TCM Putative Target References: TCMFx4077


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC1180
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5210 (nM), Ref: 22487176
Ki: 5100 (nM), Ref: 22487176
TCMC1180
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9300 (nM), Ref: 22487176
Ki: 9200 (nM), Ref: 22487176
TCMC1180
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5540 (nM), Ref: 22487176
Ki: 5630 (nM), Ref: 22487176
TCMC1180
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6590 (nM), Ref: 22487176
Ki: 6650 (nM), Ref: 22487176
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC1424
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2100 (nM), Ref: 17994701
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC1376
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 40 (nM), Ref: 11678654
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1925
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 18798681
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1201
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 3150 (nM), Ref: 8576921
TCMC1201
TCMT132 Butyrylcholinesterase Homo sapiens Ki: 6900 (nM), Ref: 19879672
TCMC1201
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1201
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 40 (nM), Ref: 20696580
TCMC1201
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1201
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1201
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 568.3 (nM), Ref: 26498393
TCMC1201
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 24.5 (nM), Ref: 26498393
TCMC1201
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 41.8 (nM), Ref: 26498393
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC469
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 100 (nM), Ref: 22921742
TCMC1015
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 4320 (nM), Ref:
TCMC2196
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 64 (nM), Ref: 22819942
IC50: 64 (nM), Ref: 23146282
TCMC2196
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 150 (nM), Ref: 22819942
TCMC2196
TCMT336 Indoleamine 2,3-dioxygenase Homo sapiens IC50: 53.7 (nM), Ref: 24099220
IC50: 7150 (nM), Ref: 24099220
Ki: 4810 (nM), Ref: 24099220
TCMC1597
TCMT807 Solute carrier family 22 member 12 Homo sapiens IC50: 2000 (nM), Ref: 17325024
Ki: 5740 (nM), Ref: 17325024
TCMC1597
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2927.18 (nM), Ref:
TCMC1597
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2988.26 (nM), Ref:
TCMC1597
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 1600 (nM), Ref: 24900447
TCMC1597
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 1600 (nM), Ref: 26322379
TCMC1597
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 4300 (nM), Ref: 26602279
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC418
TCMT223 Aldose reductase Homo sapiens IC50: 78 (nM), Ref: 22236472
TCMC418
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 240 (nM), Ref: 22236472
TCMC418
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4700 (nM), Ref: 22921742
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC183
TCMT188 Dihydrofolate reductase Homo sapiens IC50: 500 (nM), Ref: 26979156
TCMC1377
TCMT186 Monoamine oxidase B Homo sapiens Ki: 3000 (nM), Ref: 16137882
Ki: 3000 (nM), Ref: 19342233
IC50: 7943.28 (nM), Ref: 20934874
Ki: 5340 (nM), Ref: 21134756
Ki: 3000 (nM), Ref: 21778064
Ki: 2000 (nM), Ref: 24140951
TCMC1377
TCMT208 Monoamine oxidase A Homo sapiens Ki: 8380 (nM), Ref: 21134756
TCMC732
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 5900 (nM), Ref: 21561086
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC1179
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 19592245
IC50: 5900 (nM), Ref: 19592245
TCMC1179
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8 (nM), Ref: 20413308
IC50: 10000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC1179
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1890 (nM), Ref: 22487176
Ki: 1880 (nM), Ref: 22487176
TCMC1179
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8710 (nM), Ref: 22487176
Ki: 8800 (nM), Ref: 22487176
TCMC1179
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4130 (nM), Ref: 22487176
Ki: 4220 (nM), Ref: 22487176
TCMC1179
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7220 (nM), Ref: 22487176
Ki: 7330 (nM), Ref: 22487176
TCMC1179
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 1380.38 (nM), Ref: 23574272
IC50: 1400 (nM), Ref: 23574272
TCMC1179
TCMT128 Tankyrase-2 Homo sapiens IC50: 147.91 (nM), Ref: 23574272
IC50: 140 (nM), Ref: 23574272
TCMC1179
TCMT129 Tankyrase-1 Homo sapiens IC50: 323.59 (nM), Ref: 23574272
IC50: 320 (nM), Ref: 23574272
IC50: 323.59 (nM), Ref: 24116873
IC50: 330 (nM), Ref: 24116873
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC1371
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 4 (nM), Ref: 26562543
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC1175
TCMT186 Monoamine oxidase B Homo sapiens IC50: 2870 (nM), Ref: 20045650
TCMC1175
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC987
TCMT885 Lysine-specific demethylase 2A Homo sapiens Ki: 1970 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 23964788
TCMC987
TCMT965 Lysine-specific demethylase 7 Homo sapiens IC50: 2100 (nM), Ref: 22724510
TCMC987
TCMT884 Histone lysine demethylase PHF8 Homo sapiens IC50: 550 (nM), Ref: 22724510
IC50: 550 (nM), Ref: 23964788
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1174
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 850 (nM), Ref: 15689157
IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1174
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC469
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 5.4 (ug/ml), Ref: 16643034
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1801
TCMT1136 Neuraminidase Influenza A virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2383
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.96 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1424
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 27.95 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC1925
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 23.3 (ug/ml), Ref: 9748372
TCMC2459
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37.5 (ug/ml), Ref: 9748372
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2196
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 10 (ug/ml), Ref: 22819942
MIC: 0.5 (ug/ml), Ref: 26253635
TCMC2196
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 1 (ug/ml), Ref: 23360475
MIC: 1 (ug/ml), Ref: 26253635
TCMC2196
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6 (ug/ml), Ref: 26253635
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC732
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 9 (ug/ml), Ref: 9748372
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 0.087 (ug/ml), Ref: 9249972
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2655
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 IC50: 7 (ug/ml), Ref: 2828553
TCMC2655
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 IC50: 7 (ug/ml), Ref: 2828553
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2695
TCMT1251 Candida albicans Candida albicans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0135-6
TCMC582
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 16680159
TCMC1915
TCMT1347 Human rhinovirus 16 Human rhinovirus 16 IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1333 Human rhinovirus 1A Human rhinovirus 1A IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1241 Human rhinovirus 14 Human rhinovirus 14 IC50: 0.02 (ug/ml), Ref: 17116681
IC50: 100 (nM), Ref: 23977995
TCMC1801
TCMT1449 Influenza A virus Influenza A virus IC50: 1 (ug/ml), Ref: 14987066
IC50: 2.4 (nM), Ref: 19919060
IC50: 3.41 (nM), Ref: 15974612
IC50: 3.79 (nM), Ref: 16532013
IC50: 7.03 (nM), Ref: 19101157
IC50: 30 (nM), Ref: 25305333
IC50: 1.08 (nM), Ref: 9784165
IC50: 0.85 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 2.27 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 93.92 (nM), Ref: 20430633
IC50: 99.57 (nM), Ref: 20430633
IC50: 0.54 (nM), Ref: 20430633
IC50: 94.4 (nM), Ref: 20430633
IC50: 0.49 (nM), Ref: 20411974
IC50: 0.25 (nM), Ref: 20384296
IC50: 1 (nM), Ref: IC50: 95.43 (nM), Ref: 9461668
IC50: 78.12 (nM), Ref: 9461668
IC50: 75.29 (nM), Ref: 9461668
IC50: 1.84 (nM), Ref: 20166736
IC50: 1.59 (nM), Ref: 24673739
IC50: 0.34 (nM), Ref: 23675610
IC50: 0.25 (nM), Ref: 1431945
IC50: 3.64 (nM), Ref: 11170656
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC582
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 1602301
TCMC582
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 24927000
MIC: 62.5 (ug/ml), Ref: 24927000
TCMC582
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 24927000
TCMC1915
TCMT1348 Human rhinovirus 2 Human rhinovirus 2 IC50: 0.01 (ug/ml), Ref: 23920485
IC50: 100 (nM), Ref: 23977995
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1174
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 55 (ug/ml), Ref: 25564380
TCMC1174
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.6 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC1801
TCMT1162 Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1)) Ki: 1.1 (nM), Ref: IC50: 0.1 (nM), Ref: 23398362
IC50: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1164 Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1)) Ki: 4.9 (nM), Ref: 20579892
IC50: 4.9 (nM), Ref: 19708637
IC50: 3.7 (nM), Ref:
TCMC1801
TCMT1161 Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1)) Ki: 7.9 (nM), Ref: 20579892
IC50: 10.8 (nM), Ref: 10.6019/CHEMBL1201861
TCMC1801
TCMT1163 Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) IC50: 0.3 (nM), Ref: 9322359
IC50: 0.2 (nM), Ref: Ki: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/swine/Belzig/2/2001(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/New Caledonia/20/1999(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Yamagata/32/1989(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC1801
TCMT1151 Neuraminidase Influenza B virus IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Hong Kong/1/1968(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1160 Neuraminidase Influenza A virus (A/Aichi/2/1968(H3N2)) IC50: 1.55 (nM), Ref: 20185316
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/whooper swan/Mongolia/1/2009(H5N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Wisconsin/67/2005(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Shandong/LY/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/Perth/16/2009(H3N2)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1151 Neuraminidase Influenza B virus (B/Memphis/3/89) IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Sandong/Li/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC2602
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 42 (nM), Ref: 9917283
IC50: 67 (nM), Ref: 9917283
TCMC2602
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 42 (nM), Ref: 9917283
IC50: 67 (nM), Ref: 9917283
TCMC1179
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (nM), Ref: 19097788
TCMC1801
TCMT1296 Influenza A virus H3N2 Influenza A virus H3N2 IC50: 18.5 (nM), Ref: 12542349
TCMC1915
TCMT1285 Human coxsackievirus B3 Human coxsackievirus B3 IC50: 2.5 (nM), Ref: 13678412