Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT193 | Nuclear factor NF-kappa-B p65 subunit | Homo sapiens |
IC50: 250 (nM), Ref: 21513293 |
|
TCMT194 | Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens |
IC50: 80 (nM), Ref: 25529738 IC50: 11 (nM), Ref: 26481152 IC50: 8.1 (nM), Ref: 26481152 IC50: 9 (nM), Ref: 27448772 |
|
TCMT80 | MAP kinase ERK2 | Homo sapiens |
IC50: 6800 (nM), Ref: 25529738 |
|
TCMT195 | Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens |
IC50: 80 (nM), Ref: 25529738 |
|
TCMT196 | Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens |
IC50: 1300 (nM), Ref: 25529738 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
Ki: 0.208 (nM), Ref: 17004725 IC50: 800 (nM), Ref: 17270435 IC50: 3900 (nM), Ref: 26099993 |
|
TCMT566 | Nitric oxide synthase, inducible | Homo sapiens |
IC50: 6000 (nM), Ref: 18077363 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4300 (nM), Ref: 18249473 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 8500 (nM), Ref: 19128977 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2410 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 380 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4970 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9460 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 9940 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 9300 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4050 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 3480 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 6850 (nM), Ref: 20674354 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
Ki: 10000 (nM), Ref: 21237663 |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 7410 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5 IC50: 199.63 (nM), Ref: 23199480 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 8600 (nM), Ref: 23245570 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 4501 (nM), Ref: 23800686 |
|
TCMT570 | Aminopeptidase N | Homo sapiens |
IC50: 10000 (nM), Ref: 23860593 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3900 (nM), Ref: 24920381 IC50: 500 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 8100 (nM), Ref: 24920381 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 600 (nM), Ref: 24920381 IC50: 1200 (nM), Ref: 24920381 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
IC50: 1200 (nM), Ref: 24920381 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5300 (nM), Ref: 25088549 |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 25730130 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
Ki: 6800 (nM), Ref: 22752007 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 8390 (nM), Ref: 26696252 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2540 (nM), Ref: 26696252 |
|
TCMT230 | Estradiol 17-beta-dehydrogenase 3 | Homo sapiens |
IC50: 758 (nM), Ref: 11086723 IC50: 758 (nM), Ref: 16078844 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 20 (nM), Ref: 8035427 Ki: 35 (nM), Ref: 26469743 |
|
TCMT599 | Ubiquitin-conjugating enzyme E2 N | Homo sapiens | IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref: |
|
TCMT678 | Inhibitor of apoptosis protein 3 | Homo sapiens |
IC50: 4100 (nM), Ref: 15115387 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1700 (nM), Ref: 25765759 IC50: 60 (nM), Ref: 25765759 IC50: 800 (nM), Ref: 25765759 IC50: 60 (nM), Ref: 25765759 IC50: 3500 (nM), Ref: 25765759 |
|
TCMT679 | Macrophage-expressed gene 1 protein | Homo sapiens |
IC50: 210 (nM), Ref: 25765759 IC50: 210 (nM), Ref: 25765759 |
|
TCMT680 | Histone acetyltransferase PCAF | Homo sapiens |
IC50: 7200 (nM), Ref: 26701186 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 26701186 |
|
TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 710 (nM), Ref: 26819666 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 600 (nM), Ref: 6827528 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 10000 (nM), Ref: 14552748 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 3.9 (nM), Ref: 15456242 IC50: 2.7 (nM), Ref: 16309907 IC50: 4.571 (nM), Ref: 22746350 IC50: 4.17 (nM), Ref: 25646649 IC50: 4.27 (nM), Ref: 25646649 |
|
TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 14 (nM), Ref: 17149875 |
|
TCMT725 | Voltage-gated L-type calcium channel alpha-1C subunit | Homo sapiens |
IC50: 34 (nM), Ref: 22761000 IC50: 38.4 (nM), Ref: 22761000 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 10000 (nM), Ref: 14552748 IC50: 5620 (nM), Ref: 23033255 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 8290 (nM), Ref: 8917655 |
|
TCMT778 | Voltage-gated potassium channel subunit Kv1.5 | Homo sapiens |
IC50: 6100 (nM), Ref: 19004630 |
|
TCMT780 | Voltage-gated L-type calcium channel alpha-1D subunit | Homo sapiens |
IC50: 1350 (nM), Ref: 24754640 |
|
TCMT725 | Voltage-gated L-type calcium channel alpha-1C subunit | Homo sapiens |
IC50: 22 (nM), Ref: 22761000 IC50: 55 (nM), Ref: 22761000 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 2300 (nM), Ref: 23033255 |
|
TCMT31 | Cytochrome P450 2C19 | Homo sapiens |
IC50: 5420 (nM), Ref: 23033255 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4080 (nM), Ref: 23033255 |
|
TCMT220 | Cytochrome P450 2J2 | Homo sapiens |
IC50: 3060 (nM), Ref: 23033255 |
|
TCMT407 | Myosin light chain kinase, smooth muscle | Homo sapiens |
IC50: 2020 (nM), Ref: 26385444 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 3900 (nM), Ref: 10.1016/S0960-894X(97)00194-7 |
|
TCMT194 | Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens |
IC50: 1300 (nM), Ref: 26481152 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens |
IC50: 2200 (nM), Ref: 18778098 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 3430 (nM), Ref: 19097799 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 4960 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 3656 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 79.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 44.3 (nM), Ref: 26498393 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.77 (nM), Ref: 16250647 |
|
TCMT675 | Beta-1 adrenergic receptor | Homo sapiens |
IC50: 600 (nM), Ref: 18983139 Ki: 430 (nM), Ref: 18983139 IC50: 1740 (nM), Ref: 18588282 IC50: 1640 (nM), Ref: 20875743 Ki: 170 (nM), Ref: 21726069 Ki: 150 (nM), Ref: 23466604 IC50: 260 (nM), Ref: 23466604 IC50: 210 (nM), Ref: 26988801 |
|
TCMT907 | Farnesyl diphosphate synthase | Homo sapiens |
IC50: 452.9 (nM), Ref: 18327899 Ki: 82.2 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18327899 Ki: 0.36 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18434151 IC50: 300 (nM), Ref: 20801032 IC50: 11 (nM), Ref: 22390415 IC50: 860 (nM), Ref: 22390415 IC50: 11 (nM), Ref: 22884353 IC50: 10 (nM), Ref: 21780776 IC50: 5.2 (nM), Ref: 23998921 IC50: 11 (nM), Ref: 23998921 IC50: 6 (nM), Ref: 24911527 IC50: 11 (nM), Ref: 25630225 IC50: 6 (nM), Ref: 25935643 IC50: 0.36 (nM), Ref: 25815158 IC50: 82 (nM), Ref: 25815158 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 515 (nM), Ref: 12270171 IC50: 14.4 (nM), Ref: 16480284 IC50: 3.1 (nM), Ref: 16480284 IC50: 33 (nM), Ref: 16516473 IC50: 54 (nM), Ref: 16516473 IC50: 23 (nM), Ref: 16806916 IC50: 80 (nM), Ref: 16806916 IC50: 5.4 (nM), Ref: 17416531 IC50: 2753 (nM), Ref: 17416531 IC50: 22 (nM), Ref: 19170633 IC50: 33 (nM), Ref: 20304535 IC50: 70 (nM), Ref: 21353546 IC50: 1 (nM), Ref: 22101132 IC50: 1080 (nM), Ref: 22698782 IC50: 72 (nM), Ref: 22818848 IC50: 33 (nM), Ref: 23611691 IC50: 33 (nM), Ref: 23142066 IC50: 0.1 (nM), Ref: 23668441 IC50: 0.1 (nM), Ref: 23792318 IC50: 62 (nM), Ref: 23930994 IC50: 23 (nM), Ref: 23973168 IC50: 498 (nM), Ref: 23988354 IC50: 39.9 (nM), Ref: 23988354 IC50: 0.6 (nM), Ref: 23988354 IC50: 4000 (nM), Ref: 24900594 IC50: 1100 (nM), Ref: 24094432 IC50: 1 (nM), Ref: 24411123 IC50: 25 (nM), Ref: 24411123 IC50: 4000 (nM), Ref: 10.1039/C3MD00118K IC50: 70 (nM), Ref: 10.1039/C0MD00183J IC50: 1 (nM), Ref: 24588073 IC50: 0.1 (nM), Ref: 24607591 IC50: 20 (nM), Ref: 24731281 IC50: 0.45 (nM), Ref: 25468044 IC50: 0.45 (nM), Ref: 25462282 IC50: 76 (nM), Ref: 25409491 IC50: 380 (nM), Ref: 25768701 IC50: 1 (nM), Ref: 26275028 IC50: 26 (nM), Ref: 26256032 IC50: 22 (nM), Ref: 26318056 IC50: 1.3 (nM), Ref: 26706113 IC50: 22 (nM), Ref: 26451770 IC50: 13 (nM), Ref: 10.1039/C5MD00208G IC50: 15.5 (nM), Ref: 26829280 IC50: 11.8 (nM), Ref: 26879314 IC50: 2.6 (nM), Ref: 27234887 IC50: 0.509 (nM), Ref: 27288180 IC50: 127 (nM), Ref: 27288180 IC50: 76 (nM), Ref: 27387355 IC50: 0.585 (nM), Ref: 27132165 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 1604 (nM), Ref: 12270171 IC50: 343 (nM), Ref: 16480284 IC50: 599 (nM), Ref: 16480284 IC50: 280 (nM), Ref: 24411123 IC50: 1000 (nM), Ref: 25409491 IC50: 1830 (nM), Ref: 27132165 |
|
TCMT747 | ATP-binding cassette sub-family G member 2 | Homo sapiens |
IC50: 3190 (nM), Ref: 24184213 |