Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 310 (nM), Ref: 23332346 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
Ki: 122 (nM), Ref: 26125082 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 810 (nM), Ref: 20100662 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 5000 (nM), Ref: 24844534 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
Ki: 78 (nM), Ref: 26125082 |
|
TCMT37 | Serotonin 2a (5-HT2a) receptor | Homo sapiens |
Ki: 966 (nM), Ref: 25695425 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 43 (nM), Ref: 25695425 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 171 (nM), Ref: 25695425 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
Ki: 6800 (nM), Ref: 22752007 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2100 (nM), Ref: 17994701 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 85 (nM), Ref: 16562853 Ki: 314 (nM), Ref: 25695425 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 373 (nM), Ref: 25695425 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 20 (nM), Ref: 25695425 |
|
TCMT315 | Serotonin 6 (5-HT6) receptor | Homo sapiens |
Ki: 306 (nM), Ref: 25695425 |
|
TCMT646 | Serotonin 5a (5-HT5a) receptor | Homo sapiens |
Ki: 566 (nM), Ref: 25695425 |
|
TCMT313 | Serotonin 2b (5-HT2b) receptor | Homo sapiens |
Ki: 323 (nM), Ref: 25695425 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 3000 (nM), Ref: 24844534 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 152.43 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 50 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 305 (nM), Ref: 23332346 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 149 (nM), Ref: 23332346 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 10000 (nM), Ref: 14552748 IC50: 5620 (nM), Ref: 23033255 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 8290 (nM), Ref: 8917655 |
|
TCMT778 | Voltage-gated potassium channel subunit Kv1.5 | Homo sapiens |
IC50: 6100 (nM), Ref: 19004630 |
|
TCMT780 | Voltage-gated L-type calcium channel alpha-1D subunit | Homo sapiens |
IC50: 1350 (nM), Ref: 24754640 |
|
TCMT725 | Voltage-gated L-type calcium channel alpha-1C subunit | Homo sapiens |
IC50: 22 (nM), Ref: 22761000 IC50: 55 (nM), Ref: 22761000 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 2300 (nM), Ref: 23033255 |
|
TCMT31 | Cytochrome P450 2C19 | Homo sapiens |
IC50: 5420 (nM), Ref: 23033255 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4080 (nM), Ref: 23033255 |
|
TCMT220 | Cytochrome P450 2J2 | Homo sapiens |
IC50: 3060 (nM), Ref: 23033255 |
|
TCMT407 | Myosin light chain kinase, smooth muscle | Homo sapiens |
IC50: 2020 (nM), Ref: 26385444 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 22 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 214 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 1189 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 105 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 6.6 (nM), Ref: 23332346 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 22.78 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 231 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 3900 (nM), Ref: 10.1016/S0960-894X(97)00194-7 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 66 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 119 (nM), Ref: 23332346 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 6200 (nM), Ref: 22222157 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 251 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 86 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 12 (nM), Ref: 20696580 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 1100 (nM), Ref: 24844534 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 509 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 88 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 529 (nM), Ref: 23332346 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 3430 (nM), Ref: 19097799 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 4960 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 3656 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 79.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 44.3 (nM), Ref: 26498393 |
|
TCMT853 | Sigma opioid receptor | Homo sapiens |
Ki: 106 (nM), Ref: 27032890 |
|
TCMT651 | Dopamine D3 receptor | Homo sapiens |
Ki: 37 (nM), Ref: 27032890 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 102 (nM), Ref: 27032890 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 15 (nM), Ref: 27032890 |
|
TCMT643 | Alpha-1a adrenergic receptor | Homo sapiens |
Ki: 430 (nM), Ref: 15664832 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.77 (nM), Ref: 16250647 |
|
TCMT675 | Beta-1 adrenergic receptor | Homo sapiens |
IC50: 600 (nM), Ref: 18983139 Ki: 430 (nM), Ref: 18983139 IC50: 1740 (nM), Ref: 18588282 IC50: 1640 (nM), Ref: 20875743 Ki: 170 (nM), Ref: 21726069 Ki: 150 (nM), Ref: 23466604 IC50: 260 (nM), Ref: 23466604 IC50: 210 (nM), Ref: 26988801 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
Ki: 8.5 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12781197 IC50: 37 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 9873735 IC50: 37 (nM), Ref: 9784110 Ki: 35 (nM), Ref: 20510622 |
|
TCMT613 | Glucocorticoid receptor | Homo sapiens |
Ki: 30.5 (nM), Ref: 12954062 Ki: 30.5 (nM), Ref: 9873735 Ki: 30.5 (nM), Ref: 9784110 |
|
TCMT783 | Mineralocorticoid receptor | Homo sapiens |
IC50: 14 (nM), Ref: 12954062 IC50: 14 (nM), Ref: 12781197 IC50: 14 (nM), Ref: 9784110 IC50: 30 (nM), Ref: 8709117 |
|
TCMT904 | Progesterone receptor | Homo sapiens |
Ki: 3.5 (nM), Ref: 10212133 IC50: 3.5 (nM), Ref: 11859003 Ki: 3.5 (nM), Ref: 9464361 IC50: 5 (nM), Ref: 8523399 Ki: 3.8 (nM), Ref: 9667968 Ki: 3.467 (nM), Ref: 16821785 Ki: 3.4 (nM), Ref: 18553958 Ki: 5.1 (nM), Ref: 20510622 |
|
TCMT615 | Sentrin-specific protease 8 | Homo sapiens | IC50: 5470 (nM), Ref: |
|
TCMT616 | Sentrin-specific protease 7 | Homo sapiens | IC50: 4630 (nM), Ref: |
|
TCMT617 | Sentrin-specific protease 6 | Homo sapiens | IC50: 1860 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 8.35 (nM), Ref: 23199480 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 100 (nM), Ref: 26003344 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1090 (nM), Ref: 26003344 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 91 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4.5 (nM), Ref: 23332346 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 515 (nM), Ref: 12270171 IC50: 14.4 (nM), Ref: 16480284 IC50: 3.1 (nM), Ref: 16480284 IC50: 33 (nM), Ref: 16516473 IC50: 54 (nM), Ref: 16516473 IC50: 23 (nM), Ref: 16806916 IC50: 80 (nM), Ref: 16806916 IC50: 5.4 (nM), Ref: 17416531 IC50: 2753 (nM), Ref: 17416531 IC50: 22 (nM), Ref: 19170633 IC50: 33 (nM), Ref: 20304535 IC50: 70 (nM), Ref: 21353546 IC50: 1 (nM), Ref: 22101132 IC50: 1080 (nM), Ref: 22698782 IC50: 72 (nM), Ref: 22818848 IC50: 33 (nM), Ref: 23611691 IC50: 33 (nM), Ref: 23142066 IC50: 0.1 (nM), Ref: 23668441 IC50: 0.1 (nM), Ref: 23792318 IC50: 62 (nM), Ref: 23930994 IC50: 23 (nM), Ref: 23973168 IC50: 498 (nM), Ref: 23988354 IC50: 39.9 (nM), Ref: 23988354 IC50: 0.6 (nM), Ref: 23988354 IC50: 4000 (nM), Ref: 24900594 IC50: 1100 (nM), Ref: 24094432 IC50: 1 (nM), Ref: 24411123 IC50: 25 (nM), Ref: 24411123 IC50: 4000 (nM), Ref: 10.1039/C3MD00118K IC50: 70 (nM), Ref: 10.1039/C0MD00183J IC50: 1 (nM), Ref: 24588073 IC50: 0.1 (nM), Ref: 24607591 IC50: 20 (nM), Ref: 24731281 IC50: 0.45 (nM), Ref: 25468044 IC50: 0.45 (nM), Ref: 25462282 IC50: 76 (nM), Ref: 25409491 IC50: 380 (nM), Ref: 25768701 IC50: 1 (nM), Ref: 26275028 IC50: 26 (nM), Ref: 26256032 IC50: 22 (nM), Ref: 26318056 IC50: 1.3 (nM), Ref: 26706113 IC50: 22 (nM), Ref: 26451770 IC50: 13 (nM), Ref: 10.1039/C5MD00208G IC50: 15.5 (nM), Ref: 26829280 IC50: 11.8 (nM), Ref: 26879314 IC50: 2.6 (nM), Ref: 27234887 IC50: 0.509 (nM), Ref: 27288180 IC50: 127 (nM), Ref: 27288180 IC50: 76 (nM), Ref: 27387355 IC50: 0.585 (nM), Ref: 27132165 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 1604 (nM), Ref: 12270171 IC50: 343 (nM), Ref: 16480284 IC50: 599 (nM), Ref: 16480284 IC50: 280 (nM), Ref: 24411123 IC50: 1000 (nM), Ref: 25409491 IC50: 1830 (nM), Ref: 27132165 |
|
TCMT747 | ATP-binding cassette sub-family G member 2 | Homo sapiens |
IC50: 3190 (nM), Ref: 24184213 |