Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 2000 (nM), Ref: 22696418 |
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TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
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TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 4880 (nM), Ref: 15658857 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
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TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
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TCMT45 | Beta amyloid A4 protein | Homo sapiens |
Ki: 0.208 (nM), Ref: 17004725 IC50: 800 (nM), Ref: 17270435 IC50: 3900 (nM), Ref: 26099993 |
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TCMT566 | Nitric oxide synthase, inducible | Homo sapiens |
IC50: 6000 (nM), Ref: 18077363 |
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TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4300 (nM), Ref: 18249473 |
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TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 8500 (nM), Ref: 19128977 |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2410 (nM), Ref: 20674354 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 380 (nM), Ref: 20674354 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4970 (nM), Ref: 20674354 |
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TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9460 (nM), Ref: 20674354 |
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TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 9940 (nM), Ref: 20674354 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 9300 (nM), Ref: 20674354 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4050 (nM), Ref: 20674354 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 3480 (nM), Ref: 20674354 |
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TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 6850 (nM), Ref: 20674354 |
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TCMT44 | Glyoxalase I | Homo sapiens |
Ki: 10000 (nM), Ref: 21237663 |
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TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 7410 (nM), Ref: |
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TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5 IC50: 199.63 (nM), Ref: 23199480 |
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TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 8600 (nM), Ref: 23245570 |
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TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 4501 (nM), Ref: 23800686 |
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TCMT570 | Aminopeptidase N | Homo sapiens |
IC50: 10000 (nM), Ref: 23860593 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3900 (nM), Ref: 24920381 IC50: 500 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 |
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TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 8100 (nM), Ref: 24920381 |
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TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 600 (nM), Ref: 24920381 IC50: 1200 (nM), Ref: 24920381 |
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TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
IC50: 1200 (nM), Ref: 24920381 |
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TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5300 (nM), Ref: 25088549 |
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TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 25730130 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3200 (nM), Ref: 24920381 |
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TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 8390 (nM), Ref: 26696252 |
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TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2540 (nM), Ref: 26696252 |
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TCMT203 | Glucose-6-phosphate 1-dehydrogenase | Homo sapiens |
Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7370 (nM), Ref: 22892213 |
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TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 5270 (nM), Ref: 22892213 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4140 (nM), Ref: 22892213 |
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TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H |
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TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 26701186 |
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TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 710 (nM), Ref: 26819666 |
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TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1118 (nM), Ref: 20696580 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 95 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 20 (nM), Ref: 20696580 |
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TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
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TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
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TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
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TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
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TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
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TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
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TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
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TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
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TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
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TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
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TCMT320 | Matrix metalloproteinase 3 | Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
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TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
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TCMT322 | Matrix metalloproteinase 13 | Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
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TCMT422 | CaM kinase II beta | Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
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TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
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TCMT784 | Vasopressin V2 receptor | Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
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TCMT785 | Interleukin-8 receptor A | Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
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TCMT786 | C-C chemokine receptor type 4 | Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
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TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
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TCMT601 | Thrombin | Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
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TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
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TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
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TCMT791 | Protein kinase N1 | Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
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TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
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TCMT462 | Serine/threonine-protein kinase NEK6 | Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
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TCMT445 | Serine/threonine-protein kinase NEK2 | Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
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TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
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TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
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TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
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TCMT388 | Tyrosine-protein kinase receptor UFO | Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
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TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
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TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
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TCMT402 | ALK tyrosine kinase receptor | Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
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TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
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TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
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TCMT793 | Liver glycogen phosphorylase | Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
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TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
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TCMT217 | Cytochrome P450 2C8 | Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
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TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT230 | Estradiol 17-beta-dehydrogenase 3 | Homo sapiens |
IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844 |
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TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
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TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
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TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
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TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
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TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
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TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
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TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
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TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
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TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
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TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
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TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 6200 (nM), Ref: 22222157 |
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TCMT614 | Egl nine homolog 1 | Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
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TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
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TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
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TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
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TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
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TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
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TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
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TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
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TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 5900 (nM), Ref: 21561086 |
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TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 7700 (nM), Ref: 18258440 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 3370 (nM), Ref: 20696580 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1249 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 79 (nM), Ref: 20696580 |
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TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 8200 (nM), Ref: 21641214 |
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TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 3610 (nM), Ref: 22658537 |
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TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 5620 (nM), Ref: 22658537 |
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TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 980 (nM), Ref: 22658537 |
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TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 830 (nM), Ref: 23411073 |
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TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272 |
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TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272 |
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TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272 |
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TCMT223 | Aldose reductase | Homo sapiens |
IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1600 (nM), Ref: 24368208 |
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TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 6400 (nM), Ref: 24878198 |
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TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677 |
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TCMT100 | Transthyretin | Homo sapiens |
IC50: 7000 (nM), Ref: 26214366 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3691.6 (nM), Ref: 26498393 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.7 (nM), Ref: 26498393 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 60.3 (nM), Ref: 26498393 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 293 (nM), Ref: 26498393 |
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TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 9200 (nM), Ref: 26529431 |
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TCMT241 | Neuronal acetylcholine receptor protein alpha-7 subunit | Homo sapiens |
Ki: 7943.28 (nM), Ref: 22243960 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
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TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
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TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
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TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
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TCMT962 | Autotaxin | Homo sapiens |
Ki: 1890 (nM), Ref: 24387347 IC50: 1310 (nM), Ref: 16513348 |
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TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens | IC50: 257 (nM), Ref: |
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TCMT191 | Signal transducer and activator of transcription 3 | Homo sapiens |
IC50: 6000 (nM), Ref: 19128055 |
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TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 600 (nM), Ref: 22206869 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens | IC50: 5200 (nM), Ref: IC50: 800 (nM), Ref: |
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TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
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TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
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TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
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TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
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TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
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TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
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TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
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TCMT974 | G-protein coupled estrogen receptor 1 | Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |
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TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
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TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
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TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
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TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
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TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
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TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
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TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
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TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
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TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
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TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 2437 (nM), Ref: 20696580 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 140 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 29 (nM), Ref: 20696580 |
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 840 (nM), Ref: 16248836 Ki: 2500 (nM), Ref: 16248836 |
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TCMT154 | Protein kinase C delta | Homo sapiens |
Ki: 9.7 (nM), Ref: 23582444 |