Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2700 (nM), Ref: 22261024 |
|
TCMT337 | Exportin-1 | Homo sapiens |
IC50: 1600 (nM), Ref: 20493693 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 4630 (nM), Ref: 15270556 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5405 (nM), Ref: |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2100 (nM), Ref: 17994701 |
|
TCMT107 | Glutamate receptor ionotropic kainate 2 | Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
|
TCMT108 | Glutamate receptor ionotropic, AMPA 1 | Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
|
TCMT109 | Glutamate receptor ionotropic, AMPA 2 | Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
|
TCMT110 | Glutamate receptor ionotropic, AMPA 4 | Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
|
TCMT111 | Glutamate receptor ionotropic kainate 5 | Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
|
TCMT660 | Metabotropic glutamate receptor 8 | Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
|
TCMT653 | Metabotropic glutamate receptor 1 | Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT654 | Metabotropic glutamate receptor 5 | Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT657 | Metabotropic glutamate receptor 4 | Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT655 | Metabotropic glutamate receptor 2 | Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT664 | Excitatory amino acid transporter 3 | Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
|
TCMT656 | Metabotropic glutamate receptor 3 | Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT594 | Platelet activating factor receptor | Homo sapiens |
Ki: 1000 (nM), Ref: 1404229 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
|
TCMT753 | Mothers against decapentaplegic homolog 3 | Homo sapiens | IC50: 142 (nM), Ref: |
|
TCMT721 | Heat shock 70 kDa protein 1 | Homo sapiens | IC50: 760 (nM), Ref: |
|
TCMT189 | Dual specificity protein phosphatase 3 | Homo sapiens | IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
|
TCMT354 | Serine/threonine-protein kinase Aurora-A | Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
|
TCMT626 | Serine/threonine-protein kinase B-raf | Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
|
TCMT418 | Ephrin type-B receptor 4 | Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
|
TCMT457 | Vascular endothelial growth factor receptor 3 | Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
|
TCMT377 | Insulin receptor | Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
|
TCMT536 | Platelet-derived growth factor receptor beta | Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT755 | Serine/threonine-protein kinase PLK4 | Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
|
TCMT502 | Tyrosine-protein kinase TIE-2 | Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
|
TCMT756 | Mitogen-activated protein kinase kinase kinase 8 | Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 22.78 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 231 (nM), Ref: 23332346 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 610 (nM), Ref: 23062825 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 900 (nM), Ref: 17994701 |
|
TCMT302 | HMG-CoA reductase | Homo sapiens |
IC50: 5860 (nM), Ref: 25311563 IC50: 36.31 (nM), Ref: 25311563 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 100 (nM), Ref: 26003344 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1090 (nM), Ref: 26003344 |