Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
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TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
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TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5 |
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TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
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TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
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TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT1455 | Mycobacterium tuberculosis H37Rv | Mycobacterium tuberculosis H37Rv |
MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8 MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8 |
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TCMT1229 | Enterococcus faecalis | Enterococcus faecalis |
MIC: 16 (ug/ml), Ref: 23534483 |
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TCMT1176 | Streptococcus pneumoniae | Streptococcus pneumoniae |
MIC: 1 (ug/ml), Ref: 23534483 |
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TCMT1218 | Staphylococcus aureus | Staphylococcus aureus |
MIC: 2 (ug/ml), Ref: 23534483 MIC: 4 (ug/ml), Ref: 23534483 |
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TCMT1218 | Staphylococcus aureus | Staphylococcus aureus |
MIC: 0.5 (ug/ml), Ref: 15863332 |
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TCMT1093 | Enoyl-acyl-carrier protein reductase | Plasmodium falciparum |
Ki: 16 (nM), Ref: 17263522 |
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TCMT1246 | Escherichia coli | Escherichia coli |
MIC: 100 (ug/ml), Ref: 3430167 |
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TCMT1284 | Penicillium expansum | Penicillium expansum |
MIC: 50 (ug/ml), Ref: 3430167 |
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TCMT1438 | Plasmodium falciparum | Plasmodium falciparum 3D7 |
IC50: 50.1 (nM), Ref: 20349996 IC50: 28 (nM), Ref: 20349996 |
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TCMT1438 | Plasmodium falciparum | Plasmodium falciparum |
IC50: 50.1 (nM), Ref: 20349996 IC50: 28 (nM), Ref: 20349996 |