Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.

Ingredient ID & Structure	Target ID	Target Name	Target Organism	Activity Records & Reference
TCMC879	TCMT47	Apoptosis regulator Bcl-2	Homo sapiens	Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1211	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 270 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 270 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 750 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1211	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 2200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC417	TCMT127	Poly [ADP-ribose] polymerase-1	Homo sapiens	IC50: 7585.78 (nM), Ref: 23574272 IC50: 7500 (nM), Ref: 23574272
TCMC417	TCMT128	Tankyrase-2	Homo sapiens	IC50: 870.96 (nM), Ref: 23574272 IC50: 870 (nM), Ref: 23574272
TCMC417	TCMT129	Tankyrase-1	Homo sapiens	IC50: 645.65 (nM), Ref: 23574272 IC50: 630 (nM), Ref: 23574272
TCMC417	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2000 (nM), Ref: 24368208
TCMC1173	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394
TCMC1173	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394
TCMC1173	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9870 (nM), Ref: 20185318
TCMC1173	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7410 (nM), Ref: 20185318
TCMC1173	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 8450 (nM), Ref: 20185318
TCMC1173	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7040 (nM), Ref: 20185318
TCMC1173	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2400 (nM), Ref: 20185318
TCMC1173	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2890 (nM), Ref: 20185318
TCMC943	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 810 (nM), Ref: 20100662
TCMC943	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2042	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 2600 (nM), Ref: 16356713
TCMC616	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 800 (nM), Ref: 16759088 IC50: 3450 (nM), Ref: 16759088 IC50: 7138 (nM), Ref: 20851614 IC50: 7100 (nM), Ref: 21376605
TCMC616	TCMT209	11-beta-hydroxysteroid dehydrogenase 2	Homo sapiens	IC50: 201 (nM), Ref: 16759088 IC50: 6430 (nM), Ref: 16759088 IC50: 750 (nM), Ref: 20851614 IC50: 750 (nM), Ref: 21376605
TCMC616	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 3780 (nM), Ref: 16759088
TCMC2051	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 8710 (nM), Ref: 22892213
TCMC2051	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4050 (nM), Ref: 22892213
TCMC2051	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 960 (nM), Ref: 22892213
TCMC761	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 3920 (nM), Ref: 15658857
TCMC908	TCMT249	Cyclin-dependent kinase 6	Homo sapiens	IC50: 6000 (nM), Ref: 15689157 IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908	TCMT156	Cytochrome P450 19A1	Homo sapiens	Ki: 2600 (nM), Ref: 15267241 IC50: 1 (nM), Ref: 20413308 IC50: 800 (nM), Ref: 10.1039/C3MD00166K IC50: 500 (nM), Ref: 26301554
TCMC908	TCMT223	Aldose reductase	Homo sapiens	IC50: 8500 (nM), Ref: 18165015
TCMC908	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	IC50: 670 (nM), Ref: 19097799 Ki: 110 (nM), Ref: 19097799
TCMC908	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 153 (nM), Ref: 20696580 IC50: 1290 (nM), Ref: 23600958
TCMC908	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 84 (nM), Ref: 20696580 IC50: 54 (nM), Ref: 20832301 IC50: 570 (nM), Ref: 23600958
TCMC908	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 24 (nM), Ref: 20696580
TCMC908	TCMT87	Cytochrome P450 2C9	Homo sapiens	IC50: 5225 (nM), Ref: 20832301
TCMC908	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5490 (nM), Ref: 22487176 Ki: 5420 (nM), Ref: 22487176
TCMC908	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 4380 (nM), Ref: 22487176 Ki: 4310 (nM), Ref: 22487176
TCMC908	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 2650 (nM), Ref: 22487176 Ki: 2710 (nM), Ref: 22487176
TCMC908	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8960 (nM), Ref: 22487176 Ki: 9070 (nM), Ref: 22487176 Ki: 34.7 (nM), Ref: 26498393
TCMC908	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 537.75 (nM), Ref: 26498393
TCMC908	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 171.41 (nM), Ref: 26498393
TCMC959	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 2500 (nM), Ref: 21319773
TCMC948	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394
TCMC948	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394
TCMC948	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5330 (nM), Ref: 20185318
TCMC948	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 5230 (nM), Ref: 20185318
TCMC948	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6720 (nM), Ref: 20185318
TCMC948	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7760 (nM), Ref: 20185318
TCMC948	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 5960 (nM), Ref: 20185318
TCMC948	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9600 (nM), Ref: 20185318
TCMC948	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7570 (nM), Ref: 20185318
TCMC948	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 980 (nM), Ref: 20185318
TCMC948	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1070 (nM), Ref: 20185318
TCMC948	TCMT223	Aldose reductase	Homo sapiens	IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1187	TCMT151	Protein kinase C alpha	Homo sapiens	IC50: 1900 (nM), Ref: 9834166
TCMC1447	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 3000 (nM), Ref: 18565755 IC50: 2600 (nM), Ref: 18565755
TCMC1372	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 2330 (nM), Ref: 22245047
TCMC1372	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 3630 (nM), Ref: 22245047
TCMC332	TCMT231	Beta-glucosidase	Homo sapiens	Ki: 200 (nM), Ref: 10.1039/C3MD00033H
TCMC1495	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668
TCMC1495	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668
TCMC1495	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC218	TCMT307	HERG	Homo sapiens	IC50: 6025.6 (nM), Ref: 21185626
TCMC715	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC715	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC88	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 3400 (nM), Ref: 11678652
TCMC1433	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 6863.3 (nM), Ref: 26498393
TCMC1433	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 62.2 (nM), Ref: 26498393
TCMC1433	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 26.6 (nM), Ref: 26498393
TCMC1433	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 399.7 (nM), Ref: 26498393
TCMC1180	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 5210 (nM), Ref: 22487176 Ki: 5100 (nM), Ref: 22487176
TCMC1180	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9300 (nM), Ref: 22487176 Ki: 9200 (nM), Ref: 22487176
TCMC1180	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5540 (nM), Ref: 22487176 Ki: 5630 (nM), Ref: 22487176
TCMC1180	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 6590 (nM), Ref: 22487176 Ki: 6650 (nM), Ref: 22487176
TCMC1803	TCMT337	Exportin-1	Homo sapiens	IC50: 1600 (nM), Ref: 20493693
TCMC1450	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1450	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1449	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 2200 (nM), Ref: 21511472 IC50: 3400 (nM), Ref: 21511472
TCMC1449	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1449	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1369	TCMT347	Endoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase	Homo sapiens	Ki: 1260 (nM), Ref: 23151473
TCMC2037	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662
TCMC2037	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662
TCMC2037	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8800 (nM), Ref: 18579385
TCMC619	TCMT293	Muscarinic acetylcholine receptor M2	Homo sapiens	Ki: 158.49 (nM), Ref: 18077164
TCMC619	TCMT291	Muscarinic acetylcholine receptor M3	Homo sapiens	Ki: 7079.46 (nM), Ref: 18077164
TCMC619	TCMT551	Muscarinic acetylcholine receptor M4	Homo sapiens	Ki: 8511.38 (nM), Ref: 18077164
TCMC619	TCMT290	Muscarinic acetylcholine receptor M5	Homo sapiens	Ki: 9772.37 (nM), Ref: 18077164
TCMC1871	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056
TCMC1871	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662
TCMC1871	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455
TCMC1871	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455
TCMC1871	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662
TCMC87	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 400 (nM), Ref: 11678652
TCMC1397	TCMT34	Cytochrome P450 2D6	Homo sapiens	IC50: 4630 (nM), Ref: 15270556
TCMC1397	TCMT61	Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens	IC50: 5405 (nM), Ref:
TCMC619	TCMT241	Neuronal acetylcholine receptor protein alpha-7 subunit	Homo sapiens	Ki: 7943.28 (nM), Ref: 21920761
TCMC1851	TCMT560	Coagulation factor X	Homo sapiens	IC50: 170 (nM), Ref: 9834152 Ki: 570 (nM), Ref: 9834152
TCMC1851	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3760 (nM), Ref: 24835197 Ki: 5130 (nM), Ref: 24835197
TCMC1851	TCMT240	Salivary alpha-amylase	Homo sapiens	IC50: 2350 (nM), Ref: 26395057 Ki: 2600 (nM), Ref: 26395057
TCMC415	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 1800 (nM), Ref: 14592472
TCMC487	TCMT561	5'-nucleotidase	Homo sapiens	IC50: 8200 (nM), Ref: 24215819
TCMC1464	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 3900 (nM), Ref: 18565755 IC50: 8400 (nM), Ref: 18565755
TCMC2093	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 57 (nM), Ref: 17149865
TCMC2093	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 68 (nM), Ref: 17149865
TCMC795	TCMT223	Aldose reductase	Homo sapiens	IC50: 8000 (nM), Ref: 24341381
TCMC242	TCMT158	Epoxide hydratase	Homo sapiens	IC50: 52 (nM), Ref: 17616115 IC50: 52 (nM), Ref: 22079754 IC50: 25.3 (nM), Ref: 24656800 IC50: 3 (nM), Ref: 24685540 IC50: 5.1 (nM), Ref: 24685540 IC50: 25 (nM), Ref: 27096037
TCMC242	TCMT572	Epoxide hydrolase 1	Homo sapiens	IC50: 160 (nM), Ref: 10.1007/s00044-011-9953-1 IC50: 160 (nM), Ref:
TCMC1451	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 2700 (nM), Ref: 19846295
TCMC2119	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 9140 (nM), Ref: 20185318
TCMC2119	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9010 (nM), Ref: 20185318
TCMC2119	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8200 (nM), Ref: 20185318
TCMC2119	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7810 (nM), Ref: 20185318
TCMC2119	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7550 (nM), Ref: 20185318
TCMC2119	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6340 (nM), Ref: 20185318
TCMC2119	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8580 (nM), Ref: 20185318
TCMC2119	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3190 (nM), Ref: 20185318
TCMC2119	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4150 (nM), Ref: 20185318
TCMC1773	TCMT575	Phospholipase A2 group IIA	Homo sapiens	IC50: 3500 (nM), Ref: 16504502
TCMC1293	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2940 (nM), Ref: 19231207
TCMC231	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 4800 (nM), Ref: 20806783
TCMC1429	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2700 (nM), Ref: 17378609
TCMC1429	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 1050 (nM), Ref: 18533708
TCMC1429	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 360 (nM), Ref: 18533708
TCMC1429	TCMT187	Androgen Receptor	Homo sapiens	IC50: 9700 (nM), Ref: 19592245
TCMC1429	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 716 (nM), Ref: 20696580
TCMC1429	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 632 (nM), Ref: 20696580
TCMC1429	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 47 (nM), Ref: 20696580
TCMC1429	TCMT223	Aldose reductase	Homo sapiens	IC50: 10000 (nM), Ref: 22261024
TCMC1429	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 2320 (nM), Ref: 23411073
TCMC1429	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 9640 (nM), Ref: 23656512
TCMC1429	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 10000 (nM), Ref: 26322379
TCMC1429	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9525.7 (nM), Ref: 26498393
TCMC1429	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 25 (nM), Ref: 26498393
TCMC1429	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 145.9 (nM), Ref: 26498393
TCMC1429	TCMT159	Tyrosinase	Homo sapiens	IC50: 1000 (nM), Ref: 26841168
TCMC1255	TCMT33	Cytochrome P450 3A4	Homo sapiens	Ki: 7000 (nM), Ref: 16248836
TCMC920	TCMT112	Adenosine A3 receptor	Homo sapiens	Ki: 1720 (nM), Ref: 8576921
TCMC2188	TCMT223	Aldose reductase	Homo sapiens	IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 452.6 (nM), Ref: 26498393
TCMC1965	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 515 (nM), Ref: 26498393
TCMC1411	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1261 (nM), Ref: 20696580
TCMC1411	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 56 (nM), Ref: 20696580
TCMC1411	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 17 (nM), Ref: 20696580
TCMC1411	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 212.9 (nM), Ref: 26498393
TCMC1411	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.4 (nM), Ref: 26498393
TCMC1411	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 54.9 (nM), Ref: 26498393 Ki: 220 (nM), Ref: 26498393
TCMC1411	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 440 (nM), Ref: 26498393
TCMC13	TCMT23	Alkaline phosphatase, tissue-nonspecific isozyme	Homo sapiens	IC50: 407 (nM), Ref:
TCMC1620	TCMT223	Aldose reductase	Homo sapiens	IC50: 88 (nM), Ref: 22236472
TCMC1620	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 130 (nM), Ref: 22236472
TCMC2054	TCMT240	Salivary alpha-amylase	Homo sapiens	IC50: 9640 (nM), Ref: 18507367
TCMC2054	TCMT384	G protein-coupled receptor kinase 6	Homo sapiens	IC50: 6610 (nM), Ref:
TCMC2054	TCMT283	Receptor-type tyrosine-protein phosphatase S	Homo sapiens	IC50: 600 (nM), Ref: 26602279
TCMC737	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 168 (nM), Ref: 26498393
TCMC737	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 5591.2 (nM), Ref: 26498393
TCMC737	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 423.7 (nM), Ref: 26498393
TCMC737	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4.9 (nM), Ref: 26498393
TCMC1041	TCMT636	DNA polymerase alpha subunit	Homo sapiens	Ki: 830 (nM), Ref: 1705574
TCMC1041	TCMT17	DNA polymerase beta	Homo sapiens	Ki: 390 (nM), Ref: 1705574
TCMC1430	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC856	TCMT125	Beta-glucocerebrosidase	Homo sapiens	IC50: 1000 (nM), Ref: 21292481 IC50: 5100 (nM), Ref: 24657053 Ki: 3800 (nM), Ref: 24657053
TCMC949	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8900 (nM), Ref: 19911821
TCMC949	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 48 (nM), Ref: 19911821
TCMC949	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9100 (nM), Ref: 19911821
TCMC949	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3300 (nM), Ref: 19911821
TCMC949	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 2000 (nM), Ref: 19911821
TCMC949	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 5200 (nM), Ref: 19911821
TCMC949	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9400 (nM), Ref: 19911821
TCMC949	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 6800 (nM), Ref: 19911821
TCMC949	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 5600 (nM), Ref: 19911821
TCMC949	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270
TCMC949	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270
TCMC498	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 410 (nM), Ref: 26688270
TCMC498	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 6300 (nM), Ref: 26688270
TCMC1786	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900
TCMC1786	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086
TCMC1786	TCMT190	T-cell protein-tyrosine phosphatase	Homo sapiens	IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900
TCMC1786	TCMT563	Dual specificity phosphatase Cdc25B	Homo sapiens	IC50: 980 (nM), Ref: 25497963
TCMC1735	TCMT599	Ubiquitin-conjugating enzyme E2 N	Homo sapiens	IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC845	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 630 (nM), Ref: 19231207
TCMC1083	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867
TCMC1083	TCMT651	Dopamine D3 receptor	Homo sapiens	Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329
TCMC1083	TCMT635	Dopamine transporter	Homo sapiens	Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523
TCMC1083	TCMT634	Norepinephrine transporter	Homo sapiens	IC50: 6.63 (nM), Ref: 14592523
TCMC1083	TCMT648	Dopamine D4 receptor	Homo sapiens	Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965
TCMC1083	TCMT316	Melatonin receptor 1A	Homo sapiens	Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083	TCMT317	Melatonin receptor 1B	Homo sapiens	Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7
TCMC1083	TCMT27	Dopamine D1 receptor	Homo sapiens	Ki: 4470 (nM), Ref: 23134120
TCMC1083	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC315	TCMT46	Coagulation factor III	Homo sapiens	IC50: 14.98 (nM), Ref: 23199480
TCMC1376	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 40 (nM), Ref: 11678654
TCMC1501	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 2100 (nM), Ref: 18042388 IC50: 340 (nM), Ref: 18778944
TCMC1189	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9890 (nM), Ref: 22892213
TCMC1189	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7840 (nM), Ref: 22892213
TCMC1189	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 5560 (nM), Ref: 22892213
TCMC1189	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 850 (nM), Ref: 22892213
TCMC2124	TCMT39	Phosphodiesterase 5A	Homo sapiens	IC50: 4703 (nM), Ref:
TCMC2124	TCMT289	Thromboxane-A synthase	Homo sapiens	IC50: 325 (nM), Ref:
TCMC1594	TCMT197	Phosphodiesterase 4D	Homo sapiens	IC50: 2900 (nM), Ref: 22483586 IC50: 2910 (nM), Ref: 26473791
TCMC1594	TCMT698	Phosphodiesterase 4B	Homo sapiens	IC50: 4500 (nM), Ref: 22483586
TCMC1844	TCMT113	Delta opioid receptor	Homo sapiens	Ki: 8400 (nM), Ref: 26035635
TCMC1844	TCMT510	Stem cell growth factor receptor	Homo sapiens	IC50: 600 (nM), Ref: 26807861 IC50: 1500 (nM), Ref: 26807861
TCMC632	TCMT597	Solute carrier family 28 member 3	Homo sapiens	Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705
TCMC632	TCMT709	Sodium/nucleoside cotransporter 2	Homo sapiens	Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT710	Sodium/nucleoside cotransporter 1	Homo sapiens	Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705
TCMC632	TCMT296	Adenosine A1 receptor	Homo sapiens	IC50: 2.344 (nM), Ref: 26756468
TCMC632	TCMT112	Adenosine A3 receptor	Homo sapiens	IC50: 1.148 (nM), Ref: 26756468
TCMC1956	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1080 (nM), Ref: 21282059
TCMC1956	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 470 (nM), Ref: 21282059
TCMC1956	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4450 (nM), Ref: 21282059
TCMC1956	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4090 (nM), Ref: 21282059
TCMC1956	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439
TCMC1956	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 2450 (nM), Ref: 22687439
TCMC1956	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 690 (nM), Ref: 22668600
TCMC1956	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7870 (nM), Ref: 22668600
TCMC670	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 7700 (nM), Ref: 15679319
TCMC1113	TCMT47	Apoptosis regulator Bcl-2	Homo sapiens	Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC2003	TCMT82	Estrogen receptor alpha	Homo sapiens	Ki: 785 (nM), Ref: 15634023
TCMC2003	TCMT164	Cyclooxygenase-1	Homo sapiens	IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref:
TCMC2003	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006
TCMC2003	TCMT329	Quinone reductase 2	Homo sapiens	IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376
TCMC2003	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2210 (nM), Ref: 20674354
TCMC2003	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2770 (nM), Ref: 20674354
TCMC2003	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 9090 (nM), Ref: 20674354
TCMC2003	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4470 (nM), Ref: 20674354
TCMC2003	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4750 (nM), Ref: 20674354
TCMC2003	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4640 (nM), Ref: 20674354
TCMC2003	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 8070 (nM), Ref: 20674354
TCMC2003	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4350 (nM), Ref: 20674354
TCMC2003	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 810 (nM), Ref: 20674354
TCMC2003	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 950 (nM), Ref: 20674354
TCMC2003	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4090 (nM), Ref: 20674354
TCMC2003	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 830 (nM), Ref: 20674354
TCMC2003	TCMT729	PI3-kinase p110-alpha subunit	Homo sapiens	IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003	TCMT730	PI3-kinase p110-beta subunit	Homo sapiens	IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601
TCMC1591	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 4600 (nM), Ref: 11678652
TCMC577	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 190 (nM), Ref: 26688270
TCMC577	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 680 (nM), Ref: 26688270
TCMC1446	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 6300 (nM), Ref: 21641214
TCMC1758	TCMT247	Alpha-2a adrenergic receptor	Homo sapiens	Ki: 66 (nM), Ref: 8632424
TCMC1758	TCMT243	Alpha-2c adrenergic receptor	Homo sapiens	Ki: 63 (nM), Ref: 8632424
TCMC1758	TCMT559	Beta-2 adrenergic receptor	Homo sapiens	Ki: 3300 (nM), Ref: 27132867
TCMC1758	TCMT38	Dopamine D2 receptor	Homo sapiens	Ki: 1300 (nM), Ref: 27132867
TCMC1603	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 4900 (nM), Ref: 16356713
TCMC1609	TCMT44	Glyoxalase I	Homo sapiens	IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529
TCMC1609	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18778944
TCMC1609	TCMT737	DNA dC->dU-editing enzyme APOBEC-3G	Homo sapiens	IC50: 2390 (nM), Ref:
TCMC1609	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 2120 (nM), Ref: 24900447
TCMC1609	TCMT558	DNA topoisomerase II alpha	Homo sapiens	IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1690 (nM), Ref: 23411073
TCMC1609	TCMT2	Microtubule-associated protein tau	Homo sapiens	IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 3000 (nM), Ref: 25086914
TCMC1609	TCMT740	PI3-kinase p110-gamma subunit	Homo sapiens	IC50: 4720 (nM), Ref: 25050878
TCMC1609	TCMT13	DNA-(apurinic or apyrimidinic site) lyase	Homo sapiens	IC50: 320 (nM), Ref: 25280182
TCMC1399	TCMT223	Aldose reductase	Homo sapiens	IC50: 320 (nM), Ref: 22261024
TCMC575	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 2400 (nM), Ref: 26704263 Ki: 2500 (nM), Ref: 26704263
TCMC584	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 2 (nM), Ref: 20413308
TCMC1986	TCMT223	Aldose reductase	Homo sapiens	IC50: 150 (nM), Ref: 18165015 IC50: 2000 (nM), Ref: 22261024
TCMC2031	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 7500 (nM), Ref: 16610779
TCMC1102	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 40 (nM), Ref: 19414254
TCMC1102	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2320 (nM), Ref: 20185318
TCMC1102	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2180 (nM), Ref: 20185318
TCMC1102	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9080 (nM), Ref: 20185318
TCMC1102	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 7590 (nM), Ref: 20185318
TCMC1102	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7060 (nM), Ref: 20185318
TCMC1102	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213
TCMC1102	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 9370 (nM), Ref: 20185318
TCMC1102	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 8910 (nM), Ref: 20185318
TCMC1102	TCMT753	Mothers against decapentaplegic homolog 3	Homo sapiens	IC50: 142 (nM), Ref:
TCMC1102	TCMT721	Heat shock 70 kDa protein 1	Homo sapiens	IC50: 760 (nM), Ref:
TCMC1102	TCMT189	Dual specificity protein phosphatase 3	Homo sapiens	IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102	TCMT223	Aldose reductase	Homo sapiens	IC50: 200 (nM), Ref: 22261024
TCMC1102	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 510 (nM), Ref: 22377675
TCMC1102	TCMT354	Serine/threonine-protein kinase Aurora-A	Homo sapiens	IC50: 2480 (nM), Ref: 22377675
TCMC1102	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 2500 (nM), Ref: 22377675
TCMC1102	TCMT626	Serine/threonine-protein kinase B-raf	Homo sapiens	IC50: 1760 (nM), Ref: 22377675
TCMC1102	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 690 (nM), Ref: 22377675
TCMC1102	TCMT418	Ephrin type-B receptor 4	Homo sapiens	IC50: 1830 (nM), Ref: 22377675
TCMC1102	TCMT704	Receptor protein-tyrosine kinase erbB-2	Homo sapiens	IC50: 3540 (nM), Ref: 22377675
TCMC1102	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 3110 (nM), Ref: 22377675
TCMC1102	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 250 (nM), Ref: 22377675
TCMC1102	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 800 (nM), Ref: 22377675
TCMC1102	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 790 (nM), Ref: 22377675
TCMC1102	TCMT457	Vascular endothelial growth factor receptor 3	Homo sapiens	IC50: 1540 (nM), Ref: 22377675
TCMC1102	TCMT377	Insulin receptor	Homo sapiens	IC50: 340 (nM), Ref: 22377675
TCMC1102	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 22377675
TCMC1102	TCMT536	Platelet-derived growth factor receptor beta	Homo sapiens	IC50: 1300 (nM), Ref: 22377675
TCMC1102	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 3340 (nM), Ref: 22377675
TCMC1102	TCMT755	Serine/threonine-protein kinase PLK4	Homo sapiens	IC50: 2970 (nM), Ref: 22377675
TCMC1102	TCMT502	Tyrosine-protein kinase TIE-2	Homo sapiens	IC50: 260 (nM), Ref: 22377675
TCMC1102	TCMT756	Mitogen-activated protein kinase kinase kinase 8	Homo sapiens	IC50: 2370 (nM), Ref: 22377675
TCMC1102	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 100 (nM), Ref: 24900447
TCMC1102	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 8150 (nM), Ref: 22892213
TCMC1102	TCMT225	Carbonic anhydrase XIII	Homo sapiens	Ki: 4240 (nM), Ref: 22892213
TCMC1102	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3900 (nM), Ref: 24835197
TCMC1409	TCMT22	Intestinal alkaline phosphatase	Homo sapiens	IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409	TCMT223	Aldose reductase	Homo sapiens	IC50: 4500 (nM), Ref: 22261024
TCMC1409	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393
TCMC1409	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 75.7 (nM), Ref: 26498393
TCMC1409	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3.8 (nM), Ref: 26498393
TCMC1409	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393
TCMC910	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1118 (nM), Ref: 20696580
TCMC910	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 95 (nM), Ref: 20696580
TCMC910	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 20 (nM), Ref: 20696580
TCMC1982	TCMT239	Serine/threonine-protein kinase PIM1	Homo sapiens	IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302
TCMC1982	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208
TCMC1982	TCMT223	Aldose reductase	Homo sapiens	IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999
TCMC405	TCMT506	Protein tyrosine kinase 2 beta	Homo sapiens	IC50: 2324 (nM), Ref:
TCMC1982	TCMT44	Glyoxalase I	Homo sapiens	IC50: 3200 (nM), Ref: 18258440
TCMC1201	TCMT112	Adenosine A3 receptor	Homo sapiens	Ki: 3150 (nM), Ref: 8576921
TCMC1201	TCMT132	Butyrylcholinesterase	Homo sapiens	Ki: 6900 (nM), Ref: 19879672
TCMC1201	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 77 (nM), Ref: 20696580
TCMC1201	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 40 (nM), Ref: 20696580
TCMC1201	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC1201	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1201	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 568.3 (nM), Ref: 26498393
TCMC1201	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 24.5 (nM), Ref: 26498393
TCMC1201	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 41.8 (nM), Ref: 26498393
TCMC1982	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 1540 (nM), Ref: 18533708
TCMC970	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC970	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7890 (nM), Ref: 20185318
TCMC1982	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8100 (nM), Ref: 20185318
TCMC1982	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2540 (nM), Ref: 20185318
TCMC1982	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2680 (nM), Ref: 20185318
TCMC1982	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6810 (nM), Ref: 20185318
TCMC1982	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6170 (nM), Ref: 20185318
TCMC1982	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4840 (nM), Ref: 20185318
TCMC1982	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 7000 (nM), Ref: 20185318
TCMC1982	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9390 (nM), Ref: 20185318
TCMC1982	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 5410 (nM), Ref: 20185318
TCMC1158	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 3100 (nM), Ref: 24835197 Ki: 6840 (nM), Ref: 24835197
TCMC1982	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 12 (nM), Ref: 20413308
TCMC1982	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583
TCMC1982	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1191 (nM), Ref: 20696580
TCMC1982	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 77 (nM), Ref: 20696580
TCMC1982	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 6680 (nM), Ref: 22658537
TCMC1982	TCMT320	Matrix metalloproteinase 3	Homo sapiens	IC50: 5570 (nM), Ref: 22658537
TCMC1982	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 1610 (nM), Ref: 22658537
TCMC1982	TCMT322	Matrix metalloproteinase 13	Homo sapiens	IC50: 8460 (nM), Ref: 22658537
TCMC1982	TCMT422	CaM kinase II beta	Homo sapiens	IC50: 3000 (nM), Ref: 21798748
TCMC1982	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344
TCMC1982	TCMT784	Vasopressin V2 receptor	Homo sapiens	IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772
TCMC1982	TCMT785	Interleukin-8 receptor A	Homo sapiens	IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772
TCMC1982	TCMT786	C-C chemokine receptor type 4	Homo sapiens	IC50: 10000 (nM), Ref: 23437772
TCMC1982	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 590 (nM), Ref: 23411073
TCMC645	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 9200 (nM), Ref: 19846295
TCMC1982	TCMT601	Thrombin	Homo sapiens	IC50: 1500 (nM), Ref: 24610996
TCMC1982	TCMT370	Vascular endothelial growth factor receptor 2	Homo sapiens	IC50: 280 (nM), Ref: 24328302
TCMC1982	TCMT212	Tyrosine-protein kinase SRC	Homo sapiens	IC50: 120 (nM), Ref: 24328302
TCMC1982	TCMT791	Protein kinase N1	Homo sapiens	IC50: 5800 (nM), Ref: 24328302
TCMC1982	TCMT484	Serine/threonine-protein kinase PLK1	Homo sapiens	IC50: 5750 (nM), Ref: 24328302
TCMC1982	TCMT462	Serine/threonine-protein kinase NEK6	Homo sapiens	IC50: 4230 (nM), Ref: 24328302
TCMC1982	TCMT445	Serine/threonine-protein kinase NEK2	Homo sapiens	IC50: 5730 (nM), Ref: 24328302
TCMC1982	TCMT401	Hepatocyte growth factor receptor	Homo sapiens	IC50: 580 (nM), Ref: 24328302
TCMC1982	TCMT369	Insulin-like growth factor I receptor	Homo sapiens	IC50: 300 (nM), Ref: 24328302
TCMC1982	TCMT441	Focal adhesion kinase 1	Homo sapiens	IC50: 1200 (nM), Ref: 24328302
TCMC1982	TCMT388	Tyrosine-protein kinase receptor UFO	Homo sapiens	IC50: 960 (nM), Ref: 24328302
TCMC1982	TCMT374	Serine/threonine-protein kinase Aurora-B	Homo sapiens	IC50: 910 (nM), Ref: 24328302
TCMC1982	TCMT436	NUAK family SNF1-like kinase 1	Homo sapiens	IC50: 5090 (nM), Ref: 24328302
TCMC1982	TCMT402	ALK tyrosine kinase receptor	Homo sapiens	IC50: 3320 (nM), Ref: 24328302
TCMC1982	TCMT479	Serine/threonine-protein kinase AKT	Homo sapiens	IC50: 5390 (nM), Ref: 24328302
TCMC1982	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124
TCMC1982	TCMT793	Liver glycogen phosphorylase	Homo sapiens	IC50: 4800 (nM), Ref: 25092521
TCMC1982	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 2110 (nM), Ref: 22328583
TCMC1982	TCMT217	Cytochrome P450 2C8	Homo sapiens	IC50: 1390 (nM), Ref: 22328583
TCMC614	TCMT151	Protein kinase C alpha	Homo sapiens	IC50: 9300 (nM), Ref: 9834166
TCMC1982	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 8900 (nM), Ref: 26322379
TCMC1398	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 100 (nM), Ref: 11678652
TCMC1281	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 10 (nM), Ref: 19564108 IC50: 18.6 (nM), Ref: 22148241 IC50: 6 (nM), Ref: 22360639
TCMC1281	TCMT209	11-beta-hydroxysteroid dehydrogenase 2	Homo sapiens	IC50: 1 (nM), Ref: 19564108 IC50: 0.7 (nM), Ref: 22148241 IC50: 0.4 (nM), Ref: 22360639
TCMC1380	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3000 (nM), Ref: 26841168
TCMC1013	TCMT124	Alpha-L-fucosidase I	Homo sapiens	Ki: 10 (nM), Ref: 16481162 IC50: 140 (nM), Ref: 24026016
TCMC533	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 9300 (nM), Ref: 26704263 Ki: 9600 (nM), Ref: 26704263
TCMC469	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 100 (nM), Ref: 22921742
TCMC916	TCMT161	Hydroxycarboxylic acid receptor 2	Homo sapiens	Ki: 4900 (nM), Ref: 21167710
TCMC1015	TCMT318	Putative hexokinase HKDC1	Homo sapiens	IC50: 4320 (nM), Ref:
TCMC2196	TCMT30	Cyclooxygenase-2	Homo sapiens	IC50: 64 (nM), Ref: 22819942 IC50: 64 (nM), Ref: 23146282
TCMC2196	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 150 (nM), Ref: 22819942
TCMC2196	TCMT336	Indoleamine 2,3-dioxygenase	Homo sapiens	IC50: 53.7 (nM), Ref: 24099220 IC50: 7150 (nM), Ref: 24099220 Ki: 4810 (nM), Ref: 24099220
TCMC1268	TCMT278	Solute carrier organic anion transporter family member 1B1	Homo sapiens	IC50: 1400 (nM), Ref: 22587986 IC50: 2200 (nM), Ref: 22587986
TCMC1268	TCMT221	Bile salt export pump	Homo sapiens	IC50: 5300 (nM), Ref: 21965623
TCMC2105	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC22	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 1000 (nM), Ref: 15679319 Ki: 177 (nM), Ref: 16248836
TCMC1597	TCMT807	Solute carrier family 22 member 12	Homo sapiens	IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024
TCMC1597	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 2927.18 (nM), Ref:
TCMC1597	TCMT61	Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens	IC50: 2988.26 (nM), Ref:
TCMC1597	TCMT739	G-protein coupled receptor 35	Homo sapiens	IC50: 1600 (nM), Ref: 24900447
TCMC1597	TCMT261	Death-associated protein kinase 1	Homo sapiens	IC50: 1600 (nM), Ref: 26322379
TCMC1597	TCMT283	Receptor-type tyrosine-protein phosphatase S	Homo sapiens	IC50: 4300 (nM), Ref: 26602279
TCMC1830	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	IC50: 930 (nM), Ref: 15357969
TCMC1830	TCMT298	Fatty acid binding protein muscle	Homo sapiens	IC50: 2600 (nM), Ref: 15357969
TCMC1830	TCMT808	Fatty acid binding protein epidermal	Homo sapiens	IC50: 1200 (nM), Ref: 15357969
TCMC1830	TCMT809	Fatty acid binding protein intestinal	Homo sapiens	IC50: 1700 (nM), Ref: 15357969
TCMC1830	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1830	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1602	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1602	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1432	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8790.2 (nM), Ref: 26498393
TCMC1432	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 344.2 (nM), Ref: 26498393
TCMC1432	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.7 (nM), Ref: 26498393
TCMC1432	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 408.9 (nM), Ref: 26498393
TCMC596	TCMT39	Phosphodiesterase 5A	Homo sapiens	IC50: 1290 (nM), Ref: 18778098
TCMC1596	TCMT11	Hypoxia-inducible factor 1 alpha	Homo sapiens	IC50: 6.76 (nM), Ref: 21481991
TCMC2094	TCMT238	Sodium/glucose cotransporter 2	Homo sapiens	IC50: 4100 (nM), Ref: 17374486
TCMC2094	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 1100 (nM), Ref: 18565755 IC50: 5200 (nM), Ref: 18565755
TCMC846	TCMT207	Beta-secretase 1	Homo sapiens	Ki: 6200 (nM), Ref: 22222157
TCMC418	TCMT223	Aldose reductase	Homo sapiens	IC50: 78 (nM), Ref: 22236472
TCMC418	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 240 (nM), Ref: 22236472
TCMC418	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 4700 (nM), Ref: 22921742
TCMC1202	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 7030 (nM), Ref: 20185318
TCMC1202	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1202	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6990 (nM), Ref: 20185318
TCMC1202	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6070 (nM), Ref: 20185318
TCMC1202	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 6130 (nM), Ref: 20185318
TCMC1202	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9970 (nM), Ref: 20185318
TCMC1202	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1202	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9800 (nM), Ref: 20185318
TCMC1202	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 7490 (nM), Ref: 20185318
TCMC1202	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 2250 (nM), Ref: 20185318
TCMC1202	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3200 (nM), Ref: 20185318
TCMC1202	TCMT822	Alpha-(1,3)-fucosyltransferase 7	Homo sapiens	IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1869	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 4410 (nM), Ref: 15658857
TCMC606	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 251 (nM), Ref: 20696580
TCMC606	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 86 (nM), Ref: 20696580
TCMC606	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 12 (nM), Ref: 20696580
TCMC587	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 9900 (nM), Ref: 26841168
TCMC1111	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 11.78 (nM), Ref: 18242087 IC50: 13 (nM), Ref: 18653260 IC50: 778 (nM), Ref: 20851614 IC50: 778 (nM), Ref: 21376605 IC50: 8.6 (nM), Ref: 21873057 IC50: 29.1 (nM), Ref: 23747808 IC50: 29.1 (nM), Ref: 25590374
TCMC1111	TCMT209	11-beta-hydroxysteroid dehydrogenase 2	Homo sapiens	IC50: 257 (nM), Ref: 20851614 IC50: 257 (nM), Ref: 21376605 IC50: 1.22 (nM), Ref: 23747808 IC50: 1.2 (nM), Ref: 25590374
TCMC1111	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 4900 (nM), Ref: 21561086
TCMC983	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref:
TCMC983	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 7300 (nM), Ref: 21030469
TCMC983	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 718.7 (nM), Ref: 26498393
TCMC983	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.2 (nM), Ref: 26498393
TCMC983	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 56.4 (nM), Ref: 26498393
TCMC84	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 6700 (nM), Ref: 18565755
TCMC183	TCMT188	Dihydrofolate reductase	Homo sapiens	IC50: 500 (nM), Ref: 26979156
TCMC2111	TCMT614	Egl nine homolog 1	Homo sapiens	IC50: 3000 (nM), Ref: 18942826
TCMC755	TCMT3	Arachidonate 15-lipoxygenase	Homo sapiens	Ki: 600 (nM), Ref: 21739938
TCMC755	TCMT81	Arachidonate 12-lipoxygenase	Homo sapiens	Ki: 1600 (nM), Ref: 21739938
TCMC755	TCMT8	Lysine-specific demethylase 4D-like	Homo sapiens	IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755	TCMT162	UDP-glucuronosyltransferase 1-1	Homo sapiens	IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469
TCMC755	TCMT384	G protein-coupled receptor kinase 6	Homo sapiens	IC50: 8700 (nM), Ref:
TCMC1329	TCMT239	Serine/threonine-protein kinase PIM1	Homo sapiens	IC50: 2710 (nM), Ref: 26275107
TCMC1428	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 509 (nM), Ref: 20696580
TCMC1428	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 88 (nM), Ref: 20696580
TCMC1428	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC412	TCMT683	Macrophage migration inhibitory factor	Homo sapiens	Ki: 38 (nM), Ref: 19090668 IC50: 38 (nM), Ref: 27156768
TCMC1898	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 7906 (nM), Ref: 20696580
TCMC1898	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 1679 (nM), Ref: 20696580
TCMC1898	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 1491 (nM), Ref: 20696580
TCMC1898	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 900 (nM), Ref: 10.1039/C3MD00166K
TCMC1774	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 3100 (nM), Ref: 20674354 Ki: 3100 (nM), Ref: 21282059 Ki: 3400 (nM), Ref: 22137345
TCMC1774	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9300 (nM), Ref: 22137345
TCMC2204	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270
TCMC2204	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270
TCMC2239	TCMT226	3-phosphoinositide dependent protein kinase-1	Homo sapiens	IC50: 6600 (nM), Ref: 22537682
TCMC2239	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 2100 (nM), Ref: 26918635 IC50: 2900 (nM), Ref: 26918635
TCMC1118	TCMT304	Matrix metalloproteinase 14	Homo sapiens	IC50: 6800 (nM), Ref: 19524436
TCMC1118	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 9600 (nM), Ref: 19524436
TCMC1118	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 757 (nM), Ref: 22225636
TCMC1118	TCMT126	Telomerase reverse transcriptase	Homo sapiens	IC50: 1000 (nM), Ref: 22413845 IC50: 1080 (nM), Ref: 22413845 IC50: 1180 (nM), Ref: 22413845 IC50: 1000 (nM), Ref: 10.1039/C0MD00241K
TCMC1118	TCMT47	Apoptosis regulator Bcl-2	Homo sapiens	Ki: 335 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1118	TCMT2	Microtubule-associated protein tau	Homo sapiens	IC50: 1800 (nM), Ref: 23484434
TCMC1118	TCMT751	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Homo sapiens	IC50: 330 (nM), Ref: 24188002
TCMC1118	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 4600 (nM), Ref: 24878198 IC50: 3000 (nM), Ref: 24878198 IC50: 500 (nM), Ref: 25978520
TCMC1118	TCMT567	DNA (cytosine-5)-methyltransferase 1	Homo sapiens	IC50: 500 (nM), Ref: 25406944
TCMC1118	TCMT232	P-glycoprotein 1	Homo sapiens	IC50: 124.1 (nM), Ref: 25985195 IC50: 122.6 (nM), Ref: 25985195
TCMC2043	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 1600 (nM), Ref: 16356713
TCMC1839	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318
TCMC1839	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318
TCMC1839	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318
TCMC1839	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 6160 (nM), Ref: 20185318
TCMC1839	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 3730 (nM), Ref: 20185318
TCMC1839	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4080 (nM), Ref: 20185318
TCMC1839	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 5700 (nM), Ref: 20185318
TCMC1839	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 7130 (nM), Ref: 20185318
TCMC1839	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7780 (nM), Ref: 20185318
TCMC1839	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 6610 (nM), Ref: 20185318
TCMC1839	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 870 (nM), Ref: 20185318
TCMC1377	TCMT186	Monoamine oxidase B	Homo sapiens	Ki: 3000 (nM), Ref: 16137882 Ki: 3000 (nM), Ref: 19342233 IC50: 7943.28 (nM), Ref: 20934874 Ki: 5340 (nM), Ref: 21134756 Ki: 3000 (nM), Ref: 21778064 Ki: 2000 (nM), Ref: 24140951
TCMC1377	TCMT208	Monoamine oxidase A	Homo sapiens	Ki: 8380 (nM), Ref: 21134756
TCMC1105	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 2000 (nM), Ref: 19414254
TCMC1105	TCMT239	Serine/threonine-protein kinase PIM1	Homo sapiens	IC50: 2500 (nM), Ref: 27173800
TCMC1400	TCMT223	Aldose reductase	Homo sapiens	IC50: 720 (nM), Ref: 22261024
TCMC1788	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788	TCMT126	Telomerase reverse transcriptase	Homo sapiens	IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788	TCMT297	Fatty acid binding protein adipocyte	Homo sapiens	Ki: 1500 (nM), Ref: 27460668
TCMC937	TCMT232	P-glycoprotein 1	Homo sapiens	IC50: 11.5 (nM), Ref: 23332369 IC50: 6.6 (nM), Ref: 23895532
TCMC937	TCMT801	Tubulin beta-3 chain	Homo sapiens	IC50: 5.2 (nM), Ref: 23332369 IC50: 5.7 (nM), Ref: 23895532
TCMC1203	TCMT822	Alpha-(1,3)-fucosyltransferase 7	Homo sapiens	IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC804	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 2000 (nM), Ref: 21561086
TCMC1489	TCMT223	Aldose reductase	Homo sapiens	IC50: 560 (nM), Ref: 22261024
TCMC453	TCMT588	D-amino-acid oxidase	Homo sapiens	Ki: 156 (nM), Ref: 23391306 IC50: 943 (nM), Ref: 23391306 IC50: 440 (nM), Ref: 23391306 IC50: 34.67 (nM), Ref: 23631755 Ki: 13 (nM), Ref: 23631755
TCMC1204	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2500 (nM), Ref: 14592472
TCMC1516	TCMT44	Glyoxalase I	Homo sapiens	IC50: 7700 (nM), Ref: 18258440
TCMC1516	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 3370 (nM), Ref: 20696580
TCMC1516	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 1249 (nM), Ref: 20696580
TCMC1516	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 79 (nM), Ref: 20696580
TCMC1516	TCMT83	Lymphocyte differentiation antigen CD38	Homo sapiens	IC50: 8200 (nM), Ref: 21641214
TCMC1516	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 3610 (nM), Ref: 22658537
TCMC1516	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 5620 (nM), Ref: 22658537
TCMC1516	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 980 (nM), Ref: 22658537
TCMC1516	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 830 (nM), Ref: 23411073
TCMC1516	TCMT127	Poly [ADP-ribose] polymerase-1	Homo sapiens	IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272
TCMC1516	TCMT128	Tankyrase-2	Homo sapiens	IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272
TCMC1516	TCMT129	Tankyrase-1	Homo sapiens	IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272
TCMC1516	TCMT223	Aldose reductase	Homo sapiens	IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431
TCMC1516	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 1600 (nM), Ref: 24368208
TCMC1516	TCMT45	Beta amyloid A4 protein	Homo sapiens	IC50: 6400 (nM), Ref: 24878198
TCMC1516	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677
TCMC1516	TCMT100	Transthyretin	Homo sapiens	IC50: 7000 (nM), Ref: 26214366
TCMC1516	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 3691.6 (nM), Ref: 26498393
TCMC1516	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.7 (nM), Ref: 26498393
TCMC1516	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 60.3 (nM), Ref: 26498393
TCMC1516	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 293 (nM), Ref: 26498393
TCMC1516	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 9200 (nM), Ref: 26529431
TCMC1977	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 7410 (nM), Ref: 21669522
TCMC1977	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 540 (nM), Ref: 21669522
TCMC1977	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 520 (nM), Ref: 21669522
TCMC1179	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5900 (nM), Ref: 19592245 IC50: 5900 (nM), Ref: 19592245
TCMC1179	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 8 (nM), Ref: 20413308 IC50: 10000 (nM), Ref: 24345481 IC50: 8000 (nM), Ref: 26301554
TCMC1356	TCMT223	Aldose reductase	Homo sapiens	IC50: 3000 (nM), Ref: 22261024
TCMC1179	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 1890 (nM), Ref: 22487176 Ki: 1880 (nM), Ref: 22487176
TCMC1179	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8710 (nM), Ref: 22487176 Ki: 8800 (nM), Ref: 22487176
TCMC1179	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 4130 (nM), Ref: 22487176 Ki: 4220 (nM), Ref: 22487176
TCMC1179	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7220 (nM), Ref: 22487176 Ki: 7330 (nM), Ref: 22487176
TCMC1179	TCMT127	Poly [ADP-ribose] polymerase-1	Homo sapiens	IC50: 1380.38 (nM), Ref: 23574272 IC50: 1400 (nM), Ref: 23574272
TCMC1179	TCMT128	Tankyrase-2	Homo sapiens	IC50: 147.91 (nM), Ref: 23574272 IC50: 140 (nM), Ref: 23574272
TCMC1179	TCMT129	Tankyrase-1	Homo sapiens	IC50: 323.59 (nM), Ref: 23574272 IC50: 320 (nM), Ref: 23574272 IC50: 323.59 (nM), Ref: 24116873 IC50: 330 (nM), Ref: 24116873
TCMC1734	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 3430 (nM), Ref: 19097799
TCMC1734	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 4960 (nM), Ref: 18533708
TCMC1734	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469
TCMC1734	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 3656 (nM), Ref: 20696580
TCMC2228	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 6830 (nM), Ref: 21282059
TCMC2228	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 6180 (nM), Ref: 21282059
TCMC2228	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 8250 (nM), Ref: 21282059
TCMC2228	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 6700 (nM), Ref: 21282059
TCMC2228	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 6480 (nM), Ref: 22687439
TCMC2228	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 740 (nM), Ref: 22668600
TCMC2228	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 7150 (nM), Ref: 22668600
TCMC1734	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 79.5 (nM), Ref: 26498393
TCMC1734	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.3 (nM), Ref: 26498393
TCMC1734	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 44.3 (nM), Ref: 26498393
TCMC1551	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 1900 (nM), Ref: 16248836 Ki: 1900 (nM), Ref: 16248836 Ki: 800 (nM), Ref: 16248836 Ki: 250 (nM), Ref: 22696418
TCMC1551	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 760 (nM), Ref: 23746477
TCMC1551	TCMT268	Cytochrome P450 2A13	Homo sapiens	Ki: 40 (nM), Ref: 22696418
TCMC2114	TCMT683	Macrophage migration inhibitory factor	Homo sapiens	IC50: 2200 (nM), Ref: 25743213
TCMC2114	TCMT423	Epidermal growth factor receptor erbB1	Homo sapiens	IC50: 9000 (nM), Ref: 27135370
TCMC1798	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1480 (nM), Ref: 23411073
TCMC135	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 7400 (nM), Ref: 15679319
TCMC811	TCMT254	Carbonyl reductase [NADPH] 1	Homo sapiens	Ki: 2030 (nM), Ref: 19097799
TCMC811	TCMT66	Estradiol 17-beta-dehydrogenase 2	Homo sapiens	IC50: 9900 (nM), Ref: 18533708
TCMC811	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10.2 (nM), Ref: 20413308
TCMC811	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 7078.5 (nM), Ref: 26498393
TCMC811	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 371.5 (nM), Ref: 26498393
TCMC811	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 52.5 (nM), Ref: 26498393
TCMC1496	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496	TCMT164	Cyclooxygenase-1	Homo sapiens	Ki: 4000 (nM), Ref: 24088053
TCMC1123	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 1284 (nM), Ref: 20696580
TCMC1123	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 72.8 (nM), Ref: 26498393
TCMC1123	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 4.3 (nM), Ref: 26498393
TCMC1123	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 31.1 (nM), Ref: 26498393
TCMC847	TCMT135	Carbonic anhydrase XIV	Homo sapiens	Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394
TCMC847	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394
TCMC847	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 7870 (nM), Ref: 20185318
TCMC847	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 6420 (nM), Ref: 20185318
TCMC847	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 7330 (nM), Ref: 20185318
TCMC847	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 9080 (nM), Ref: 20185318
TCMC847	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 6490 (nM), Ref: 20185318
TCMC847	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 10000 (nM), Ref: 20185318
TCMC847	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1610 (nM), Ref: 20185318
TCMC847	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2380 (nM), Ref: 20185318
TCMC847	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3060 (nM), Ref: 19476336
TCMC847	TCMT321	Matrix metalloproteinase 9	Homo sapiens	IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794
TCMC847	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 24.26 (nM), Ref: 23375794
TCMC847	TCMT295	Matrix metalloproteinase-1	Homo sapiens	IC50: 238.91 (nM), Ref: 23375794
TCMC847	TCMT130	Arachidonate 5-lipoxygenase	Homo sapiens	IC50: 8500 (nM), Ref: 26197161
TCMC1562	TCMT210	Carboxylesterase 2	Homo sapiens	IC50: 5610 (nM), Ref: 26900660
TCMC2201	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8700 (nM), Ref: 21332115
TCMC1873	TCMT210	Carboxylesterase 2	Homo sapiens	Ki: 1840 (nM), Ref: 15828829 Ki: 1840 (nM), Ref: 21733699
TCMC1873	TCMT211	Acyl coenzyme A:cholesterol acyltransferase	Homo sapiens	Ki: 5270 (nM), Ref: 15828829 Ki: 5270 (nM), Ref: 21733699
TCMC1371	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 4 (nM), Ref: 26562543
TCMC1205	TCMT47	Apoptosis regulator Bcl-2	Homo sapiens	Ki: 235 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1611	TCMT810	Toll-like receptor 2	Homo sapiens	IC50: 5000 (nM), Ref: 16509590
TCMC1611	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1003	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 15 (nM), Ref: 20413308
TCMC897	TCMT223	Aldose reductase	Homo sapiens	IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024
TCMC897	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	IC50: 7900 (nM), Ref: 22236472
TCMC1320	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 2786 (nM), Ref: 20696580
TCMC1320	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 511 (nM), Ref: 20696580
TCMC1320	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 102.1 (nM), Ref: 26498393
TCMC1320	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 3.3 (nM), Ref: 26498393
TCMC1320	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 454.1 (nM), Ref: 26498393
TCMC18	TCMT11	Hypoxia-inducible factor 1 alpha	Homo sapiens	IC50: 6.76 (nM), Ref: 21481991
TCMC1832	TCMT63	Peroxisome proliferator-activated receptor alpha	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT64	Peroxisome proliferator-activated receptor delta	Homo sapiens	IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832	TCMT67	Peroxisome proliferator-activated receptor gamma	Homo sapiens	IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1090	TCMT118	Maltase-glucoamylase	Homo sapiens	IC50: 40 (nM), Ref: 15771446
TCMC1090	TCMT18	Lysosomal alpha-glucosidase	Homo sapiens	IC50: 1000 (nM), Ref: 18595718 IC50: 60 (nM), Ref: 18595718 IC50: 1500 (nM), Ref: 19853441
TCMC1940	TCMT187	Androgen Receptor	Homo sapiens	Ki: 8.5 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12954062 IC50: 37 (nM), Ref: 12781197 IC50: 37 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 8627601 Ki: 8.5 (nM), Ref: 9873735 IC50: 37 (nM), Ref: 9784110 Ki: 35 (nM), Ref: 20510622
TCMC1940	TCMT613	Glucocorticoid receptor	Homo sapiens	Ki: 30.5 (nM), Ref: 12954062 Ki: 30.5 (nM), Ref: 9873735 Ki: 30.5 (nM), Ref: 9784110
TCMC1940	TCMT783	Mineralocorticoid receptor	Homo sapiens	IC50: 14 (nM), Ref: 12954062 IC50: 14 (nM), Ref: 12781197 IC50: 14 (nM), Ref: 9784110 IC50: 30 (nM), Ref: 8709117
TCMC1940	TCMT904	Progesterone receptor	Homo sapiens	Ki: 3.5 (nM), Ref: 10212133 IC50: 3.5 (nM), Ref: 11859003 Ki: 3.5 (nM), Ref: 9464361 IC50: 5 (nM), Ref: 8523399 Ki: 3.8 (nM), Ref: 9667968 Ki: 3.467 (nM), Ref: 16821785 Ki: 3.4 (nM), Ref: 18553958 Ki: 5.1 (nM), Ref: 20510622
TCMC1237	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7300 (nM), Ref: 22668600
TCMC1237	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 6600 (nM), Ref: 22668600
TCMC1237	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 4100 (nM), Ref: 22668600
TCMC1237	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 4200 (nM), Ref: 22668600
TCMC1175	TCMT186	Monoamine oxidase B	Homo sapiens	IC50: 2870 (nM), Ref: 20045650
TCMC1175	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 8000 (nM), Ref: 24345481 IC50: 8000 (nM), Ref: 26301554
TCMC2137	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 5750 (nM), Ref: 22658537
TCMC2137	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 9098.2 (nM), Ref: 26498393
TCMC2137	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 493.1 (nM), Ref: 26498393
TCMC2137	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 32.5 (nM), Ref: 26498393
TCMC1267	TCMT159	Tyrosinase	Homo sapiens	IC50: 154 (nM), Ref: 26841168
TCMC1236	TCMT236	Estrogen receptor beta	Homo sapiens	IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref:
TCMC1236	TCMT82	Estrogen receptor alpha	Homo sapiens	IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref:
TCMC1236	TCMT591	Estrogen-related receptor alpha	Homo sapiens	IC50: 10 (nM), Ref: 17482813
TCMC1236	TCMT910	Estrogen-related receptor beta	Homo sapiens	IC50: 395 (nM), Ref: 17482813
TCMC1236	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 2210 (nM), Ref: 18533708
TCMC1236	TCMT344	Aldehyde oxidase	Homo sapiens	IC50: 340 (nM), Ref: 20853847
TCMC1236	TCMT289	Thromboxane-A synthase	Homo sapiens	IC50: 7720 (nM), Ref:
TCMC1048	TCMT33	Cytochrome P450 3A4	Homo sapiens	IC50: 9500 (nM), Ref: 15679319 Ki: 142 (nM), Ref: 16248836
TCMC90	TCMT207	Beta-secretase 1	Homo sapiens	IC50: 2400 (nM), Ref: 14592472
TCMC1521	TCMT306	Matrix metalloproteinase-2	Homo sapiens	IC50: 3880 (nM), Ref: 22658537
TCMC1521	TCMT734	Matrix metalloproteinase 12	Homo sapiens	IC50: 1200 (nM), Ref: 22658537
TCMC1521	TCMT322	Matrix metalloproteinase 13	Homo sapiens	IC50: 7620 (nM), Ref: 22658537
TCMC2055	TCMT747	ATP-binding cassette sub-family G member 2	Homo sapiens	IC50: 10000 (nM), Ref: 22822035
TCMC987	TCMT885	Lysine-specific demethylase 2A	Homo sapiens	Ki: 1970 (nM), Ref: 22724510 IC50: 1500 (nM), Ref: 22724510 IC50: 1500 (nM), Ref: 22724510 IC50: 1500 (nM), Ref: 23964788
TCMC987	TCMT965	Lysine-specific demethylase 7	Homo sapiens	IC50: 2100 (nM), Ref: 22724510
TCMC987	TCMT884	Histone lysine demethylase PHF8	Homo sapiens	IC50: 550 (nM), Ref: 22724510 IC50: 550 (nM), Ref: 23964788
TCMC33	TCMT11	Hypoxia-inducible factor 1 alpha	Homo sapiens	IC50: 0.65 (nM), Ref: 25461329
TCMC710	TCMT249	Cyclin-dependent kinase 6	Homo sapiens	IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554
TCMC710	TCMT65	Estradiol 17-beta-dehydrogenase 1	Homo sapiens	IC50: 710 (nM), Ref: 18533708
TCMC710	TCMT752	Casein kinase II alpha	Homo sapiens	IC50: 800 (nM), Ref: 19414254
TCMC710	TCMT187	Androgen Receptor	Homo sapiens	IC50: 5200 (nM), Ref: 19592245
TCMC710	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 795 (nM), Ref: 20696580
TCMC710	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 427 (nM), Ref: 20696580
TCMC710	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 25 (nM), Ref: 20696580
TCMC710	TCMT265	Glycogen synthase kinase-3 beta	Homo sapiens	IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710	TCMT260	Tyrosine-protein kinase receptor FLT3	Homo sapiens	IC50: 1450 (nM), Ref: 23411073
TCMC710	TCMT128	Tankyrase-2	Homo sapiens	IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272
TCMC710	TCMT129	Tankyrase-1	Homo sapiens	IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272
TCMC710	TCMT592	Xanthine dehydrogenase	Homo sapiens	Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844
TCMC710	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431
TCMC1961	TCMT206	Cytochrome P450 2A6	Homo sapiens	Ki: 600 (nM), Ref: 16248836
TCMC1961	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 6480 (nM), Ref: 23746477
TCMC1174	TCMT249	Cyclin-dependent kinase 6	Homo sapiens	IC50: 850 (nM), Ref: 15689157 IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1174	TCMT131	Acetylcholinesterase	Homo sapiens	IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC2216	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168
TCMC2216	TCMT174	11-beta-hydroxysteroid dehydrogenase 1	Homo sapiens	IC50: 1900 (nM), Ref: 20100662
TCMC2216	TCMT102	Low molecular weight phosphotyrosine protein phosphatase	Homo sapiens	IC50: 7200 (nM), Ref: 21453996
TCMC2216	TCMT103	Receptor-type tyrosine-protein phosphatase F (LAR)	Homo sapiens	IC50: 3800 (nM), Ref: 21453996
TCMC2216	TCMT280	Aldo-keto reductase family 1 member B10	Homo sapiens	Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086
TCMC2216	TCMT190	T-cell protein-tyrosine phosphatase	Homo sapiens	IC50: 2400 (nM), Ref: 23387824
TCMC2216	TCMT150	Nuclear receptor ROR-gamma	Homo sapiens	IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616
TCMC1064	TCMT219	Cytochrome P450 1A2	Homo sapiens	IC50: 2437 (nM), Ref: 20696580
TCMC1064	TCMT215	Cytochrome P450 1A1	Homo sapiens	IC50: 140 (nM), Ref: 20696580
TCMC1064	TCMT257	Cytochrome P450 1B1	Homo sapiens	IC50: 29 (nM), Ref: 20696580
TCMC2180	TCMT302	HMG-CoA reductase	Homo sapiens	IC50: 5860 (nM), Ref: 25311563 IC50: 36.31 (nM), Ref: 25311563
TCMC1403	TCMT223	Aldose reductase	Homo sapiens	IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1266	TCMT159	Tyrosinase	Homo sapiens	IC50: 177 (nM), Ref: 26841168
TCMC700	TCMT101	Protein-tyrosine phosphatase 1B	Homo sapiens	IC50: 400 (nM), Ref: 26841168
TCMC702	TCMT206	Cytochrome P450 2A6	Homo sapiens	IC50: 5150 (nM), Ref: 15658857
TCMC646	TCMT156	Cytochrome P450 19A1	Homo sapiens	IC50: 7500 (nM), Ref: 11678652
TCMC878	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 2420 (nM), Ref: 20674354
TCMC878	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 1840 (nM), Ref: 20674354
TCMC878	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 3580 (nM), Ref: 20674354
TCMC878	TCMT142	Carbonic anhydrase IV	Homo sapiens	Ki: 4900 (nM), Ref: 20674354
TCMC878	TCMT141	Carbonic anhydrase VA	Homo sapiens	Ki: 4210 (nM), Ref: 20674354
TCMC878	TCMT140	Carbonic anhydrase VB	Homo sapiens	Ki: 4020 (nM), Ref: 20674354
TCMC878	TCMT139	Carbonic anhydrase VI	Homo sapiens	Ki: 4910 (nM), Ref: 20674354
TCMC878	TCMT138	Carbonic anhydrase VII	Homo sapiens	Ki: 450 (nM), Ref: 20674354
TCMC878	TCMT137	Carbonic anhydrase IX	Homo sapiens	Ki: 5030 (nM), Ref: 20674354
TCMC878	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 4720 (nM), Ref: 20674354
TCMC1834	TCMT133	Carbonic anhydrase I	Homo sapiens	Ki: 9060 (nM), Ref: 21402476
TCMC1834	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 8030 (nM), Ref: 21402476
TCMC770	TCMT588	D-amino-acid oxidase	Homo sapiens	Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755
TCMC1601	TCMT132	Butyrylcholinesterase	Homo sapiens	IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1601	TCMT131	Acetylcholinesterase	Homo sapiens	Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1343	TCMT134	Carbonic anhydrase II	Homo sapiens	Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385
TCMC1343	TCMT136	Carbonic anhydrase XII	Homo sapiens	Ki: 7800 (nM), Ref: 18579385
TCMC1343	TCMT143	Carbonic anhydrase III	Homo sapiens	Ki: 8200 (nM), Ref: 18579385