TCM Putative Target References: TCMFx1294


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1803
TCMT337 Exportin-1 Homo sapiens IC50: 1600 (nM), Ref: 20493693
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC2021
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 6200 (nM), Ref: 25907369
Ki: 6800 (nM), Ref: 25907369
TCMC1985
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6367.7 (nM), Ref: 26498393
TCMC1985
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 67.3 (nM), Ref: 26498393
TCMC1985
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.9 (nM), Ref: 26498393
TCMC1985
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 43.5 (nM), Ref: 26498393
TCMC680
TCMT666 Transitional endoplasmic reticulum ATPase Homo sapiens IC50: 8984 (nM), Ref:
TCMC680
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 1634.07 (nM), Ref:
TCMC680
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7400 (nM), Ref: 25907369
Ki: 7800 (nM), Ref: 25907369
TCMC1396
TCMT689 Protein-glutamine gamma-glutamyltransferase Homo sapiens IC50: 8000 (nM), Ref: 21215619
TCMC2242
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7710 (nM), Ref: 22892213
TCMC2242
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6270 (nM), Ref: 22892213
TCMC2242
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 3150 (nM), Ref: 22892213
TCMC2242
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC2242
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 740 (nM), Ref: 22892213
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1986
TCMT223 Aldose reductase Homo sapiens IC50: 150 (nM), Ref: 18165015
IC50: 2000 (nM), Ref: 22261024
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC961
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 9600 (nM), Ref: 25907369
TCMC846
TCMT207 Beta-secretase 1 Homo sapiens Ki: 6200 (nM), Ref: 22222157
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC804
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 2000 (nM), Ref: 21561086
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC341
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 19231207
TCMC2121
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 5400 (nM), Ref: 25907369
Ki: 4500 (nM), Ref: 25907369
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC273
TCMT332 Amine oxidase, copper containing Homo sapiens IC50: 4100 (nM), Ref: 23664164
TCMC2057
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens Ki: 3000 (nM), Ref: 24195447
IC50: 4600 (nM), Ref: 10.6019/CHEMBL1201861
TCMC2058
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens Ki: 8900 (nM), Ref: 24195447
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1803
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 2 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1986
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 75.2 (ug/ml), Ref: 9461665
TCMC1324
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 41.8 (ug/ml), Ref: 20116898
TCMC2233
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.85 (ug/ml), Ref: 20116898
TCMC1866
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1802
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 2 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC1514
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 2.1 (ug/ml), Ref: 19515569
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2315
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 64 (ug/ml), Ref: 12608857
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC1803
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 23369537
TCMC1985
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 84.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 26112067
TCMC1986
TCMT1442 Leishmania donovani Leishmania donovani IC50: 17.7 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2481
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 12.5 (ug/ml), Ref: 17027268
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC1515
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC804
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC687
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 5 (ug/ml), Ref: 9428161
MIC: 0.03 (ug/ml), Ref: 19524330
MIC: 64 (ug/ml), Ref: 19237648
MIC: 64 (ug/ml), Ref: 19237648
MIC: 0.0005 (ug/ml), Ref: 20805400
MIC: 0.25 (ug/ml), Ref: 21855181
TCMC687
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 5 (ug/ml), Ref: 9428161
MIC: 0.03 (ug/ml), Ref: 19524330
MIC: 64 (ug/ml), Ref: 19237648
MIC: 64 (ug/ml), Ref: 19237648
MIC: 0.0005 (ug/ml), Ref: 20805400
MIC: 0.25 (ug/ml), Ref: 21855181
TCMC687
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 0.16 (ug/ml), Ref: 19828313
MIC: 0.0005 (ug/ml), Ref: 20805400
MIC: 0.2 (ug/ml), Ref: 21855181
MIC: 0.3 (ug/ml), Ref: 27072906
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001