TCM Putative Target References: TCMF7259


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1372
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2330 (nM), Ref: 22245047
TCMC1372
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3630 (nM), Ref: 22245047
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC244
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 7900 (nM), Ref: 15916432
TCMC244
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 8300 (nM), Ref: 15658857
IC50: 8298.51 (nM), Ref: 19110342
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC1851
TCMT560 Coagulation factor X Homo sapiens IC50: 170 (nM), Ref: 9834152
Ki: 570 (nM), Ref: 9834152
TCMC1851
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3760 (nM), Ref: 24835197
Ki: 5130 (nM), Ref: 24835197
TCMC1851
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 2350 (nM), Ref: 26395057
Ki: 2600 (nM), Ref: 26395057
TCMC795
TCMT223 Aldose reductase Homo sapiens IC50: 8000 (nM), Ref: 24341381
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC450
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 5157.65 (nM), Ref:
TCMC231
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 4800 (nM), Ref: 20806783
TCMC891
TCMT598 DNA topoisomerase I Homo sapiens IC50: 50 (nM), Ref: 1324981
IC50: 100 (nM), Ref: 1324981
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC837
TCMT690 Histone deacetylase 3 Homo sapiens IC50: 9000 (nM), Ref: 21874153
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC963
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 500 (nM), Ref: 15357993
Ki: 500 (nM), Ref: 15454240
Ki: 500 (nM), Ref: 15501038
Ki: 500 (nM), Ref: 21208801
Ki: 500 (nM), Ref: 26525863
Ki: 500 (nM), Ref: 26853167
Ki: 500 (nM), Ref: 27283786
TCMC963
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4000 (nM), Ref: 15501038
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1399
TCMT223 Aldose reductase Homo sapiens IC50: 320 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1361
TCMT39 Phosphodiesterase 5A Homo sapiens IC50: 160 (nM), Ref: 18778098
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1886
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 670 (nM), Ref: 26498394
TCMC1886
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 770 (nM), Ref: 26498394
TCMC1886
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 620 (nM), Ref: 26498394
TCMC1886
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8470 (nM), Ref: 26498394
TCMC1886
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 720 (nM), Ref: 26498394
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC829
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 8100 (nM), Ref: 20493686
TCMC829
TCMT236 Estrogen receptor beta Homo sapiens IC50: 1800 (nM), Ref: 20493686
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1168
TCMT117 Kappa opioid receptor Homo sapiens Ki: 2515 (nM), Ref: 18166466
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1105
TCMT752 Casein kinase II alpha Homo sapiens IC50: 2000 (nM), Ref: 19414254
TCMC1105
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2500 (nM), Ref: 27173800
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC1008
TCMT186 Monoamine oxidase B Homo sapiens IC50: 8.61 (nM), Ref: 21405131
IC50: 8709.64 (nM), Ref: 24169316
TCMC392
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 2400 (nM), Ref: 15658857
IC50: 2398.83 (nM), Ref: 19110342
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC1551
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1900 (nM), Ref: 16248836
Ki: 1900 (nM), Ref: 16248836
Ki: 800 (nM), Ref: 16248836
Ki: 250 (nM), Ref: 22696418
TCMC1551
TCMT131 Acetylcholinesterase Homo sapiens IC50: 760 (nM), Ref: 23746477
TCMC1551
TCMT268 Cytochrome P450 2A13 Homo sapiens Ki: 40 (nM), Ref: 22696418
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1742
TCMT637 NAD-dependent deacetylase sirtuin 3 Homo sapiens IC50: 6200 (nM), Ref: 25275824
TCMC1742
TCMT638 NAD-dependent deacetylase sirtuin 2 Homo sapiens IC50: 6300 (nM), Ref: 25549554
IC50: 1200 (nM), Ref: 26696402
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC1961
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 600 (nM), Ref: 16248836
TCMC1961
TCMT131 Acetylcholinesterase Homo sapiens IC50: 6480 (nM), Ref: 23746477
TCMC1403
TCMT223 Aldose reductase Homo sapiens IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1851
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28 (ug/ml), Ref: 9461665
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC1399
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1136 Neuraminidase Influenza A virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1121 Sialidase Clostridium perfringens IC50: 11.28 (ug/ml), Ref: 21123068
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC2233
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.85 (ug/ml), Ref: 20116898
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC2288
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 55 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC2123
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1793
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1251 Candida albicans Candida albicans MIC: 12.5 (ug/ml), Ref: 9392889
TCMC1793
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 61.5 (ug/ml), Ref: 20218656
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC2332
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 13 (ug/ml), Ref: 16392829
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2351
TCMT1190 Plasmodium falciparum (isolate FcB1 / Columbia) Plasmodium falciparum FcB1/Columbia IC50: 16.7 (ug/ml), Ref: 21985060
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC795
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.6 (ug/ml), Ref: 15844943
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC2415
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14 (ug/ml), Ref: 16392829
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1399
TCMT1286 Bacillus cereus Bacillus cereus MIC: 62.5 (ug/ml), Ref: 18951808
TCMC1399
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 18951808
MIC: 31.25 (ug/ml), Ref: 22169259
MIC: 62.5 (ug/ml), Ref: 22169259
MIC: 15.6 (ug/ml), Ref: 25137491
TCMC2482
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC887
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 10395496
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC2519
TCMT1283 Human enterovirus 71 Human enterovirus 71 IC50: 10 (ug/ml), Ref: 22342145
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2548
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 20 (ug/ml), Ref: 16392829
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC1117
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 10425115
TCMC1117
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.89 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2578
TCMT1251 Candida albicans Candida albicans IC50: 82.98 (ug/ml), Ref: 25686593
TCMC2581
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC2593
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 17601740
TCMC1168
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 9392889
MIC: 2.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 9392889
TCMC1168
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
MIC: 25 (ug/ml), Ref: 10217726
TCMC1168
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 9392889
TCMC1168
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.2 (ug/ml), Ref: 20218656
TCMC1105
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1105
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 23534483
TCMC1105
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1 (ug/ml), Ref: 23534483
TCMC1105
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 23534483
MIC: 4 (ug/ml), Ref: 23534483
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC348
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 62 (ug/ml), Ref: 25813159
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1033
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2661
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 11 (ug/ml), Ref: 19904996
TCMC1551
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 20832915
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2681
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 16 (ug/ml), Ref: 19904996
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC2714
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 1.4 (ug/ml), Ref: 22280816
TCMC2714
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25.3 (ug/ml), Ref: 22280816
TCMC1961
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 6.25 (ug/ml), Ref: 20832915
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1403
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC1117
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 17.56 (nM), Ref: 17263522