Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
Ki: 2.5 (nM), Ref: 11327599 Ki: 6.4 (nM), Ref: 21596562 |
|
TCMT152 | Protein kinase C beta | Homo sapiens |
Ki: 1.8 (nM), Ref: 11327599 |
|
TCMT153 | Protein kinase C gamma | Homo sapiens |
Ki: 4.9 (nM), Ref: 11327599 |
|
TCMT154 | Protein kinase C delta | Homo sapiens |
Ki: 0.8 (nM), Ref: 11327599 |
|
TCMT155 | Protein kinase C epsilon | Homo sapiens |
Ki: 0.45 (nM), Ref: 11327599 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT193 | Nuclear factor NF-kappa-B p65 subunit | Homo sapiens |
IC50: 250 (nM), Ref: 21513293 |
|
TCMT194 | Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens |
IC50: 80 (nM), Ref: 25529738 IC50: 11 (nM), Ref: 26481152 IC50: 8.1 (nM), Ref: 26481152 IC50: 9 (nM), Ref: 27448772 |
|
TCMT80 | MAP kinase ERK2 | Homo sapiens |
IC50: 6800 (nM), Ref: 25529738 |
|
TCMT195 | Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens |
IC50: 80 (nM), Ref: 25529738 |
|
TCMT196 | Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens |
IC50: 1300 (nM), Ref: 25529738 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 1800 (nM), Ref: 14592472 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
Ki: 0.208 (nM), Ref: 17004725 IC50: 800 (nM), Ref: 17270435 IC50: 3900 (nM), Ref: 26099993 |
|
TCMT566 | Nitric oxide synthase, inducible | Homo sapiens |
IC50: 6000 (nM), Ref: 18077363 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4300 (nM), Ref: 18249473 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 8500 (nM), Ref: 19128977 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2410 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 380 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4970 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9460 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 9940 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 9300 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4050 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 3480 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 6850 (nM), Ref: 20674354 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
Ki: 10000 (nM), Ref: 21237663 |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 7410 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5 IC50: 199.63 (nM), Ref: 23199480 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 8600 (nM), Ref: 23245570 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 4501 (nM), Ref: 23800686 |
|
TCMT570 | Aminopeptidase N | Homo sapiens |
IC50: 10000 (nM), Ref: 23860593 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3900 (nM), Ref: 24920381 IC50: 500 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 8100 (nM), Ref: 24920381 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 600 (nM), Ref: 24920381 IC50: 1200 (nM), Ref: 24920381 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
IC50: 1200 (nM), Ref: 24920381 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5300 (nM), Ref: 25088549 |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 25730130 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9140 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9010 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8200 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7550 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6340 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8580 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3190 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 4150 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT23 | Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | IC50: 407 (nM), Ref: |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 8390 (nM), Ref: 26696252 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2540 (nM), Ref: 26696252 |
|
TCMT203 | Glucose-6-phosphate 1-dehydrogenase | Homo sapiens |
Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561 |
|
TCMT292 | Muscarinic acetylcholine receptor M1 | Homo sapiens |
Ki: 14 (nM), Ref: 10891110 IC50: 115 (nM), Ref: 11597415 |
|
TCMT293 | Muscarinic acetylcholine receptor M2 | Homo sapiens |
Ki: 40 (nM), Ref: 10891110 Ki: 40 (nM), Ref: 9622546 Ki: 2454.71 (nM), Ref: 18182302 |
|
TCMT551 | Muscarinic acetylcholine receptor M4 | Homo sapiens |
Ki: 2400 (nM), Ref: 10891110 Ki: 26 (nM), Ref: 10891110 Ki: 2400 (nM), Ref: 9622546 |
|
TCMT571 | Adenosine A2b receptor | Homo sapiens |
Ki: 8200 (nM), Ref: 15084123 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 680 (nM), Ref: 15084123 |
|
TCMT230 | Estradiol 17-beta-dehydrogenase 3 | Homo sapiens |
IC50: 758 (nM), Ref: 11086723 IC50: 758 (nM), Ref: 16078844 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 20 (nM), Ref: 8035427 Ki: 35 (nM), Ref: 26469743 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens | IC50: 4703 (nM), Ref: |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 325 (nM), Ref: |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 26701186 |
|
TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 710 (nM), Ref: 26819666 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 600 (nM), Ref: 6827528 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 10000 (nM), Ref: 14552748 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 3.9 (nM), Ref: 15456242 IC50: 2.7 (nM), Ref: 16309907 IC50: 4.571 (nM), Ref: 22746350 IC50: 4.17 (nM), Ref: 25646649 IC50: 4.27 (nM), Ref: 25646649 |
|
TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 14 (nM), Ref: 17149875 |
|
TCMT725 | Voltage-gated L-type calcium channel alpha-1C subunit | Homo sapiens |
IC50: 34 (nM), Ref: 22761000 IC50: 38.4 (nM), Ref: 22761000 |
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT230 | Estradiol 17-beta-dehydrogenase 3 | Homo sapiens |
IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844 |
|
TCMT194 | Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens |
IC50: 1300 (nM), Ref: 26481152 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2500 (nM), Ref: 14592472 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT637 | NAD-dependent deacetylase sirtuin 3 | Homo sapiens |
IC50: 6200 (nM), Ref: 25275824 |
|
TCMT638 | NAD-dependent deacetylase sirtuin 2 | Homo sapiens |
IC50: 6300 (nM), Ref: 25549554 IC50: 1200 (nM), Ref: 26696402 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 8500 (nM), Ref: 23869482 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
|
TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
|
TCMT974 | G-protein coupled estrogen receptor 1 | Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |