Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2700 (nM), Ref: 22261024 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 452.6 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 515 (nM), Ref: 26498393 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2100 (nM), Ref: 17994701 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 4100 (nM), Ref: 22668600 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 820 (nM), Ref: 22668600 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5500 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 780 (nM), Ref: 22668600 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3400 (nM), Ref: 22668600 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2600 (nM), Ref: 22668600 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 22.78 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 231 (nM), Ref: 23332346 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref: |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 7300 (nM), Ref: 21030469 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 718.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.2 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 56.4 (nM), Ref: 26498393 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT307 | HERG | Homo sapiens |
IC50: 4897.79 (nM), Ref: 21185626 |
|
TCMT707 | Adenosine A2a receptor | Homo sapiens |
Ki: 5011.87 (nM), Ref: 21661720 Ki: 9560 (nM), Ref: 23200243 Ki: 2480 (nM), Ref: 23200243 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 7250 (nM), Ref: 23791077 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5900 (nM), Ref: 19592245 IC50: 5900 (nM), Ref: 19592245 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 8 (nM), Ref: 20413308 IC50: 10000 (nM), Ref: 24345481 IC50: 8000 (nM), Ref: 26301554 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1890 (nM), Ref: 22487176 Ki: 1880 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8710 (nM), Ref: 22487176 Ki: 8800 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4130 (nM), Ref: 22487176 Ki: 4220 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7220 (nM), Ref: 22487176 Ki: 7330 (nM), Ref: 22487176 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 1380.38 (nM), Ref: 23574272 IC50: 1400 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 147.91 (nM), Ref: 23574272 IC50: 140 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 323.59 (nM), Ref: 23574272 IC50: 320 (nM), Ref: 23574272 IC50: 323.59 (nM), Ref: 24116873 IC50: 330 (nM), Ref: 24116873 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 610 (nM), Ref: 23062825 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 900 (nM), Ref: 17994701 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref: |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 10 (nM), Ref: 17482813 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 395 (nM), Ref: 17482813 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 2210 (nM), Ref: 18533708 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 340 (nM), Ref: 20853847 |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 7720 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 100 (nM), Ref: 26003344 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1090 (nM), Ref: 26003344 |