Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 7585.78 (nM), Ref: 23574272 IC50: 7500 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 870.96 (nM), Ref: 23574272 IC50: 870 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 645.65 (nM), Ref: 23574272 IC50: 630 (nM), Ref: 23574272 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2000 (nM), Ref: 24368208 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 810 (nM), Ref: 20100662 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 7000 (nM), Ref: 22940448 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 800 (nM), Ref: 16759088 IC50: 3450 (nM), Ref: 16759088 IC50: 7138 (nM), Ref: 20851614 IC50: 7100 (nM), Ref: 21376605 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 201 (nM), Ref: 16759088 IC50: 6430 (nM), Ref: 16759088 IC50: 750 (nM), Ref: 20851614 IC50: 750 (nM), Ref: 21376605 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 3780 (nM), Ref: 16759088 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 5930 (nM), Ref: 19846303 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 630 (nM), Ref: 21561086 |
|
TCMT231 | Beta-glucosidase | Homo sapiens |
Ki: 200 (nM), Ref: 10.1039/C3MD00033H |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
Ki: 78 (nM), Ref: 26125082 |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4000 (nM), Ref: 21030469 IC50: 3600 (nM), Ref: 21030469 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 9550 (nM), Ref: |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 400 (nM), Ref: 11678652 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 4630 (nM), Ref: 15270556 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5405 (nM), Ref: |
|
TCMT560 | Coagulation factor X | Homo sapiens |
IC50: 170 (nM), Ref: 9834152 Ki: 570 (nM), Ref: 9834152 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3760 (nM), Ref: 24835197 Ki: 5130 (nM), Ref: 24835197 |
|
TCMT240 | Salivary alpha-amylase | Homo sapiens |
IC50: 2350 (nM), Ref: 26395057 Ki: 2600 (nM), Ref: 26395057 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 57 (nM), Ref: 17149865 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 68 (nM), Ref: 17149865 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8000 (nM), Ref: 24341381 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9140 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9010 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8200 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7550 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6340 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8580 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3190 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 4150 (nM), Ref: 20185318 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 4500 (nM), Ref: 14592472 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
Ki: 7000 (nM), Ref: 16248836 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 452.6 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 515 (nM), Ref: 26498393 |
|
TCMT23 | Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | IC50: 407 (nM), Ref: |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 168 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 5591.2 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 423.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4.9 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8900 (nM), Ref: 19911821 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 48 (nM), Ref: 19911821 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9100 (nM), Ref: 19911821 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3300 (nM), Ref: 19911821 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 2000 (nM), Ref: 19911821 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 5200 (nM), Ref: 19911821 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9400 (nM), Ref: 19911821 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 6800 (nM), Ref: 19911821 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 5600 (nM), Ref: 19911821 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
|
TCMT599 | Ubiquitin-conjugating enzyme E2 N | Homo sapiens | IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2100 (nM), Ref: 18042388 IC50: 340 (nM), Ref: 18778944 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens | IC50: 4703 (nM), Ref: |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 325 (nM), Ref: |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 26701186 |
|
TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 710 (nM), Ref: 26819666 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
Ki: 785 (nM), Ref: 15634023 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref: |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006 |
|
TCMT329 | Quinone reductase 2 | Homo sapiens |
IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2210 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2770 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 9090 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4470 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4750 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4640 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8070 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4350 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 810 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 950 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4090 (nM), Ref: 20674354 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 830 (nM), Ref: 20674354 |
|
TCMT729 | PI3-kinase p110-alpha subunit | Homo sapiens |
IC50: 250 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT730 | PI3-kinase p110-beta subunit | Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 35 (nM), Ref: 16000002 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 290 (nM), Ref: 22257892 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 4200 (nM), Ref: 19481465 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 5610 (nM), Ref: 24900561 Ki: 5.61 (nM), Ref: 27078864 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 6460 (nM), Ref: 24900561 Ki: 6.46 (nM), Ref: 27078864 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 1610 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 320 (nM), Ref: 22261024 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 2400 (nM), Ref: 26704263 Ki: 2500 (nM), Ref: 26704263 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2 (nM), Ref: 20413308 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 9510 (nM), Ref: 19028102 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
|
TCMT753 | Mothers against decapentaplegic homolog 3 | Homo sapiens | IC50: 142 (nM), Ref: |
|
TCMT721 | Heat shock 70 kDa protein 1 | Homo sapiens | IC50: 760 (nM), Ref: |
|
TCMT189 | Dual specificity protein phosphatase 3 | Homo sapiens | IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
|
TCMT354 | Serine/threonine-protein kinase Aurora-A | Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
|
TCMT626 | Serine/threonine-protein kinase B-raf | Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
|
TCMT418 | Ephrin type-B receptor 4 | Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
|
TCMT457 | Vascular endothelial growth factor receptor 3 | Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
|
TCMT377 | Insulin receptor | Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
|
TCMT536 | Platelet-derived growth factor receptor beta | Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT755 | Serine/threonine-protein kinase PLK4 | Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
|
TCMT502 | Tyrosine-protein kinase TIE-2 | Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
|
TCMT756 | Mitogen-activated protein kinase kinase kinase 8 | Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 5000 (nM), Ref: 22257892 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1118 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 95 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 20 (nM), Ref: 20696580 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
|
TCMT506 | Protein tyrosine kinase 2 beta | Homo sapiens | IC50: 2324 (nM), Ref: |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 8576921 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
Ki: 6900 (nM), Ref: 19879672 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 40 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 568.3 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 24.5 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 41.8 (nM), Ref: 26498393 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 5.9 (nM), Ref: 19744859 IC50: 12.29 (nM), Ref: 22748706 Ki: 6.23 (nM), Ref: 22748706 Ki: 3.4 (nM), Ref: 23332346 Ki: 12.29 (nM), Ref: 25308766 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 974 (nM), Ref: 19744859 IC50: 105.41 (nM), Ref: 22748706 Ki: 56.17 (nM), Ref: 22748706 Ki: 11 (nM), Ref: 23332346 Ki: 105.41 (nM), Ref: 25308766 IC50: 4380 (nM), Ref: 25308766 |
|
TCMT648 | Dopamine D4 receptor | Homo sapiens |
Ki: 3748 (nM), Ref: 19744859 |
|
TCMT649 | Dopamine D5 receptor | Homo sapiens |
Ki: 4.4 (nM), Ref: 19744859 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 104.58 (nM), Ref: 23199480 |
|
TCMT651 | Dopamine D3 receptor | Homo sapiens |
Ki: 90.02 (nM), Ref: 25308766 Ki: 30 (nM), Ref: 27032890 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3100 (nM), Ref: 24835197 Ki: 6840 (nM), Ref: 24835197 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
|
TCMT320 | Matrix metalloproteinase 3 | Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
|
TCMT322 | Matrix metalloproteinase 13 | Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
|
TCMT422 | CaM kinase II beta | Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
|
TCMT784 | Vasopressin V2 receptor | Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
|
TCMT785 | Interleukin-8 receptor A | Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
|
TCMT786 | C-C chemokine receptor type 4 | Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
|
TCMT601 | Thrombin | Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
|
TCMT791 | Protein kinase N1 | Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
|
TCMT462 | Serine/threonine-protein kinase NEK6 | Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
|
TCMT445 | Serine/threonine-protein kinase NEK2 | Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
|
TCMT388 | Tyrosine-protein kinase receptor UFO | Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
|
TCMT402 | ALK tyrosine kinase receptor | Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
|
TCMT793 | Liver glycogen phosphorylase | Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
|
TCMT217 | Cytochrome P450 2C8 | Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 100 (nM), Ref: 11678652 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 10 (nM), Ref: 19564108 IC50: 18.6 (nM), Ref: 22148241 IC50: 6 (nM), Ref: 22360639 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 1 (nM), Ref: 19564108 IC50: 0.7 (nM), Ref: 22148241 IC50: 0.4 (nM), Ref: 22360639 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3000 (nM), Ref: 26841168 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9910 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 20185318 Ki: 9900 (nM), Ref: 22245047 Ki: 9900 (nM), Ref: 26073005 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4200 (nM), Ref: 18579385 Ki: 4200 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8900 (nM), Ref: 18579385 Ki: 8900 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 9300 (nM), Ref: 26704263 Ki: 9600 (nM), Ref: 26704263 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens |
IC50: 1290 (nM), Ref: 18778098 |
|
TCMT646 | Serotonin 5a (5-HT5a) receptor | Homo sapiens |
Ki: 126 (nM), Ref: 12825922 IC50: 180 (nM), Ref: 18983139 Ki: 110 (nM), Ref: 18983139 IC50: 184 (nM), Ref: 18588282 Ki: 170 (nM), Ref: 21726069 IC50: 280 (nM), Ref: 23582449 Ki: 82 (nM), Ref: 23466604 IC50: 160 (nM), Ref: 23466604 IC50: 180 (nM), Ref: 26988801 |
|
TCMT315 | Serotonin 6 (5-HT6) receptor | Homo sapiens |
Ki: 65 (nM), Ref: 12825922 Ki: 100 (nM), Ref: 15357994 IC50: 200 (nM), Ref: 18983139 Ki: 93 (nM), Ref: 18983139 IC50: 262 (nM), Ref: 18588282 IC50: 27.5 (nM), Ref: 20170099 Ki: 84 (nM), Ref: 21726069 Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8 IC50: 180 (nM), Ref: 23582449 Ki: 50 (nM), Ref: 23466604 IC50: 100 (nM), Ref: 23466604 Ki: 33 (nM), Ref: 24805037 Ki: 33 (nM), Ref: 25557493 IC50: 120 (nM), Ref: 26988801 Ki: 100 (nM), Ref: 26996373 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 8.1 (nM), Ref: 12825922 IC50: 0.61 (nM), Ref: 18983139 Ki: 0.22 (nM), Ref: 18983139 IC50: 2.55 (nM), Ref: 12713409 IC50: 1.5 (nM), Ref: 18588282 Ki: 0.13 (nM), Ref: 21726069 IC50: 0.49 (nM), Ref: 23582449 Ki: 0.11 (nM), Ref: 23466604 IC50: 0.29 (nM), Ref: 23466604 Ki: 1.4 (nM), Ref: 24763360 Ki: 0.8 (nM), Ref: 24805037 Ki: 0.8 (nM), Ref: 25557493 IC50: 0.25 (nM), Ref: 26988801 |
|
TCMT37 | Serotonin 2a (5-HT2a) receptor | Homo sapiens |
Ki: 14 (nM), Ref: 15081042 Ki: 8.2 (nM), Ref: 16392816 Ki: 14 (nM), Ref: 16257207 Ki: 120 (nM), Ref: 18468904 Ki: 160 (nM), Ref: 18468904 Ki: 130 (nM), Ref: 18468904 Ki: 150 (nM), Ref: 18468904 Ki: 320 (nM), Ref: 11975483 Ki: 690 (nM), Ref: 17067154 Ki: 323.59 (nM), Ref: 23301527 Ki: 320 (nM), Ref: 23301527 |
|
TCMT313 | Serotonin 2b (5-HT2b) receptor | Homo sapiens |
Ki: 12 (nM), Ref: 15081042 Ki: 13 (nM), Ref: 12954071 Ki: 13 (nM), Ref: 16392816 Ki: 12 (nM), Ref: 16257207 Ki: 13.49 (nM), Ref: 24582985 |
|
TCMT314 | Serotonin 2c (5-HT2c) receptor | Homo sapiens |
Ki: 6.9 (nM), Ref: 15081042 Ki: 8.3 (nM), Ref: 12954071 Ki: 8.3 (nM), Ref: 16392816 Ki: 6.9 (nM), Ref: 16257207 Ki: 130 (nM), Ref: 11975483 Ki: 20 (nM), Ref: 17067154 Ki: 79.43 (nM), Ref: 23301527 Ki: 79 (nM), Ref: 23301527 |
|
TCMT815 | Serotonin 1d (5-HT1d) receptor | Homo sapiens |
Ki: 5.5 (nM), Ref: 8071931 Ki: 0.5 (nM), Ref: 18507369 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 2.5 (nM), Ref: 7658447 IC50: 1.2 (nM), Ref: 12954071 Ki: 1.259 (nM), Ref: 18433113 Ki: 10000 (nM), Ref: 18433113 Ki: 0.62 (nM), Ref: 22748706 Ki: 0.9 (nM), Ref: 23332346 Ki: 9.5 (nM), Ref: 24161678 Ki: 2.08 (nM), Ref: 25128671 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 79 (nM), Ref: 16250647 |
|
TCMT816 | Serotonin 1b (5-HT1b) receptor | Homo sapiens |
Ki: 1.1 (nM), Ref: 18507369 IC50: 29 (nM), Ref: 18983139 Ki: 18 (nM), Ref: 18983139 Ki: 14 (nM), Ref: 21726069 IC50: 12 (nM), Ref: 23582449 Ki: 4 (nM), Ref: 23466604 IC50: 6.5 (nM), Ref: 23466604 |
|
TCMT817 | Serotonin 4 (5-HT4) receptor | Homo sapiens |
Ki: 1049 (nM), Ref: 19334715 Ki: 500 (nM), Ref: 17067154 Ki: 29.51 (nM), Ref: 19223092 Ki: 109.65 (nM), Ref: 19223092 |
|
TCMT645 | Serotonin 1e (5-HT1e) receptor | Homo sapiens |
Ki: 10.72 (nM), Ref: 24365159 Ki: 11 (nM), Ref: 24365159 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 9900 (nM), Ref: 26841168 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 11.78 (nM), Ref: 18242087 IC50: 13 (nM), Ref: 18653260 IC50: 778 (nM), Ref: 20851614 IC50: 778 (nM), Ref: 21376605 IC50: 8.6 (nM), Ref: 21873057 IC50: 29.1 (nM), Ref: 23747808 IC50: 29.1 (nM), Ref: 25590374 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 257 (nM), Ref: 20851614 IC50: 257 (nM), Ref: 21376605 IC50: 1.22 (nM), Ref: 23747808 IC50: 1.2 (nM), Ref: 25590374 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4900 (nM), Ref: 21561086 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref: |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 7300 (nM), Ref: 21030469 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 718.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.2 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 56.4 (nM), Ref: 26498393 |
|
TCMT614 | Egl nine homolog 1 | Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
Ki: 600 (nM), Ref: 21739938 |
|
TCMT81 | Arachidonate 12-lipoxygenase | Homo sapiens |
Ki: 1600 (nM), Ref: 21739938 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 8700 (nM), Ref: |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3100 (nM), Ref: 20674354 Ki: 3100 (nM), Ref: 21282059 Ki: 3400 (nM), Ref: 22137345 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9300 (nM), Ref: 22137345 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 720 (nM), Ref: 22261024 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 8000 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 2000 (nM), Ref: 21561086 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 560 (nM), Ref: 22261024 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3500 (nM), Ref: 18798681 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 5320 (nM), Ref: 10.1007/s00044-010-9529-5 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 7410 (nM), Ref: 21669522 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 540 (nM), Ref: 21669522 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 520 (nM), Ref: 21669522 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 3000 (nM), Ref: 22261024 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 3430 (nM), Ref: 19097799 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 4960 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 3656 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 79.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 44.3 (nM), Ref: 26498393 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 9000 (nM), Ref: 23791077 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 1440 (nM), Ref: 24900561 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 24900561 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 6000 (nM), Ref: 14592472 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 5610 (nM), Ref: 26900660 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 800 (nM), Ref: 10.1039/C3MD00317E Ki: 2100 (nM), Ref: 10.1039/C0MD00242A |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
Ki: 160 (nM), Ref: 10.1039/C0MD00242A |
|
TCMT508 | Tyrosine-protein kinase SYK | Homo sapiens |
IC50: 10000 (nM), Ref: 23917087 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT317 | Melatonin receptor 1B | Homo sapiens |
Ki: 0.3 (nM), Ref: 15203165 Ki: 0.41 (nM), Ref: 12646022 Ki: 0.29 (nM), Ref: 10.1016/S0960-894X(97)00444-7 Ki: 0.195 (nM), Ref: 12213063 Ki: 0.31 (nM), Ref: 11960497 Ki: 0.7 (nM), Ref: 15713384 Ki: 0.7 (nM), Ref: 15380218 Ki: 0.2818 (nM), Ref: 15293992 Ki: 0.2818 (nM), Ref: 15943478 Ki: 0.35 (nM), Ref: 16759094 Ki: 0.257 (nM), Ref: 17149869 Ki: 0.3 (nM), Ref: 17481904 Ki: 0.3548 (nM), Ref: 17346859 Ki: 0.3388 (nM), Ref: 17459711 Ki: 0.2399 (nM), Ref: 18052314 IC50: 0.53 (nM), Ref: 18372181 Ki: 0.41 (nM), Ref: 18778943 Ki: 0.955 (nM), Ref: 19193160 Ki: 0.741 (nM), Ref: 18657980 Ki: 0.429 (nM), Ref: 20227878 Ki: 0.6166 (nM), Ref: 20674373 Ki: 0.34 (nM), Ref: 21420861 IC50: 0.53 (nM), Ref: 21377769 Ki: 0.21 (nM), Ref: 21473625 Ki: 0.35 (nM), Ref: 21392858 Ki: 0.21 (nM), Ref: 21568291 Ki: 0.3388 (nM), Ref: 21775151 Ki: 0.34 (nM), Ref: 21764185 Ki: 0.5 (nM), Ref: 23265885 Ki: 0.429 (nM), Ref: 23228808 Ki: 0.955 (nM), Ref: 10.1039/C1MD00149C Ki: 0.41 (nM), Ref: 25232966 Ki: 0.15 (nM), Ref: 26023814 Ki: 0.15 (nM), Ref: 26367450 Ki: 0.955 (nM), Ref: 10.1039/C5MD00190K Ki: 0.52 (nM), Ref: 26820449 Ki: 0.34 (nM), Ref: 26785296 |
|
TCMT316 | Melatonin receptor 1A | Homo sapiens |
Ki: 0.14 (nM), Ref: 12646022 Ki: 0.2 (nM), Ref: 10.1016/S0960-894X(97)00444-7 Ki: 0.0823 (nM), Ref: 12213063 Ki: 0.12 (nM), Ref: 11960497 Ki: 0.3 (nM), Ref: 15713384 Ki: 0.3 (nM), Ref: 15380218 Ki: 0.2884 (nM), Ref: 15293992 Ki: 0.2884 (nM), Ref: 15943478 Ki: 0.39 (nM), Ref: 16759094 Ki: 0.3236 (nM), Ref: 17149869 Ki: 0.2 (nM), Ref: 17481904 Ki: 0.389 (nM), Ref: 17346859 Ki: 0.263 (nM), Ref: 17459711 Ki: 0.1413 (nM), Ref: 18052314 IC50: 0.2 (nM), Ref: 18372181 IC50: 0.18 (nM), Ref: 18983139 Ki: 0.11 (nM), Ref: 18983139 Ki: 0.14 (nM), Ref: 18778943 Ki: 0.4571 (nM), Ref: 19193160 Ki: 0.525 (nM), Ref: 18657980 Ki: 0.296 (nM), Ref: 20227878 Ki: 0.3311 (nM), Ref: 20674373 Ki: 0.25 (nM), Ref: 21420861 IC50: 0.2 (nM), Ref: 21377769 Ki: 0.24 (nM), Ref: 21473625 Ki: 0.22 (nM), Ref: 21392858 Ki: 0.24 (nM), Ref: 21568291 Ki: 0.37 (nM), Ref: 21726069 Ki: 0.263 (nM), Ref: 21775151 Ki: 0.25 (nM), Ref: 21764185 Ki: 0.2 (nM), Ref: 23265885 Ki: 0.296 (nM), Ref: 23228808 IC50: 0.53 (nM), Ref: 23582449 Ki: 0.35 (nM), Ref: 23466604 IC50: 0.44 (nM), Ref: 23466604 Ki: 0.4571 (nM), Ref: 10.1039/C1MD00149C Ki: 0.14 (nM), Ref: 25232966 Ki: 0.091 (nM), Ref: 26023814 Ki: 0.091 (nM), Ref: 26367450 Ki: 0.4571 (nM), Ref: 10.1039/C5MD00190K Ki: 0.23 (nM), Ref: 26820449 Ki: 0.25 (nM), Ref: 26785296 IC50: 0.11 (nM), Ref: 26988801 |
|
TCMT329 | Quinone reductase 2 | Homo sapiens |
IC50: 64.6 (nM), Ref: 21377769 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 154 (nM), Ref: 26841168 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref: |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 10 (nM), Ref: 17482813 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 395 (nM), Ref: 17482813 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 2210 (nM), Ref: 18533708 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 340 (nM), Ref: 20853847 |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 7720 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2400 (nM), Ref: 14592472 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 850 (nM), Ref: 15689157 IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3600 (nM), Ref: 17489632 IC50: 3100 (nM), Ref: 18798681 IC50: 3600 (nM), Ref: 19008110 IC50: 3600 (nM), Ref: 17125223 IC50: 3800 (nM), Ref: 19846295 IC50: 3900 (nM), Ref: 19632832 IC50: 3600 (nM), Ref: 19836230 IC50: 3100 (nM), Ref: 21555221 IC50: 3600 (nM), Ref: 21571537 IC50: 3100 (nM), Ref: 22940448 IC50: 2300 (nM), Ref: 21453996 Ki: 3400 (nM), Ref: 21453996 IC50: 3600 (nM), Ref: 23022281 IC50: 3080 (nM), Ref: 23141910 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2750 (nM), Ref: 23387824 IC50: 4120 (nM), Ref: 24224843 IC50: 4000 (nM), Ref: 24953600 IC50: 3500 (nM), Ref: 25559759 IC50: 3400 (nM), Ref: 25907369 Ki: 6400 (nM), Ref: 25907369 IC50: 5200 (nM), Ref: 26841168 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 1900 (nM), Ref: 20100662 |
|
TCMT102 | Low molecular weight phosphotyrosine protein phosphatase | Homo sapiens |
IC50: 7200 (nM), Ref: 21453996 |
|
TCMT103 | Receptor-type tyrosine-protein phosphatase F (LAR) | Homo sapiens |
IC50: 3800 (nM), Ref: 21453996 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 21561086 Ki: 3700 (nM), Ref: 21561086 Ki: 2100 (nM), Ref: 21561086 Ki: 2800 (nM), Ref: 21561086 Ki: 2000 (nM), Ref: 21561086 IC50: 4000 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 2400 (nM), Ref: 23387824 |
|
TCMT150 | Nuclear receptor ROR-gamma | Homo sapiens |
IC50: 680 (nM), Ref: 10.1039/C3MD00005B IC50: 130 (nM), Ref: 24704616 IC50: 1060 (nM), Ref: 24704616 IC50: 9410 (nM), Ref: 24704616 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 177 (nM), Ref: 26841168 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 400 (nM), Ref: 26841168 |
|
TCMT632 | Purine nucleoside phosphorylase | Homo sapiens |
Ki: 5000 (nM), Ref: 31484 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |
|
TCMT588 | D-amino-acid oxidase | Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7800 (nM), Ref: 18579385 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8200 (nM), Ref: 18579385 |