TCM Putative Target References: TCMFx6317


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC879
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC550
TCMT113 Delta opioid receptor Homo sapiens Ki: 3100 (nM), Ref: 26035635
TCMC206
TCMT131 Acetylcholinesterase Homo sapiens IC50: 27 (nM), Ref: 16570913
TCMC206
TCMT132 Butyrylcholinesterase Homo sapiens IC50: 4 (nM), Ref: 16570913
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC704
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4000 (nM), Ref: 21030469
IC50: 3600 (nM), Ref: 21030469
TCMC2126
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 1410 (nM), Ref: 23286284
TCMC2126
TCMT171 Protein-tyrosine phosphatase 1C Homo sapiens IC50: 1970 (nM), Ref: 23957426
TCMC2126
TCMT233 Protein-tyrosine phosphatase 2C Homo sapiens IC50: 2570 (nM), Ref: 23957426
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC1397
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 4630 (nM), Ref: 15270556
TCMC1397
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 5405 (nM), Ref:
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC920
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 1720 (nM), Ref: 8576921
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC1985
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6367.7 (nM), Ref: 26498393
TCMC1985
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 67.3 (nM), Ref: 26498393
TCMC1985
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.9 (nM), Ref: 26498393
TCMC1985
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 43.5 (nM), Ref: 26498393
TCMC1582
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1582
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 820 (nM), Ref: 22668600
TCMC1582
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5500 (nM), Ref: 22668600
TCMC1582
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 780 (nM), Ref: 22668600
TCMC1582
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3400 (nM), Ref: 22668600
TCMC1582
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2600 (nM), Ref: 22668600
TCMC1041
TCMT636 DNA polymerase alpha subunit Homo sapiens Ki: 830 (nM), Ref: 1705574
TCMC1041
TCMT17 DNA polymerase beta Homo sapiens Ki: 390 (nM), Ref: 1705574
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC1104
TCMT678 Inhibitor of apoptosis protein 3 Homo sapiens IC50: 4100 (nM), Ref: 15115387
TCMC1104
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1700 (nM), Ref: 25765759
IC50: 60 (nM), Ref: 25765759
IC50: 800 (nM), Ref: 25765759
IC50: 60 (nM), Ref: 25765759
IC50: 3500 (nM), Ref: 25765759
TCMC1104
TCMT679 Macrophage-expressed gene 1 protein Homo sapiens IC50: 210 (nM), Ref: 25765759
IC50: 210 (nM), Ref: 25765759
TCMC1104
TCMT680 Histone acetyltransferase PCAF Homo sapiens IC50: 7200 (nM), Ref: 26701186
TCMC2124
TCMT39 Phosphodiesterase 5A Homo sapiens IC50: 4703 (nM), Ref:
TCMC2124
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 325 (nM), Ref:
TCMC2242
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7710 (nM), Ref: 22892213
TCMC2242
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6270 (nM), Ref: 22892213
TCMC2242
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 3150 (nM), Ref: 22892213
TCMC2242
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC2242
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 740 (nM), Ref: 22892213
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC2003
TCMT82 Estrogen receptor alpha Homo sapiens Ki: 785 (nM), Ref: 15634023
TCMC2003
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 2840 (nM), Ref: 16814546
IC50: 4120 (nM), Ref: 18063374
IC50: 625 (nM), Ref:
TCMC2003
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 996 (nM), Ref: 17604631
IC50: 750 (nM), Ref: 20527891
IC50: 996 (nM), Ref: 26850006
TCMC2003
TCMT329 Quinone reductase 2 Homo sapiens IC50: 960 (nM), Ref: 19265439
IC50: 450 (nM), Ref: 20036559
IC50: 450 (nM), Ref: 20356739
IC50: 960 (nM), Ref: 21261296
IC50: 6900 (nM), Ref: 23953689
Ki: 88 (nM), Ref: 23953689
IC50: 1400 (nM), Ref: 26854376
IC50: 913 (nM), Ref: 26854376
TCMC2003
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2210 (nM), Ref: 20674354
TCMC2003
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2770 (nM), Ref: 20674354
TCMC2003
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9090 (nM), Ref: 20674354
TCMC2003
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4470 (nM), Ref: 20674354
TCMC2003
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4750 (nM), Ref: 20674354
TCMC2003
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4640 (nM), Ref: 20674354
TCMC2003
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8070 (nM), Ref: 20674354
TCMC2003
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4350 (nM), Ref: 20674354
TCMC2003
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 20674354
TCMC2003
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 950 (nM), Ref: 20674354
TCMC2003
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4090 (nM), Ref: 20674354
TCMC2003
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 830 (nM), Ref: 20674354
TCMC2003
TCMT729 PI3-kinase p110-alpha subunit Homo sapiens IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT730 PI3-kinase p110-beta subunit Homo sapiens IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4100 (nM), Ref: 27190601
IC50: 2600 (nM), Ref: 27190601
TCMC2225
TCMT594 Platelet activating factor receptor Homo sapiens Ki: 1000 (nM), Ref: 1404229
TCMC706
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 9510 (nM), Ref: 19028102
TCMC1986
TCMT223 Aldose reductase Homo sapiens IC50: 150 (nM), Ref: 18165015
IC50: 2000 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1199
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 1000 (nM), Ref: 10.1016/0960-894X(95)00282-X
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC880
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9910 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 20185318
Ki: 9900 (nM), Ref: 22245047
Ki: 9900 (nM), Ref: 26073005
Ki: 9900 (nM), Ref: 26520662
TCMC880
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4200 (nM), Ref: 18579385
Ki: 4200 (nM), Ref: 20185318
TCMC880
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 18579385
Ki: 8900 (nM), Ref: 20185318
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC336
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6500 (nM), Ref: 22668600
TCMC336
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7200 (nM), Ref: 22668600
TCMC336
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5900 (nM), Ref: 22668600
TCMC336
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC336
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5200 (nM), Ref: 22668600
TCMC336
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5700 (nM), Ref: 22668600
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC751
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8980 (nM), Ref: 22892213
TCMC751
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 8460 (nM), Ref: 22892213
TCMC751
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 780 (nM), Ref: 22892213
TCMC751
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 770 (nM), Ref: 22892213
TCMC536
TCMT466 c-Jun N-terminal kinase 2 Homo sapiens IC50: 2500 (nM), Ref: 23002419
TCMC412
TCMT683 Macrophage migration inhibitory factor Homo sapiens Ki: 38 (nM), Ref: 19090668
IC50: 38 (nM), Ref: 27156768
TCMC1190
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9280 (nM), Ref: 22892213
TCMC1190
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6580 (nM), Ref: 22892213
TCMC1190
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1190
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9.7 (nM), Ref: 22892213
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1105
TCMT752 Casein kinase II alpha Homo sapiens IC50: 2000 (nM), Ref: 19414254
TCMC1105
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2500 (nM), Ref: 27173800
TCMC2245
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9180 (nM), Ref: 22892213
TCMC2245
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 8360 (nM), Ref: 22892213
TCMC2245
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7510 (nM), Ref: 22892213
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1551
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1900 (nM), Ref: 16248836
Ki: 1900 (nM), Ref: 16248836
Ki: 800 (nM), Ref: 16248836
Ki: 250 (nM), Ref: 22696418
TCMC1551
TCMT131 Acetylcholinesterase Homo sapiens IC50: 760 (nM), Ref: 23746477
TCMC1551
TCMT268 Cytochrome P450 2A13 Homo sapiens Ki: 40 (nM), Ref: 22696418
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC1892
TCMT508 Tyrosine-protein kinase SYK Homo sapiens IC50: 10000 (nM), Ref: 23917087
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1958
TCMT899 Aldehyde dehydrogenase Homo sapiens Ki: 450 (nM), Ref: 18613661
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC557
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7660 (nM), Ref: 22892213
TCMC557
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 790 (nM), Ref: 22892213
TCMC557
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 650 (nM), Ref: 22892213
TCMC557
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 620 (nM), Ref: 22892213
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC2180
TCMT302 HMG-CoA reductase Homo sapiens IC50: 5860 (nM), Ref: 25311563
IC50: 36.31 (nM), Ref: 25311563
TCMC1998
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2500 (nM), Ref: 25765759
IC50: 220 (nM), Ref: 25765759
IC50: 4700 (nM), Ref: 25765759
TCMC1998
TCMT679 Macrophage-expressed gene 1 protein Homo sapiens IC50: 900 (nM), Ref: 25765759
TCMC702
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 5150 (nM), Ref: 15658857
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC998
TCMT154 Protein kinase C delta Homo sapiens Ki: 9.7 (nM), Ref: 23582444
TCMC1343
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 90 (nM), Ref: 18501600
Ki: 90 (nM), Ref: 18579385
TCMC1343
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7800 (nM), Ref: 18579385
TCMC1343
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8200 (nM), Ref: 18579385

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC2257
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 15.46 (ug/ml), Ref: 20116898
TCMC2124
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 50 (ug/ml), Ref: 1710653
TCMC2264
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 13.01 (ug/ml), Ref: 22552195
IC50: 11.54 (ug/ml), Ref: 22552195
IC50: 22.45 (ug/ml), Ref: 22552195
IC50: 23.54 (ug/ml), Ref: 22552195
TCMC2264
TCMT1136 Neuraminidase Influenza A virus IC50: 13.01 (ug/ml), Ref: 22552195
IC50: 11.54 (ug/ml), Ref: 22552195
IC50: 22.45 (ug/ml), Ref: 22552195
IC50: 23.54 (ug/ml), Ref: 22552195
TCMC2269
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 13.41 (ug/ml), Ref: 22552195
IC50: 24.77 (ug/ml), Ref: 22552195
IC50: 26.81 (ug/ml), Ref: 22552195
IC50: 9.14 (ug/ml), Ref: 22552195
TCMC2269
TCMT1136 Neuraminidase Influenza A virus IC50: 13.41 (ug/ml), Ref: 22552195
IC50: 24.77 (ug/ml), Ref: 22552195
IC50: 26.81 (ug/ml), Ref: 22552195
IC50: 9.14 (ug/ml), Ref: 22552195
TCMC1986
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 75.2 (ug/ml), Ref: 9461665
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC1491
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00423 (ug/ml), Ref: 21334901
IC50: 0.00211 (ug/ml), Ref: 21334901
TCMC2123
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC2305
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 12.8 (ug/ml), Ref: 22552195
IC50: 9.33 (ug/ml), Ref: 22552195
IC50: 25.59 (ug/ml), Ref: 22552195
IC50: 28.42 (ug/ml), Ref: 22552195
TCMC2305
TCMT1136 Neuraminidase Influenza A virus IC50: 12.8 (ug/ml), Ref: 22552195
IC50: 9.33 (ug/ml), Ref: 22552195
IC50: 25.59 (ug/ml), Ref: 22552195
IC50: 28.42 (ug/ml), Ref: 22552195
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC2363
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 22537683
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC920
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 31.25 (ug/ml), Ref: 6677714
TCMC920
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 6677714
TCMC920
TCMT1246 Escherichia coli Escherichia coli MIC: 45 (ug/ml), Ref: 6677714
TCMC920
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 45 (ug/ml), Ref: 6677714
TCMC920
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 31.25 (ug/ml), Ref: 6677714
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1985
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 84.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1582
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 18539361
TCMC1582
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 12.5 (ug/ml), Ref: 18539361
TCMC1582
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 25 (ug/ml), Ref: 18539361
TCMC1210
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC1104
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1104
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 35.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 49 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 14.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2257
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 37.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 59.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2439
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 2 (ug/ml), Ref: 9784148
TCMC2444
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 5.8 (ug/ml), Ref: 8786363
IC50: 3.65 (ug/ml), Ref: 8786363
TCMC2444
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.8 (ug/ml), Ref: 8786363
IC50: 3.65 (ug/ml), Ref: 8786363
TCMC2444
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 25372601
TCMC2454
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 19.6 (ug/ml), Ref: 10425115
TCMC2003
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1251 Candida albicans Candida albicans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1246 Escherichia coli Escherichia coli MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12036362
TCMC2003
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
TCMC2003
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 25 (ug/ml), Ref: 20022753
TCMC1986
TCMT1442 Leishmania donovani Leishmania donovani IC50: 17.7 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC1848
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 22280816
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC2554
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 20702006
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC1936
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 14 (ug/ml), Ref: 10425115
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2576
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 1.24 (ug/ml), Ref: 8786363
IC50: 1.68 (ug/ml), Ref: 8786363
TCMC2576
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 1.24 (ug/ml), Ref: 8786363
IC50: 1.68 (ug/ml), Ref: 8786363
TCMC2580
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 12398535
TCMC2580
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 17.2 (ug/ml), Ref: 10425115
TCMC2595
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 25462220
TCMC1105
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1105
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 23534483
TCMC1105
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1 (ug/ml), Ref: 23534483
TCMC1105
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 23534483
MIC: 4 (ug/ml), Ref: 23534483
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2617
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 29.9 (ug/ml), Ref: 10425115
TCMC2622
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 3430167
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2625
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6 (ug/ml), Ref: 3430167
TCMC2625
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3 (ug/ml), Ref: 3430167
TCMC2625
TCMT1246 Escherichia coli Escherichia coli MIC: 6 (ug/ml), Ref: 3430167
TCMC2625
TCMT1251 Candida albicans Candida albicans MIC: 50 (ug/ml), Ref: 3430167
TCMC946
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 14510592
TCMC1033
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC2633
TCMT1286 Bacillus cereus Bacillus cereus MIC: 100 (ug/ml), Ref: 10425115
TCMC2633
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 5.8 (ug/ml), Ref: 10425115
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1939
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 4.3 (ug/ml), Ref: 10425115
TCMC2648
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 31.2 (ug/ml), Ref: 20702006
MIC: 31.2 (ug/ml), Ref: 24300736
TCMC2648
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 31.2 (ug/ml), Ref: 20702006
MIC: 31.2 (ug/ml), Ref: 24300736
TCMC2648
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 62.5 (ug/ml), Ref: 20702006
MIC: 62.5 (ug/ml), Ref: 24300736
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2014
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 10 (ug/ml), Ref: 17220400
TCMC1551
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 20832915
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2086
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC2086
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1892
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1892
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1491
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 0.92 (ug/ml), Ref: 21334901
TCMC1491
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 1.07 (ug/ml), Ref: 21334901
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC1889
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2709
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 59.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1998
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 65 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1998
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 35 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850