References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC486
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 9500 (nM), Ref: 18579385 |
TCMC1480
|
TCMT107 |
Glutamate receptor ionotropic kainate 2 |
Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
TCMC1480
|
TCMT108 |
Glutamate receptor ionotropic, AMPA 1 |
Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
TCMC1480
|
TCMT109 |
Glutamate receptor ionotropic, AMPA 2 |
Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
TCMC1480
|
TCMT110 |
Glutamate receptor ionotropic, AMPA 4 |
Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
TCMC1480
|
TCMT111 |
Glutamate receptor ionotropic kainate 5 |
Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
TCMC1480
|
TCMT660 |
Metabotropic glutamate receptor 8 |
Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
TCMC1480
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
TCMC1480
|
TCMT653 |
Metabotropic glutamate receptor 1 |
Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT654 |
Metabotropic glutamate receptor 5 |
Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT657 |
Metabotropic glutamate receptor 4 |
Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT655 |
Metabotropic glutamate receptor 2 |
Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT664 |
Excitatory amino acid transporter 3 |
Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
TCMC1480
|
TCMT656 |
Metabotropic glutamate receptor 3 |
Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
TCMC949
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8900 (nM), Ref: 19911821 |
TCMC949
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 48 (nM), Ref: 19911821 |
TCMC949
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9100 (nM), Ref: 19911821 |
TCMC949
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 3300 (nM), Ref: 19911821 |
TCMC949
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 2000 (nM), Ref: 19911821 |
TCMC949
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 5200 (nM), Ref: 19911821 |
TCMC949
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9400 (nM), Ref: 19911821 |
TCMC949
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 6800 (nM), Ref: 19911821 |
TCMC949
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 5600 (nM), Ref: 19911821 |
TCMC949
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270 |
TCMC949
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270 |
TCMC1083
|
TCMT38 |
Dopamine D2 receptor |
Homo sapiens |
Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867 |
TCMC1083
|
TCMT651 |
Dopamine D3 receptor |
Homo sapiens |
Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329 |
TCMC1083
|
TCMT635 |
Dopamine transporter |
Homo sapiens |
Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523 |
TCMC1083
|
TCMT634 |
Norepinephrine transporter |
Homo sapiens |
IC50: 6.63 (nM), Ref: 14592523 |
TCMC1083
|
TCMT648 |
Dopamine D4 receptor |
Homo sapiens |
Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965 |
TCMC1083
|
TCMT316 |
Melatonin receptor 1A |
Homo sapiens |
Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
TCMC1083
|
TCMT317 |
Melatonin receptor 1B |
Homo sapiens |
Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
TCMC1083
|
TCMT27 |
Dopamine D1 receptor |
Homo sapiens |
Ki: 4470 (nM), Ref: 23134120 |
TCMC1083
|
TCMT8 |
Lysine-specific demethylase 4D-like |
Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC706
|
TCMT563 |
Dual specificity phosphatase Cdc25B |
Homo sapiens |
IC50: 9510 (nM), Ref: 19028102 |
TCMC405
|
TCMT506 |
Protein tyrosine kinase 2 beta |
Homo sapiens |
IC50: 2324 (nM), Ref: |
TCMC226
|
TCMT38 |
Dopamine D2 receptor |
Homo sapiens |
Ki: 3900 (nM), Ref: 10.1016/S0960-894X(97)00194-7 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1839
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
TCMC1839
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
TCMC1839
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
TCMC1839
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
TCMC1839
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
TCMC1839
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1839
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
TCMC1839
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
TCMC1839
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1839
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
TCMC1839
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
TCMC437
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 7200 (nM), Ref: 22668600 |
TCMC437
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 7700 (nM), Ref: 22668600 |
TCMC437
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4900 (nM), Ref: 22668600 |
TCMC437
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 5900 (nM), Ref: 22668600 |
TCMC437
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 4700 (nM), Ref: 22668600 |
TCMC437
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 4900 (nM), Ref: 22668600 |
TCMC49
|
TCMT651 |
Dopamine D3 receptor |
Homo sapiens |
Ki: 500 (nM), Ref: 24559070 |
TCMC49
|
TCMT38 |
Dopamine D2 receptor |
Homo sapiens |
Ki: 5000 (nM), Ref: 24559070 |
TCMC1228
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 5200 (nM), Ref: 18558747 |
TCMC878
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
TCMC878
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
TCMC878
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
TCMC878
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
TCMC878
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
TCMC878
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
TCMC878
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
TCMC878
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
TCMC878
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
TCMC878
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |