Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 9500 (nM), Ref: 18579385 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 810 (nM), Ref: 20100662 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 5000 (nM), Ref: 24844534 |
|
TCMT636 | DNA polymerase alpha subunit | Homo sapiens |
Ki: 830 (nM), Ref: 1705574 |
|
TCMT17 | DNA polymerase beta | Homo sapiens |
Ki: 390 (nM), Ref: 1705574 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 3000 (nM), Ref: 24844534 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens | IC50: 4703 (nM), Ref: |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 325 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
Ki: 785 (nM), Ref: 15634023 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref: |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006 |
|
TCMT329 | Quinone reductase 2 | Homo sapiens |
IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2210 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2770 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 9090 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4470 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4750 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4640 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8070 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4350 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 810 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 950 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4090 (nM), Ref: 20674354 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 830 (nM), Ref: 20674354 |
|
TCMT729 | PI3-kinase p110-alpha subunit | Homo sapiens |
IC50: 250 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT730 | PI3-kinase p110-beta subunit | Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 3900 (nM), Ref: 10.1016/S0960-894X(97)00194-7 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 251 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 86 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 12 (nM), Ref: 20696580 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 1100 (nM), Ref: 24844534 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7200 (nM), Ref: 22668600 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7700 (nM), Ref: 22668600 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4900 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5900 (nM), Ref: 22668600 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 4700 (nM), Ref: 22668600 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 4900 (nM), Ref: 22668600 |
|
TCMT651 | Dopamine D3 receptor | Homo sapiens |
Ki: 500 (nM), Ref: 24559070 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 5000 (nM), Ref: 24559070 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
Ki: 8.5 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12781197 IC50: 37 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 9873735 IC50: 37 (nM), Ref: 9784110 Ki: 35 (nM), Ref: 20510622 |
|
TCMT613 | Glucocorticoid receptor | Homo sapiens |
Ki: 30.5 (nM), Ref: 12954062 Ki: 30.5 (nM), Ref: 9873735 Ki: 30.5 (nM), Ref: 9784110 |
|
TCMT783 | Mineralocorticoid receptor | Homo sapiens |
IC50: 14 (nM), Ref: 12954062 IC50: 14 (nM), Ref: 12781197 IC50: 14 (nM), Ref: 9784110 IC50: 30 (nM), Ref: 8709117 |
|
TCMT904 | Progesterone receptor | Homo sapiens |
Ki: 3.5 (nM), Ref: 10212133 IC50: 3.5 (nM), Ref: 11859003 Ki: 3.5 (nM), Ref: 9464361 IC50: 5 (nM), Ref: 8523399 Ki: 3.8 (nM), Ref: 9667968 Ki: 3.467 (nM), Ref: 16821785 Ki: 3.4 (nM), Ref: 18553958 Ki: 5.1 (nM), Ref: 20510622 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |