Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 3100 (nM), Ref: 26035635 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 7585.78 (nM), Ref: 23574272 IC50: 7500 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 870.96 (nM), Ref: 23574272 IC50: 870 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 645.65 (nM), Ref: 23574272 IC50: 630 (nM), Ref: 23574272 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2000 (nM), Ref: 24368208 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 800 (nM), Ref: 16759088 IC50: 3450 (nM), Ref: 16759088 IC50: 7138 (nM), Ref: 20851614 IC50: 7100 (nM), Ref: 21376605 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 201 (nM), Ref: 16759088 IC50: 6430 (nM), Ref: 16759088 IC50: 750 (nM), Ref: 20851614 IC50: 750 (nM), Ref: 21376605 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 3780 (nM), Ref: 16759088 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 340 (nM), Ref: 19072652 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 6000 (nM), Ref: 15689157 IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 2600 (nM), Ref: 15267241 IC50: 1 (nM), Ref: 20413308 IC50: 800 (nM), Ref: 10.1039/C3MD00166K IC50: 500 (nM), Ref: 26301554 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8500 (nM), Ref: 18165015 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
IC50: 670 (nM), Ref: 19097799 Ki: 110 (nM), Ref: 19097799 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 153 (nM), Ref: 20696580 IC50: 1290 (nM), Ref: 23600958 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 84 (nM), Ref: 20696580 IC50: 54 (nM), Ref: 20832301 IC50: 570 (nM), Ref: 23600958 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 24 (nM), Ref: 20696580 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 5225 (nM), Ref: 20832301 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 5490 (nM), Ref: 22487176 Ki: 5420 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 4380 (nM), Ref: 22487176 Ki: 4310 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 2650 (nM), Ref: 22487176 Ki: 2710 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8960 (nM), Ref: 22487176 Ki: 9070 (nM), Ref: 22487176 Ki: 34.7 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 537.75 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 171.41 (nM), Ref: 26498393 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 2000 (nM), Ref: 22696418 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT231 | Beta-glucosidase | Homo sapiens |
Ki: 200 (nM), Ref: 10.1039/C3MD00033H |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 4630 (nM), Ref: 26425784 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2700 (nM), Ref: 22261024 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 5210 (nM), Ref: 22487176 Ki: 5100 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9300 (nM), Ref: 22487176 Ki: 9200 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5540 (nM), Ref: 22487176 Ki: 5630 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 6590 (nM), Ref: 22487176 Ki: 6650 (nM), Ref: 22487176 |
|
TCMT337 | Exportin-1 | Homo sapiens |
IC50: 1600 (nM), Ref: 20493693 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
|
TCMT293 | Muscarinic acetylcholine receptor M2 | Homo sapiens |
Ki: 158.49 (nM), Ref: 18077164 |
|
TCMT291 | Muscarinic acetylcholine receptor M3 | Homo sapiens |
Ki: 7079.46 (nM), Ref: 18077164 |
|
TCMT551 | Muscarinic acetylcholine receptor M4 | Homo sapiens |
Ki: 8511.38 (nM), Ref: 18077164 |
|
TCMT290 | Muscarinic acetylcholine receptor M5 | Homo sapiens |
Ki: 9772.37 (nM), Ref: 18077164 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 400 (nM), Ref: 11678652 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 4630 (nM), Ref: 15270556 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5405 (nM), Ref: |
|
TCMT241 | Neuronal acetylcholine receptor protein alpha-7 subunit | Homo sapiens |
Ki: 7943.28 (nM), Ref: 21920761 |
|
TCMT561 | 5'-nucleotidase | Homo sapiens |
IC50: 8200 (nM), Ref: 24215819 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 57 (nM), Ref: 17149865 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 68 (nM), Ref: 17149865 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8000 (nM), Ref: 24341381 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
Ki: 0.208 (nM), Ref: 17004725 IC50: 800 (nM), Ref: 17270435 IC50: 3900 (nM), Ref: 26099993 |
|
TCMT566 | Nitric oxide synthase, inducible | Homo sapiens |
IC50: 6000 (nM), Ref: 18077363 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 4300 (nM), Ref: 18249473 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 8500 (nM), Ref: 19128977 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2410 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 380 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4970 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9460 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 9940 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 9300 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4050 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 3480 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 6850 (nM), Ref: 20674354 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
Ki: 10000 (nM), Ref: 21237663 |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 7410 (nM), Ref: |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5 IC50: 199.63 (nM), Ref: 23199480 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 8600 (nM), Ref: 23245570 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 4501 (nM), Ref: 23800686 |
|
TCMT570 | Aminopeptidase N | Homo sapiens |
IC50: 10000 (nM), Ref: 23860593 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3900 (nM), Ref: 24920381 IC50: 500 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 IC50: 600 (nM), Ref: 24920381 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 8100 (nM), Ref: 24920381 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 600 (nM), Ref: 24920381 IC50: 1200 (nM), Ref: 24920381 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
IC50: 1200 (nM), Ref: 24920381 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5300 (nM), Ref: 25088549 |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 25730130 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9140 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9010 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8200 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7550 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6340 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8580 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3190 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 4150 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT588 | D-amino-acid oxidase | Homo sapiens |
IC50: 2000 (nM), Ref: 23683589 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 9150 (nM), Ref: 26386819 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 4000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT308 | Oxoeicosanoid receptor 1 | Homo sapiens |
IC50: 2000 (nM), Ref: 24351031 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
Ki: 7000 (nM), Ref: 16248836 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 1720 (nM), Ref: 8576921 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 452.6 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 515 (nM), Ref: 26498393 |
|
TCMT23 | Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | IC50: 407 (nM), Ref: |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 3200 (nM), Ref: 24920381 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2100 (nM), Ref: 17994701 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 8390 (nM), Ref: 26696252 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2540 (nM), Ref: 26696252 |
|
TCMT240 | Salivary alpha-amylase | Homo sapiens |
IC50: 9640 (nM), Ref: 18507367 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 6610 (nM), Ref: |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 600 (nM), Ref: 26602279 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 168 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 5591.2 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 423.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4.9 (nM), Ref: 26498393 |
|
TCMT636 | DNA polymerase alpha subunit | Homo sapiens |
Ki: 830 (nM), Ref: 1705574 |
|
TCMT17 | DNA polymerase beta | Homo sapiens |
Ki: 390 (nM), Ref: 1705574 |
|
TCMT571 | Adenosine A2b receptor | Homo sapiens |
Ki: 8200 (nM), Ref: 15084123 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 680 (nM), Ref: 15084123 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8900 (nM), Ref: 19911821 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 48 (nM), Ref: 19911821 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9100 (nM), Ref: 19911821 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3300 (nM), Ref: 19911821 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 2000 (nM), Ref: 19911821 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 5200 (nM), Ref: 19911821 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9400 (nM), Ref: 19911821 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 6800 (nM), Ref: 19911821 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 5600 (nM), Ref: 19911821 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
|
TCMT599 | Ubiquitin-conjugating enzyme E2 N | Homo sapiens | IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref: |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 630 (nM), Ref: 19231207 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 14.98 (nM), Ref: 23199480 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2100 (nM), Ref: 18042388 IC50: 340 (nM), Ref: 18778944 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens | IC50: 4703 (nM), Ref: |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 325 (nM), Ref: |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 7710 (nM), Ref: 22892213 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6270 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 3150 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 740 (nM), Ref: 22892213 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 441.49 (nM), Ref: |
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT301 | Prostaglandin E synthase | Homo sapiens |
IC50: 220 (nM), Ref: 26588603 IC50: 200 (nM), Ref: 10.1039/C5MD00278H |
|
TCMT565 | Histone acetyltransferase p300 | Homo sapiens |
IC50: 6500 (nM), Ref: 26701186 |
|
TCMT208 | Monoamine oxidase A | Homo sapiens |
Ki: 710 (nM), Ref: 26819666 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3100 (nM), Ref: 27190601 IC50: 1500 (nM), Ref: 27190601 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 35 (nM), Ref: 16000002 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085 |
|
TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 6300 (nM), Ref: 21641214 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 4200 (nM), Ref: 19481465 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 5610 (nM), Ref: 24900561 Ki: 5.61 (nM), Ref: 27078864 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 6460 (nM), Ref: 24900561 Ki: 6.46 (nM), Ref: 27078864 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18778944 |
|
TCMT737 | DNA dC->dU-editing enzyme APOBEC-3G | Homo sapiens | IC50: 2390 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 2120 (nM), Ref: 24900447 |
|
TCMT558 | DNA topoisomerase II alpha | Homo sapiens |
IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1690 (nM), Ref: 23411073 |
|
TCMT2 | Microtubule-associated protein tau | Homo sapiens |
IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3000 (nM), Ref: 25086914 |
|
TCMT740 | PI3-kinase p110-gamma subunit | Homo sapiens |
IC50: 4720 (nM), Ref: 25050878 |
|
TCMT13 | DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens |
IC50: 320 (nM), Ref: 25280182 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 320 (nM), Ref: 22261024 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 2400 (nM), Ref: 26704263 Ki: 2500 (nM), Ref: 26704263 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2 (nM), Ref: 20413308 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 150 (nM), Ref: 18165015 IC50: 2000 (nM), Ref: 22261024 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
|
TCMT753 | Mothers against decapentaplegic homolog 3 | Homo sapiens | IC50: 142 (nM), Ref: |
|
TCMT721 | Heat shock 70 kDa protein 1 | Homo sapiens | IC50: 760 (nM), Ref: |
|
TCMT189 | Dual specificity protein phosphatase 3 | Homo sapiens | IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
|
TCMT354 | Serine/threonine-protein kinase Aurora-A | Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
|
TCMT626 | Serine/threonine-protein kinase B-raf | Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
|
TCMT418 | Ephrin type-B receptor 4 | Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
|
TCMT457 | Vascular endothelial growth factor receptor 3 | Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
|
TCMT377 | Insulin receptor | Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
|
TCMT536 | Platelet-derived growth factor receptor beta | Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT755 | Serine/threonine-protein kinase PLK4 | Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
|
TCMT502 | Tyrosine-protein kinase TIE-2 | Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
|
TCMT756 | Mitogen-activated protein kinase kinase kinase 8 | Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens |
IC50: 160 (nM), Ref: 18778098 |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1118 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 95 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 20 (nM), Ref: 20696580 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
|
TCMT506 | Protein tyrosine kinase 2 beta | Homo sapiens | IC50: 2324 (nM), Ref: |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 8576921 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
Ki: 6900 (nM), Ref: 19879672 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 40 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 568.3 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 24.5 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 41.8 (nM), Ref: 26498393 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
|
TCMT320 | Matrix metalloproteinase 3 | Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
|
TCMT322 | Matrix metalloproteinase 13 | Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
|
TCMT422 | CaM kinase II beta | Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1400 (nM), Ref: 20590092 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1110 (nM), Ref: 20590092 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 112 (nM), Ref: 20590092 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 1220 (nM), Ref: 20590092 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 1440 (nM), Ref: 20590092 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 1410 (nM), Ref: 20590092 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 1230 (nM), Ref: 20590092 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 1370 (nM), Ref: 20590092 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 1000 (nM), Ref: 20590092 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
|
TCMT784 | Vasopressin V2 receptor | Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
|
TCMT785 | Interleukin-8 receptor A | Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
|
TCMT786 | C-C chemokine receptor type 4 | Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
|
TCMT601 | Thrombin | Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
|
TCMT791 | Protein kinase N1 | Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
|
TCMT462 | Serine/threonine-protein kinase NEK6 | Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
|
TCMT445 | Serine/threonine-protein kinase NEK2 | Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
|
TCMT388 | Tyrosine-protein kinase receptor UFO | Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
|
TCMT402 | ALK tyrosine kinase receptor | Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
|
TCMT793 | Liver glycogen phosphorylase | Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
|
TCMT217 | Cytochrome P450 2C8 | Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 100 (nM), Ref: 11678652 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 10 (nM), Ref: 19564108 IC50: 18.6 (nM), Ref: 22148241 IC50: 6 (nM), Ref: 22360639 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 1 (nM), Ref: 19564108 IC50: 0.7 (nM), Ref: 22148241 IC50: 0.4 (nM), Ref: 22360639 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3000 (nM), Ref: 26841168 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 9300 (nM), Ref: 26704263 Ki: 9600 (nM), Ref: 26704263 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
|
TCMT278 | Solute carrier organic anion transporter family member 1B1 | Homo sapiens |
IC50: 1400 (nM), Ref: 22587986 IC50: 2200 (nM), Ref: 22587986 |
|
TCMT221 | Bile salt export pump | Homo sapiens |
IC50: 5300 (nM), Ref: 21965623 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT46 | Coagulation factor III | Homo sapiens |
IC50: 22.78 (nM), Ref: 23199480 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 231 (nM), Ref: 23332346 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT39 | Phosphodiesterase 5A | Homo sapiens |
IC50: 1290 (nM), Ref: 18778098 |
|
TCMT287 | Taste receptor type 2 member 31 | Homo sapiens |
IC50: 3600 (nM), Ref: 21650152 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 8100 (nM), Ref: 20493686 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 1800 (nM), Ref: 20493686 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 251 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 86 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 12 (nM), Ref: 20696580 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 9900 (nM), Ref: 26841168 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 11.78 (nM), Ref: 18242087 IC50: 13 (nM), Ref: 18653260 IC50: 778 (nM), Ref: 20851614 IC50: 778 (nM), Ref: 21376605 IC50: 8.6 (nM), Ref: 21873057 IC50: 29.1 (nM), Ref: 23747808 IC50: 29.1 (nM), Ref: 25590374 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 257 (nM), Ref: 20851614 IC50: 257 (nM), Ref: 21376605 IC50: 1.22 (nM), Ref: 23747808 IC50: 1.2 (nM), Ref: 25590374 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4900 (nM), Ref: 21561086 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref: |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 7300 (nM), Ref: 21030469 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 718.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.2 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 56.4 (nM), Ref: 26498393 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
Ki: 600 (nM), Ref: 21739938 |
|
TCMT81 | Arachidonate 12-lipoxygenase | Homo sapiens |
Ki: 1600 (nM), Ref: 21739938 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 8700 (nM), Ref: |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 509 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 88 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 9180 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 8360 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7510 (nM), Ref: 22892213 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 720 (nM), Ref: 22261024 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT232 | P-glycoprotein 1 | Homo sapiens |
IC50: 11.5 (nM), Ref: 23332369 IC50: 6.6 (nM), Ref: 23895532 |
|
TCMT801 | Tubulin beta-3 chain | Homo sapiens |
IC50: 5.2 (nM), Ref: 23332369 IC50: 5.7 (nM), Ref: 23895532 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 8000 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 560 (nM), Ref: 22261024 |
|
TCMT308 | Oxoeicosanoid receptor 1 | Homo sapiens |
IC50: 2000 (nM), Ref: 24351031 |
|
TCMT186 | Monoamine oxidase B | Homo sapiens |
IC50: 8.61 (nM), Ref: 21405131 IC50: 8709.64 (nM), Ref: 24169316 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 7700 (nM), Ref: 18258440 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 3370 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1249 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 79 (nM), Ref: 20696580 |
|
TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 8200 (nM), Ref: 21641214 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 3610 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 5620 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 980 (nM), Ref: 22658537 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 830 (nM), Ref: 23411073 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1600 (nM), Ref: 24368208 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 6400 (nM), Ref: 24878198 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677 |
|
TCMT100 | Transthyretin | Homo sapiens |
IC50: 7000 (nM), Ref: 26214366 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3691.6 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 60.3 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 293 (nM), Ref: 26498393 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 9200 (nM), Ref: 26529431 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 3000 (nM), Ref: 22261024 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 3430 (nM), Ref: 19097799 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 4960 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 3656 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 79.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 44.3 (nM), Ref: 26498393 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 1440 (nM), Ref: 24900561 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 24900561 |
|
TCMT683 | Macrophage migration inhibitory factor | Homo sapiens |
IC50: 2200 (nM), Ref: 25743213 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 9000 (nM), Ref: 27135370 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1480 (nM), Ref: 23411073 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1284 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 72.8 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 31.1 (nM), Ref: 26498393 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 5610 (nM), Ref: 26900660 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 610 (nM), Ref: 23062825 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 2786 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 511 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 102.1 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 454.1 (nM), Ref: 26498393 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 800 (nM), Ref: 22668600 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 490 (nM), Ref: 22668600 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 610 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 850 (nM), Ref: 22668600 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 710 (nM), Ref: 22668600 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 320 (nM), Ref: 22668600 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 900 (nM), Ref: 17994701 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 52 (nM), Ref: 20590092 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 44 (nM), Ref: 20590092 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 540 (nM), Ref: 20590092 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 740 (nM), Ref: 20590092 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 420 (nM), Ref: 20590092 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 380 (nM), Ref: 20590092 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 450 (nM), Ref: 20590092 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT637 | NAD-dependent deacetylase sirtuin 3 | Homo sapiens |
IC50: 6200 (nM), Ref: 25275824 |
|
TCMT638 | NAD-dependent deacetylase sirtuin 2 | Homo sapiens |
IC50: 6300 (nM), Ref: 25549554 IC50: 1200 (nM), Ref: 26696402 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 154 (nM), Ref: 26841168 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref: |
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TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 10 (nM), Ref: 17482813 |
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TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 395 (nM), Ref: 17482813 |
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TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 2210 (nM), Ref: 18533708 |
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TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 340 (nM), Ref: 20853847 |
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TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 7720 (nM), Ref: |
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TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: |
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TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: |
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TCMT962 | Autotaxin | Homo sapiens |
Ki: 1890 (nM), Ref: 24387347 IC50: 1310 (nM), Ref: 16513348 |
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TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens | IC50: 257 (nM), Ref: |
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TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 2020 (nM), Ref: 10879539 Ki: 1760 (nM), Ref: 16872140 |
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TCMT747 | ATP-binding cassette sub-family G member 2 | Homo sapiens |
IC50: 10000 (nM), Ref: 22822035 |
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TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
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TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
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TCMT191 | Signal transducer and activator of transcription 3 | Homo sapiens |
IC50: 6000 (nM), Ref: 19128055 |
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TCMT601 | Thrombin | Homo sapiens |
IC50: 250 (nM), Ref: 24610996 |
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TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 600 (nM), Ref: 22206869 |
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TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 4720 (nM), Ref: 12027740 |
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TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 4580 (nM), Ref: 20438092 |
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TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens | IC50: 5200 (nM), Ref: IC50: 800 (nM), Ref: |
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TCMT210 | Carboxylesterase 2 | Homo sapiens |
IC50: 8680 (nM), Ref: 15332848 |
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TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
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TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
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TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
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TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
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TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
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TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
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TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
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TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
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TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
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TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
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TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
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TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
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TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
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TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 850 (nM), Ref: 15689157 IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5 |
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TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
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TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 100 (nM), Ref: 26003344 |
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TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1090 (nM), Ref: 26003344 |
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TCMT159 | Tyrosinase | Homo sapiens |
IC50: 177 (nM), Ref: 26841168 |
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TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 400 (nM), Ref: 26841168 |
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 5150 (nM), Ref: 15658857 |
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TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 840 (nM), Ref: 16248836 Ki: 2500 (nM), Ref: 16248836 |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
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TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
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TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
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TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
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TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
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TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
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TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
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TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
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TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |
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TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9060 (nM), Ref: 21402476 |
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TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8030 (nM), Ref: 21402476 |
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TCMT588 | D-amino-acid oxidase | Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |
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TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
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TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |