
TCMC216	TCMT945	Sphingosine 1-phosphate receptor Edg-1	Homo sapiens	IC50: 0.16 (nM), Ref: 15149705 IC50: 0.67 (nM), Ref: 15615513 IC50: 0.47 (nM), Ref: 19081720 IC50: 0.78 (nM), Ref: 20304639
TCMC216	TCMT946	Sphingosine 1-phosphate receptor Edg-3	Homo sapiens	IC50: 0.04 (nM), Ref: 15149705 IC50: 0.26 (nM), Ref: 15615513 IC50: 0.66 (nM), Ref: 19081720 IC50: 0.92 (nM), Ref: 20304639
TCMC216	TCMT947	Sphingosine 1-phosphate receptor Edg-6	Homo sapiens	IC50: 23 (nM), Ref: 15149705 IC50: 34 (nM), Ref: 15615513 IC50: 2.4 (nM), Ref: 19081720 IC50: 1.04 (nM), Ref: 20304639 IC50: 2.9 (nM), Ref: 20446681
TCMC216	TCMT948	Sphingosine 1-phosphate receptor Edg-5	Homo sapiens	IC50: 0.23 (nM), Ref: 15149705 IC50: 0.35 (nM), Ref: 15615513
TCMC216	TCMT949	Sphingosine 1-phosphate receptor Edg-8	Homo sapiens	IC50: 0.55 (nM), Ref: 15615513 IC50: 1.1 (nM), Ref: 19081720 IC50: 2 (nM), Ref: 20304639
TCMC854	TCMT279	Vitamin D receptor	Homo sapiens	IC50: 0.7 (nM), Ref: 17149880 IC50: 0.8 (nM), Ref: 17924616 IC50: 9.3 (nM), Ref: 24035340 IC50: 0.08 (nM), Ref: 24742174 IC50: 0.06 (nM), Ref: 26515040 IC50: 0.35 (nM), Ref: 26613420 IC50: 0.1 (nM), Ref: 26613420 IC50: 1.13 (nM), Ref: 26562542
TCMC826	TCMT951	Bradykinin B2 receptor	Homo sapiens	Ki: 0.11 (nM), Ref: 10882364 Ki: 1.1 (nM), Ref: 23403082 IC50: 1.8 (nM), Ref: 23403082
TCMC1029	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 12 (nM), Ref: 16250647
TCMC129	TCMT81	Arachidonate 12-lipoxygenase	Homo sapiens	IC50: 1000 (nM), Ref: 24924423
TCMC1822	TCMT760	Oxytocin receptor	Homo sapiens	Ki: 0.8 (nM), Ref: 12036367 IC50: 2.7 (nM), Ref: 17316912 Ki: 0.79 (nM), Ref: 25642985 Ki: 9.53 (nM), Ref: 25642985 Ki: 6.6 (nM), Ref: 25642985 Ki: 0.79 (nM), Ref: 25642985 Ki: 0.8 (nM), Ref: 26741855 Ki: 0.44 (nM), Ref: 27297999
TCMC1822	TCMT918	Vasopressin V1a receptor	Homo sapiens	Ki: 120 (nM), Ref: 12036367 Ki: 120 (nM), Ref: 25642985
TCMC1822	TCMT784	Vasopressin V2 receptor	Homo sapiens	Ki: 3500 (nM), Ref: 12036367 Ki: 1544 (nM), Ref: 25642985
TCMC1822	TCMT672	Vasopressin V1b receptor	Homo sapiens	Ki: 1782 (nM), Ref: 25642985
TCMC2174	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 500 (nM), Ref: 15771438 Ki: 430 (nM), Ref: 15771438 Ki: 9600 (nM), Ref: 15771438 Ki: 7700 (nM), Ref: 15771438 Ki: 5 (nM), Ref: 15686895 Ki: 5 (nM), Ref: 15686894 Ki: 5 (nM), Ref: 15686931 Ki: 5000 (nM), Ref: 15546717 Ki: 10.3 (nM), Ref: 15837316 Ki: 5 (nM), Ref: 16134940 Ki: 10 (nM), Ref: 16302824 Ki: 10 (nM), Ref: 16539401 Ki: 10 (nM), Ref: 16459077 Ki: 10 (nM), Ref: 17125255 Ki: 10 (nM), Ref: 17228881 Ki: 10 (nM), Ref: 17376683 Ki: 10 (nM), Ref: 17475500 Ki: 450 (nM), Ref: 18363349 Ki: 10 (nM), Ref: 19317447 Ki: 10 (nM), Ref: 19124253 Ki: 10 (nM), Ref: 19193158 Ki: 10 (nM), Ref: 18990571 Ki: 10 (nM), Ref: 19338333 Ki: 10 (nM), Ref: 18640037 Ki: 10 (nM), Ref: 18644716 Ki: 10 (nM), Ref: 19398204 Ki: 10 (nM), Ref: 19520577 Ki: 10 (nM), Ref: 19539481 Ki: 5 (nM), Ref: 19827837 Ki: 10 (nM), Ref: 19846301 Ki: 10 (nM), Ref: 20028100 IC50: 2100 (nM), Ref: 19388676 Ki: 300 (nM), Ref: 19388676 Ki: 5 (nM), Ref: 20201556 Ki: 10 (nM), Ref: 20472429 Ki: 10 (nM), Ref: 20624682 Ki: 10 (nM), Ref: 21208801 Ki: 10 (nM), Ref: 21251841 Ki: 10 (nM), Ref: 21300547 Ki: 5 (nM), Ref: 21314129 Ki: 10 (nM), Ref: 21332115 Ki: 10 (nM), Ref: 19435663 Ki: 10 (nM), Ref: 21506569 Ki: 5 (nM), Ref: 21723123 Ki: 10 (nM), Ref: 21757360 Ki: 10 (nM), Ref: 22285172 Ki: 10 (nM), Ref: 22386980 Ki: 10 (nM), Ref: 22424239 Ki: 10 (nM), Ref: 22443141 Ki: 10 (nM), Ref: 23391336 Ki: 10 (nM), Ref: 22883029 Ki: 10 (nM), Ref: 23867389 Ki: 10 (nM), Ref: 23965175 Ki: 300 (nM), Ref: 24205976 IC50: 500 (nM), Ref: 24205976 Ki: 10 (nM), Ref: 24314394 Ki: 10 (nM), Ref: 24513184 Ki: 10 (nM), Ref: 24792813 Ki: 10 (nM), Ref: 25129169 Ki: 10 (nM), Ref: 25533402 Ki: 10 (nM), Ref: 25773015 Ki: 10 (nM), Ref: 25882523 Ki: 10 (nM), Ref: 26174556 Ki: 10 (nM), Ref: 26525863 Ki: 10 (nM), Ref: 26691758 Ki: 10 (nM), Ref: 26850377 Ki: 10 (nM), Ref: 26832216 Ki: 10 (nM), Ref: 26920803
TCMC2174	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 1590 (nM), Ref: 16039848 Ki: 58 (nM), Ref: 16134940 Ki: 58 (nM), Ref: 17125255 Ki: 1590 (nM), Ref: 17125255 Ki: 1590 (nM), Ref: 17228881 Ki: 58 (nM), Ref: 17228881 Ki: 1590 (nM), Ref: 17376683 Ki: 58 (nM), Ref: 17475500 Ki: 58 (nM), Ref: 19193158 Ki: 58 (nM), Ref: 18640037 Ki: 58 (nM), Ref: 19398204 Ki: 58 (nM), Ref: 19827837 Ki: 58 (nM), Ref: 20028100 Ki: 58 (nM), Ref: 20201556 Ki: 58 (nM), Ref: 20472429 Ki: 58 (nM), Ref: 21314129 Ki: 58 (nM), Ref: 21723123 Ki: 58 (nM), Ref: 22443141 Ki: 58 (nM), Ref: 23965175 Ki: 58 (nM), Ref: 24513184
TCMC2174	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 3800 (nM), Ref: 16039848 Ki: 3.8 (nM), Ref: 15686894 Ki: 3.8 (nM), Ref: 17125255 Ki: 3.8 (nM), Ref: 17475500 Ki: 3.8 (nM), Ref: 18640037 Ki: 3800 (nM), Ref: 18406497 Ki: 3.8 (nM), Ref: 19827837 Ki: 3.8 (nM), Ref: 20028100 Ki: 3.8 (nM), Ref: 20201556 Ki: 3.8 (nM), Ref: 20472429 Ki: 3.8 (nM), Ref: 21314129 Ki: 3.8 (nM), Ref: 21723123 Ki: 3.8 (nM), Ref: 23965175 Ki: 3.8 (nM), Ref: 24513184
TCMC2174	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 1460 (nM), Ref: 16039848 Ki: 1460 (nM), Ref: 17125255 Ki: 1460 (nM), Ref: 17376683 Ki: 1460 (nM), Ref: 17475500 Ki: 1460 (nM), Ref: 18640037 Ki: 1460 (nM), Ref: 18406497 Ki: 1460 (nM), Ref: 19398204 Ki: 1460 (nM), Ref: 20028100 Ki: 1460 (nM), Ref: 20472429 Ki: 1460 (nM), Ref: 21506569 Ki: 1460 (nM), Ref: 22443141
TCMC2174	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 250 (nM), Ref: 15686895 Ki: 250 (nM), Ref: 15686894 Ki: 250 (nM), Ref: 15686931 Ki: 250 (nM), Ref: 15546717 Ki: 250 (nM), Ref: 16539401 Ki: 250 (nM), Ref: 16459077 Ki: 250 (nM), Ref: 17125255 Ki: 250 (nM), Ref: 17228881 Ki: 250 (nM), Ref: 17376683 Ki: 250 (nM), Ref: 17475500 Ki: 250 (nM), Ref: 19317447 Ki: 250 (nM), Ref: 19124253 Ki: 250 (nM), Ref: 19193158 Ki: 250 (nM), Ref: 18990571 Ki: 250 (nM), Ref: 19338333 Ki: 250 (nM), Ref: 18640037 Ki: 250 (nM), Ref: 18644716 Ki: 250 (nM), Ref: 19398204 Ki: 250 (nM), Ref: 19450983 Ki: 250 (nM), Ref: 19520577 Ki: 250 (nM), Ref: 19539481 Ki: 250 (nM), Ref: 19827837 Ki: 250 (nM), Ref: 20028100 Ki: 250 (nM), Ref: 20201556 Ki: 250 (nM), Ref: 20472429 Ki: 250 (nM), Ref: 20624682 Ki: 250 (nM), Ref: 21208801 Ki: 250 (nM), Ref: 21251841 Ki: 250 (nM), Ref: 21300547 Ki: 250 (nM), Ref: 21314129 Ki: 250 (nM), Ref: 21332115 Ki: 250 (nM), Ref: 19435663 Ki: 250 (nM), Ref: 21506569 Ki: 250 (nM), Ref: 21723123 Ki: 250 (nM), Ref: 21757360 Ki: 250 (nM), Ref: 22285172 Ki: 250 (nM), Ref: 22443141 Ki: 250 (nM), Ref: 23391336 Ki: 250 (nM), Ref: 22883029 Ki: 250 (nM), Ref: 23867389 Ki: 250 (nM), Ref: 23965175 Ki: 250 (nM), Ref: 24513184 Ki: 250 (nM), Ref: 24792813 Ki: 250 (nM), Ref: 25129169 Ki: 250 (nM), Ref: 25533402 Ki: 250 (nM), Ref: 25773015 Ki: 250 (nM), Ref: 25882523 Ki: 250 (nM), Ref: 26525863 Ki: 250 (nM), Ref: 26691758 Ki: 250 (nM), Ref: 26850377 Ki: 250 (nM), Ref: 26920803
TCMC2174	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 0.87 (nM), Ref: 15686895 Ki: 0.9 (nM), Ref: 17125255 Ki: 0.9 (nM), Ref: 17376683 Ki: 0.9 (nM), Ref: 17475500 Ki: 0.9 (nM), Ref: 18640037 Ki: 0.87 (nM), Ref: 18406497 Ki: 0.9 (nM), Ref: 20028100 Ki: 0.9 (nM), Ref: 20472429 Ki: 0.9 (nM), Ref: 21395315 Ki: 0.9 (nM), Ref: 19435663 Ki: 0.9 (nM), Ref: 21506569 Ki: 0.9 (nM), Ref: 22443141 Ki: 0.9 (nM), Ref: 23867389 Ki: 0.9 (nM), Ref: 23965175 Ki: 0.9 (nM), Ref: 24287559
TCMC2174	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4900 (nM), Ref: 15686931 Ki: 4900 (nM), Ref: 17125255 Ki: 4900 (nM), Ref: 17376683 Ki: 4900 (nM), Ref: 17475500 Ki: 4900 (nM), Ref: 18990571 Ki: 4900 (nM), Ref: 18640037 Ki: 4900 (nM), Ref: 20028100 Ki: 4900 (nM), Ref: 20472429
TCMC2174	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 63 (nM), Ref: 16302824 Ki: 63 (nM), Ref: 17125255 Ki: 63 (nM), Ref: 17376683 Ki: 63 (nM), Ref: 17475500 Ki: 63 (nM), Ref: 18640037 Ki: 63 (nM), Ref: 18644716 Ki: 63 (nM), Ref: 19539481 Ki: 63 (nM), Ref: 20028100 Ki: 63 (nM), Ref: 20472429 Ki: 63 (nM), Ref: 21300547
TCMC2174	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 30 (nM), Ref: 16302824 Ki: 30 (nM), Ref: 17125255 Ki: 30 (nM), Ref: 17475500 Ki: 30 (nM), Ref: 18640037 Ki: 30 (nM), Ref: 18644716 Ki: 30 (nM), Ref: 19539481 Ki: 30 (nM), Ref: 20028100 Ki: 30 (nM), Ref: 20472429 Ki: 30 (nM), Ref: 21300547
TCMC2174	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 45 (nM), Ref: 17228881 Ki: 45 (nM), Ref: 17475500 Ki: 45 (nM), Ref: 19193158 Ki: 45 (nM), Ref: 18640037 Ki: 45 (nM), Ref: 20028100 Ki: 45 (nM), Ref: 20472429 Ki: 45 (nM), Ref: 21208801
TCMC2174	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 47 (nM), Ref: 20028100
TCMC654	TCMT915	Retinoid X receptor gamma	Homo sapiens	Ki: 27 (nM), Ref: 10.1016/S0960-894X(97)00420-4 Ki: 14 (nM), Ref: 8765503 Ki: 11 (nM), Ref: 9435893
TCMC654	TCMT735	Retinoid X receptor alpha	Homo sapiens	Ki: 8 (nM), Ref: 8765503 Ki: 12 (nM), Ref: 9435893 IC50: 29 (nM), Ref: 15317450
TCMC654	TCMT914	Retinoid X receptor beta	Homo sapiens	Ki: 9 (nM), Ref: 8765503 Ki: 3.8 (nM), Ref: 9435893
TCMC654	TCMT912	Retinoic acid receptor gamma	Homo sapiens	Ki: 1 (nM), Ref: 9435893
TCMC1820	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 1000 (nM), Ref: 25060641 Ki: 35 (nM), Ref: 25060641
TCMC1472	TCMT105	Solute carrier family 15 member 2	Homo sapiens	Ki: 10000 (nM), Ref: 21741846 Ki: 10000 (nM), Ref: 21741846
TCMC950	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref:
TCMC950	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref:
TCMC806	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8600 (nM), Ref: 15664814
TCMC260	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 1160 (nM), Ref: 24074876
TCMC260	TCMT209	11-beta-hydroxysteroid dehydrogenase 2	Homo sapiens	IC50: 490 (nM), Ref: 24074876
TCMC2032	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 5950 (nM), Ref: 18042384 Ki: 5950 (nM), Ref: 19317447 Ki: 5950 (nM), Ref: 19124253 Ki: 5950 (nM), Ref: 19338333 Ki: 5950 (nM), Ref: 19520577 Ki: 5950 (nM), Ref: 19846301 Ki: 5959 (nM), Ref: 20624682 Ki: 5950 (nM), Ref: 21208801 Ki: 5950 (nM), Ref: 21377369 Ki: 5950 (nM), Ref: 21757360 Ki: 5950 (nM), Ref: 22285172 Ki: 5959 (nM), Ref: 22386980 Ki: 5959 (nM), Ref: 23181552 Ki: 5959 (nM), Ref: 23391336 Ki: 5950 (nM), Ref: 22974493 Ki: 5959 (nM), Ref: 22883029 Ki: 5959 (nM), Ref: 24314394 Ki: 5950 (nM), Ref: 24560739 Ki: 5950 (nM), Ref: 24689792 Ki: 5959 (nM), Ref: 24792813 Ki: 5959 (nM), Ref: 25129169 Ki: 5959 (nM), Ref: 25773015 Ki: 5959 (nM), Ref: 25882523 Ki: 5959 (nM), Ref: 26174556 Ki: 5950 (nM), Ref: 26525863 Ki: 5959 (nM), Ref: 26691758 Ki: 5959 (nM), Ref: 26850377 Ki: 5950 (nM), Ref: 26810710 Ki: 5959 (nM), Ref: 26832216 Ki: 5959 (nM), Ref: 26920803
TCMC2032	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 103 (nM), Ref: 18042384 Ki: 103 (nM), Ref: 22974493 Ki: 103 (nM), Ref: 24560739 Ki: 103 (nM), Ref: 24689792 Ki: 103 (nM), Ref: 26810710
TCMC2032	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 633 (nM), Ref: 18042384 Ki: 633 (nM), Ref: 24560739 Ki: 633 (nM), Ref: 24689792 Ki: 633 (nM), Ref: 26810710
TCMC2032	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 935 (nM), Ref: 21208801 Ki: 935 (nM), Ref: 24689792
TCMC2032	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7920 (nM), Ref: 24689792
TCMC2032	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7210 (nM), Ref: 24689792
TCMC2032	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 10 (nM), Ref: 24689792
TCMC2032	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 773 (nM), Ref: 24689792
TCMC2032	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 3600 (nM), Ref: 25537270
TCMC698	TCMT794	Type-1 angiotensin II receptor	Homo sapiens	Ki: 0.9 (nM), Ref: 20146480 Ki: 0.24 (nM), Ref: 26824643 IC50: 0.7244 (nM), Ref: 26824643 Ki: 0.16 (nM), Ref: 26824643
TCMC698	TCMT957	Angiotensin II type 2 (AT-2) receptor	Homo sapiens	Ki: 0.2 (nM), Ref: 26810314
TCMC1789	TCMT115	Cannabinoid CB1 receptor	Homo sapiens	Ki: 1100 (nM), Ref: 16570929 Ki: 1100 (nM), Ref: 19361197
TCMC566	TCMT308	Oxoeicosanoid receptor 1	Homo sapiens	IC50: 3 (nM), Ref: 21377873
TCMC1437	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 330 (nM), Ref: 18667313 IC50: 14 (nM), Ref:
TCMC1437	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 690 (nM), Ref: 18667313 IC50: 3800 (nM), Ref: 25221653 IC50: 61 (nM), Ref: 26487917
TCMC929	TCMT116	Mu opioid receptor	Homo sapiens	Ki: 6300 (nM), Ref: 17616524
TCMC2209	TCMT597	Solute carrier family 28 member 3	Homo sapiens	Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705
TCMC2209	TCMT710	Sodium/nucleoside cotransporter 1	Homo sapiens	Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705
TCMC1542	TCMT336	Indoleamine 2,3-dioxygenase	Homo sapiens	IC50: 1000 (nM), Ref: 18318466
TCMC1542	TCMT563	Dual specificity phosphatase Cdc25B	Homo sapiens	IC50: 3380 (nM), Ref: 19028102
TCMC1542	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 200 (nM), Ref: 20853847 Ki: 1500 (nM), Ref: 22996261 Ki: 470 (nM), Ref: 22996261
TCMC1542	TCMT186	Monoamine oxidase B	Homo sapiens	Ki: 400 (nM), Ref: 22071524
TCMC1813	TCMT36	Serotonin 1a (5-HT1a) receptor	Homo sapiens	Ki: 0.91 (nM), Ref: 25759032 Ki: 1.8 (nM), Ref: 26227779
TCMC1813	TCMT160	Serotonin 7 (5-HT7) receptor	Homo sapiens	Ki: 2.12 (nM), Ref: 25759032
TCMC583	TCMT855	Nuclear receptor ROR-alpha	Homo sapiens	Ki: 12 (nM), Ref: 10.1039/C3MD00005B
TCMC583	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	Ki: 10 (nM), Ref: 10.1039/C3MD00005B
TCMC1133	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030
TCMC1133	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030
TCMC1133	TCMT187	Androgen Receptor	Homo sapiens	IC50: 19.1 (nM), Ref: 16309907
TCMC1133	TCMT99	Testis-specific androgen-binding protein	Homo sapiens	IC50: 50 (nM), Ref: 17149875
TCMC1133	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346
TCMC1133	TCMT910	Estrogen-related receptor beta	Homo sapiens	IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346
TCMC1133	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261
TCMC1133	TCMT974	G-protein coupled estrogen receptor 1	Homo sapiens	Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A
TCMC1471	TCMT976	Leukotriene B4 receptor 1	Homo sapiens	IC50: 32 (nM), Ref: 10.1016/S0960-894X(01)80853-2
TCMC710	TCMT249	Cyclin-dependent kinase 6	Homo sapiens	IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554
TCMC710	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 710 (nM), Ref: 18533708
TCMC710	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 800 (nM), Ref: 19414254
TCMC710	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5200 (nM), Ref: 19592245
TCMC710	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 795 (nM), Ref: 20696580
TCMC710	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 427 (nM), Ref: 20696580
TCMC710	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC710	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1450 (nM), Ref: 23411073
TCMC710	TCMT128	Tankyrase-2	Homo sapiens	IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272
TCMC710	TCMT129	Tankyrase-1	Homo sapiens	IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272
TCMC710	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844
TCMC710	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431
TCMC349	TCMT203	Glucose-6-phosphate 1-dehydrogenase	Homo sapiens	IC50: 5300 (nM), Ref: 22506561
TCMC784	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 100 (nM), Ref: 26003344
TCMC784	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1090 (nM), Ref: 26003344
TCMC2100	TCMT599	Ubiquitin-conjugating enzyme E2 N	Homo sapiens	IC50: 6425 (nM), Ref: IC50: 6200 (nM), Ref:
TCMC1543	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 840 (nM), Ref: 16248836 Ki: 2500 (nM), Ref: 16248836
TCMC1297	TCMT632	Purine nucleoside phosphorylase	Homo sapiens	Ki: 5000 (nM), Ref: 31484
TCMC1834	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9060 (nM), Ref: 21402476
TCMC1834	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8030 (nM), Ref: 21402476
TCMC770	TCMT588	D-amino-acid oxidase	Homo sapiens	Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755
TCMC1343	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385
TCMC1343	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7800 (nM), Ref: 18579385
TCMC1343	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8200 (nM), Ref: 18579385