TCM Putative Target References: TCMF5461


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1881
TCMT151 Protein kinase C alpha Homo sapiens Ki: 2.5 (nM), Ref: 11327599
Ki: 6.4 (nM), Ref: 21596562
TCMC1881
TCMT152 Protein kinase C beta Homo sapiens Ki: 1.8 (nM), Ref: 11327599
TCMC1881
TCMT153 Protein kinase C gamma Homo sapiens Ki: 4.9 (nM), Ref: 11327599
TCMC1881
TCMT154 Protein kinase C delta Homo sapiens Ki: 0.8 (nM), Ref: 11327599
TCMC1881
TCMT155 Protein kinase C epsilon Homo sapiens Ki: 0.45 (nM), Ref: 11327599
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC159
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 2000 (nM), Ref: 22696418
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1372
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2330 (nM), Ref: 22245047
TCMC1372
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3630 (nM), Ref: 22245047
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC244
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 7900 (nM), Ref: 15916432
TCMC244
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 8300 (nM), Ref: 15658857
IC50: 8298.51 (nM), Ref: 19110342
TCMC2013
TCMT223 Aldose reductase Homo sapiens IC50: 2700 (nM), Ref: 22261024
TCMC37
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC715
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1180
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5210 (nM), Ref: 22487176
Ki: 5100 (nM), Ref: 22487176
TCMC1180
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9300 (nM), Ref: 22487176
Ki: 9200 (nM), Ref: 22487176
TCMC1180
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5540 (nM), Ref: 22487176
Ki: 5630 (nM), Ref: 22487176
TCMC1180
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6590 (nM), Ref: 22487176
Ki: 6650 (nM), Ref: 22487176
TCMC1803
TCMT337 Exportin-1 Homo sapiens IC50: 1600 (nM), Ref: 20493693
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC962
TCMT45 Beta amyloid A4 protein Homo sapiens Ki: 0.208 (nM), Ref: 17004725
IC50: 800 (nM), Ref: 17270435
IC50: 3900 (nM), Ref: 26099993
TCMC962
TCMT566 Nitric oxide synthase, inducible Homo sapiens IC50: 6000 (nM), Ref: 18077363
TCMC962
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 4300 (nM), Ref: 18249473
TCMC962
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 8500 (nM), Ref: 19128977
TCMC962
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2410 (nM), Ref: 20674354
TCMC962
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 380 (nM), Ref: 20674354
TCMC962
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4970 (nM), Ref: 20674354
TCMC962
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9460 (nM), Ref: 20674354
TCMC962
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 9940 (nM), Ref: 20674354
TCMC962
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9300 (nM), Ref: 20674354
TCMC962
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4050 (nM), Ref: 20674354
TCMC962
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3480 (nM), Ref: 20674354
TCMC962
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 6850 (nM), Ref: 20674354
TCMC962
TCMT44 Glyoxalase I Homo sapiens Ki: 10000 (nM), Ref: 21237663
TCMC962
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 7410 (nM), Ref:
TCMC962
TCMT46 Coagulation factor III Homo sapiens IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5
IC50: 199.63 (nM), Ref: 23199480
TCMC962
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 8600 (nM), Ref: 23245570
TCMC962
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 4501 (nM), Ref: 23800686
TCMC962
TCMT570 Aminopeptidase N Homo sapiens IC50: 10000 (nM), Ref: 23860593
TCMC962
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 3900 (nM), Ref: 24920381
IC50: 500 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
TCMC962
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 8100 (nM), Ref: 24920381
TCMC962
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 600 (nM), Ref: 24920381
IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5300 (nM), Ref: 25088549
TCMC962
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 25730130
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC416
TCMT207 Beta-secretase 1 Homo sapiens IC50: 4500 (nM), Ref: 14592472
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1439
TCMT588 D-amino-acid oxidase Homo sapiens IC50: 2000 (nM), Ref: 23683589
TCMC1439
TCMT159 Tyrosinase Homo sapiens IC50: 9150 (nM), Ref: 26386819
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1411
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1261 (nM), Ref: 20696580
TCMC1411
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 56 (nM), Ref: 20696580
TCMC1411
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 17 (nM), Ref: 20696580
TCMC1411
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 212.9 (nM), Ref: 26498393
TCMC1411
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.4 (nM), Ref: 26498393
TCMC1411
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 54.9 (nM), Ref: 26498393
Ki: 220 (nM), Ref: 26498393
TCMC1411
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 440 (nM), Ref: 26498393
TCMC895
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 8990 (nM), Ref:
TCMC895
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 3012 (nM), Ref: IC50: 2197 (nM), Ref:
TCMC895
TCMT608 Solute carrier family 22 member 3 Homo sapiens IC50: 410 (nM), Ref: 23241029
TCMC895
TCMT213 Solute carrier family 22 member 1 Homo sapiens IC50: 210 (nM), Ref: 23241029
TCMC895
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 400 (nM), Ref: 23241029
TCMC895
TCMT310 Multidrug and toxin extrusion protein 2 Homo sapiens IC50: 500 (nM), Ref: 23241029
TCMC895
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 700 (nM), Ref: 23241029
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC2148
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 3200 (nM), Ref: 24920381
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC42
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 8390 (nM), Ref: 26696252
TCMC42
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2540 (nM), Ref: 26696252
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC1041
TCMT636 DNA polymerase alpha subunit Homo sapiens Ki: 830 (nM), Ref: 1705574
TCMC1041
TCMT17 DNA polymerase beta Homo sapiens Ki: 390 (nM), Ref: 1705574
TCMC1480
TCMT107 Glutamate receptor ionotropic kainate 2 Homo sapiens Ki: 1106 (nM), Ref: 10821708
TCMC1480
TCMT108 Glutamate receptor ionotropic, AMPA 1 Homo sapiens Ki: 1360 (nM), Ref: 9357531
TCMC1480
TCMT109 Glutamate receptor ionotropic, AMPA 2 Homo sapiens Ki: 940 (nM), Ref: 9357531
TCMC1480
TCMT110 Glutamate receptor ionotropic, AMPA 4 Homo sapiens Ki: 868 (nM), Ref: 9357531
TCMC1480
TCMT111 Glutamate receptor ionotropic kainate 5 Homo sapiens Ki: 701 (nM), Ref: 9357531
TCMC1480
TCMT660 Metabotropic glutamate receptor 8 Homo sapiens IC50: 5.7 (nM), Ref: 15603952
TCMC1480
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 613 (nM), Ref: 16250647
TCMC1480
TCMT653 Metabotropic glutamate receptor 1 Homo sapiens Ki: 250 (nM), Ref: 17725337
Ki: 570 (nM), Ref: 19042134
Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT654 Metabotropic glutamate receptor 5 Homo sapiens Ki: 390 (nM), Ref: 17725337
Ki: 1160 (nM), Ref: 19042134
Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT657 Metabotropic glutamate receptor 4 Homo sapiens Ki: 2400 (nM), Ref: 17725337
Ki: 1400 (nM), Ref: 19042134
Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT655 Metabotropic glutamate receptor 2 Homo sapiens Ki: 6400 (nM), Ref: 19042134
Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H
TCMC1480
TCMT664 Excitatory amino acid transporter 3 Homo sapiens Ki: 51 (nM), Ref: 18578477
TCMC1480
TCMT656 Metabotropic glutamate receptor 3 Homo sapiens Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H
TCMC949
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 19911821
TCMC949
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 48 (nM), Ref: 19911821
TCMC949
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9100 (nM), Ref: 19911821
TCMC949
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3300 (nM), Ref: 19911821
TCMC949
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 2000 (nM), Ref: 19911821
TCMC949
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 5200 (nM), Ref: 19911821
TCMC949
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9400 (nM), Ref: 19911821
TCMC949
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 6800 (nM), Ref: 19911821
TCMC949
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 5600 (nM), Ref: 19911821
TCMC949
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3100 (nM), Ref: 19911821
Ki: 3100 (nM), Ref: 21067924
Ki: 3100 (nM), Ref: 22137345
Ki: 3100 (nM), Ref: 22077347
Ki: 3100 (nM), Ref: 22365761
Ki: 3100 (nM), Ref: 22377674
Ki: 3100 (nM), Ref: 23241068
Ki: 3100 (nM), Ref: 22892213
Ki: 3100 (nM), Ref: 26688270
TCMC949
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9200 (nM), Ref: 21067924
Ki: 9200 (nM), Ref: 22137345
Ki: 9200 (nM), Ref: 22077347
Ki: 9200 (nM), Ref: 22365761
Ki: 9200 (nM), Ref: 22377674
Ki: 9200 (nM), Ref: 23241068
Ki: 9200 (nM), Ref: 22892213
Ki: 9200 (nM), Ref: 26688270
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC1104
TCMT678 Inhibitor of apoptosis protein 3 Homo sapiens IC50: 4100 (nM), Ref: 15115387
TCMC1104
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1700 (nM), Ref: 25765759
IC50: 60 (nM), Ref: 25765759
IC50: 800 (nM), Ref: 25765759
IC50: 60 (nM), Ref: 25765759
IC50: 3500 (nM), Ref: 25765759
TCMC1104
TCMT679 Macrophage-expressed gene 1 protein Homo sapiens IC50: 210 (nM), Ref: 25765759
IC50: 210 (nM), Ref: 25765759
TCMC1104
TCMT680 Histone acetyltransferase PCAF Homo sapiens IC50: 7200 (nM), Ref: 26701186
TCMC845
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 630 (nM), Ref: 19231207
TCMC662
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 250 (nM), Ref: 25743213
IC50: 1100 (nM), Ref: 25743213
TCMC315
TCMT46 Coagulation factor III Homo sapiens IC50: 14.98 (nM), Ref: 23199480
TCMC1396
TCMT689 Protein-glutamine gamma-glutamyltransferase Homo sapiens IC50: 8000 (nM), Ref: 21215619
TCMC837
TCMT690 Histone deacetylase 3 Homo sapiens IC50: 9000 (nM), Ref: 21874153
TCMC2124
TCMT39 Phosphodiesterase 5A Homo sapiens IC50: 4703 (nM), Ref:
TCMC2124
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 325 (nM), Ref:
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1113
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC43
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 220 (nM), Ref: 26588603
IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 26701186
TCMC43
TCMT208 Monoamine oxidase A Homo sapiens Ki: 710 (nM), Ref: 26819666
TCMC43
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3100 (nM), Ref: 27190601
IC50: 1500 (nM), Ref: 27190601
TCMC2003
TCMT82 Estrogen receptor alpha Homo sapiens Ki: 785 (nM), Ref: 15634023
TCMC2003
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 2840 (nM), Ref: 16814546
IC50: 4120 (nM), Ref: 18063374
IC50: 625 (nM), Ref:
TCMC2003
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 996 (nM), Ref: 17604631
IC50: 750 (nM), Ref: 20527891
IC50: 996 (nM), Ref: 26850006
TCMC2003
TCMT329 Quinone reductase 2 Homo sapiens IC50: 960 (nM), Ref: 19265439
IC50: 450 (nM), Ref: 20036559
IC50: 450 (nM), Ref: 20356739
IC50: 960 (nM), Ref: 21261296
IC50: 6900 (nM), Ref: 23953689
Ki: 88 (nM), Ref: 23953689
IC50: 1400 (nM), Ref: 26854376
IC50: 913 (nM), Ref: 26854376
TCMC2003
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2210 (nM), Ref: 20674354
TCMC2003
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2770 (nM), Ref: 20674354
TCMC2003
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9090 (nM), Ref: 20674354
TCMC2003
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4470 (nM), Ref: 20674354
TCMC2003
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4750 (nM), Ref: 20674354
TCMC2003
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4640 (nM), Ref: 20674354
TCMC2003
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8070 (nM), Ref: 20674354
TCMC2003
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4350 (nM), Ref: 20674354
TCMC2003
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 20674354
TCMC2003
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 950 (nM), Ref: 20674354
TCMC2003
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4090 (nM), Ref: 20674354
TCMC2003
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 830 (nM), Ref: 20674354
TCMC2003
TCMT729 PI3-kinase p110-alpha subunit Homo sapiens IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT730 PI3-kinase p110-beta subunit Homo sapiens IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4100 (nM), Ref: 27190601
IC50: 2600 (nM), Ref: 27190601
TCMC876
TCMT560 Coagulation factor X Homo sapiens IC50: 720 (nM), Ref: 9834152
Ki: 450 (nM), Ref: 9834152
TCMC2070
TCMT327 Vanilloid receptor Homo sapiens IC50: 290 (nM), Ref: 22257892
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC2225
TCMT594 Platelet activating factor receptor Homo sapiens Ki: 1000 (nM), Ref: 1404229
TCMC1986
TCMT223 Aldose reductase Homo sapiens IC50: 150 (nM), Ref: 18165015
IC50: 2000 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1199
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 1000 (nM), Ref: 10.1016/0960-894X(95)00282-X
TCMC1248
TCMT759 SUMO-activating enzyme subunit 1 Homo sapiens IC50: 3000 (nM), Ref: 23360215
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1964
TCMT726 Bcr/Abl fusion protein Homo sapiens IC50: 10000 (nM), Ref: 16686543
TCMC1964
TCMT329 Quinone reductase 2 Homo sapiens IC50: 5100 (nM), Ref: 23953689
TCMC1964
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1400 (nM), Ref: 10.1039/C3MD00317E
Ki: 900 (nM), Ref: 10.1039/C0MD00242A
TCMC1964
TCMT215 Cytochrome P450 1A1 Homo sapiens Ki: 570 (nM), Ref: 10.1039/C0MD00242A
TCMC910
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1118 (nM), Ref: 20696580
TCMC910
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 95 (nM), Ref: 20696580
TCMC910
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 20 (nM), Ref: 20696580
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1201
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 3150 (nM), Ref: 8576921
TCMC1201
TCMT132 Butyrylcholinesterase Homo sapiens Ki: 6900 (nM), Ref: 19879672
TCMC1201
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1201
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 40 (nM), Ref: 20696580
TCMC1201
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1201
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1201
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 568.3 (nM), Ref: 26498393
TCMC1201
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 24.5 (nM), Ref: 26498393
TCMC1201
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 41.8 (nM), Ref: 26498393
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC2106
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 5.9 (nM), Ref: 19744859
IC50: 12.29 (nM), Ref: 22748706
Ki: 6.23 (nM), Ref: 22748706
Ki: 3.4 (nM), Ref: 23332346
Ki: 12.29 (nM), Ref: 25308766
TCMC2106
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 974 (nM), Ref: 19744859
IC50: 105.41 (nM), Ref: 22748706
Ki: 56.17 (nM), Ref: 22748706
Ki: 11 (nM), Ref: 23332346
Ki: 105.41 (nM), Ref: 25308766
IC50: 4380 (nM), Ref: 25308766
TCMC2106
TCMT648 Dopamine D4 receptor Homo sapiens Ki: 3748 (nM), Ref: 19744859
TCMC2106
TCMT649 Dopamine D5 receptor Homo sapiens Ki: 4.4 (nM), Ref: 19744859
TCMC2106
TCMT46 Coagulation factor III Homo sapiens IC50: 104.58 (nM), Ref: 23199480
TCMC2106
TCMT651 Dopamine D3 receptor Homo sapiens Ki: 90.02 (nM), Ref: 25308766
Ki: 30 (nM), Ref: 27032890
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1158
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3100 (nM), Ref: 24835197
Ki: 6840 (nM), Ref: 24835197
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1526
TCMT131 Acetylcholinesterase Homo sapiens IC50: 1840 (nM), Ref: 27236720
Ki: 4330 (nM), Ref: 27236720
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC880
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9910 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 20185318
Ki: 9900 (nM), Ref: 22245047
Ki: 9900 (nM), Ref: 26073005
Ki: 9900 (nM), Ref: 26520662
TCMC880
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4200 (nM), Ref: 18579385
Ki: 4200 (nM), Ref: 20185318
TCMC880
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 18579385
Ki: 8900 (nM), Ref: 20185318
TCMC469
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 100 (nM), Ref: 22921742
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1886
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 670 (nM), Ref: 26498394
TCMC1886
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 770 (nM), Ref: 26498394
TCMC1886
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 620 (nM), Ref: 26498394
TCMC1886
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8470 (nM), Ref: 26498394
TCMC1886
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 720 (nM), Ref: 26498394
TCMC1597
TCMT807 Solute carrier family 22 member 12 Homo sapiens IC50: 2000 (nM), Ref: 17325024
Ki: 5740 (nM), Ref: 17325024
TCMC1597
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2927.18 (nM), Ref:
TCMC1597
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2988.26 (nM), Ref:
TCMC1597
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 1600 (nM), Ref: 24900447
TCMC1597
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 1600 (nM), Ref: 26322379
TCMC1597
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 4300 (nM), Ref: 26602279
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC846
TCMT207 Beta-secretase 1 Homo sapiens Ki: 6200 (nM), Ref: 22222157
TCMC418
TCMT223 Aldose reductase Homo sapiens IC50: 78 (nM), Ref: 22236472
TCMC418
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 240 (nM), Ref: 22236472
TCMC418
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4700 (nM), Ref: 22921742
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1143
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 860 (nM), Ref: 22668600
TCMC1143
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 830 (nM), Ref: 22668600
TCMC1143
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 780 (nM), Ref: 22668600
TCMC1143
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 750 (nM), Ref: 22668600
TCMC1143
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 610 (nM), Ref: 22668600
TCMC1143
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 650 (nM), Ref: 22668600
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC536
TCMT466 c-Jun N-terminal kinase 2 Homo sapiens IC50: 2500 (nM), Ref: 23002419
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC1329
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2710 (nM), Ref: 26275107
TCMC1428
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 509 (nM), Ref: 20696580
TCMC1428
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 88 (nM), Ref: 20696580
TCMC1428
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1527
TCMT131 Acetylcholinesterase Homo sapiens IC50: 1940 (nM), Ref: 27236720
Ki: 5860 (nM), Ref: 27236720
TCMC1774
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3100 (nM), Ref: 20674354
Ki: 3100 (nM), Ref: 21282059
Ki: 3400 (nM), Ref: 22137345
TCMC1774
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9300 (nM), Ref: 22137345
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1168
TCMT117 Kappa opioid receptor Homo sapiens Ki: 2515 (nM), Ref: 18166466
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC850
TCMT307 HERG Homo sapiens IC50: 4897.79 (nM), Ref: 21185626
TCMC850
TCMT707 Adenosine A2a receptor Homo sapiens Ki: 5011.87 (nM), Ref: 21661720
Ki: 9560 (nM), Ref: 23200243
Ki: 2480 (nM), Ref: 23200243
TCMC850
TCMT131 Acetylcholinesterase Homo sapiens IC50: 7250 (nM), Ref: 23791077
TCMC2139
TCMT560 Coagulation factor X Homo sapiens IC50: 210 (nM), Ref: 9834152
Ki: 440 (nM), Ref: 9834152
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC1203
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC804
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 2000 (nM), Ref: 21561086
TCMC1078
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC392
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 2400 (nM), Ref: 15658857
IC50: 2398.83 (nM), Ref: 19110342
TCMC1179
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 19592245
IC50: 5900 (nM), Ref: 19592245
TCMC1179
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8 (nM), Ref: 20413308
IC50: 10000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1179
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1890 (nM), Ref: 22487176
Ki: 1880 (nM), Ref: 22487176
TCMC1179
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8710 (nM), Ref: 22487176
Ki: 8800 (nM), Ref: 22487176
TCMC1179
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4130 (nM), Ref: 22487176
Ki: 4220 (nM), Ref: 22487176
TCMC1179
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7220 (nM), Ref: 22487176
Ki: 7330 (nM), Ref: 22487176
TCMC1179
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 1380.38 (nM), Ref: 23574272
IC50: 1400 (nM), Ref: 23574272
TCMC1179
TCMT128 Tankyrase-2 Homo sapiens IC50: 147.91 (nM), Ref: 23574272
IC50: 140 (nM), Ref: 23574272
TCMC1179
TCMT129 Tankyrase-1 Homo sapiens IC50: 323.59 (nM), Ref: 23574272
IC50: 320 (nM), Ref: 23574272
IC50: 323.59 (nM), Ref: 24116873
IC50: 330 (nM), Ref: 24116873
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC4
TCMT207 Beta-secretase 1 Homo sapiens IC50: 6000 (nM), Ref: 14592472
TCMC341
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 19231207
TCMC1032
TCMT131 Acetylcholinesterase Homo sapiens IC50: 2310 (nM), Ref: 26386602
IC50: 627 (nM), Ref: 26386602
TCMC1551
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1900 (nM), Ref: 16248836
Ki: 1900 (nM), Ref: 16248836
Ki: 800 (nM), Ref: 16248836
Ki: 250 (nM), Ref: 22696418
TCMC1551
TCMT131 Acetylcholinesterase Homo sapiens IC50: 760 (nM), Ref: 23746477
TCMC1551
TCMT268 Cytochrome P450 2A13 Homo sapiens Ki: 40 (nM), Ref: 22696418
TCMC2114
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 2200 (nM), Ref: 25743213
TCMC2114
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 9000 (nM), Ref: 27135370
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC1892
TCMT508 Tyrosine-protein kinase SYK Homo sapiens IC50: 10000 (nM), Ref: 23917087
TCMC2201
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8700 (nM), Ref: 21332115
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1148
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 800 (nM), Ref: 22668600
TCMC1148
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 490 (nM), Ref: 22668600
TCMC1148
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 610 (nM), Ref: 22668600
TCMC1148
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 850 (nM), Ref: 22668600
TCMC1148
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 710 (nM), Ref: 22668600
TCMC1148
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 320 (nM), Ref: 22668600
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC740
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.77 (nM), Ref: 16250647
TCMC740
TCMT675 Beta-1 adrenergic receptor Homo sapiens IC50: 600 (nM), Ref: 18983139
Ki: 430 (nM), Ref: 18983139
IC50: 1740 (nM), Ref: 18588282
IC50: 1640 (nM), Ref: 20875743
Ki: 170 (nM), Ref: 21726069
Ki: 150 (nM), Ref: 23466604
IC50: 260 (nM), Ref: 23466604
IC50: 210 (nM), Ref: 26988801
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC1175
TCMT186 Monoamine oxidase B Homo sapiens IC50: 2870 (nM), Ref: 20045650
TCMC1175
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC273
TCMT332 Amine oxidase, copper containing Homo sapiens IC50: 4100 (nM), Ref: 23664164
TCMC1946
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 1900 (nM), Ref: 15993593
IC50: 5011.87 (nM), Ref: 26565745
TCMC1946
TCMT559 Beta-2 adrenergic receptor Homo sapiens Ki: 3.69 (nM), Ref: 24326276
Ki: 0.46 (nM), Ref: 24326276
IC50: 50.12 (nM), Ref: 26565745
TCMC1946
TCMT48 Sodium channel protein type V alpha subunit Homo sapiens IC50: 2100 (nM), Ref: 21300721
TCMC1946
TCMT675 Beta-1 adrenergic receptor Homo sapiens IC50: 251.19 (nM), Ref: 26565745
TCMC1946
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens IC50: 3981.07 (nM), Ref: 26565745
TCMC1945
TCMT131 Acetylcholinesterase Homo sapiens IC50: 2300 (nM), Ref: 26386602
IC50: 590 (nM), Ref: 26386602
TCMC939
TCMT962 Autotaxin Homo sapiens Ki: 1890 (nM), Ref: 24387347
IC50: 1310 (nM), Ref: 16513348
TCMC249
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 257 (nM), Ref:
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC987
TCMT885 Lysine-specific demethylase 2A Homo sapiens Ki: 1970 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 23964788
TCMC987
TCMT965 Lysine-specific demethylase 7 Homo sapiens IC50: 2100 (nM), Ref: 22724510
TCMC987
TCMT884 Histone lysine demethylase PHF8 Homo sapiens IC50: 550 (nM), Ref: 22724510
IC50: 550 (nM), Ref: 23964788
TCMC249
TCMT191 Signal transducer and activator of transcription 3 Homo sapiens IC50: 6000 (nM), Ref: 19128055
TCMC249
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 600 (nM), Ref: 22206869
TCMC249
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 5200 (nM), Ref: IC50: 800 (nM), Ref:
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1961
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 600 (nM), Ref: 16248836
TCMC1961
TCMT131 Acetylcholinesterase Homo sapiens IC50: 6480 (nM), Ref: 23746477
TCMC1174
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 850 (nM), Ref: 15689157
IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1174
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC2180
TCMT302 HMG-CoA reductase Homo sapiens IC50: 5860 (nM), Ref: 25311563
IC50: 36.31 (nM), Ref: 25311563
TCMC1403
TCMT223 Aldose reductase Homo sapiens IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC702
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 5150 (nM), Ref: 15658857
TCMC1543
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 840 (nM), Ref: 16248836
Ki: 2500 (nM), Ref: 16248836
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC1343
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 90 (nM), Ref: 18501600
Ki: 90 (nM), Ref: 18579385
TCMC1343
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7800 (nM), Ref: 18579385
TCMC1343
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8200 (nM), Ref: 18579385

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC1803
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 2 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC962
TCMT1104 Sortase Staphylococcus aureus IC50: 13.8 (ug/ml), Ref: 19269184
TCMC962
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 51.3 (ug/ml), Ref: 16643034
TCMC962
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 1 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2257
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 15.46 (ug/ml), Ref: 20116898
TCMC2124
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 50 (ug/ml), Ref: 1710653
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC1986
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 75.2 (ug/ml), Ref: 9461665
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC469
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 5.4 (ug/ml), Ref: 16643034
TCMC2233
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.85 (ug/ml), Ref: 20116898
TCMC1866
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC2281
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00342 (ug/ml), Ref: 21334901
IC50: 0.00356 (ug/ml), Ref: 21334901
TCMC1329
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.9 (ug/ml), Ref: 20116898
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1203
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.5 (ug/ml), Ref: 9461665
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC2123
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC819
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 20691508
TCMC1711
TCMT1257 Colletotrichum lagenarium Colletotrichum lagenarium MIC: 12.5 (ug/ml), Ref: 17190464
TCMC1793
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1251 Candida albicans Candida albicans MIC: 12.5 (ug/ml), Ref: 9392889
TCMC1793
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 61.5 (ug/ml), Ref: 20218656
TCMC23
TCMT1251 Candida albicans Candida albicans MIC: 8 (ug/ml), Ref: 10.1021/np50053a042
MIC: 7.5 (ug/ml), Ref: 12444675
TCMC23
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 7.5 (ug/ml), Ref: 12444675
TCMC23
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 7.5 (ug/ml), Ref: 12444675
TCMC23
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 MIC: 3.6 (ug/ml), Ref: 12444675
MIC: 1.8 (ug/ml), Ref: 12444675
TCMC23
TCMT1438 Plasmodium falciparum Plasmodium falciparum MIC: 3.6 (ug/ml), Ref: 12444675
MIC: 1.8 (ug/ml), Ref: 12444675
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2328
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 16 (ug/ml), Ref: 11473422
MIC: 32 (ug/ml), Ref: 11473422
TCMC2328
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 11473422
TCMC2328
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 11473422
TCMC2328
TCMT1246 Escherichia coli Escherichia coli MIC: 32 (ug/ml), Ref: 11473422
TCMC2328
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 32 (ug/ml), Ref: 11473422
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC2013
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2351
TCMT1190 Plasmodium falciparum (isolate FcB1 / Columbia) Plasmodium falciparum FcB1/Columbia IC50: 16.7 (ug/ml), Ref: 21985060
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC1803
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 23369537
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC962
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 5 (ug/ml), Ref: 19204190
MIC: 15 (ug/ml), Ref: 19204190
MIC: 50 (ug/ml), Ref: 19204190
MIC: 30 (ug/ml), Ref: 19204190
TCMC962
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 30 (ug/ml), Ref: 18284200
TCMC2382
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 20022753
TCMC2382
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 12.5 (ug/ml), Ref: 20022753
TCMC962
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 25938986
MIC: 32 (ug/ml), Ref: 25938986
TCMC2383
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.96 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1170
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 25.16 (ug/ml), Ref: 10.1007/s00044-011-9767-1
IC50: 10.51 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC221
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 1955885
TCMC221
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 32 (ug/ml), Ref: 1955885
TCMC221
TCMT1312 Enterococcus durans Enterococcus durans MIC: 32 (ug/ml), Ref: 1955885
TCMC221
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 1955885
TCMC2402
TCMT1251 Candida albicans Candida albicans MIC: 31.25 (ug/ml), Ref: 8254344
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC895
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.2 (ug/ml), Ref: 6492075
TCMC895
TCMT1246 Escherichia coli Escherichia coli MIC: 0.5 (ug/ml), Ref: 6492075
MIC: 1 (ug/ml), Ref: 6492075
MIC: 2 (ug/ml), Ref: 19770280
MIC: 4 (ug/ml), Ref: 19770280
TCMC895
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 3.9 (ug/ml), Ref: 6492075
TCMC895
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 15.6 (ug/ml), Ref: 6492075
TCMC895
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 15.6 (ug/ml), Ref: 6492075
MIC: 10 (ug/ml), Ref: 18838593
MIC: 2.5 (ug/ml), Ref: 18838593
MIC: 1.25 (ug/ml), Ref: 18838593
MIC: 0.625 (ug/ml), Ref: 18838593
MIC: 5 (ug/ml), Ref: 18838593
MIC: 20 (ug/ml), Ref: 18838593
TCMC895
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 2 (ug/ml), Ref: 17220400
MIC: 0.312 (ug/ml), Ref: 10543897
TCMC895
TCMT1251 Candida albicans Candida albicans MIC: 1.5 (ug/ml), Ref: 19841146
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1412
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 8463795
TCMC2148
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 20691508
TCMC2411
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 16 (ug/ml), Ref: 11141098
TCMC2411
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 64 (ug/ml), Ref: 12608857
TCMC2417
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 16 (ug/ml), Ref: 25760525
MIC: 32 (ug/ml), Ref: 25760525
TCMC2417
TCMT1187 Enterococcus faecalis ATCC 29212 Enterococcus faecalis ATCC 29212 MIC: 16 (ug/ml), Ref: 25760525
TCMC2417
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 16 (ug/ml), Ref: 25760525
TCMC2417
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 8 (ug/ml), Ref: 25760525
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC1322
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1104
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1104
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 35.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 49 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 14.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2257
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 37.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 59.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2439
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 2 (ug/ml), Ref: 9784148
TCMC845
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 1522419
MIC: 6.25 (ug/ml), Ref: 1522419
TCMC845
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 1522419
MIC: 1.57 (ug/ml), Ref: 1522419
TCMC2454
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 19.6 (ug/ml), Ref: 10425115
TCMC1113
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 15863332
TCMC2003
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1251 Candida albicans Candida albicans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1246 Escherichia coli Escherichia coli MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12036362
TCMC2003
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
TCMC2003
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 25 (ug/ml), Ref: 20022753
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2477
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 72.5 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1986
TCMT1442 Leishmania donovani Leishmania donovani IC50: 17.7 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2482
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC2487
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 11.4 (ug/ml), Ref: 23294378
TCMC1248
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 6.25 (ug/ml), Ref: 17959274
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2490
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 4 (ug/ml), Ref: 11975515
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC887
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 10395496
TCMC2496
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1006
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 20691508
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1515
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC1848
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 22280816
TCMC1526
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1 (ug/ml), Ref: 1955885
TCMC1526
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 1 (ug/ml), Ref: 1955885
TCMC1526
TCMT1312 Enterococcus durans Enterococcus durans MIC: 1 (ug/ml), Ref: 1955885
MIC: 2 (ug/ml), Ref: 1955885
TCMC1526
TCMT1251 Candida albicans Candida albicans MIC: 4 (ug/ml), Ref: 1955885
MIC: 8 (ug/ml), Ref: 1955885
MIC: 16 (ug/ml), Ref: 1955885
TCMC2516
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 1.43 (ug/ml), Ref: 1955879
TCMC2516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 10.82 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1791
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 70.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2534
TCMT1251 Candida albicans Candida albicans MIC: 64 (ug/ml), Ref: 22424614
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC1171
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 14.71 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC724
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC724
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
IC50: 36 (ug/ml), Ref: 9748372
TCMC724
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 21288041
TCMC724
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 64 (ug/ml), Ref: 21288041
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2578
TCMT1251 Candida albicans Candida albicans IC50: 82.98 (ug/ml), Ref: 25686593
TCMC915
TCMT1246 Escherichia coli Escherichia coli MIC: 1 (ug/ml), Ref: 25791674
TCMC915
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.5 (ug/ml), Ref: 25791674
TCMC915
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.25 (ug/ml), Ref: 25791674
TCMC2580
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 12398535
TCMC2580
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 17.2 (ug/ml), Ref: 10425115
TCMC2581
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC2281
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 13 (ug/ml), Ref: 21334901
TCMC2281
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 3.98 (ug/ml), Ref: 21334901
TCMC1329
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1428
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1286 Bacillus cereus Bacillus cereus MIC: 25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 32.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 26 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2590
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 62.5 (ug/ml), Ref: 15974602
MIC: 31.3 (ug/ml), Ref: 15974602
TCMC1527
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2 (ug/ml), Ref: 1955885
TCMC1527
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 4 (ug/ml), Ref: 1955885
MIC: 8 (ug/ml), Ref: 1955885
TCMC1527
TCMT1312 Enterococcus durans Enterococcus durans MIC: 4 (ug/ml), Ref: 1955885
MIC: 8 (ug/ml), Ref: 1955885
TCMC1527
TCMT1251 Candida albicans Candida albicans MIC: 8 (ug/ml), Ref: 1955885
MIC: 32 (ug/ml), Ref: 1955885
TCMC899
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 52 (ug/ml), Ref: 22902032
TCMC899
TCMT1251 Candida albicans Candida albicans MIC: 0.5 (ug/ml), Ref: 23489634
MIC: 0.7 (ug/ml), Ref: 24044873
TCMC899
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 23489634
MIC: 1.3 (ug/ml), Ref: 24044873
TCMC899
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 1.7 (ug/ml), Ref: 24044873
TCMC899
TCMT1246 Escherichia coli Escherichia coli MIC: 0.5 (ug/ml), Ref: 24044873
TCMC1168
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 9392889
MIC: 2.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 9392889
TCMC1168
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
MIC: 25 (ug/ml), Ref: 10217726
TCMC1168
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 9392889
TCMC1168
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.2 (ug/ml), Ref: 20218656
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC348
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 62 (ug/ml), Ref: 25813159
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2617
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 29.9 (ug/ml), Ref: 10425115
TCMC1203
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 22.6 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC804
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC946
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 14510592
TCMC1033
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1939
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 4.3 (ug/ml), Ref: 10425115
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2655
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 IC50: 7 (ug/ml), Ref: 2828553
TCMC2655
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 IC50: 7 (ug/ml), Ref: 2828553
TCMC2660
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 6.25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2667
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 15104489
MIC: 100 (ug/ml), Ref: 20542692
TCMC1551
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 20832915
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC2675
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 8.3 (ug/ml), Ref: 10425115
TCMC1892
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1892
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC2676
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 18.49 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2688
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 14969530
TCMC2688
TCMT1282 Colletotrichum orbiculare Colletotrichum orbiculare MIC: 30 (ug/ml), Ref: 14969530
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC2714
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 1.4 (ug/ml), Ref: 22280816
TCMC2714
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25.3 (ug/ml), Ref: 22280816
TCMC2723
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 4 (ug/ml), Ref: 11975483
MIC: 4 (ug/ml), Ref: 23102654
TCMC2730
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 23806014
MIC: 32 (ug/ml), Ref: 20303770
TCMC2731
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 31.3 (ug/ml), Ref:
TCMC2731
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 7.8 (ug/ml), Ref: MIC: 7.8 (ug/ml), Ref: 8699183
MIC: 7.8 (ug/ml), Ref: 15711537
MIC: 7.8 (ug/ml), Ref:
TCMC2723
TCMT1312 Enterococcus durans Enterococcus durans MIC: 4 (ug/ml), Ref: 15332848
MIC: 2 (ug/ml), Ref: 23964704
TCMC2723
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 4 (ug/ml), Ref: 8759163
MIC: 4 (ug/ml), Ref:
TCMC2730
TCMT1312 Enterococcus durans Enterococcus durans MIC: 32 (ug/ml), Ref: 20303770
TCMC2730
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 32 (ug/ml), Ref: 21703733
TCMC2730
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 22880631
TCMC2739
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 22880631
MIC: 32 (ug/ml), Ref: 25322455
MIC: 32 (ug/ml), Ref: 25499882
TCMC2739
TCMT1312 Enterococcus durans Enterococcus durans MIC: 32 (ug/ml), Ref: 22880631
MIC: 32 (ug/ml), Ref: 25322455
TCMC2739
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 32 (ug/ml), Ref: 22880631
MIC: 32 (ug/ml), Ref: 25322455
TCMC2739
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 20346682
MIC: 32 (ug/ml), Ref: 25322455
TCMC2760
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 19.8 (ug/ml), Ref: 18227183
TCMC2723
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 25499882
MIC: 32 (ug/ml), Ref: 25322455
TCMC2763
TCMT1251 Candida albicans Candida albicans MIC: 8 (ug/ml), Ref: 12713401
MIC: 8 (ug/ml), Ref: MIC: 16 (ug/ml), Ref: 16038534
MIC: 16 (ug/ml), Ref: 7400822
MIC: 8 (ug/ml), Ref: 14640516
MIC: 8 (ug/ml), Ref: 17988094
TCMC2763
TCMT1312 Enterococcus durans Enterococcus durans MIC: 8 (ug/ml), Ref: 23869482
MIC: 4 (ug/ml), Ref: 19344127
TCMC2766
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 8411013
MIC: 32 (ug/ml), Ref: 8411013
MIC: 32 (ug/ml), Ref: 12713415
MIC: 32 (ug/ml), Ref: 17269824
TCMC2767
TCMT1312 Enterococcus durans Enterococcus durans MIC: 32 (ug/ml), Ref: 8411013
TCMC2767
TCMT1251 Candida albicans Candida albicans MIC: 32 (ug/ml), Ref: 8411013
TCMC2767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 8411013
TCMC2767
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 32 (ug/ml), Ref: 8411013
TCMC2768
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 15.6 (ug/ml), Ref: 22647719
MIC: 7.8 (ug/ml), Ref: 22647719
MIC: 15.6 (ug/ml), Ref: MIC: 31.3 (ug/ml), Ref: MIC: 7.8 (ug/ml), Ref: MIC: 15.6 (ug/ml), Ref: 22472691
MIC: 7.8 (ug/ml), Ref: 22472691
TCMC2766
TCMT1312 Enterococcus durans Enterococcus durans MIC: 8 (ug/ml), Ref: 22424239
MIC: 16 (ug/ml), Ref: 7400822
TCMC2766
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 16 (ug/ml), Ref: 7400822
MIC: 8 (ug/ml), Ref: 10.6019/CHEMBL1201861
TCMC582
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 16680159
TCMC2763
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 4 (ug/ml), Ref: 19344127
MIC: 4 (ug/ml), Ref: 15679329
TCMC2763
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 4 (ug/ml), Ref: 19344127
MIC: 4 (ug/ml), Ref: 2158562
TCMC2766
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 4 (ug/ml), Ref: 15679329
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC582
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 1602301
TCMC582
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 24927000
MIC: 62.5 (ug/ml), Ref: 24927000
TCMC582
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 24927000
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2768
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 31.3 (ug/ml), Ref: 23398362
TCMC1961
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 6.25 (ug/ml), Ref: 20832915
TCMC1174
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 55 (ug/ml), Ref: 25564380
TCMC1174
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.6 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1403
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2817
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 12.5 (ug/ml), Ref: 20691508
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1113
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 16 (nM), Ref: 17263522
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC4
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 40 (nM), Ref: 16722653
TCMC1032
TCMT1114 Acetylcholinesterase Anopheles gambiae IC50: 60.1 (nM), Ref: 26386602
TCMC1945
TCMT1114 Acetylcholinesterase Anopheles gambiae IC50: 43.6 (nM), Ref: 26386602
TCMC962
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 10.2 (nM), Ref: 17503850
TCMC962
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37 (nM), Ref: 20034711
TCMC962
TCMT1313 Human immunodeficiency virus 2 Human immunodeficiency virus type 2 (ISOLATE ROD) IC50: 37 (nM), Ref: 20034711
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1179
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (nM), Ref: 19097788