Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2330 (nM), Ref: 22245047 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 3630 (nM), Ref: 22245047 |
|
TCMT107 | Glutamate receptor ionotropic kainate 2 | Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
|
TCMT108 | Glutamate receptor ionotropic, AMPA 1 | Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
|
TCMT109 | Glutamate receptor ionotropic, AMPA 2 | Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
|
TCMT110 | Glutamate receptor ionotropic, AMPA 4 | Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
|
TCMT111 | Glutamate receptor ionotropic kainate 5 | Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
|
TCMT660 | Metabotropic glutamate receptor 8 | Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
|
TCMT653 | Metabotropic glutamate receptor 1 | Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT654 | Metabotropic glutamate receptor 5 | Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT657 | Metabotropic glutamate receptor 4 | Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT655 | Metabotropic glutamate receptor 2 | Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT664 | Excitatory amino acid transporter 3 | Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
|
TCMT656 | Metabotropic glutamate receptor 3 | Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 410 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 6300 (nM), Ref: 26688270 |
|
TCMT689 | Protein-glutamine gamma-glutamyltransferase | Homo sapiens |
IC50: 8000 (nM), Ref: 21215619 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 4400 (nM), Ref: 15634016 |
|
TCMT241 | Neuronal acetylcholine receptor protein alpha-7 subunit | Homo sapiens |
Ki: 7200 (nM), Ref: 15686879 Ki: 6300 (nM), Ref: 15908213 Ki: 630 (nM), Ref: 16171993 Ki: 10000 (nM), Ref: 17722904 Ki: 1000 (nM), Ref: 19331415 Ki: 1023.29 (nM), Ref: 20828128 Ki: 1000 (nM), Ref: 21920761 Ki: 1000 (nM), Ref: 22243960 Ki: 3000 (nM), Ref: 22793665 Ki: 3000 (nM), Ref: 23126648 Ki: 3800 (nM), Ref: 23561269 IC50: 7600 (nM), Ref: 23561269 Ki: 3000 (nM), Ref: 23692872 |
|
TCMT552 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens |
IC50: 45 (nM), Ref: 11312774 |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 64 (nM), Ref: 22819942 IC50: 64 (nM), Ref: 23146282 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 150 (nM), Ref: 22819942 |
|
TCMT336 | Indoleamine 2,3-dioxygenase | Homo sapiens |
IC50: 53.7 (nM), Ref: 24099220 IC50: 7150 (nM), Ref: 24099220 Ki: 4810 (nM), Ref: 24099220 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270 |
|
TCMT186 | Monoamine oxidase B | Homo sapiens |
Ki: 3000 (nM), Ref: 16137882 Ki: 3000 (nM), Ref: 19342233 IC50: 7943.28 (nM), Ref: 20934874 Ki: 5340 (nM), Ref: 21134756 Ki: 3000 (nM), Ref: 21778064 Ki: 2000 (nM), Ref: 24140951 |
|
TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 8380 (nM), Ref: 21134756 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 5900 (nM), Ref: 21561086 |
|
TCMT605 | Endothelin receptor ET-A | Homo sapiens |
Ki: 18 (nM), Ref: 10.1016/0960-894X(95)00019-P |
|
TCMT118 | Maltase-glucoamylase | Homo sapiens |
IC50: 40 (nM), Ref: 15771446 |
|
TCMT18 | Lysosomal alpha-glucosidase | Homo sapiens |
IC50: 1000 (nM), Ref: 18595718 IC50: 60 (nM), Ref: 18595718 IC50: 1500 (nM), Ref: 19853441 |
|
TCMT907 | Farnesyl diphosphate synthase | Homo sapiens |
IC50: 452.9 (nM), Ref: 18327899 Ki: 82.2 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18327899 Ki: 0.36 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18434151 IC50: 300 (nM), Ref: 20801032 IC50: 11 (nM), Ref: 22390415 IC50: 860 (nM), Ref: 22390415 IC50: 11 (nM), Ref: 22884353 IC50: 10 (nM), Ref: 21780776 IC50: 5.2 (nM), Ref: 23998921 IC50: 11 (nM), Ref: 23998921 IC50: 6 (nM), Ref: 24911527 IC50: 11 (nM), Ref: 25630225 IC50: 6 (nM), Ref: 25935643 IC50: 0.36 (nM), Ref: 25815158 IC50: 82 (nM), Ref: 25815158 |
|
TCMT588 | D-amino-acid oxidase | Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |