Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867 |
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TCMT651 | Dopamine D3 receptor | Homo sapiens |
Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329 |
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TCMT635 | Dopamine transporter | Homo sapiens |
Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523 |
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TCMT634 | Norepinephrine transporter | Homo sapiens |
IC50: 6.63 (nM), Ref: 14592523 |
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TCMT648 | Dopamine D4 receptor | Homo sapiens |
Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965 |
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TCMT316 | Melatonin receptor 1A | Homo sapiens |
Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
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TCMT317 | Melatonin receptor 1B | Homo sapiens |
Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
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TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4470 (nM), Ref: 23134120 |
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TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
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TCMT290 | Muscarinic acetylcholine receptor M5 | Homo sapiens |
Ki: 0.14 (nM), Ref: 23707254 Ki: 0.3388 (nM), Ref: 24365159 Ki: 0.34 (nM), Ref: 24365159 Ki: 3.02 (nM), Ref: 25051097 |
Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
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TCMT1465 | Entamoeba histolytica | Entamoeba histolytica |
IC50: 25.16 (ug/ml), Ref: 10.1007/s00044-011-9767-1 IC50: 10.51 (ug/ml), Ref: 10.1007/s00044-011-9767-1 |
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TCMT1246 | Escherichia coli | Escherichia coli |
MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7 MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7 MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7 |
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TCMT1412 | Salmonella typhimurium | Salmonella enterica subsp. enterica serovar Typhimurium |
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7 |
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TCMT1249 | Dengue virus 2 | Dengue virus 2 |
IC50: 55 (ug/ml), Ref: 25564380 |
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TCMT1442 | Leishmania donovani | Leishmania donovani |
IC50: 0.6 (ug/ml), Ref: 10.1039/C5MD00481K |
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TCMT1438 | Plasmodium falciparum | Plasmodium falciparum |
IC50: 2 (nM), Ref: 19097788 |
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TCMT1178 | Actinomyces viscosus | Actinomyces viscosus |
MIC: 78 (ug/ml), Ref: 8904847 |
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TCMT1438 | Plasmodium falciparum | Plasmodium falciparum |
IC50: 14.8 (ug/ml), Ref: 15844943 |
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TCMT1108 | Integrase | Human immunodeficiency virus 1 |
IC50: 28.5 (ug/ml), Ref: 9461665 |
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TCMT1465 | Entamoeba histolytica | Entamoeba histolytica |
IC50: 22.6 (ug/ml), Ref: 10.1007/s00044-011-9767-1 |