References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC619
|
TCMT293 |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki: 158.49 (nM), Ref: 18077164 |
TCMC619
|
TCMT291 |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
Ki: 7079.46 (nM), Ref: 18077164 |
TCMC619
|
TCMT551 |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki: 8511.38 (nM), Ref: 18077164 |
TCMC619
|
TCMT290 |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
Ki: 9772.37 (nM), Ref: 18077164 |
TCMC619
|
TCMT241 |
Neuronal acetylcholine receptor protein alpha-7 subunit |
Homo sapiens |
Ki: 7943.28 (nM), Ref: 21920761 |
TCMC1330
|
TCMT246 |
Histamine H4 receptor |
Homo sapiens |
Ki: 14.45 (nM), Ref: 14640553 Ki: 7.943 (nM), Ref: 15454206 Ki: 12.02 (nM), Ref: 18357976 Ki: 13.4 (nM), Ref: 18459760 Ki: 12.02 (nM), Ref: 20192225 Ki: 60 (nM), Ref: 20452213 Ki: 7.943 (nM), Ref: 21044842 Ki: 12.59 (nM), Ref: 21044842 Ki: 12.02 (nM), Ref: 21348462 Ki: 15.85 (nM), Ref: 22003888 Ki: 9 (nM), Ref: 22153663 Ki: 19.95 (nM), Ref: 10.1039/C2MD20212C Ki: 4.8 (nM), Ref: 25993395 Ki: 8 (nM), Ref: 25993395 Ki: 15.85 (nM), Ref: 10.1039/C5MD00022J |
TCMC1330
|
TCMT242 |
Histamine H3 receptor |
Homo sapiens |
Ki: 5.2 (nM), Ref: 20384344 Ki: 10 (nM), Ref: 21044842 Ki: 11.75 (nM), Ref: 21348462 Ki: 6.31 (nM), Ref: 22003888 Ki: 16 (nM), Ref: 25993395 |
TCMC1330
|
TCMT245 |
Histamine H2 receptor |
Homo sapiens |
Ki: 5000 (nM), Ref: 25993395 |
TCMC1330
|
TCMT244 |
Histamine H1 receptor |
Homo sapiens |
Ki: 6000 (nM), Ref: 25993395 |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC1102
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
TCMC1102
|
TCMT752 |
Casein kinase II alpha |
Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
TCMC1102
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
TCMC1102
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
TCMC1102
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC1102
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
TCMC1102
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
TCMC1102
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
TCMC1102
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
TCMC1102
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
TCMC1102
|
TCMT753 |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
IC50: 142 (nM), Ref: |
TCMC1102
|
TCMT721 |
Heat shock 70 kDa protein 1 |
Homo sapiens |
IC50: 760 (nM), Ref: |
TCMC1102
|
TCMT189 |
Dual specificity protein phosphatase 3 |
Homo sapiens |
IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
TCMC1102
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
TCMC1102
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
TCMC1102
|
TCMT354 |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
TCMC1102
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
TCMC1102
|
TCMT626 |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
TCMC1102
|
TCMT423 |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
TCMC1102
|
TCMT418 |
Ephrin type-B receptor 4 |
Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
TCMC1102
|
TCMT704 |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
TCMC1102
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
TCMC1102
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
TCMC1102
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
TCMC1102
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
TCMC1102
|
TCMT457 |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
TCMC1102
|
TCMT377 |
Insulin receptor |
Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
TCMC1102
|
TCMT536 |
Platelet-derived growth factor receptor beta |
Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
TCMC1102
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
TCMC1102
|
TCMT755 |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
TCMC1102
|
TCMT502 |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
TCMC1102
|
TCMT756 |
Mitogen-activated protein kinase kinase kinase 8 |
Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
TCMC1102
|
TCMT739 |
G-protein coupled receptor 35 |
Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
TCMC1102
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
TCMC1102
|
TCMT225 |
Carbonic anhydrase XIII |
Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
TCMC1102
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1566
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 830 (nM), Ref: 22668600 |
TCMC1566
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 810 (nM), Ref: 22668600 |
TCMC1566
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 850 (nM), Ref: 22668600 |
TCMC1566
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 820 (nM), Ref: 22668600 |
TCMC1566
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 800 (nM), Ref: 22668600 |
TCMC1566
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 780 (nM), Ref: 22668600 |
TCMC878
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
TCMC878
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
TCMC878
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
TCMC878
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
TCMC878
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
TCMC878
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
TCMC878
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
TCMC878
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
TCMC878
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
TCMC878
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |
TCMC1378
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
TCMC1378
|
TCMT734 |
Matrix metalloproteinase 12 |
Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |