Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2700 (nM), Ref: 22261024 |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4000 (nM), Ref: 21030469 IC50: 3600 (nM), Ref: 21030469 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 9550 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8000 (nM), Ref: 24341381 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1970 (nM), Ref: 23062825 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 4500 (nM), Ref: 14592472 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT23 | Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | IC50: 407 (nM), Ref: |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2100 (nM), Ref: 17994701 |
|
TCMT203 | Glucose-6-phosphate 1-dehydrogenase | Homo sapiens |
Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561 |
|
TCMT599 | Ubiquitin-conjugating enzyme E2 N | Homo sapiens | IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
Ki: 785 (nM), Ref: 15634023 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref: |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006 |
|
TCMT329 | Quinone reductase 2 | Homo sapiens |
IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2210 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2770 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 9090 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4470 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4750 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4640 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8070 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4350 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 810 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 950 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4090 (nM), Ref: 20674354 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 830 (nM), Ref: 20674354 |
|
TCMT729 | PI3-kinase p110-alpha subunit | Homo sapiens |
IC50: 250 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT730 | PI3-kinase p110-beta subunit | Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 4200 (nM), Ref: 19481465 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 5610 (nM), Ref: 24900561 Ki: 5.61 (nM), Ref: 27078864 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 6460 (nM), Ref: 24900561 Ki: 6.46 (nM), Ref: 27078864 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18778944 |
|
TCMT737 | DNA dC->dU-editing enzyme APOBEC-3G | Homo sapiens | IC50: 2390 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 2120 (nM), Ref: 24900447 |
|
TCMT558 | DNA topoisomerase II alpha | Homo sapiens |
IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1690 (nM), Ref: 23411073 |
|
TCMT2 | Microtubule-associated protein tau | Homo sapiens |
IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3000 (nM), Ref: 25086914 |
|
TCMT740 | PI3-kinase p110-gamma subunit | Homo sapiens |
IC50: 4720 (nM), Ref: 25050878 |
|
TCMT13 | DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens |
IC50: 320 (nM), Ref: 25280182 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 1610 (nM), Ref: |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 9510 (nM), Ref: 19028102 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 10 (nM), Ref: 19564108 IC50: 18.6 (nM), Ref: 22148241 IC50: 6 (nM), Ref: 22360639 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 1 (nM), Ref: 19564108 IC50: 0.7 (nM), Ref: 22148241 IC50: 0.4 (nM), Ref: 22360639 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 22.78 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 231 (nM), Ref: 23332346 |
|
TCMT230 | Estradiol 17-beta-dehydrogenase 3 | Homo sapiens |
IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT646 | Serotonin 5a (5-HT5a) receptor | Homo sapiens |
Ki: 126 (nM), Ref: 12825922 IC50: 180 (nM), Ref: 18983139 Ki: 110 (nM), Ref: 18983139 IC50: 184 (nM), Ref: 18588282 Ki: 170 (nM), Ref: 21726069 IC50: 280 (nM), Ref: 23582449 Ki: 82 (nM), Ref: 23466604 IC50: 160 (nM), Ref: 23466604 IC50: 180 (nM), Ref: 26988801 |
|
TCMT315 | Serotonin 6 (5-HT6) receptor | Homo sapiens |
Ki: 65 (nM), Ref: 12825922 Ki: 100 (nM), Ref: 15357994 IC50: 200 (nM), Ref: 18983139 Ki: 93 (nM), Ref: 18983139 IC50: 262 (nM), Ref: 18588282 IC50: 27.5 (nM), Ref: 20170099 Ki: 84 (nM), Ref: 21726069 Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8 IC50: 180 (nM), Ref: 23582449 Ki: 50 (nM), Ref: 23466604 IC50: 100 (nM), Ref: 23466604 Ki: 33 (nM), Ref: 24805037 Ki: 33 (nM), Ref: 25557493 IC50: 120 (nM), Ref: 26988801 Ki: 100 (nM), Ref: 26996373 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 8.1 (nM), Ref: 12825922 IC50: 0.61 (nM), Ref: 18983139 Ki: 0.22 (nM), Ref: 18983139 IC50: 2.55 (nM), Ref: 12713409 IC50: 1.5 (nM), Ref: 18588282 Ki: 0.13 (nM), Ref: 21726069 IC50: 0.49 (nM), Ref: 23582449 Ki: 0.11 (nM), Ref: 23466604 IC50: 0.29 (nM), Ref: 23466604 Ki: 1.4 (nM), Ref: 24763360 Ki: 0.8 (nM), Ref: 24805037 Ki: 0.8 (nM), Ref: 25557493 IC50: 0.25 (nM), Ref: 26988801 |
|
TCMT37 | Serotonin 2a (5-HT2a) receptor | Homo sapiens |
Ki: 14 (nM), Ref: 15081042 Ki: 8.2 (nM), Ref: 16392816 Ki: 14 (nM), Ref: 16257207 Ki: 120 (nM), Ref: 18468904 Ki: 160 (nM), Ref: 18468904 Ki: 130 (nM), Ref: 18468904 Ki: 150 (nM), Ref: 18468904 Ki: 320 (nM), Ref: 11975483 Ki: 690 (nM), Ref: 17067154 Ki: 323.59 (nM), Ref: 23301527 Ki: 320 (nM), Ref: 23301527 |
|
TCMT313 | Serotonin 2b (5-HT2b) receptor | Homo sapiens |
Ki: 12 (nM), Ref: 15081042 Ki: 13 (nM), Ref: 12954071 Ki: 13 (nM), Ref: 16392816 Ki: 12 (nM), Ref: 16257207 Ki: 13.49 (nM), Ref: 24582985 |
|
TCMT314 | Serotonin 2c (5-HT2c) receptor | Homo sapiens |
Ki: 6.9 (nM), Ref: 15081042 Ki: 8.3 (nM), Ref: 12954071 Ki: 8.3 (nM), Ref: 16392816 Ki: 6.9 (nM), Ref: 16257207 Ki: 130 (nM), Ref: 11975483 Ki: 20 (nM), Ref: 17067154 Ki: 79.43 (nM), Ref: 23301527 Ki: 79 (nM), Ref: 23301527 |
|
TCMT815 | Serotonin 1d (5-HT1d) receptor | Homo sapiens |
Ki: 5.5 (nM), Ref: 8071931 Ki: 0.5 (nM), Ref: 18507369 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 2.5 (nM), Ref: 7658447 IC50: 1.2 (nM), Ref: 12954071 Ki: 1.259 (nM), Ref: 18433113 Ki: 10000 (nM), Ref: 18433113 Ki: 0.62 (nM), Ref: 22748706 Ki: 0.9 (nM), Ref: 23332346 Ki: 9.5 (nM), Ref: 24161678 Ki: 2.08 (nM), Ref: 25128671 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 79 (nM), Ref: 16250647 |
|
TCMT816 | Serotonin 1b (5-HT1b) receptor | Homo sapiens |
Ki: 1.1 (nM), Ref: 18507369 IC50: 29 (nM), Ref: 18983139 Ki: 18 (nM), Ref: 18983139 Ki: 14 (nM), Ref: 21726069 IC50: 12 (nM), Ref: 23582449 Ki: 4 (nM), Ref: 23466604 IC50: 6.5 (nM), Ref: 23466604 |
|
TCMT817 | Serotonin 4 (5-HT4) receptor | Homo sapiens |
Ki: 1049 (nM), Ref: 19334715 Ki: 500 (nM), Ref: 17067154 Ki: 29.51 (nM), Ref: 19223092 Ki: 109.65 (nM), Ref: 19223092 |
|
TCMT645 | Serotonin 1e (5-HT1e) receptor | Homo sapiens |
Ki: 10.72 (nM), Ref: 24365159 Ki: 11 (nM), Ref: 24365159 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT614 | Egl nine homolog 1 | Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
Ki: 600 (nM), Ref: 21739938 |
|
TCMT81 | Arachidonate 12-lipoxygenase | Homo sapiens |
Ki: 1600 (nM), Ref: 21739938 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 8700 (nM), Ref: |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 5900 (nM), Ref: 21561086 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 8000 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3500 (nM), Ref: 18798681 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 1440 (nM), Ref: 24900561 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 24900561 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 6000 (nM), Ref: 14592472 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 610 (nM), Ref: 23062825 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 800 (nM), Ref: 10.1039/C3MD00317E Ki: 2100 (nM), Ref: 10.1039/C0MD00242A |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
Ki: 160 (nM), Ref: 10.1039/C0MD00242A |
|
TCMT508 | Tyrosine-protein kinase SYK | Homo sapiens |
IC50: 10000 (nM), Ref: 23917087 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 900 (nM), Ref: 17994701 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 52 (nM), Ref: 20590092 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 44 (nM), Ref: 20590092 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 540 (nM), Ref: 20590092 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 740 (nM), Ref: 20590092 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 420 (nM), Ref: 20590092 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 380 (nM), Ref: 20590092 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 450 (nM), Ref: 20590092 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
|
TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
|
TCMT974 | G-protein coupled estrogen receptor 1 | Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 1900 (nM), Ref: 20100662 |
|
TCMT102 | Low molecular weight phosphotyrosine protein phosphatase | Homo sapiens |
IC50: 7200 (nM), Ref: 21453996 |
|
TCMT103 | Receptor-type tyrosine-protein phosphatase F (LAR) | Homo sapiens |
IC50: 3800 (nM), Ref: 21453996 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 2400 (nM), Ref: 23387824 |
|
TCMT150 | Nuclear receptor ROR-gamma | Homo sapiens |
IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 100 (nM), Ref: 26003344 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1090 (nM), Ref: 26003344 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 91 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4.5 (nM), Ref: 23332346 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 5150 (nM), Ref: 15658857 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |