References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1881
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
Ki: 2.5 (nM), Ref: 11327599 Ki: 6.4 (nM), Ref: 21596562 |
TCMC1881
|
TCMT152 |
Protein kinase C beta |
Homo sapiens |
Ki: 1.8 (nM), Ref: 11327599 |
TCMC1881
|
TCMT153 |
Protein kinase C gamma |
Homo sapiens |
Ki: 4.9 (nM), Ref: 11327599 |
TCMC1881
|
TCMT154 |
Protein kinase C delta |
Homo sapiens |
Ki: 0.8 (nM), Ref: 11327599 |
TCMC1881
|
TCMT155 |
Protein kinase C epsilon |
Homo sapiens |
Ki: 0.45 (nM), Ref: 11327599 |
TCMC2080
|
TCMT87 |
Cytochrome P450 2C9 |
Homo sapiens |
IC50: 8200 (nM), Ref: 23260576 |
TCMC2080
|
TCMT278 |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
IC50: 8500 (nM), Ref: 23401473 |
TCMC2080
|
TCMT277 |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
IC50: 5000 (nM), Ref: 23401473 |
TCMC2080
|
TCMT276 |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
IC50: 800 (nM), Ref: 23401473 |
TCMC1495
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
TCMC1495
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
TCMC1495
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC715
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC715
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC715
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC619
|
TCMT293 |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki: 158.49 (nM), Ref: 18077164 |
TCMC619
|
TCMT291 |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
Ki: 7079.46 (nM), Ref: 18077164 |
TCMC619
|
TCMT551 |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki: 8511.38 (nM), Ref: 18077164 |
TCMC619
|
TCMT290 |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
Ki: 9772.37 (nM), Ref: 18077164 |
TCMC619
|
TCMT241 |
Neuronal acetylcholine receptor protein alpha-7 subunit |
Homo sapiens |
Ki: 7943.28 (nM), Ref: 21920761 |
TCMC487
|
TCMT561 |
5'-nucleotidase |
Homo sapiens |
IC50: 8200 (nM), Ref: 24215819 |
TCMC2079
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1490 (nM), Ref: 20674354 |
TCMC2079
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2510 (nM), Ref: 20674354 |
TCMC2079
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6430 (nM), Ref: 20674354 |
TCMC2079
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 8960 (nM), Ref: 20674354 |
TCMC2079
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4080 (nM), Ref: 20674354 |
TCMC2079
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 4560 (nM), Ref: 20674354 |
TCMC2079
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 9700 (nM), Ref: 20674354 |
TCMC2079
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4710 (nM), Ref: 20674354 |
TCMC2079
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9050 (nM), Ref: 20674354 |
TCMC2079
|
TCMT225 |
Carbonic anhydrase XIII |
Homo sapiens |
Ki: 4820 (nM), Ref: 20674354 |
TCMC2079
|
TCMT87 |
Cytochrome P450 2C9 |
Homo sapiens |
Ki: 5000 (nM), Ref: 16248836 |
TCMC2079
|
TCMT278 |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
IC50: 9700 (nM), Ref: 23401473 |
TCMC2079
|
TCMT277 |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
IC50: 2700 (nM), Ref: 23401473 |
TCMC2079
|
TCMT276 |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
IC50: 4500 (nM), Ref: 23401473 |
TCMC1480
|
TCMT107 |
Glutamate receptor ionotropic kainate 2 |
Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
TCMC1480
|
TCMT108 |
Glutamate receptor ionotropic, AMPA 1 |
Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
TCMC1480
|
TCMT109 |
Glutamate receptor ionotropic, AMPA 2 |
Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
TCMC1480
|
TCMT110 |
Glutamate receptor ionotropic, AMPA 4 |
Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
TCMC1480
|
TCMT111 |
Glutamate receptor ionotropic kainate 5 |
Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
TCMC1480
|
TCMT660 |
Metabotropic glutamate receptor 8 |
Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
TCMC1480
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
TCMC1480
|
TCMT653 |
Metabotropic glutamate receptor 1 |
Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT654 |
Metabotropic glutamate receptor 5 |
Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT657 |
Metabotropic glutamate receptor 4 |
Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT655 |
Metabotropic glutamate receptor 2 |
Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT664 |
Excitatory amino acid transporter 3 |
Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
TCMC1480
|
TCMT656 |
Metabotropic glutamate receptor 3 |
Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
TCMC1982
|
TCMT239 |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
TCMC1982
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
TCMC1982
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
TCMC1982
|
TCMT44 |
Glyoxalase I |
Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
TCMC1982
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
TCMC1982
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
TCMC1982
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
TCMC1982
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
TCMC1982
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
TCMC1982
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
TCMC1982
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
TCMC1982
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
TCMC1982
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
TCMC1982
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
TCMC1982
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
TCMC1982
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
TCMC1982
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
TCMC1982
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
TCMC1982
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
TCMC1982
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
TCMC1982
|
TCMT320 |
Matrix metalloproteinase 3 |
Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
TCMC1982
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
TCMC1982
|
TCMT322 |
Matrix metalloproteinase 13 |
Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
TCMC1982
|
TCMT422 |
CaM kinase II beta |
Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
TCMC1982
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1982
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
TCMC1982
|
TCMT784 |
Vasopressin V2 receptor |
Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
TCMC1982
|
TCMT785 |
Interleukin-8 receptor A |
Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
TCMC1982
|
TCMT786 |
C-C chemokine receptor type 4 |
Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
TCMC1982
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
TCMC1982
|
TCMT601 |
Thrombin |
Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
TCMC1982
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
TCMC1982
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
TCMC1982
|
TCMT791 |
Protein kinase N1 |
Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
TCMC1982
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
TCMC1982
|
TCMT462 |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
TCMC1982
|
TCMT445 |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
TCMC1982
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
TCMC1982
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
TCMC1982
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
TCMC1982
|
TCMT388 |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
TCMC1982
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
TCMC1982
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
TCMC1982
|
TCMT402 |
ALK tyrosine kinase receptor |
Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
TCMC1982
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
TCMC1982
|
TCMT592 |
Xanthine dehydrogenase |
Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
TCMC1982
|
TCMT793 |
Liver glycogen phosphorylase |
Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
TCMC1982
|
TCMT33 |
Cytochrome P450 3A4 |
Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
TCMC1982
|
TCMT217 |
Cytochrome P450 2C8 |
Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
TCMC1982
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
TCMC2105
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2105
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1428
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 509 (nM), Ref: 20696580 |
TCMC1428
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 88 (nM), Ref: 20696580 |
TCMC1428
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
TCMC1788
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT126 |
Telomerase reverse transcriptase |
Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
TCMC1788
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
TCMC2081
|
TCMT278 |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
IC50: 9000 (nM), Ref: 23401473 |
TCMC2081
|
TCMT276 |
Solute carrier organic anion transporter family member 2B1 |
Homo sapiens |
IC50: 3600 (nM), Ref: 23401473 |
TCMC1496
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1496
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1496
|
TCMT164 |
Cyclooxygenase-1 |
Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
TCMC1611
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1611
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |