Structure

Physi-Chem Properties

Molecular Weight:  679.42
Volume:  732.348
LogP:  7.853
LogD:  4.948
LogS:  -4.176
# Rotatable Bonds:  5
TPSA:  80.92
# H-Bond Aceptor:  6
# H-Bond Donor:  2
# Rings:  8
# Heavy Atoms:  6

MedChem Properties

QED Drug-Likeness Score:  0.146
Synthetic Accessibility Score:  5.839
Fsp3:  0.614
Lipinski Rule-of-5:  Rejected
Pfizer Rule:  Accepted
GSK Rule:  Rejected
BMS Rule:  0
Golden Triangle Rule:  Rejected
Chelating Alert:  0
PAINS Alert:  0

ADMET Properties (ADMETlab2.0)

ADMET: Absorption

Caco-2 Permeability:  -5.485
MDCK Permeability:  2.034136741713155e-05
Pgp-inhibitor:  1.0
Pgp-substrate:  0.954
Human Intestinal Absorption (HIA):  0.013
20% Bioavailability (F20%):  0.573
30% Bioavailability (F30%):  0.884

ADMET: Distribution

Blood-Brain-Barrier Penetration (BBB):  0.825
Plasma Protein Binding (PPB):  96.06407928466797%
Volume Distribution (VD):  2.569
Pgp-substrate:  7.00372838973999%

ADMET: Metabolism

CYP1A2-inhibitor:  0.039
CYP1A2-substrate:  0.893
CYP2C19-inhibitor:  0.363
CYP2C19-substrate:  0.852
CYP2C9-inhibitor:  0.694
CYP2C9-substrate:  0.344
CYP2D6-inhibitor:  0.798
CYP2D6-substrate:  0.147
CYP3A4-inhibitor:  0.962
CYP3A4-substrate:  0.923

ADMET: Excretion

Clearance (CL):  8.156
Half-life (T1/2):  0.008

ADMET: Toxicity

hERG Blockers:  0.841
Human Hepatotoxicity (H-HT):  0.509
Drug-inuced Liver Injury (DILI):  0.092
AMES Toxicity:  0.014
Rat Oral Acute Toxicity:  0.923
Maximum Recommended Daily Dose:  0.991
Skin Sensitization:  0.093
Carcinogencity:  0.925
Eye Corrosion:  0.003
Eye Irritation:  0.006
Respiratory Toxicity:  0.946

Download Data

Data Type Select
General Info & Identifiers & Properties  
Structure MOL file  
Source Organisms  
Biological Activities  
Similar NPs/Drugs  

  Natural Product: NPC469308

Natural Product ID:  NPC469308
Common Name*:   Sb-203580
IUPAC Name:   4-[4-(4-fluorophenyl)-2-(4-methylsulfinylphenyl)-1H-imidazol-5-yl]pyridine
Synonyms:   SB-203580
Standard InCHIKey:  CDMGBJANTYXAIV-UHFFFAOYSA-N
Standard InCHI:  InChI=1S/C21H16FN3OS/c1-27(26)18-8-4-16(5-9-18)21-24-19(14-2-6-17(22)7-3-14)20(25-21)15-10-12-23-13-11-15/h2-13H,1H3,(H,24,25)
SMILES:  Fc1ccc(cc1)c1[nH]c(nc1c1ccncc1)c1ccc(cc1)S(=O)C
Synthetic Gene Cluster:   n.a.
ChEMBL Identifier:   CHEMBL10
PubChem CID:   176155
Chemical Classification**:  
  • CHEMONTID:0000000 [Organic compounds]
    • [CHEMONTID:0000002] Organoheterocyclic compounds
      • [CHEMONTID:0000436] Azoles
        • [CHEMONTID:0000078] Imidazoles
          • [CHEMONTID:0002310] Substituted imidazoles
            • [CHEMONTID:0002327] Phenylimidazoles

*Note: the InCHIKey will be temporarily assigned as the "Common Name" if no IUPAC name or alternative short name is available.
**Note: the Chemical Classification was calculated by NPClassifier Version 1.5. Reference: PMID:34662515.

  Species Source

Organism ID Organism Name Taxonomy Level Family SuperKingdom Isolation Part Collection Location Collection Time Reference
NPO29834 Acanthopanax koreanum n.a. n.a. n.a. n.a. n.a. n.a. PMID[20621475]
NPO29834 Acanthopanax koreanum n.a. n.a. n.a. steamed leaves n.a. n.a. PMID[20932756]
NPO27826 Sinularia maxima Species Alcyoniidae Eukaryota n.a. n.a. n.a. PMID[23200246]
NPO33245 asterina batheri Species n.a. Eukaryota n.a. n.a. n.a. PMID[23395633]
NPO5842 Annulohypoxylon truncatum Species n.a. Eukaryota n.a. n.a. n.a. PMID[28009172]
NPO29834 Acanthopanax koreanum n.a. n.a. n.a. n.a. n.a. n.a. Database[HerDing]
NPO27826 Sinularia maxima Species Alcyoniidae Eukaryota n.a. n.a. n.a. Database[UNPD]
NPO5842 Annulohypoxylon truncatum Species n.a. Eukaryota n.a. n.a. n.a. Database[UNPD]

☑ Note for Reference:
In addition to directly collecting NP source organism data from primary literature (where reference will provided as NCBI PMID or DOI links), NPASS also integrated them from below databases:
UNPD: Universal Natural Products Database [PMID: 23638153].
StreptomeDB: a database of streptomycetes natural products [PMID: 33051671].
TM-MC: a database of medicinal materials and chemical compounds in Northeast Asian traditional medicine [PMID: 26156871].
TCM@Taiwan: a Traditional Chinese Medicine database [PMID: 21253603].
TCMID: a Traditional Chinese Medicine database [PMID: 29106634].
TCMSP: The traditional Chinese medicine systems pharmacology database and analysis platform [PMID: 24735618].
HerDing: a herb recommendation system to treat diseases using genes and chemicals [PMID: 26980517].
MetaboLights: a metabolomics database [PMID: 27010336].
FooDB: a database of constituents, chemistry and biology of food species [www.foodb.ca].

  NP Quantity Composition/Concentration

Organism ID NP ID Organism Material Preparation Organism Part NP Quantity (Standard) NP Quantity (Minimum) NP Quantity (Maximum) Quantity Unit Reference

☑ Note for Reference:
In addition to directly collecting NP quantitative data from primary literature (where reference will provided as NCBI PMID or DOI links), NPASS also integrated NP quantitative records for specific NP domains (e.g., NPS from foods or herbs) from domain-specific databases. These databases include:
DUKE: Dr. Duke's Phytochemical and Ethnobotanical Databases.
PHENOL EXPLORER: is the first comprehensive database on polyphenol content in foods [PMID: 24103452], its homepage can be accessed at here.
FooDB: a database of constituents, chemistry and biology of food species [www.foodb.ca].

  Biological Activity

Target ID Target Type Target Name Target Organism Activity Type Activity Relation Value Unit Reference
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 290.0 nM PMID[532298]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 72.0 nM PMID[532299]
NPT6452 Individual Protein MAP kinase p38 alpha Mus musculus Kd = 20.0 nM PMID[532301]
NPT6452 Individual Protein MAP kinase p38 alpha Mus musculus Tm = 46.6 degrees C PMID[532301]
NPT927 Cell Line PBMC Homo sapiens IC50 = 25.0 nM PMID[532303]
NPT927 Cell Line PBMC Homo sapiens IC50 = 48.0 nM PMID[532303]
NPT927 Cell Line PBMC Homo sapiens IC50 = 160.0 nM PMID[532303]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Inhibition = 55.0 % PMID[532303]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Inhibition = 54.0 % PMID[532303]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Inhibition = 22.0 % PMID[532303]
NPT30 Individual Protein Cyclooxygenase-1 Homo sapiens IC50 > 5000.0 nM PMID[532303]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens IC50 = 30000.0 nM PMID[532304]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 38.0 nM PMID[532305]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens IC50 = 330.0 nM PMID[532306]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 290.0 nM PMID[532306]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 1900.0 nM PMID[532306]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens IC50 = 3450.0 nM PMID[532306]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens IC50 = 96000.0 nM PMID[532306]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens Inhibition = 61.0 % PMID[532307]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens Inhibition = 75.0 % PMID[532307]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens Inhibition = 85.0 % PMID[532307]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Inhibition = 67.0 % PMID[532307]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Inhibition = 61.0 % PMID[532307]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 39.0 nM PMID[532308]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens IC50 = 78.0 nM PMID[532308]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Inhibition = 46.0 % PMID[532308]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens IC50 = 370.0 nM PMID[532308]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Inhibition = 50.0 % PMID[532308]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 280.0 nM PMID[532308]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 1920.0 nM PMID[532308]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 20.0 nM PMID[532309]
NPT3089 Cell Line SW1353 Homo sapiens IC50 = 50.0 nM PMID[532309]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 20.0 nM PMID[532311]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 20.0 nM PMID[532312]
NPT3089 Cell Line SW1353 Homo sapiens IC50 = 50.0 nM PMID[532312]
NPT570 Individual Protein Arachidonate 5-lipoxygenase Homo sapiens IC50 = 80.0 nM PMID[532315]
NPT183 Individual Protein Arachidonate 5-lipoxygenase Rattus norvegicus IC50 = 58000.0 nM PMID[532315]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens IC50 = 6000.0 nM PMID[532316]
NPT30 Individual Protein Cyclooxygenase-1 Homo sapiens IC50 = 2000.0 nM PMID[532317]
NPT1814 Individual Protein Glucagon receptor Homo sapiens Inhibition = 18.0 % PMID[532318]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532319]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 20.0 nM PMID[532320]
NPT3089 Cell Line SW1353 Homo sapiens IC50 = 50.0 nM PMID[532320]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 72000.0 nM PMID[532321]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 136000.0 nM PMID[532321]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 20.0 nM PMID[532322]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 10.0 nM PMID[532323]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens IC50 > 33000.0 nM PMID[532323]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 72.0 nM PMID[532325]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532325]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Kd = 6800.0 nM PMID[532326]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens IC50 = 7800.0 nM PMID[532326]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Inhibition = 86.5 % PMID[532326]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 16.0 nM PMID[532327]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens IC50 = 135.0 nM PMID[532327]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens IC50 = 124.0 nM PMID[532327]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens IC50 = 2000.0 nM PMID[532327]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 11000.0 nM PMID[532327]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens IC50 = 5000.0 nM PMID[532327]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 38.0 nM PMID[532327]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens IC50 = 500.0 nM PMID[532327]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 72.0 nM PMID[532329]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Kd = 4400.0 nM PMID[532330]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Kd = 45.0 nM PMID[532330]
NPT3208 Individual Protein Serine/threonine-protein kinase 36 Homo sapiens Kd = 860.0 nM PMID[532330]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Kd = 9000.0 nM PMID[532330]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Kd = 95.0 nM PMID[532330]
NPT1706 Individual Protein Serine/threonine-protein kinase 2 Homo sapiens Kd = 4600.0 nM PMID[532330]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Kd = 2100.0 nM PMID[532330]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens Kd = 39.0 nM PMID[532330]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 2900.0 nM PMID[532330]
NPT1712 Individual Protein TRAF2- and NCK-interacting kinase Homo sapiens Kd = 1500.0 nM PMID[532330]
NPT3226 Individual Protein Casein kinase I epsilon Homo sapiens Kd = 220.0 nM PMID[532330]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Kd = 1200.0 nM PMID[532330]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Kd = 1700.0 nM PMID[532330]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Kd = 250.0 nM PMID[532330]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 17.0 nM PMID[532330]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 290.0 nM PMID[532331]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 72.0 nM PMID[532332]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens Inhibition = 92.0 % PMID[532333]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Inhibition = 73.0 % PMID[532333]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Inhibition = 77.0 % PMID[532333]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 68.0 nM PMID[532333]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 30.0 nM PMID[532334]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens IC50 = 790.0 nM PMID[532334]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 462.0 nM PMID[532335]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens Inhibition = 61.0 % PMID[532335]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens Inhibition = 75.0 % PMID[532335]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens Inhibition = 85.0 % PMID[532335]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Inhibition = 67.0 % PMID[532335]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Inhibition = 61.0 % PMID[532335]
NPT2576 Individual Protein Tyrosine-protein kinase TIE-2 Homo sapiens IC50 = 20000.0 nM PMID[532337]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Ki = 18.0 nM PMID[532340]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Ki = 90.0 nM PMID[532340]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 16.0 nM PMID[532341]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 39.0 nM PMID[532341]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 6000.0 nM PMID[532341]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens IC50 = 330.0 nM PMID[532342]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 50.0 nM PMID[532343]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 45.0 nM PMID[532344]
NPT150 Individual Protein Anthrax lethal factor Bacillus anthracis FC = 4.3 n.a. PMID[532346]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 62.0 nM PMID[532347]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens Inhibition = 85.0 % PMID[532347]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Inhibition = 15.0 % PMID[532347]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Inhibition = 0.0 % PMID[532347]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Inhibition = 32.0 % PMID[532347]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Inhibition = 86.0 % PMID[532347]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Inhibition = 98.0 % PMID[532347]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Inhibition = 90.0 % PMID[532347]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Inhibition = 4.0 % PMID[532347]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Inhibition = 7.0 % PMID[532347]
NPT182 Individual Protein Protein kinase C alpha Homo sapiens Inhibition = 11.0 % PMID[532347]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Inhibition = 34.0 % PMID[532347]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Inhibition = 23.0 % PMID[532347]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Inhibition = 68.0 % PMID[532347]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens Inhibition = 38.0 % PMID[532347]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens Inhibition = 87.0 % PMID[532347]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens Inhibition = 92.0 % PMID[532347]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Inhibition = 73.0 % PMID[532347]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Inhibition = 77.0 % PMID[532347]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 50.0 nM PMID[532349]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 7000.0 nM PMID[532350]
NPT6239 Individual Protein Mitogen-activated protein kinase 1 Toxoplasma gondii IC50 = 100.0 nM PMID[532350]
NPT1650 Individual Protein Tyrosine-protein kinase receptor FLT3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2573 Individual Protein Vascular endothelial growth factor receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Kd = 1500.0 nM PMID[532352]
NPT3247 Individual Protein Serine/threonine-protein kinase PAK 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3250 Individual Protein Serine/threonine-protein kinase PCTAIRE-2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3251 Individual Protein Serine/threonine-protein kinase PCTAIRE-3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3252 Individual Protein Serine/threonine-protein kinase PFTAIRE-1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3224 Individual Protein Phosphorylase kinase gamma subunit 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3253 Individual Protein Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Kd = 250.0 nM PMID[532352]
NPT3255 Individual Protein Myosin light chain kinase family member 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3277 Individual Protein Tyrosine-protein kinase receptor TYRO3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1478 Individual Protein Vascular endothelial growth factor receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3256 Individual Protein Serine/threonine-protein kinase WEE1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3257 Individual Protein Serine/threonine-protein kinase 32C Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1663 Individual Protein Tyrosine-protein kinase YES Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1717 Individual Protein Serine/threonine-protein kinase 25 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3258 Individual Protein Mixed lineage kinase 7 Homo sapiens Kd = 4400.0 nM PMID[532352]
NPT3259 Individual Protein Tyrosine-protein kinase ZAP-70 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Activity = 73.0 % PMID[532353]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Activity = 52.0 % PMID[532353]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Activity = 13.0 % PMID[532353]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Activity = 107.0 % PMID[532353]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Activity = 104.0 % PMID[532353]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Activity = 86.0 % PMID[532353]
NPT3260 Individual Protein Phosphatidylinositol-5-phosphate 4-kinase type-2 beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3261 Individual Protein cAMP-dependent protein kinase beta-1 catalytic subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3262 Individual Protein Serine/threonine-protein kinase PRKX Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3263 Individual Protein Protein tyrosine kinase 2 beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1681 Individual Protein Dual specificty protein kinase CLK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1683 Individual Protein Dual specificity protein kinase CLK3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3113 Individual Protein Tyrosine-protein kinase CSK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3265 Individual Protein Casein kinase I isoform alpha-like Homo sapiens Kd = 1700.0 nM PMID[532352]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Kd = 37.0 nM PMID[532352]
NPT3226 Individual Protein Casein kinase I epsilon Homo sapiens Kd = 100.0 nM PMID[532352]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Selectivity = 0.0242 n.a. PMID[532352]
NPT3356 Individual Protein Tyrosine-protein kinase receptor Tie-1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2576 Individual Protein Tyrosine-protein kinase TIE-2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3268 Individual Protein Serine/threonine-protein kinase tousled-like 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3269 Individual Protein Serine/threonine-protein kinase tousled-like 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1712 Individual Protein TRAF2- and NCK-interacting kinase Homo sapiens Kd = 820.0 nM PMID[532352]
NPT3245 Individual Protein Tyrosine kinase non-receptor protein 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3239 Individual Protein Nerve growth factor receptor Trk-A Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3270 Individual Protein Neurotrophic tyrosine kinase receptor type 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3271 Individual Protein NT-3 growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3238 Individual Protein Dual specificity protein kinase TTK Homo sapiens Kd = 2500.0 nM PMID[532352]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Activity = 89.0 % PMID[532353]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Activity = 83.0 % PMID[532353]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Activity = 81.0 % PMID[532353]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Activity = 82.0 % PMID[532353]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1598 Individual Protein Casein kinase II alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3273 Individual Protein Casein kinase II alpha (prime) Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3236 Individual Protein Death-associated protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3230 Individual Protein Serine/threonine-protein kinase 17B Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3274 Individual Protein Dual specificity tyrosine-phosphorylation-regulated kinase 1B Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Kd = 1700.0 nM PMID[532352]
NPT3275 Individual Protein Inhibitor of nuclear factor kappa B kinase epsilon subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3272 Individual Protein Tyrosine-protein kinase TXK Homo sapiens Kd = 4500.0 nM PMID[532352]
NPT3276 Individual Protein Tyrosine-protein kinase TYK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Activity = 97.0 % PMID[532353]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Activity = 81.0 % PMID[532353]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Activity = 89.0 % PMID[532353]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Activity = 90.0 % PMID[532353]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Kd = 1100.0 nM PMID[532352]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Kd = 130.0 nM PMID[532352]
NPT3242 Individual Protein LIM domain kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3278 Individual Protein LIM domain kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3279 Individual Protein Serine/threonine-protein kinase 11 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3280 Individual Protein Serine/threonine-protein kinase c-TAK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1690 Individual Protein Dual specificity mitogen-activated protein kinase kinase 2 Homo sapiens Kd = 9600.0 nM PMID[532352]
NPT3281 Individual Protein Dual specificity mitogen-activated protein kinase kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3283 Individual Protein MAP kinase-interacting serine/threonine-protein kinase MNK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT182 Individual Protein Protein kinase C alpha Homo sapiens Activity = 86.0 % PMID[532353]
NPT3455 Individual Protein Protein kinase C zeta Homo sapiens Activity = 89.0 % PMID[532353]
NPT3364 Individual Protein Protein kinase C mu Homo sapiens Activity = 78.0 % PMID[532353]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Activity = 91.0 % PMID[532353]
NPT3228 Individual Protein Adaptor-associated kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1711 Individual Protein Serine/threonine-protein kinase MST1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1693 Individual Protein Serine/threonine-protein kinase MST4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3284 Individual Protein Serine/threonine-protein kinase NEK7 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3285 Individual Protein Serine/threonine protein kinase NLK Homo sapiens Kd = 25.0 nM PMID[532352]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 12.0 nM PMID[532352]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Kd = 70.0 nM PMID[532352]
NPT3301 Individual Protein Eukaryotic translation initiation factor 2-alpha kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2574 Individual Protein Insulin receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3286 Individual Protein Insulin receptor-related protein Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3214 Individual Protein Tyrosine-protein kinase ABL2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Activity = 93.0 % PMID[532353]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Activity = 80.0 % PMID[532353]
NPT3288 Individual Protein Interleukin-1 receptor-associated kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1439 Individual Protein Tyrosine-protein kinase ITK/TSK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1689 Individual Protein Tyrosine-protein kinase JAK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3246 Individual Protein Tyrosine-protein kinase JAK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1440 Individual Protein Tyrosine-protein kinase JAK3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Kd = 35.0 nM PMID[532352]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3264 Individual Protein Serine/threonine-protein kinase RIO1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3289 Individual Protein Serine/threonine-protein kinase RIO3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3290 Individual Protein Serine/threonine-protein kinase SIK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1448 Individual Protein Serine/threonine-protein kinase Sgk1 Homo sapiens Activity = 91.0 % PMID[532353]
NPT2626 Individual Protein Myosin light chain kinase, smooth muscle Homo sapiens Activity = 85.0 % PMID[532353]
NPT3813 Individual Protein Tyrosine-protein kinase SRC Gallus gallus Activity = 73.0 % PMID[532353]
NPT3287 Individual Protein Activin receptor type-1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3293 Individual Protein Activin receptor type-1B Homo sapiens Kd = 3000.0 nM PMID[532352]
NPT3294 Individual Protein Activin receptor type-2A Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3295 Individual Protein Activin receptor type-2B Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3292 Individual Protein Serine/threonine-protein kinase SRPK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3296 Individual Protein Serine/threonine-protein kinase 33 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3297 Individual Protein Non-receptor tyrosine-protein kinase TNK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3298 Individual Protein Serine/threonine-protein kinase TNNI3K Homo sapiens Kd = 3500.0 nM PMID[532352]
NPT3299 Individual Protein Testis-specific serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3300 Individual Protein Serine/threonine-protein kinase 32B Homo sapiens Kd = 2100.0 nM PMID[532352]
NPT14 Individual Protein Tyrosine-protein kinase FYN Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens Kd = 19.0 nM PMID[532352]
NPT1661 Individual Protein ALK tyrosine kinase receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3222 Individual Protein AMP-activated protein kinase, alpha-1 subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1671 Individual Protein AMP-activated protein kinase, alpha-2 subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3342 Individual Protein Epithelial discoidin domain-containing receptor 1 Homo sapiens Kd = 1000.0 nM PMID[532352]
NPT3303 Individual Protein Discoidin domain-containing receptor 2 Homo sapiens Kd = 5000.0 nM PMID[532352]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3304 Individual Protein Serine/threonine-protein kinase receptor R3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3305 Individual Protein Chaperone activity of bc1 complex-like, mitochondrial Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2546 Individual Protein Serine/threonine-protein kinase AKT3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3307 Individual Protein Serine/threonine-protein kinase LATS1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3308 Individual Protein Serine/threonine-protein kinase LATS2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Kd = 2800.0 nM PMID[532352]
NPT1707 Individual Protein Serine/threonine-protein kinase 10 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3309 Individual Protein Leukocyte tyrosine kinase receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3111 Individual Protein Tyrosine-protein kinase Lyn Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3209 Individual Protein Mitogen-activated protein kinase kinase kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1431 Individual Protein Mitogen-activated protein kinase kinase kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1698 Individual Protein Serine/threonine-protein kinase PCTAIRE-1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Activity = 85.0 % PMID[532353]
NPT3206 Individual Protein Serine/threonine-protein kinase Aurora-C Homo sapiens Activity = 92.0 % PMID[532353]
NPT3344 Individual Protein BR serine/threonine-protein kinase 2 Homo sapiens Activity = 86.0 % PMID[532353]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Activity = 86.0 % PMID[532353]
NPT3306 Individual Protein Serine/threonine-protein kinase MRCK gamma Homo sapiens Kd = 400.0 nM PMID[532352]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1700.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 340.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 710.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1300.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1600.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1500.0 nM PMID[532352]
NPT3302 Individual Protein Ankyrin repeat and protein kinase domain-containing protein 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1660 Individual Protein NUAK family SNF1-like kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3020 Individual Protein Platelet-derived growth factor receptor alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2575 Individual Protein Platelet-derived growth factor receptor beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3223 Individual Protein Phosphorylase kinase gamma subunit 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1444 Individual Protein PI3-kinase p110-alpha subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3310 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3311 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3248 Individual Protein CaM-kinase kinase alpha Homo sapiens Activity = 106.0 % PMID[532353]
NPT1678 Individual Protein CaM-kinase kinase beta Homo sapiens Activity = 99.0 % PMID[532353]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Activity = 66.0 % PMID[532353]
NPT1680 Individual Protein Serine/threonine-protein kinase Chk2 Homo sapiens Activity = 92.0 % PMID[532353]
NPT1432 Individual Protein Serine/threonine-protein kinase Aurora-A Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1659 Individual Protein Tyrosine-protein kinase receptor UFO Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3210 Individual Protein BMP-2-inducible protein kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3312 Individual Protein Tyrosine-protein kinase BLK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3313 Individual Protein Bone morphogenetic protein receptor type-1A Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3314 Individual Protein Bone morphogenetic protein receptor type-2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1434 Individual Protein Serine/threonine-protein kinase B-raf Homo sapiens Kd = 710.0 nM PMID[532352]
NPT1434 Individual Protein Serine/threonine-protein kinase B-raf Homo sapiens Kd = 530.0 nM PMID[532352]
NPT3315 Individual Protein BR serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1673 Individual Protein CaM kinase I gamma Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3316 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 4 Homo sapiens Kd = 3700.0 nM PMID[532352]
NPT3109 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3317 Individual Protein Serine/threonine-protein kinase MARK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3235 Individual Protein MAP/microtubule affinity-regulating kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3318 Individual Protein MAP/microtubule affinity-regulating kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3319 Individual Protein Dual specificity mitogen-activated protein kinase kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1691 Individual Protein Dual specificity mitogen-activated protein kinase kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3320 Individual Protein Proto-oncogene tyrosine-protein kinase MER Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Activity = 8.0 % PMID[532353]
NPT3113 Individual Protein Tyrosine-protein kinase CSK Homo sapiens Activity = 69.0 % PMID[532353]
NPT3114 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 1A Homo sapiens Activity = 84.0 % PMID[532353]
NPT3399 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 2 Homo sapiens Activity = 97.0 % PMID[532353]
NPT1674 Individual Protein CaM kinase II alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1677 Individual Protein CaM kinase IV Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3248 Individual Protein CaM-kinase kinase alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1678 Individual Protein CaM-kinase kinase beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3321 Individual Protein PITSLRE serine/threonine-protein kinase CDC2L1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3322 Individual Protein PITSLRE serine/threonine-protein kinase CDC2L2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3323 Individual Protein Cell division cycle 2-like protein kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3324 Individual Protein Cell division protein kinase 8 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3325 Individual Protein Myosin light chain kinase, smooth muscle Gallus gallus Kd > 10000.0 nM PMID[532352]
NPT3326 Individual Protein Mitogen-activated protein kinase kinase kinase 9 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3327 Individual Protein Mitogen-activated protein kinase kinase kinase 10 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3328 Individual Protein Mitogen-activated protein kinase kinase kinase 11 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3329 Individual Protein Serine/threonine-protein kinase MRCK-A Homo sapiens Kd = 6200.0 nM PMID[532352]
NPT3330 Individual Protein Serine/threonine-protein kinase MRCK beta Homo sapiens Kd = 2700.0 nM PMID[532352]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3332 Individual Protein Serine/threonine-protein kinase 24 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3333 Individual Protein Muscle, skeletal receptor tyrosine protein kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2626 Individual Protein Myosin light chain kinase, smooth muscle Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3460 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 3 Homo sapiens Activity = 112.0 % PMID[532353]
NPT1344 Individual Protein Serine/threonine-protein kinase EEF2K Homo sapiens Activity = 98.0 % PMID[532353]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Activity = 89.0 % PMID[532353]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Activity = 83.0 % PMID[532353]
NPT3363 Individual Protein Mitogen-activated protein kinase 15 Homo sapiens Activity = 93.0 % PMID[532353]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens Activity = 25.0 % PMID[532353]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3334 Individual Protein Citron Rho-interacting kinase Homo sapiens Kd = 420.0 nM PMID[532352]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3231 Individual Protein Dual specificity protein kinase CLK4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3267 Individual Protein Macrophage colony stimulating factor receptor Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1721 Individual Protein Death-associated protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3335 Individual Protein Serine/threonine-protein kinase DCLK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3336 Individual Protein Serine/threonine-protein kinase DCLK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3337 Individual Protein Serine/threonine-protein kinase DCLK3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3243 Individual Protein myosin light chain kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3338 Individual Protein Myosin IIIA Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3339 Individual Protein Myosin-IIIB Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3233 Individual Protein Serine/threonine-protein kinase 38-like Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3340 Individual Protein Serine/threonine-protein kinase Nek1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3341 Individual Protein Serine/threonine-protein kinase Nek5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3241 Individual Protein Serine/threonine-protein kinase NEK9 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3120 Individual Protein Serine/threonine-protein kinase PAK 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1442 Individual Protein Serine/threonine-protein kinase PAK 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Activity = 86.0 % PMID[532353]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Activity = 81.0 % PMID[532353]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Activity = 98.0 % PMID[532353]
NPT3284 Individual Protein Serine/threonine-protein kinase NEK7 Homo sapiens Activity = 96.0 % PMID[532353]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Activity = 9.0 % PMID[532353]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Kd = 1800.0 nM PMID[532352]
NPT3343 Individual Protein Uncharacterized aarF domain-containing protein kinase 4 Homo sapiens Kd = 3100.0 nM PMID[532352]
NPT3206 Individual Protein Serine/threonine-protein kinase Aurora-C Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2750 Individual Protein Tyrosine-protein kinase BMX Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3344 Individual Protein BR serine/threonine-protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1371 Individual Protein Cyclin-dependent kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3345 Individual Protein Cyclin-dependent kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3240 Individual Protein Cyclin-dependent kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3346 Individual Protein Cyclin-dependent kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1706 Individual Protein Serine/threonine-protein kinase 2 Homo sapiens Kd = 3700.0 nM PMID[532352]
NPT3348 Individual Protein NUAK family SNF1-like kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3349 Individual Protein Serine/threonine-protein kinase SIK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Kd = 5300.0 nM PMID[532352]
NPT3350 Individual Protein Tyrosine-protein kinase Srms Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1708 Individual Protein Serine/threonine-protein kinase 16 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3208 Individual Protein Serine/threonine-protein kinase 36 Homo sapiens Kd = 1300.0 nM PMID[532352]
NPT1449 Individual Protein Tyrosine-protein kinase SYK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3351 Individual Protein Tyrosine-protein kinase TEC Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3352 Individual Protein Dual specificity testis-specific protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens Kd = 7100.0 nM PMID[532352]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Activity = 34.0 % PMID[532353]
NPT3432 Individual Protein Homeodomain-interacting protein kinase 2 Homo sapiens Activity = 86.0 % PMID[532353]
NPT3409 Individual Protein Homeodomain-interacting protein kinase 3 Homo sapiens Activity = 96.0 % PMID[532353]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Activity = 95.0 % PMID[532353]
NPT3347 Individual Protein Cyclin-dependent kinase 9 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1900.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 3200.0 nM PMID[532352]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 2000.0 nM PMID[532352]
NPT3354 Individual Protein Ephrin type-A receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3225 Individual Protein Ephrin type-A receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3217 Individual Protein Ephrin type-A receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3218 Individual Protein Ephrin type-A receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3219 Individual Protein Ephrin type-A receptor 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3220 Individual Protein Ephrin type-A receptor 6 Homo sapiens Kd = 1200.0 nM PMID[532352]
NPT3211 Individual Protein Ephrin type-A receptor 7 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3355 Individual Protein TGF-beta receptor type II Homo sapiens Kd = 1800.0 nM PMID[532352]
NPT3249 Individual Protein Tyrosine- and threonine-specific cdc2-inhibitory kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1656 Individual Protein Protein kinase N1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3358 Individual Protein Serine/threonine-protein kinase PLK3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1702 Individual Protein Serine/threonine-protein kinase PLK4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3124 Individual Protein Protein kinase C eta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Activity = 60.0 % PMID[532353]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Activity = 72.0 % PMID[532353]
NPT3815 Individual Protein Tyrosine-protein kinase LCK Mus musculus Activity = 56.0 % PMID[532353]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Activity = 84.0 % PMID[532353]
NPT3461 Individual Protein MAP kinase-activated protein kinase 3 Homo sapiens Activity = 120.0 % PMID[532353]
NPT3216 Individual Protein Ephrin type-A receptor 8 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3212 Individual Protein Ephrin type-B receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3359 Individual Protein Ephrin type-B receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2572 Individual Protein Ephrin type-B receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT286 Individual Protein Receptor protein-tyrosine kinase erbB-2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3360 Individual Protein Tubulin alpha-1 chain Rattus norvegicus Kd > 10000.0 nM PMID[532352]
NPT1692 Individual Protein Mitogen-activated protein kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3361 Individual Protein Mitogen-activated protein kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3362 Individual Protein Mitogen-activated protein kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3363 Individual Protein Mitogen-activated protein kinase 15 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3244 Individual Protein Tyrosine-protein kinase FER Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3364 Individual Protein Protein kinase C mu Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3365 Individual Protein Serine/threonine-protein kinase D2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3366 Individual Protein Protein kinase C nu Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3368 Individual Protein cGMP-dependent protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3369 Individual Protein Interferon-induced, double-stranded RNA-activated protein kinase Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1436 Individual Protein Focal adhesion kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Kd = 3900.0 nM PMID[532352]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens Kd = 980.0 nM PMID[532352]
NPT3370 Individual Protein Tyrosine-protein kinase receptor RET Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3280 Individual Protein Serine/threonine-protein kinase c-TAK1 Homo sapiens Activity = 98.0 % PMID[532353]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Activity = 83.0 % PMID[532353]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Activity = 85.0 % PMID[532353]
NPT3283 Individual Protein MAP kinase-interacting serine/threonine-protein kinase MNK1 Homo sapiens Activity = 109.0 % PMID[532353]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Activity = 107.0 % PMID[532353]
NPT1437 Individual Protein Tyrosine-protein kinase FES Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1480 Individual Protein Fibroblast growth factor receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1481 Individual Protein Fibroblast growth factor receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3227 Individual Protein Fibroblast growth factor receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3372 Individual Protein Fibroblast growth factor receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3112 Individual Protein Tyrosine-protein kinase FGR Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT301 Individual Protein Vascular endothelial growth factor receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3371 Individual Protein Receptor-interacting serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Kd = 24.0 nM PMID[532352]
NPT3373 Individual Protein Proto-oncogene tyrosine-protein kinase ROS Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Kd = 320.0 nM PMID[532352]
NPT3234 Individual Protein Ribosomal protein S6 kinase alpha 2 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT3374 Individual Protein Ribosomal protein S6 kinase alpha 4 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Activity = 91.0 % PMID[532353]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Activity = 96.0 % PMID[532353]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Activity = 95.0 % PMID[532353]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Activity = 7.0 % PMID[532353]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens IC50 = 290.0 nM PMID[532354]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Inhibition = 78.0 % PMID[532355]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens IC50 = 120.0 nM PMID[532356]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Inhibition = 92.0 % PMID[532356]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 40.0 nM PMID[532356]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532357]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 70.0 nM PMID[532358]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 = 320.0 nM PMID[532358]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532359]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 44.0 nM PMID[532360]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 39.0 nM PMID[532361]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 6000.0 nM PMID[532361]
NPT306 Cell Line PC-3 Homo sapiens FC = 0.721 n.a. PMID[532363]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Inhibition = 95.0 % PMID[532364]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Inhibition = 32.0 % PMID[532364]
NPT1610 Individual Protein Rho-associated protein kinase 2 Rattus norvegicus Inhibition = 77.0 % PMID[532364]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Inhibition = 66.0 % PMID[532364]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Inhibition = 87.0 % PMID[532364]
NPT1448 Individual Protein Serine/threonine-protein kinase Sgk1 Homo sapiens Inhibition = 83.0 % PMID[532364]
NPT1443 Individual Protein Pyruvate dehydrogenase kinase isoform 1 Homo sapiens Inhibition = 89.0 % PMID[532364]
NPT182 Individual Protein Protein kinase C alpha Homo sapiens Inhibition = 89.0 % PMID[532364]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Inhibition = 112.0 % PMID[532364]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Inhibition = 86.0 % PMID[532364]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Inhibition = 93.0 % PMID[532364]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Inhibition = 93.0 % PMID[532364]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Inhibition = 96.0 % PMID[532364]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Inhibition = 10.0 % PMID[532364]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Inhibition = 2.0 % PMID[532364]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Inhibition = 101.0 % PMID[532364]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Inhibition = 85.0 % PMID[532364]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Ki = 57.0 nM PMID[532365]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 4.1 nM PMID[532365]
NPT149 Individual Protein Endoplasmic reticulum-associated amyloid beta-peptide-binding protein Homo sapiens Potency = 19952.6 nM PMID[532369]
NPT149 Individual Protein Endoplasmic reticulum-associated amyloid beta-peptide-binding protein Homo sapiens Potency = 39810.7 nM PMID[532368]
NPT48 Individual Protein Lysine-specific demethylase 4D-like Homo sapiens Potency = 35481.3 nM PMID[532369]
NPT48 Individual Protein Lysine-specific demethylase 4D-like Homo sapiens Potency = 25118.9 nM PMID[532368]
NPT210 Individual Protein Thyroid stimulating hormone receptor Homo sapiens Potency = 39810.7 nM PMID[532369]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens Potency = 39.8 nM PMID[532369]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Potency = 25118.9 nM PMID[532369]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Potency = 12589.3 nM PMID[532368]
NPT150 Individual Protein Anthrax lethal factor Bacillus anthracis Potency = 12589.3 nM PMID[532368]
NPT150 Individual Protein Anthrax lethal factor Bacillus anthracis Potency = 31622.8 nM PMID[532369]
NPT151 Individual Protein 15-hydroxyprostaglandin dehydrogenase [NAD+] Homo sapiens Potency = 31622.8 nM PMID[532368]
NPT151 Individual Protein 15-hydroxyprostaglandin dehydrogenase [NAD+] Homo sapiens Potency = 25118.9 nM PMID[532369]
NPT149 Individual Protein Endoplasmic reticulum-associated amyloid beta-peptide-binding protein Homo sapiens Potency = 39810.7 nM PMID[532369]
NPT149 Individual Protein Endoplasmic reticulum-associated amyloid beta-peptide-binding protein Homo sapiens Potency = 31622.8 nM PMID[532368]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Potency = 501.2 nM PMID[532368]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens Potency = 39810.7 nM PMID[532369]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens Potency = 1258.9 nM PMID[532369]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens Potency = 1995.3 nM PMID[532369]
NPT1139 Individual Protein Arachidonate 15-lipoxygenase, type II Homo sapiens Potency n.a. 25118.9 nM PMID[532369]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens AC50 = 39810.72 nM PMID[532369]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens AC50 = 1995.26 nM PMID[532369]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens AC50 = 501.19 nM PMID[532368]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens AC50 = 630.96 nM PMID[532368]
NPT109 Individual Protein Cytochrome P450 3A4 Homo sapiens AC50 = 1258.93 nM PMID[532369]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens AC50 = 3981.07 nM PMID[532369]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens AC50 = 39.81 nM PMID[532369]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 15.0 nM PMID[532372]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 1230.0 nM PMID[532372]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532373]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 55.0 nM PMID[532374]
NPT198 Individual Protein Vitamin D receptor Homo sapiens Potency n.a. 70794.6 nM PMID[532369]
NPT199 Individual Protein DNA polymerase kappa Homo sapiens Potency n.a. 7943.3 nM PMID[532369]
NPT444 Individual Protein Ubiquitin carboxyl-terminal hydrolase 1 Homo sapiens Potency n.a. 56234.1 nM PMID[532369]
NPT1681 Individual Protein Dual specificty protein kinase CLK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3271 Individual Protein NT-3 growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Kd = 1500.0 nM PMID[532375]
NPT3320 Individual Protein Proto-oncogene tyrosine-protein kinase MER Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3292 Individual Protein Serine/threonine-protein kinase SRPK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3206 Individual Protein Serine/threonine-protein kinase Aurora-C Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3269 Individual Protein Serine/threonine-protein kinase tousled-like 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3222 Individual Protein AMP-activated protein kinase, alpha-1 subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3378 Individual Protein Serine/threonine-protein kinase SIK3 Homo sapiens Kd = 3900.0 nM PMID[532375]
NPT1708 Individual Protein Serine/threonine-protein kinase 16 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3250 Individual Protein Serine/threonine-protein kinase PCTAIRE-2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3303 Individual Protein Discoidin domain-containing receptor 2 Homo sapiens Kd = 5000.0 nM PMID[532375]
NPT3304 Individual Protein Serine/threonine-protein kinase receptor R3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2213 Individual Protein Cyclin-dependent kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3227 Individual Protein Fibroblast growth factor receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2574 Individual Protein Insulin receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1440 Individual Protein Tyrosine-protein kinase JAK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Kd = 7900.0 nM PMID[532375]
NPT3223 Individual Protein Phosphorylase kinase gamma subunit 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3279 Individual Protein Serine/threonine-protein kinase 11 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2576 Individual Protein Tyrosine-protein kinase TIE-2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3379 Individual Protein Mitogen-activated protein kinase kinase kinase 15 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1680 Individual Protein Serine/threonine-protein kinase Chk2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT286 Individual Protein Receptor protein-tyrosine kinase erbB-2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3234 Individual Protein Ribosomal protein S6 kinase alpha 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3374 Individual Protein Ribosomal protein S6 kinase alpha 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3245 Individual Protein Tyrosine kinase non-receptor protein 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3239 Individual Protein Nerve growth factor receptor Trk-A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3255 Individual Protein Myosin light chain kinase family member 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3301 Individual Protein Eukaryotic translation initiation factor 2-alpha kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3380 Individual Protein Serine/threonine-protein kinase SBK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3381 Individual Protein Misshapen-like kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3336 Individual Protein Serine/threonine-protein kinase DCLK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1435 Individual Protein Receptor protein-tyrosine kinase erbB-4 Homo sapiens Kd = 4800.0 nM PMID[532375]
NPT3310 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3220 Individual Protein Ephrin type-A receptor 6 Homo sapiens Kd = 1200.0 nM PMID[532375]
NPT3339 Individual Protein Myosin-IIIB Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3382 Individual Protein Serine/threonine-protein kinase ULK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3287 Individual Protein Activin receptor type-1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3295 Individual Protein Activin receptor type-2B Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3383 Individual Protein Serine/threonine-protein kinase 32A Homo sapiens Kd = 1300.0 nM PMID[532375]
NPT3384 Individual Protein Cyclin-dependent kinase-like 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3283 Individual Protein MAP kinase-interacting serine/threonine-protein kinase MNK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3253 Individual Protein Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3385 Individual Protein Bone morphogenetic protein receptor type-1B Homo sapiens Kd = 3300.0 nM PMID[532375]
NPT3314 Individual Protein Bone morphogenetic protein receptor type-2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3345 Individual Protein Cyclin-dependent kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3324 Individual Protein Cell division protein kinase 8 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3347 Individual Protein Cyclin-dependent kinase 9 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1890 Individual Protein Serine/threonine-protein kinase/endoribonuclease IRE1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3386 Individual Protein Interleukin-1 receptor-associated kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3294 Individual Protein Activin receptor type-2A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1659 Individual Protein Tyrosine-protein kinase receptor UFO Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3312 Individual Protein Tyrosine-protein kinase BLK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2750 Individual Protein Tyrosine-protein kinase BMX Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1677 Individual Protein CaM kinase IV Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1371 Individual Protein Cyclin-dependent kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3346 Individual Protein Cyclin-dependent kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3168 Individual Protein Casein kinase I alpha Homo sapiens Kd = 75.0 nM PMID[532375]
NPT3226 Individual Protein Casein kinase I epsilon Homo sapiens Kd = 100.0 nM PMID[532375]
NPT1598 Individual Protein Casein kinase II alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3273 Individual Protein Casein kinase II alpha (prime) Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3342 Individual Protein Epithelial discoidin domain-containing receptor 1 Homo sapiens Kd = 1000.0 nM PMID[532375]
NPT3387 Individual Protein Receptor tyrosine-protein kinase erbB-3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1437 Individual Protein Tyrosine-protein kinase FES Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT301 Individual Protein Vascular endothelial growth factor receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2573 Individual Protein Vascular endothelial growth factor receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Kd = 1800.0 nM PMID[532375]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Kd = 1700.0 nM PMID[532375]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1689 Individual Protein Tyrosine-protein kinase JAK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1478 Individual Protein Vascular endothelial growth factor receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3242 Individual Protein LIM domain kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3111 Individual Protein Tyrosine-protein kinase Lyn Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3280 Individual Protein Serine/threonine-protein kinase c-TAK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3388 Individual Protein Tyrosine-protein kinase CTK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3389 Individual Protein Mitogen-activated protein kinase kinase kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3328 Individual Protein Mitogen-activated protein kinase kinase kinase 11 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3327 Individual Protein Mitogen-activated protein kinase kinase kinase 10 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3390 Individual Protein Macrophage-stimulating protein receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3391 Individual Protein Serine/threonine-protein kinase Nek3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3120 Individual Protein Serine/threonine-protein kinase PAK 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1442 Individual Protein Serine/threonine-protein kinase PAK 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3247 Individual Protein Serine/threonine-protein kinase PAK 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3251 Individual Protein Serine/threonine-protein kinase PCTAIRE-3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2575 Individual Protein Platelet-derived growth factor receptor beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3392 Individual Protein Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1445 Individual Protein PI3-kinase p110-gamma subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3393 Individual Protein PI4-kinase beta subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3261 Individual Protein cAMP-dependent protein kinase beta-1 catalytic subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3394 Individual Protein Protein kinase C iota Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3364 Individual Protein Protein kinase C mu Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3361 Individual Protein Mitogen-activated protein kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1692 Individual Protein Mitogen-activated protein kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3362 Individual Protein Mitogen-activated protein kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Kd = 1100.0 nM PMID[532375]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Kd = 70.0 nM PMID[532375]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Kd = 35.0 nM PMID[532375]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3281 Individual Protein Dual specificity mitogen-activated protein kinase kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1691 Individual Protein Dual specificity mitogen-activated protein kinase kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3369 Individual Protein Interferon-induced, double-stranded RNA-activated protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens Kd = 980.0 nM PMID[532375]
NPT3395 Individual Protein Rhodopsin kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3373 Individual Protein Proto-oncogene tyrosine-protein kinase ROS Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Kd = 320.0 nM PMID[532375]
NPT3319 Individual Protein Dual specificity mitogen-activated protein kinase kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3396 Individual Protein Serine/threonine-protein kinase Nek4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3397 Individual Protein Cyclin-dependent kinase-like 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1449 Individual Protein Tyrosine-protein kinase SYK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3351 Individual Protein Tyrosine-protein kinase TEC Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3355 Individual Protein TGF-beta receptor type II Homo sapiens Kd = 1800.0 nM PMID[532375]
NPT3238 Individual Protein Dual specificity protein kinase TTK Homo sapiens Kd = 2500.0 nM PMID[532375]
NPT3272 Individual Protein Tyrosine-protein kinase TXK Homo sapiens Kd = 4500.0 nM PMID[532375]
NPT3276 Individual Protein Tyrosine-protein kinase TYK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3276 Individual Protein Tyrosine-protein kinase TYK2 Homo sapiens Kd = 2000.0 nM PMID[532375]
NPT3256 Individual Protein Serine/threonine-protein kinase WEE1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3260 Individual Protein Phosphatidylinositol-5-phosphate 4-kinase type-2 beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3398 Individual Protein Serine/threonine-protein kinase ULK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3332 Individual Protein Serine/threonine-protein kinase 24 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3399 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1432 Individual Protein Serine/threonine-protein kinase Aurora-A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3329 Individual Protein Serine/threonine-protein kinase MRCK-A Homo sapiens Kd = 6200.0 nM PMID[532375]
NPT3311 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3400 Individual Protein Peripheral plasma membrane protein CASK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3401 Individual Protein Cyclin-dependent kinase 13 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3371 Individual Protein Receptor-interacting serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Kd = 24.0 nM PMID[532375]
NPT3289 Individual Protein Serine/threonine-protein kinase RIO3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3402 Individual Protein Serine/threonine-protein kinase PRP4 homolog Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3403 Individual Protein Cyclin-dependent kinase-like 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3344 Individual Protein BR serine/threonine-protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3297 Individual Protein Non-receptor tyrosine-protein kinase TNK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1683 Individual Protein Dual specificity protein kinase CLK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3358 Individual Protein Serine/threonine-protein kinase PLK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1650 Individual Protein Tyrosine-protein kinase receptor FLT3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1679 Individual Protein Cyclin-dependent kinase-like 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3230 Individual Protein Serine/threonine-protein kinase 17B Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3293 Individual Protein Activin receptor type-1B Homo sapiens Kd = 3000.0 nM PMID[532375]
NPT1661 Individual Protein ALK tyrosine kinase receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3313 Individual Protein Bone morphogenetic protein receptor type-1A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1434 Individual Protein Serine/threonine-protein kinase B-raf Homo sapiens Kd = 710.0 nM PMID[532375]
NPT1434 Individual Protein Serine/threonine-protein kinase B-raf Homo sapiens Kd = 530.0 nM PMID[532375]
NPT3113 Individual Protein Tyrosine-protein kinase CSK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3225 Individual Protein Ephrin type-A receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3218 Individual Protein Ephrin type-A receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3211 Individual Protein Ephrin type-A receptor 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3212 Individual Protein Ephrin type-B receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3359 Individual Protein Ephrin type-B receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2572 Individual Protein Ephrin type-B receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3404 Individual Protein Ephrin type-B receptor 6 Homo sapiens Kd = 3100.0 nM PMID[532375]
NPT3405 Individual Protein Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3406 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens Kd = 7100.0 nM PMID[532375]
NPT3407 Individual Protein Mitogen-activated protein kinase kinase kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3307 Individual Protein Serine/threonine-protein kinase LATS1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3274 Individual Protein Dual specificity tyrosine-phosphorylation-regulated kinase 1B Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3408 Individual Protein Mitogen-activated protein kinase kinase kinase 13 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3335 Individual Protein Serine/threonine-protein kinase DCLK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3240 Individual Protein Cyclin-dependent kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1721 Individual Protein Death-associated protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3246 Individual Protein Tyrosine-protein kinase JAK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1446 Individual Protein PI3-kinase p110-delta subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3262 Individual Protein Serine/threonine-protein kinase PRKX Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1694 Individual Protein Serine/threonine-protein kinase OSR1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Kd = 2600.0 nM PMID[532375]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Kd = 3900.0 nM PMID[532375]
NPT3214 Individual Protein Tyrosine-protein kinase ABL2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3267 Individual Protein Macrophage colony stimulating factor receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1700.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 340.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 710.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1300.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1600.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1500.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 1900.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 3200.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 2000.0 nM PMID[532375]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Kd = 2500.0 nM PMID[532375]
NPT3354 Individual Protein Ephrin type-A receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3217 Individual Protein Ephrin type-A receptor 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3244 Individual Protein Tyrosine-protein kinase FER Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3112 Individual Protein Tyrosine-protein kinase FGR Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens Kd = 19.0 nM PMID[532375]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Kd = 2800.0 nM PMID[532375]
NPT592 Individual Protein Rho-associated protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Kd = 5300.0 nM PMID[532375]
NPT3356 Individual Protein Tyrosine-protein kinase receptor Tie-1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1663 Individual Protein Tyrosine-protein kinase YES Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2546 Individual Protein Serine/threonine-protein kinase AKT3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1439 Individual Protein Tyrosine-protein kinase ITK/TSK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3278 Individual Protein LIM domain kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3333 Individual Protein Muscle, skeletal receptor tyrosine protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3409 Individual Protein Homeodomain-interacting protein kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3366 Individual Protein Protein kinase C nu Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3410 Individual Protein Serine/threonine-protein kinase MAK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3411 Individual Protein Mitogen-activated protein kinase kinase kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3209 Individual Protein Mitogen-activated protein kinase kinase kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1431 Individual Protein Mitogen-activated protein kinase kinase kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Kd = 3900.0 nM PMID[532375]
NPT1707 Individual Protein Serine/threonine-protein kinase 10 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3330 Individual Protein Serine/threonine-protein kinase MRCK beta Homo sapiens Kd = 2700.0 nM PMID[532375]
NPT3270 Individual Protein Neurotrophic tyrosine kinase receptor type 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1698 Individual Protein Serine/threonine-protein kinase PCTAIRE-1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3020 Individual Protein Platelet-derived growth factor receptor alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3224 Individual Protein Phosphorylase kinase gamma subunit 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1444 Individual Protein PI3-kinase p110-alpha subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3376 Individual Protein PI3-kinase p110-beta subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1671 Individual Protein AMP-activated protein kinase, alpha-2 subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3124 Individual Protein Protein kinase C eta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3368 Individual Protein cGMP-dependent protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1711 Individual Protein Serine/threonine-protein kinase MST1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3352 Individual Protein Dual specificity testis-specific protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3277 Individual Protein Tyrosine-protein kinase receptor TYRO3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1715 Individual Protein Serine/threonine-protein kinase VRK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3412 Individual Protein Mitogen-activated protein kinase kinase kinase 12 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1717 Individual Protein Serine/threonine-protein kinase 25 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1678 Individual Protein CaM-kinase kinase beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3109 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3413 Individual Protein Mitogen-activated protein kinase kinase kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3414 Individual Protein Serine/threonine-protein kinase PLK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3334 Individual Protein Citron Rho-interacting kinase Homo sapiens Kd = 420.0 nM PMID[532375]
NPT3288 Individual Protein Interleukin-1 receptor-associated kinase 3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1710 Individual Protein Serine/threonine-protein kinase 38 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3340 Individual Protein Serine/threonine-protein kinase Nek1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3268 Individual Protein Serine/threonine-protein kinase tousled-like 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3252 Individual Protein Serine/threonine-protein kinase PFTAIRE-1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3415 Individual Protein Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma Homo sapiens Kd = 2600.0 nM PMID[532375]
NPT3416 Individual Protein STE20/SPS1-related proline-alanine-rich protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3417 Individual Protein Serine/threonine-protein kinase TBK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3418 Individual Protein Serine/threonine-protein kinase Sgk3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3275 Individual Protein Inhibitor of nuclear factor kappa B kinase epsilon subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3286 Individual Protein Insulin receptor-related protein Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1702 Individual Protein Serine/threonine-protein kinase PLK4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3236 Individual Protein Death-associated protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3419 Individual Protein Serine/threonine-protein kinase SRPK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3420 Individual Protein Eukaryotic translation initiation factor 2-alpha kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Kd = 250.0 nM PMID[532375]
NPT3308 Individual Protein Serine/threonine-protein kinase LATS2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3421 Individual Protein Hormonally up-regulated neu tumor-associated kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3422 Individual Protein Serine/threonine-protein kinase ULK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1706 Individual Protein Serine/threonine-protein kinase 2 Homo sapiens Kd = 3700.0 nM PMID[532375]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1660 Individual Protein NUAK family SNF1-like kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3228 Individual Protein Adaptor-associated kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3423 Individual Protein Serine/threonine-protein kinase ICK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3424 Individual Protein Microtubule-associated serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3233 Individual Protein Serine/threonine-protein kinase 38-like Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1712 Individual Protein TRAF2- and NCK-interacting kinase Homo sapiens Kd = 820.0 nM PMID[532375]
NPT3323 Individual Protein Cell division cycle 2-like protein kinase 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3290 Individual Protein Serine/threonine-protein kinase SIK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3208 Individual Protein Serine/threonine-protein kinase 36 Homo sapiens Kd = 1300.0 nM PMID[532375]
NPT3298 Individual Protein Serine/threonine-protein kinase TNNI3K Homo sapiens Kd = 3500.0 nM PMID[532375]
NPT3425 Individual Protein Interleukin-1 receptor-associated kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3426 Individual Protein Serine/threonine-protein kinase TAO2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3285 Individual Protein Serine/threonine protein kinase NLK Homo sapiens Kd = 25.0 nM PMID[532375]
NPT3427 Individual Protein Serine/threonine-protein kinase TAO3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3365 Individual Protein Serine/threonine-protein kinase D2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1693 Individual Protein Serine/threonine-protein kinase MST4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3338 Individual Protein Myosin IIIA Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3235 Individual Protein MAP/microtubule affinity-regulating kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3306 Individual Protein Serine/threonine-protein kinase MRCK gamma Homo sapiens Kd = 400.0 nM PMID[532375]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3210 Individual Protein BMP-2-inducible protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3428 Individual Protein Transient receptor potential cation channel subfamily M member 6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3429 Individual Protein SNF-related serine/threonine-protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1704 Individual Protein Serine/threonine-protein kinase RIO2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3300 Individual Protein Serine/threonine-protein kinase 32B Homo sapiens Kd = 2100.0 nM PMID[532375]
NPT3317 Individual Protein Serine/threonine-protein kinase MARK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3305 Individual Protein Chaperone activity of bc1 complex-like, mitochondrial Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1673 Individual Protein CaM kinase I gamma Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3216 Individual Protein Ephrin type-A receptor 8 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3370 Individual Protein Tyrosine-protein kinase receptor RET Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3430 Individual Protein Receptor-interacting serine/threonine-protein kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3231 Individual Protein Dual specificity protein kinase CLK4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3431 Individual Protein Serine/threonine-protein kinase TAO1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3432 Individual Protein Homeodomain-interacting protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3372 Individual Protein Fibroblast growth factor receptor 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1481 Individual Protein Fibroblast growth factor receptor 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1480 Individual Protein Fibroblast growth factor receptor 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3322 Individual Protein PITSLRE serine/threonine-protein kinase CDC2L2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3433 Individual Protein Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3343 Individual Protein Uncharacterized aarF domain-containing protein kinase 4 Homo sapiens Kd = 3100.0 nM PMID[532375]
NPT3434 Individual Protein SPS1/STE20-related protein kinase YSK4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1690 Individual Protein Dual specificity mitogen-activated protein kinase kinase 2 Homo sapiens Kd = 9600.0 nM PMID[532375]
NPT3296 Individual Protein Serine/threonine-protein kinase 33 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3348 Individual Protein NUAK family SNF1-like kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3318 Individual Protein MAP/microtubule affinity-regulating kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3264 Individual Protein Serine/threonine-protein kinase RIO1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3299 Individual Protein Testis-specific serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3248 Individual Protein CaM-kinase kinase alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3315 Individual Protein BR serine/threonine-protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3241 Individual Protein Serine/threonine-protein kinase NEK9 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3243 Individual Protein myosin light chain kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3326 Individual Protein Mitogen-activated protein kinase kinase kinase 9 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3337 Individual Protein Serine/threonine-protein kinase DCLK3 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3435 Individual Protein Serine/threonine-protein kinase pknB Mycobacterium tuberculosis Kd > 10000.0 nM PMID[532375]
NPT3321 Individual Protein PITSLRE serine/threonine-protein kinase CDC2L1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2626 Individual Protein Myosin light chain kinase, smooth muscle Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3350 Individual Protein Tyrosine-protein kinase Srms Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3436 Individual Protein Serine/threonine-protein kinase 35 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3114 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 1A Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3284 Individual Protein Serine/threonine-protein kinase NEK7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3258 Individual Protein Mixed lineage kinase 7 Homo sapiens Kd = 4400.0 nM PMID[532375]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 12.0 nM PMID[532375]
NPT3363 Individual Protein Mitogen-activated protein kinase 15 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Kd = 37.0 nM PMID[532375]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Kd = 130.0 nM PMID[532375]
NPT3437 Individual Protein Serine/threonine-protein kinase PFTAIRE-2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3438 Individual Protein G protein-coupled receptor kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3439 Individual Protein Homeodomain-interacting protein kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3440 Individual Protein Dual specificity mitogen-activated protein kinase kinase 5 Homo sapiens Kd = 1400.0 nM PMID[532375]
NPT3441 Individual Protein Dual specificity mitogen-activated protein kinase kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3265 Individual Protein Casein kinase I isoform alpha-like Homo sapiens Kd = 1700.0 nM PMID[532375]
NPT3442 Individual Protein Mitogen-activated protein kinase kinase kinase 7 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3316 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 4 Homo sapiens Kd = 3700.0 nM PMID[532375]
NPT3443 Individual Protein Serine/threonine-protein kinase Nek11 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3444 Individual Protein Homeodomain-interacting protein kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT14 Individual Protein Tyrosine-protein kinase FYN Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3445 Individual Protein Serine/threonine-protein kinase NIM1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1436 Individual Protein Focal adhesion kinase 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1674 Individual Protein CaM kinase II alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3263 Individual Protein Protein tyrosine kinase 2 beta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3349 Individual Protein Serine/threonine-protein kinase SIK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3257 Individual Protein Serine/threonine-protein kinase 32C Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3302 Individual Protein Ankyrin repeat and protein kinase domain-containing protein 1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3219 Individual Protein Ephrin type-A receptor 5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3446 Individual Protein Myosin light chain kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3249 Individual Protein Tyrosine- and threonine-specific cdc2-inhibitory kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3447 Individual Protein G protein-coupled receptor kinase 4 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3448 Individual Protein Leucine-rich repeat serine/threonine-protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3341 Individual Protein Serine/threonine-protein kinase Nek5 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3309 Individual Protein Leukocyte tyrosine kinase receptor Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3259 Individual Protein Tyrosine-protein kinase ZAP-70 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT1656 Individual Protein Protein kinase N1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3449 Individual Protein Wee1-like protein kinase 2 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3450 Individual Protein Putative uncharacterized serine/threonine-protein kinase SgK110 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3451 Individual Protein Dual serine/threonine and tyrosine protein kinase Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT3452 Individual Protein Calcium-dependent protein kinase 1 Plasmodium falciparum (isolate 3D7) Kd = 850.0 nM PMID[532375]
NPT3453 Individual Protein Cell division control protein 2 homolog Plasmodium falciparum (isolate 3D7) Kd > 10000.0 nM PMID[532375]
NPT216 Individual Protein Adenosine A1 receptor Homo sapiens IC50 = 2950.0 nM PMID[532376]
NPT216 Individual Protein Adenosine A1 receptor Homo sapiens Ki = 1721.0 nM PMID[532376]
NPT217 Individual Protein Adenosine A2a receptor Homo sapiens IC50 = 6068.0 nM PMID[532376]
NPT217 Individual Protein Adenosine A2a receptor Homo sapiens Ki = 3407.0 nM PMID[532376]
NPT208 Individual Protein Cytochrome P450 1A2 Homo sapiens IC50 = 2000.0 nM PMID[532376]
NPT213 Individual Protein Cytochrome P450 2C19 Homo sapiens IC50 = 800.0 nM PMID[532376]
NPT212 Individual Protein Cytochrome P450 2C9 Homo sapiens IC50 = 1000.0 nM PMID[532376]
NPT110 Individual Protein Cytochrome P450 2D6 Homo sapiens IC50 = 2000.0 nM PMID[532376]
NPT262 Individual Protein Muscarinic acetylcholine receptor M1 Homo sapiens IC50 = 10666.0 nM PMID[532376]
NPT262 Individual Protein Muscarinic acetylcholine receptor M1 Homo sapiens Ki = 2569.0 nM PMID[532376]
NPT273 Individual Protein Phosphodiesterase 5A Homo sapiens IC50 = 11476.0 nM PMID[532376]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 159.0 nM PMID[532376]
NPT286 Individual Protein Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50 = 18896.0 nM PMID[532376]
NPT293 Individual Protein Serotonin 4 (5-HT4) receptor Cavia porcellus IC50 = 10553.0 nM PMID[532376]
NPT293 Individual Protein Serotonin 4 (5-HT4) receptor Cavia porcellus Ki = 1759.0 nM PMID[532376]
NPT300 Individual Protein Thromboxane-A synthase Homo sapiens IC50 = 494.0 nM PMID[532376]
NPT3275 Individual Protein Inhibitor of nuclear factor kappa B kinase epsilon subunit Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3358 Individual Protein Serine/threonine-protein kinase PLK3 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3329 Individual Protein Serine/threonine-protein kinase MRCK-A Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Ki = 25.12 nM PMID[532379]
NPT3327 Individual Protein Mitogen-activated protein kinase kinase kinase 10 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1674 Individual Protein CaM kinase II alpha Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3390 Individual Protein Macrophage-stimulating protein receptor Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT3417 Individual Protein Serine/threonine-protein kinase TBK1 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1661 Individual Protein ALK tyrosine kinase receptor Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1449 Individual Protein Tyrosine-protein kinase SYK Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3318 Individual Protein MAP/microtubule affinity-regulating kinase 4 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT1659 Individual Protein Tyrosine-protein kinase receptor UFO Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3246 Individual Protein Tyrosine-protein kinase JAK2 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT2546 Individual Protein Serine/threonine-protein kinase AKT3 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT1702 Individual Protein Serine/threonine-protein kinase PLK4 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1344 Individual Protein Serine/threonine-protein kinase EEF2K Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3267 Individual Protein Macrophage colony stimulating factor receptor Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3309 Individual Protein Leukocyte tyrosine kinase receptor Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3271 Individual Protein NT-3 growth factor receptor Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3388 Individual Protein Tyrosine-protein kinase CTK Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3455 Individual Protein Protein kinase C zeta Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3370 Individual Protein Tyrosine-protein kinase receptor RET Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT3315 Individual Protein BR serine/threonine-protein kinase 1 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3222 Individual Protein AMP-activated protein kinase, alpha-1 subunit Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1713 Individual Protein PDZ-binding kinase Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT1690 Individual Protein Dual specificity mitogen-activated protein kinase kinase 2 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Ki = 19.95 nM PMID[532379]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Ki = 251.19 nM PMID[532379]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3368 Individual Protein cGMP-dependent protein kinase 2 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3365 Individual Protein Serine/threonine-protein kinase D2 Homo sapiens Ki = 6309.57 nM PMID[532379]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3316 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 4 Homo sapiens Ki = 398.11 nM PMID[532379]
NPT3223 Individual Protein Phosphorylase kinase gamma subunit 2 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3114 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 1A Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1678 Individual Protein CaM-kinase kinase beta Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3274 Individual Protein Dual specificity tyrosine-phosphorylation-regulated kinase 1B Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3448 Individual Protein Leucine-rich repeat serine/threonine-protein kinase 2 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3242 Individual Protein LIM domain kinase 1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3456 Individual Protein Serine/threonine-protein kinase Sgk2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3280 Individual Protein Serine/threonine-protein kinase c-TAK1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3350 Individual Protein Tyrosine-protein kinase Srms Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT1478 Individual Protein Vascular endothelial growth factor receptor 2 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3258 Individual Protein Mixed lineage kinase 7 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3245 Individual Protein Tyrosine kinase non-receptor protein 2 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3262 Individual Protein Serine/threonine-protein kinase PRKX Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1371 Individual Protein Cyclin-dependent kinase 2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1432 Individual Protein Serine/threonine-protein kinase Aurora-A Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT2575 Individual Protein Platelet-derived growth factor receptor beta Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3457 Individual Protein G protein-coupled receptor kinase 5 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Ki = 5011.87 nM PMID[532379]
NPT1598 Individual Protein Casein kinase II alpha Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3111 Individual Protein Tyrosine-protein kinase Lyn Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3431 Individual Protein Serine/threonine-protein kinase TAO1 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Ki = 39.81 nM PMID[532379]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3239 Individual Protein Nerve growth factor receptor Trk-A Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3290 Individual Protein Serine/threonine-protein kinase SIK2 Homo sapiens Ki = 1000.0 nM PMID[532379]
NPT1436 Individual Protein Focal adhesion kinase 1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1480 Individual Protein Fibroblast growth factor receptor 1 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3373 Individual Protein Proto-oncogene tyrosine-protein kinase ROS Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1437 Individual Protein Tyrosine-protein kinase FES Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Ki = 199.53 nM PMID[532379]
NPT3276 Individual Protein Tyrosine-protein kinase TYK2 Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1650 Individual Protein Tyrosine-protein kinase receptor FLT3 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT3240 Individual Protein Cyclin-dependent kinase 5 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT3381 Individual Protein Misshapen-like kinase 1 Homo sapiens Ki = 2511.89 nM PMID[532379]
NPT3277 Individual Protein Tyrosine-protein kinase receptor TYRO3 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3386 Individual Protein Interleukin-1 receptor-associated kinase 1 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3312 Individual Protein Tyrosine-protein kinase BLK Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Ki > 1258.93 nM PMID[532379]
NPT3406 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 2 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3396 Individual Protein Serine/threonine-protein kinase Nek4 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Ki = 1258.93 nM PMID[532379]
NPT3168 Individual Protein Casein kinase I alpha Homo sapiens Ki = 316.23 nM PMID[532379]
NPT1439 Individual Protein Tyrosine-protein kinase ITK/TSK Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT2574 Individual Protein Insulin receptor Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT286 Individual Protein Receptor protein-tyrosine kinase erbB-2 Homo sapiens Ki > 1258.93 nM PMID[532379]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT3225 Individual Protein Ephrin type-A receptor 2 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3366 Individual Protein Protein kinase C nu Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1680 Individual Protein Serine/threonine-protein kinase Chk2 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3458 Individual Protein Cell division cycle 7-related protein kinase Homo sapiens Ki > 1258.93 nM PMID[532379]
NPT3299 Individual Protein Testis-specific serine/threonine-protein kinase 1 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3263 Individual Protein Protein tyrosine kinase 2 beta Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3287 Individual Protein Activin receptor type-1 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3374 Individual Protein Ribosomal protein S6 kinase alpha 4 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3120 Individual Protein Serine/threonine-protein kinase PAK 1 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT3460 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 3 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3459 Individual Protein Dual specificity tyrosine-phosphorylation-regulated kinase 4 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1440 Individual Protein Tyrosine-protein kinase JAK3 Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3461 Individual Protein MAP kinase-activated protein kinase 3 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT3394 Individual Protein Protein kinase C iota Homo sapiens Ki > 5011.87 nM PMID[532379]
NPT3020 Individual Protein Platelet-derived growth factor receptor alpha Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT3462 Individual Protein Testis-specific serine/threonine-protein kinase 2 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT3432 Individual Protein Homeodomain-interacting protein kinase 2 Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3235 Individual Protein MAP/microtubule affinity-regulating kinase 2 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT2573 Individual Protein Vascular endothelial growth factor receptor 3 Homo sapiens Ki = 6309.57 nM PMID[532379]
NPT3439 Individual Protein Homeodomain-interacting protein kinase 4 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3324 Individual Protein Cell division protein kinase 8 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3346 Individual Protein Cyclin-dependent kinase 7 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1423 Individual Protein Cyclin-dependent kinase 1 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Ki = 1584.89 nM PMID[532379]
NPT592 Individual Protein Rho-associated protein kinase 1 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3347 Individual Protein Cyclin-dependent kinase 9 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT3425 Individual Protein Interleukin-1 receptor-associated kinase 4 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT3244 Individual Protein Tyrosine-protein kinase FER Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Ki > 1584.89 nM PMID[532379]
NPT301 Individual Protein Vascular endothelial growth factor receptor 1 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT1706 Individual Protein Serine/threonine-protein kinase 2 Homo sapiens Ki = 1995.26 nM PMID[532379]
NPT3270 Individual Protein Neurotrophic tyrosine kinase receptor type 2 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT3109 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 5 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT3335 Individual Protein Serine/threonine-protein kinase DCLK1 Homo sapiens Ki > 10000.0 nM PMID[532379]
NPT3227 Individual Protein Fibroblast growth factor receptor 3 Homo sapiens Ki > 1995.26 nM PMID[532379]
NPT1435 Individual Protein Receptor protein-tyrosine kinase erbB-4 Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT3231 Individual Protein Dual specificity protein kinase CLK4 Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT14 Individual Protein Tyrosine-protein kinase FYN Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 100.0 nM PMID[532380]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens IC50 = 430.0 nM PMID[532380]
NPT116 Cell Line HL-60 Homo sapiens Inhibition = 22.4 % PMID[532382]
NPT116 Cell Line HL-60 Homo sapiens IC50 = 50500.0 nM PMID[532382]
NPT116 Cell Line HL-60 Homo sapiens Inhibition = 50.6 % PMID[532382]
NPT116 Cell Line HL-60 Homo sapiens IC50 = 52200.0 nM PMID[532382]
NPT116 Cell Line HL-60 Homo sapiens Activity = 0.0 % PMID[532382]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 40.0 nM PMID[532383]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 2000.0 nM PMID[532383]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 37.0 nM PMID[532384]
NPT3317 Individual Protein Serine/threonine-protein kinase MARK1 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3317 Individual Protein Serine/threonine-protein kinase MARK1 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3419 Individual Protein Serine/threonine-protein kinase SRPK3 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3284 Individual Protein Serine/threonine-protein kinase NEK7 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3214 Individual Protein Tyrosine-protein kinase ABL2 Homo sapiens Residual Activity = 55.0 % PMID[532385]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Residual Activity = 68.0 % PMID[532385]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Residual Activity = 11.0 % PMID[532385]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT1721 Individual Protein Death-associated protein kinase 1 Homo sapiens Residual Activity = 85.0 % PMID[532385]
NPT3218 Individual Protein Ephrin type-A receptor 4 Homo sapiens Residual Activity = 80.0 % PMID[532385]
NPT3219 Individual Protein Ephrin type-A receptor 5 Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT3227 Individual Protein Fibroblast growth factor receptor 3 Homo sapiens Residual Activity = 99.0 % PMID[532385]
NPT14 Individual Protein Tyrosine-protein kinase FYN Homo sapiens Residual Activity = 76.0 % PMID[532385]
NPT14 Individual Protein Tyrosine-protein kinase FYN Homo sapiens Residual Activity = 35.0 % PMID[532385]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Residual Activity = 61.0 % PMID[532385]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Residual Activity = 20.0 % PMID[532385]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens Residual Activity = 1.0 % PMID[532385]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT3419 Individual Protein Serine/threonine-protein kinase SRPK3 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT1711 Individual Protein Serine/threonine-protein kinase MST1 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3284 Individual Protein Serine/threonine-protein kinase NEK7 Homo sapiens Residual Activity = 116.0 % PMID[532385]
NPT3285 Individual Protein Serine/threonine protein kinase NLK Homo sapiens Residual Activity = 62.0 % PMID[532385]
NPT1432 Individual Protein Serine/threonine-protein kinase Aurora-A Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT1432 Individual Protein Serine/threonine-protein kinase Aurora-A Homo sapiens Residual Activity = 118.0 % PMID[532385]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens Residual Activity = 5.0 % PMID[532385]
NPT1721 Individual Protein Death-associated protein kinase 1 Homo sapiens Residual Activity = 84.0 % PMID[532385]
NPT3219 Individual Protein Ephrin type-A receptor 5 Homo sapiens Residual Activity = 48.0 % PMID[532385]
NPT3372 Individual Protein Fibroblast growth factor receptor 4 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3372 Individual Protein Fibroblast growth factor receptor 4 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT3406 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 2 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT1478 Individual Protein Vascular endothelial growth factor receptor 2 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT491 Individual Protein Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1711 Individual Protein Serine/threonine-protein kinase MST1 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3285 Individual Protein Serine/threonine protein kinase NLK Homo sapiens Residual Activity = 24.0 % PMID[532385]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3236 Individual Protein Death-associated protein kinase 2 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT3236 Individual Protein Death-associated protein kinase 2 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3211 Individual Protein Ephrin type-A receptor 7 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3211 Individual Protein Ephrin type-A receptor 7 Homo sapiens Residual Activity = 65.0 % PMID[532385]
NPT3244 Individual Protein Tyrosine-protein kinase FER Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT3406 Individual Protein Mitogen-activated protein kinase kinase kinase kinase 2 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3457 Individual Protein G protein-coupled receptor kinase 5 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT2574 Individual Protein Insulin receptor Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT1478 Individual Protein Vascular endothelial growth factor receptor 2 Homo sapiens Residual Activity = 60.0 % PMID[532385]
NPT3242 Individual Protein LIM domain kinase 1 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3282 Individual Protein Maternal embryonic leucine zipper kinase Homo sapiens Residual Activity = 84.0 % PMID[532385]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT3331 Individual Protein Serine/threonine-protein kinase MST2 Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT1442 Individual Protein Serine/threonine-protein kinase PAK 2 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT1442 Individual Protein Serine/threonine-protein kinase PAK 2 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT1433 Individual Protein Serine/threonine-protein kinase Aurora-B Homo sapiens Residual Activity = 80.0 % PMID[532385]
NPT3206 Individual Protein Serine/threonine-protein kinase Aurora-C Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT3273 Individual Protein Casein kinase II alpha (prime) Homo sapiens Residual Activity = 122.0 % PMID[532385]
NPT3336 Individual Protein Serine/threonine-protein kinase DCLK2 Homo sapiens Residual Activity = 132.0 % PMID[532385]
NPT3216 Individual Protein Ephrin type-A receptor 8 Homo sapiens Residual Activity = 91.0 % PMID[532385]
NPT3457 Individual Protein G protein-coupled receptor kinase 5 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT2574 Individual Protein Insulin receptor Homo sapiens Residual Activity = 129.0 % PMID[532385]
NPT2574 Individual Protein Insulin receptor Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3242 Individual Protein LIM domain kinase 1 Homo sapiens Residual Activity = 82.0 % PMID[532385]
NPT3381 Individual Protein Misshapen-like kinase 1 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT3381 Individual Protein Misshapen-like kinase 1 Homo sapiens Residual Activity = 63.0 % PMID[532385]
NPT3332 Individual Protein Serine/threonine-protein kinase 24 Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT3247 Individual Protein Serine/threonine-protein kinase PAK 3 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT3206 Individual Protein Serine/threonine-protein kinase Aurora-C Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3273 Individual Protein Casein kinase II alpha (prime) Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT3336 Individual Protein Serine/threonine-protein kinase DCLK2 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3303 Individual Protein Discoidin domain-containing receptor 2 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3216 Individual Protein Ephrin type-A receptor 8 Homo sapiens Residual Activity = 43.0 % PMID[532385]
NPT3212 Individual Protein Ephrin type-B receptor 1 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT4088 Individual Protein G protein-coupled receptor kinase 6 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT4088 Individual Protein G protein-coupled receptor kinase 6 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT2574 Individual Protein Insulin receptor Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT3279 Individual Protein Serine/threonine-protein kinase 11 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3279 Individual Protein Serine/threonine-protein kinase 11 Homo sapiens Residual Activity = 85.0 % PMID[532385]
NPT1691 Individual Protein Dual specificity mitogen-activated protein kinase kinase 6 Homo sapiens Residual Activity = 43.0 % PMID[532385]
NPT3332 Individual Protein Serine/threonine-protein kinase 24 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3320 Individual Protein Proto-oncogene tyrosine-protein kinase MER Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT3245 Individual Protein Tyrosine kinase non-receptor protein 2 Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT1659 Individual Protein Tyrosine-protein kinase receptor UFO Homo sapiens Residual Activity = 122.0 % PMID[532385]
NPT1659 Individual Protein Tyrosine-protein kinase receptor UFO Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3303 Individual Protein Discoidin domain-containing receptor 2 Homo sapiens Residual Activity = 46.0 % PMID[532385]
NPT3212 Individual Protein Ephrin type-B receptor 1 Homo sapiens Residual Activity = 56.0 % PMID[532385]
NPT3438 Individual Protein G protein-coupled receptor kinase 7 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3386 Individual Protein Interleukin-1 receptor-associated kinase 1 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3386 Individual Protein Interleukin-1 receptor-associated kinase 1 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT1707 Individual Protein Serine/threonine-protein kinase 10 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT1691 Individual Protein Dual specificity mitogen-activated protein kinase kinase 6 Homo sapiens Residual Activity = 3.0 % PMID[532385]
NPT3441 Individual Protein Dual specificity mitogen-activated protein kinase kinase 7 Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT3320 Individual Protein Proto-oncogene tyrosine-protein kinase MER Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3245 Individual Protein Tyrosine kinase non-receptor protein 2 Homo sapiens Residual Activity = 39.0 % PMID[532385]
NPT1661 Individual Protein ALK tyrosine kinase receptor Homo sapiens Residual Activity = 122.0 % PMID[532385]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Residual Activity = 59.0 % PMID[532385]
NPT1683 Individual Protein Dual specificity protein kinase CLK3 Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens Residual Activity = 122.0 % PMID[532385]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT2941 Individual Protein Ephrin type-B receptor 2 Homo sapiens Residual Activity = 61.0 % PMID[532385]
NPT3438 Individual Protein G protein-coupled receptor kinase 7 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3425 Individual Protein Interleukin-1 receptor-associated kinase 4 Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT1707 Individual Protein Serine/threonine-protein kinase 10 Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT3441 Individual Protein Dual specificity mitogen-activated protein kinase kinase 7 Homo sapiens Residual Activity = 68.0 % PMID[532385]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Residual Activity = 123.0 % PMID[532385]
NPT1337 Individual Protein Hepatocyte growth factor receptor Homo sapiens Residual Activity = 68.0 % PMID[532385]
NPT1661 Individual Protein ALK tyrosine kinase receptor Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT3293 Individual Protein Activin receptor type-1B Homo sapiens Residual Activity = 87.0 % PMID[532385]
NPT3215 Individual Protein Tyrosine-protein kinase BRK Homo sapiens Residual Activity = 7.0 % PMID[532385]
NPT3113 Individual Protein Tyrosine-protein kinase CSK Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Residual Activity = 123.0 % PMID[532385]
NPT3359 Individual Protein Ephrin type-B receptor 3 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT3244 Individual Protein Tyrosine-protein kinase FER Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3425 Individual Protein Interleukin-1 receptor-associated kinase 4 Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Residual Activity = 27.0 % PMID[532385]
NPT2626 Individual Protein Myosin light chain kinase, smooth muscle Homo sapiens Residual Activity = 118.0 % PMID[532385]
NPT2626 Individual Protein Myosin light chain kinase, smooth muscle Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3293 Individual Protein Activin receptor type-1B Homo sapiens Residual Activity = 23.0 % PMID[532385]
NPT3113 Individual Protein Tyrosine-protein kinase CSK Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3399 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 2 Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT3359 Individual Protein Ephrin type-B receptor 3 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT2572 Individual Protein Ephrin type-B receptor 4 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1437 Individual Protein Tyrosine-protein kinase FES Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT1437 Individual Protein Tyrosine-protein kinase FES Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Residual Activity = 34.0 % PMID[532385]
NPT3286 Individual Protein Insulin receptor-related protein Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3286 Individual Protein Insulin receptor-related protein Homo sapiens Residual Activity = 56.0 % PMID[532385]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Residual Activity = 91.0 % PMID[532385]
NPT13 Individual Protein Tyrosine-protein kinase LCK Homo sapiens Residual Activity = 32.0 % PMID[532385]
NPT3326 Individual Protein Mitogen-activated protein kinase kinase kinase 9 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3213 Individual Protein MAP kinase signal-integrating kinase 2 Homo sapiens Residual Activity = 87.0 % PMID[532385]
NPT3333 Individual Protein Muscle, skeletal receptor tyrosine protein kinase Homo sapiens Residual Activity = 143.0 % PMID[532385]
NPT3312 Individual Protein Tyrosine-protein kinase BLK Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3312 Individual Protein Tyrosine-protein kinase BLK Homo sapiens Residual Activity = 55.0 % PMID[532385]
NPT3232 Individual Protein CaM kinase I alpha Homo sapiens Residual Activity = 99.0 % PMID[532385]
NPT3399 Individual Protein Dual-specificity tyrosine-phosphorylation regulated kinase 2 Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT2572 Individual Protein Ephrin type-B receptor 4 Homo sapiens Residual Activity = 41.0 % PMID[532385]
NPT3112 Individual Protein Tyrosine-protein kinase FGR Homo sapiens Residual Activity = 87.0 % PMID[532385]
NPT3444 Individual Protein Homeodomain-interacting protein kinase 1 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT1439 Individual Protein Tyrosine-protein kinase ITK/TSK Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3111 Individual Protein Tyrosine-protein kinase Lyn Homo sapiens Residual Activity = 47.0 % PMID[532385]
NPT3326 Individual Protein Mitogen-activated protein kinase kinase kinase 9 Homo sapiens Residual Activity = 71.0 % PMID[532385]
NPT3329 Individual Protein Serine/threonine-protein kinase MRCK-A Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT3333 Individual Protein Muscle, skeletal receptor tyrosine protein kinase Homo sapiens Residual Activity = 95.0 % PMID[532385]
NPT2750 Individual Protein Tyrosine-protein kinase BMX Homo sapiens Residual Activity = 81.0 % PMID[532385]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1608 Individual Protein Serine/threonine-protein kinase Chk1 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Residual Activity = 1.0 % PMID[532385]
NPT285 Individual Protein Epidermal growth factor receptor erbB1 Homo sapiens Residual Activity = -1.0 % PMID[532385]
NPT1435 Individual Protein Receptor protein-tyrosine kinase erbB-4 Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT1435 Individual Protein Receptor protein-tyrosine kinase erbB-4 Homo sapiens Residual Activity = 82.0 % PMID[532385]
NPT3112 Individual Protein Tyrosine-protein kinase FGR Homo sapiens Residual Activity = 51.0 % PMID[532385]
NPT301 Individual Protein Vascular endothelial growth factor receptor 1 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3444 Individual Protein Homeodomain-interacting protein kinase 1 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT3432 Individual Protein Homeodomain-interacting protein kinase 2 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT1439 Individual Protein Tyrosine-protein kinase ITK/TSK Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT3246 Individual Protein Tyrosine-protein kinase JAK2 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT3111 Individual Protein Tyrosine-protein kinase Lyn Homo sapiens Residual Activity = 13.0 % PMID[532385]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Residual Activity = 124.0 % PMID[532385]
NPT3329 Individual Protein Serine/threonine-protein kinase MRCK-A Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT3443 Individual Protein Serine/threonine-protein kinase Nek11 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT3443 Individual Protein Serine/threonine-protein kinase Nek11 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT1660 Individual Protein NUAK family SNF1-like kinase 1 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT2750 Individual Protein Tyrosine-protein kinase BMX Homo sapiens Residual Activity = 36.0 % PMID[532385]
NPT3315 Individual Protein BR serine/threonine-protein kinase 1 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1680 Individual Protein Serine/threonine-protein kinase Chk2 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3354 Individual Protein Ephrin type-A receptor 1 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1436 Individual Protein Focal adhesion kinase 1 Homo sapiens Residual Activity = 125.0 % PMID[532385]
NPT301 Individual Protein Vascular endothelial growth factor receptor 1 Homo sapiens Residual Activity = 39.0 % PMID[532385]
NPT3432 Individual Protein Homeodomain-interacting protein kinase 2 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3246 Individual Protein Tyrosine-protein kinase JAK2 Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3330 Individual Protein Serine/threonine-protein kinase MRCK beta Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT1660 Individual Protein NUAK family SNF1-like kinase 1 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3315 Individual Protein BR serine/threonine-protein kinase 1 Homo sapiens Residual Activity = 91.0 % PMID[532385]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3354 Individual Protein Ephrin type-A receptor 1 Homo sapiens Residual Activity = 26.0 % PMID[532385]
NPT3225 Individual Protein Ephrin type-A receptor 2 Homo sapiens Residual Activity = 95.0 % PMID[532385]
NPT1436 Individual Protein Focal adhesion kinase 1 Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT1650 Individual Protein Tyrosine-protein kinase receptor FLT3 Homo sapiens Residual Activity = 91.0 % PMID[532385]
NPT1650 Individual Protein Tyrosine-protein kinase receptor FLT3 Homo sapiens Residual Activity = 82.0 % PMID[532385]
NPT3409 Individual Protein Homeodomain-interacting protein kinase 3 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3409 Individual Protein Homeodomain-interacting protein kinase 3 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT1440 Individual Protein Tyrosine-protein kinase JAK3 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1440 Individual Protein Tyrosine-protein kinase JAK3 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Residual Activity = 118.0 % PMID[532385]
NPT282 Individual Protein MAP kinase ERK2 Homo sapiens Residual Activity = 95.0 % PMID[532385]
NPT3330 Individual Protein Serine/threonine-protein kinase MRCK beta Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Residual Activity = 118.0 % PMID[532385]
NPT3391 Individual Protein Serine/threonine-protein kinase Nek3 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1431 Individual Protein Mitogen-activated protein kinase kinase kinase 5 Homo sapiens Residual Activity = 138.0 % PMID[532385]
NPT1431 Individual Protein Mitogen-activated protein kinase kinase kinase 5 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3344 Individual Protein BR serine/threonine-protein kinase 2 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3344 Individual Protein BR serine/threonine-protein kinase 2 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Residual Activity = 61.0 % PMID[532385]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT3225 Individual Protein Ephrin type-A receptor 2 Homo sapiens Residual Activity = 62.0 % PMID[532385]
NPT1480 Individual Protein Fibroblast growth factor receptor 1 Homo sapiens Residual Activity = 142.0 % PMID[532385]
NPT1480 Individual Protein Fibroblast growth factor receptor 1 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT2573 Individual Protein Vascular endothelial growth factor receptor 3 Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT4093 Individual Protein Serine/threonine-protein kinase haspin Homo sapiens Residual Activity = 88.0 % PMID[532385]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1613 Individual Protein Ribosomal protein S6 kinase alpha 5 Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Residual Activity = 120.0 % PMID[532385]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Residual Activity = 71.0 % PMID[532385]
NPT1677 Individual Protein CaM kinase IV Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT1677 Individual Protein CaM kinase IV Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT3217 Individual Protein Ephrin type-A receptor 3 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3217 Individual Protein Ephrin type-A receptor 3 Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT1481 Individual Protein Fibroblast growth factor receptor 2 Homo sapiens Residual Activity = 99.0 % PMID[532385]
NPT2573 Individual Protein Vascular endothelial growth factor receptor 3 Homo sapiens Residual Activity = 42.0 % PMID[532385]
NPT3267 Individual Protein Macrophage colony stimulating factor receptor Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT4093 Individual Protein Serine/threonine-protein kinase haspin Homo sapiens Residual Activity = 35.0 % PMID[532385]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT1426 Individual Protein c-Jun N-terminal kinase 1 Homo sapiens Residual Activity = 95.0 % PMID[532385]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Residual Activity = 74.0 % PMID[532385]
NPT1441 Individual Protein MAP kinase-activated protein kinase 2 Homo sapiens Residual Activity = 133.0 % PMID[532385]
NPT3461 Individual Protein MAP kinase-activated protein kinase 3 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT3374 Individual Protein Ribosomal protein S6 kinase alpha 4 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT3374 Individual Protein Ribosomal protein S6 kinase alpha 4 Homo sapiens Residual Activity = 81.0 % PMID[532385]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT2729 Individual Protein Tyrosine-protein kinase ABL Homo sapiens Residual Activity = 72.0 % PMID[532385]
NPT3214 Individual Protein Tyrosine-protein kinase ABL2 Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Residual Activity = 125.0 % PMID[532385]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Residual Activity = 138.0 % PMID[532385]
NPT3218 Individual Protein Ephrin type-A receptor 4 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT1481 Individual Protein Fibroblast growth factor receptor 2 Homo sapiens Residual Activity = 81.0 % PMID[532385]
NPT3227 Individual Protein Fibroblast growth factor receptor 3 Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT3267 Individual Protein Macrophage colony stimulating factor receptor Homo sapiens Residual Activity = 52.0 % PMID[532385]
NPT3205 Individual Protein Tyrosine-protein kinase HCK Homo sapiens Residual Activity = 52.0 % PMID[532385]
NPT1438 Individual Protein Insulin-like growth factor I receptor Homo sapiens Residual Activity = 122.0 % PMID[532385]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens Residual Activity = 30.0 % PMID[532385]
NPT3461 Individual Protein MAP kinase-activated protein kinase 3 Homo sapiens Residual Activity = 92.0 % PMID[532385]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3124 Individual Protein Protein kinase C eta Homo sapiens Residual Activity = 77.0 % PMID[532385]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT3277 Individual Protein Tyrosine-protein kinase receptor TYRO3 Homo sapiens Residual Activity = 95.0 % PMID[532385]
NPT3349 Individual Protein Serine/threonine-protein kinase SIK1 Homo sapiens Residual Activity = 132.0 % PMID[532385]
NPT3349 Individual Protein Serine/threonine-protein kinase SIK1 Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT3269 Individual Protein Serine/threonine-protein kinase tousled-like 2 Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT3269 Individual Protein Serine/threonine-protein kinase tousled-like 2 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT4094 Individual Protein Serine/threonine-protein kinase WNK3 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT4094 Individual Protein Serine/threonine-protein kinase WNK3 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Residual Activity = 71.0 % PMID[532385]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT3106 Individual Protein Ribosomal protein S6 kinase alpha 1 Homo sapiens Residual Activity = 80.0 % PMID[532385]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT3299 Individual Protein Testis-specific serine/threonine-protein kinase 1 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT1663 Individual Protein Tyrosine-protein kinase YES Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3394 Individual Protein Protein kinase C iota Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3394 Individual Protein Protein kinase C iota Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3291 Individual Protein Serine/threonine-protein kinase SRPK1 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3292 Individual Protein Serine/threonine-protein kinase SRPK2 Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT3299 Individual Protein Testis-specific serine/threonine-protein kinase 1 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3462 Individual Protein Testis-specific serine/threonine-protein kinase 2 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT1663 Individual Protein Tyrosine-protein kinase YES Homo sapiens Residual Activity = 45.0 % PMID[532385]
NPT3259 Individual Protein Tyrosine-protein kinase ZAP-70 Homo sapiens Residual Activity = 124.0 % PMID[532385]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT3364 Individual Protein Protein kinase C mu Homo sapiens Residual Activity = 123.0 % PMID[532385]
NPT3358 Individual Protein Serine/threonine-protein kinase PLK3 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT3234 Individual Protein Ribosomal protein S6 kinase alpha 2 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT3292 Individual Protein Serine/threonine-protein kinase SRPK2 Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT3462 Individual Protein Testis-specific serine/threonine-protein kinase 2 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3259 Individual Protein Tyrosine-protein kinase ZAP-70 Homo sapiens Residual Activity = 130.0 % PMID[532385]
NPT1430 Individual Protein Serine/threonine-protein kinase AKT2 Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT2546 Individual Protein Serine/threonine-protein kinase AKT3 Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT3364 Individual Protein Protein kinase C mu Homo sapiens Residual Activity = 66.0 % PMID[532385]
NPT3365 Individual Protein Serine/threonine-protein kinase D2 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3358 Individual Protein Serine/threonine-protein kinase PLK3 Homo sapiens Residual Activity = 92.0 % PMID[532385]
NPT3234 Individual Protein Ribosomal protein S6 kinase alpha 2 Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT3296 Individual Protein Serine/threonine-protein kinase 33 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT3296 Individual Protein Serine/threonine-protein kinase 33 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3351 Individual Protein Tyrosine-protein kinase TEC Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3351 Individual Protein Tyrosine-protein kinase TEC Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT3247 Individual Protein Serine/threonine-protein kinase PAK 3 Homo sapiens Residual Activity = 78.0 % PMID[532385]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT2546 Individual Protein Serine/threonine-protein kinase AKT3 Homo sapiens Residual Activity = 75.0 % PMID[532385]
NPT3365 Individual Protein Serine/threonine-protein kinase D2 Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT3262 Individual Protein Serine/threonine-protein kinase PRKX Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT3262 Individual Protein Serine/threonine-protein kinase PRKX Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT3254 Individual Protein Ribosomal protein S6 kinase alpha 6 Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT3414 Individual Protein Serine/threonine-protein kinase PLK2 Homo sapiens Residual Activity = 116.0 % PMID[532385]
NPT2576 Individual Protein Tyrosine-protein kinase TIE-2 Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens Residual Activity = 17.0 % PMID[532385]
NPT182 Individual Protein Protein kinase C alpha Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT182 Individual Protein Protein kinase C alpha Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Residual Activity = 99.0 % PMID[532385]
NPT3263 Individual Protein Protein tyrosine kinase 2 beta Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Residual Activity = 5.0 % PMID[532385]
NPT3414 Individual Protein Serine/threonine-protein kinase PLK2 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT1449 Individual Protein Tyrosine-protein kinase SYK Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT2576 Individual Protein Tyrosine-protein kinase TIE-2 Homo sapiens Residual Activity = 62.0 % PMID[532385]
NPT3239 Individual Protein Nerve growth factor receptor Trk-A Homo sapiens Residual Activity = 121.0 % PMID[532385]
NPT1424 Individual Protein Serine/threonine-protein kinase RAF Homo sapiens Residual Activity = 3.0 % PMID[532385]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Residual Activity = 125.0 % PMID[532385]
NPT3263 Individual Protein Protein tyrosine kinase 2 beta Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Residual Activity = 24.0 % PMID[532385]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Residual Activity = 2.0 % PMID[532385]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Residual Activity = 24.0 % PMID[532385]
NPT1449 Individual Protein Tyrosine-protein kinase SYK Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3239 Individual Protein Nerve growth factor receptor Trk-A Homo sapiens Residual Activity = 115.0 % PMID[532385]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT1479 Individual Protein Stem cell growth factor receptor Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3367 Individual Protein cGMP-dependent protein kinase 1 beta Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Residual Activity = 145.0 % PMID[532385]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Residual Activity = 21.0 % PMID[532385]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Residual Activity = 2.0 % PMID[532385]
NPT3442 Individual Protein Mitogen-activated protein kinase kinase kinase 7 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT3442 Individual Protein Mitogen-activated protein kinase kinase kinase 7 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3270 Individual Protein Neurotrophic tyrosine kinase receptor type 2 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT3270 Individual Protein Neurotrophic tyrosine kinase receptor type 2 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Residual Activity = 112.0 % PMID[532385]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3235 Individual Protein MAP/microtubule affinity-regulating kinase 2 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT1612 Individual Protein MAP kinase-activated protein kinase 5 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT592 Individual Protein Rho-associated protein kinase 1 Homo sapiens Residual Activity = 70.0 % PMID[532385]
NPT592 Individual Protein Rho-associated protein kinase 1 Homo sapiens Residual Activity = 74.0 % PMID[532385]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT1615 Individual Protein MAP kinase p38 gamma Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT3431 Individual Protein Serine/threonine-protein kinase TAO1 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3272 Individual Protein Tyrosine-protein kinase TXK Homo sapiens Residual Activity = 77.0 % PMID[532385]
NPT36 Individual Protein Tyrosine-protein kinase SRC Homo sapiens Residual Activity = 65.0 % PMID[532385]
NPT1344 Individual Protein Serine/threonine-protein kinase EEF2K Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3235 Individual Protein MAP/microtubule affinity-regulating kinase 2 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Residual Activity = 119.0 % PMID[532385]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3431 Individual Protein Serine/threonine-protein kinase TAO1 Homo sapiens Residual Activity = 77.0 % PMID[532385]
NPT3426 Individual Protein Serine/threonine-protein kinase TAO2 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3272 Individual Protein Tyrosine-protein kinase TXK Homo sapiens Residual Activity = 42.0 % PMID[532385]
NPT3422 Individual Protein Serine/threonine-protein kinase ULK2 Homo sapiens Residual Activity = 120.0 % PMID[532385]
NPT1344 Individual Protein Serine/threonine-protein kinase EEF2K Homo sapiens Residual Activity = 91.0 % PMID[532385]
NPT3454 Individual Protein PAS domain-containing serine/threonine-protein kinase Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT3357 Individual Protein Protein kinase N2 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Residual Activity = 71.0 % PMID[532385]
NPT3107 Individual Protein Rho-associated protein kinase 2 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT3370 Individual Protein Tyrosine-protein kinase receptor RET Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT1448 Individual Protein Serine/threonine-protein kinase Sgk1 Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT3426 Individual Protein Serine/threonine-protein kinase TAO2 Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT3422 Individual Protein Serine/threonine-protein kinase ULK2 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3020 Individual Protein Platelet-derived growth factor receptor alpha Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3204 Individual Protein Tyrosine-protein kinase FRK Homo sapiens Residual Activity = 17.0 % PMID[532385]
NPT3370 Individual Protein Tyrosine-protein kinase receptor RET Homo sapiens Residual Activity = 46.0 % PMID[532385]
NPT1448 Individual Protein Serine/threonine-protein kinase Sgk1 Homo sapiens Residual Activity = 124.0 % PMID[532385]
NPT3427 Individual Protein Serine/threonine-protein kinase TAO3 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3427 Individual Protein Serine/threonine-protein kinase TAO3 Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT3382 Individual Protein Serine/threonine-protein kinase ULK3 Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT3020 Individual Protein Platelet-derived growth factor receptor alpha Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3223 Individual Protein Phosphorylase kinase gamma subunit 2 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3223 Individual Protein Phosphorylase kinase gamma subunit 2 Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT3390 Individual Protein Macrophage-stimulating protein receptor Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT3390 Individual Protein Macrophage-stimulating protein receptor Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT3456 Individual Protein Serine/threonine-protein kinase Sgk2 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT3417 Individual Protein Serine/threonine-protein kinase TBK1 Homo sapiens Residual Activity = 124.0 % PMID[532385]
NPT1715 Individual Protein Serine/threonine-protein kinase VRK2 Homo sapiens Residual Activity = 114.0 % PMID[532385]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT2575 Individual Protein Platelet-derived growth factor receptor beta Homo sapiens Residual Activity = 120.0 % PMID[532385]
NPT3455 Individual Protein Protein kinase C zeta Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT3455 Individual Protein Protein kinase C zeta Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Residual Activity = 84.0 % PMID[532385]
NPT3373 Individual Protein Proto-oncogene tyrosine-protein kinase ROS Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT3456 Individual Protein Serine/threonine-protein kinase Sgk2 Homo sapiens Residual Activity = 81.0 % PMID[532385]
NPT3418 Individual Protein Serine/threonine-protein kinase Sgk3 Homo sapiens Residual Activity = 120.0 % PMID[532385]
NPT3417 Individual Protein Serine/threonine-protein kinase TBK1 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens Residual Activity = 130.0 % PMID[532385]
NPT1715 Individual Protein Serine/threonine-protein kinase VRK2 Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT4096 Individual Protein Serine/threonine-protein kinase WNK2 Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT1611 Individual Protein Ribosomal protein S6 kinase 1 Homo sapiens Residual Activity = 87.0 % PMID[532385]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT3124 Individual Protein Protein kinase C eta Homo sapiens Residual Activity = 79.0 % PMID[532385]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Residual Activity = 97.0 % PMID[532385]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Residual Activity = 125.0 % PMID[532385]
NPT3373 Individual Protein Proto-oncogene tyrosine-protein kinase ROS Homo sapiens Residual Activity = 110.0 % PMID[532385]
NPT3277 Individual Protein Tyrosine-protein kinase receptor TYRO3 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT3418 Individual Protein Serine/threonine-protein kinase Sgk3 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT3353 Individual Protein TGF-beta receptor type I Homo sapiens Residual Activity = 77.0 % PMID[532385]
NPT4096 Individual Protein Serine/threonine-protein kinase WNK2 Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 273.0 nM PMID[532386]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532386]
NPT927 Cell Line PBMC Homo sapiens Inhibition < 40.0 % PMID[532387]
NPT927 Cell Line PBMC Homo sapiens Inhibition = 80.0 % PMID[532387]
NPT927 Cell Line PBMC Homo sapiens IC50 > 10000.0 nM PMID[532387]
NPT927 Cell Line PBMC Homo sapiens IC50 = 340.0 nM PMID[532387]
NPT927 Cell Line PBMC Homo sapiens IC50 = 1000.0 nM PMID[532387]
NPT3464 Individual Protein Myelin transcription factor 1 Homo sapiens Activity < 5.0 % PMID[532391]
NPT50 Individual Protein Tyrosyl-DNA phosphodiesterase 1 Homo sapiens Potency n.a. 33498.3 nM PMID[532369]
NPT50 Individual Protein Tyrosyl-DNA phosphodiesterase 1 Homo sapiens Potency n.a. 14963.1 nM PMID[532368]
NPT50 Individual Protein Tyrosyl-DNA phosphodiesterase 1 Homo sapiens Potency n.a. 29855.4 nM PMID[532368]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 25.0 nM PMID[532393]
NPT116 Cell Line HL-60 Homo sapiens Inhibition = 68.1 % PMID[532394]
NPT116 Cell Line HL-60 Homo sapiens IC50 = 8600.0 nM PMID[532394]
NPT116 Cell Line HL-60 Homo sapiens Inhibition = 8.4 % PMID[532394]
NPT116 Cell Line HL-60 Homo sapiens IC50 = 52200.0 nM PMID[532394]
NPT116 Cell Line HL-60 Homo sapiens Activity = 0.0 % PMID[532394]
NPT1814 Individual Protein Glucagon receptor Homo sapiens IC50 = 37.07 nM PMID[532398]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 723.0 nM PMID[532399]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 48.0 nM PMID[532399]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 40.0 nM PMID[532400]
NPT1663 Individual Protein Tyrosine-protein kinase YES Homo sapiens Potency n.a. 10909.6 nM PMID[532368]
NPT49 Individual Protein DNA-(apurinic or apyrimidinic site) lyase Homo sapiens Potency n.a. 12589.3 nM PMID[532368]
NPT49 Individual Protein DNA-(apurinic or apyrimidinic site) lyase Homo sapiens Potency n.a. 39810.7 nM PMID[532370]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 19.0 nM PMID[532402]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 35.0 nM PMID[532403]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens IC50 = 105.0 nM PMID[532406]
NPT1699 Individual Protein 3-phosphoinositide dependent protein kinase-1 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1265 Individual Protein Serine/threonine-protein kinase PIM1 Homo sapiens Thermal melting change = -2.1 degrees C PMID[532343]
NPT1700 Individual Protein Serine/threonine-protein kinase PIM2 Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1701 Individual Protein Serine/threonine-protein kinase PIM3 Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1702 Individual Protein Serine/threonine-protein kinase PLK4 Homo sapiens Thermal melting change = 0.7 degrees C PMID[532343]
NPT1703 Individual Protein cAMP-dependent protein kinase alpha-catalytic subunit Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1704 Individual Protein Serine/threonine-protein kinase RIO2 Homo sapiens Thermal melting change = -0.2 degrees C PMID[532343]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Thermal melting change = 0.3 degrees C PMID[532343]
NPT1705 Individual Protein Ribosomal protein S6 kinase alpha 3 Homo sapiens Thermal melting change = -0.2 degrees C PMID[532343]
NPT1706 Individual Protein Serine/threonine-protein kinase 2 Homo sapiens Thermal melting change = 3.9 degrees C PMID[532343]
NPT1707 Individual Protein Serine/threonine-protein kinase 10 Homo sapiens Thermal melting change = 2.7 degrees C PMID[532343]
NPT1708 Individual Protein Serine/threonine-protein kinase 16 Homo sapiens Thermal melting change = 0.4 degrees C PMID[532343]
NPT1709 Individual Protein Serine/threonine-protein kinase 17A Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1710 Individual Protein Serine/threonine-protein kinase 38 Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT1693 Individual Protein Serine/threonine-protein kinase MST4 Homo sapiens Thermal melting change = -0.4 degrees C PMID[532343]
NPT1711 Individual Protein Serine/threonine-protein kinase MST1 Homo sapiens Thermal melting change = 1.0 degrees C PMID[532343]
NPT1712 Individual Protein TRAF2- and NCK-interacting kinase Homo sapiens Thermal melting change = 2.0 degrees C PMID[532343]
NPT1713 Individual Protein PDZ-binding kinase Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT1715 Individual Protein Serine/threonine-protein kinase VRK2 Homo sapiens Thermal melting change = 0.6 degrees C PMID[532343]
NPT1717 Individual Protein Serine/threonine-protein kinase 25 Homo sapiens Thermal melting change = 0.9 degrees C PMID[532343]
NPT1671 Individual Protein AMP-activated protein kinase, alpha-2 subunit Homo sapiens Thermal melting change = -0.9 degrees C PMID[532343]
NPT1672 Individual Protein CaM kinase I delta Homo sapiens Thermal melting change = -0.2 degrees C PMID[532343]
NPT1673 Individual Protein CaM kinase I gamma Homo sapiens Thermal melting change = -0.2 degrees C PMID[532343]
NPT1674 Individual Protein CaM kinase II alpha Homo sapiens Thermal melting change = 0.3 degrees C PMID[532343]
NPT1630 Individual Protein CaM kinase II beta Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1675 Individual Protein CaM kinase II delta Homo sapiens Thermal melting change = -0.3 degrees C PMID[532343]
NPT1676 Individual Protein CaM kinase II gamma Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1677 Individual Protein CaM kinase IV Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1678 Individual Protein CaM-kinase kinase beta Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1371 Individual Protein Cyclin-dependent kinase 2 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1571 Individual Protein Cyclin-dependent kinase 6 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1679 Individual Protein Cyclin-dependent kinase-like 1 Homo sapiens Thermal melting change = -0.4 degrees C PMID[532343]
NPT1680 Individual Protein Serine/threonine-protein kinase Chk2 Homo sapiens Thermal melting change = -0.5 degrees C PMID[532343]
NPT1681 Individual Protein Dual specificty protein kinase CLK1 Homo sapiens Thermal melting change = -0.3 degrees C PMID[532343]
NPT1682 Individual Protein Dual specificity protein kinase CLK2 Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT1683 Individual Protein Dual specificity protein kinase CLK3 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1684 Individual Protein Casein kinase I gamma 1 Homo sapiens Thermal melting change = 0.8 degrees C PMID[532343]
NPT1685 Individual Protein Casein kinase I gamma 2 Homo sapiens Thermal melting change = 0.7 degrees C PMID[532343]
NPT1686 Individual Protein Casein kinase I isoform gamma-3 Homo sapiens Thermal melting change = 0.4 degrees C PMID[532343]
NPT1687 Individual Protein Death-associated protein kinase 3 Homo sapiens Thermal melting change = -0.4 degrees C PMID[532343]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens Thermal melting change = 0.1 degrees C PMID[532343]
NPT591 Individual Protein Glycogen synthase kinase-3 beta Homo sapiens Thermal melting change = 3.5 degrees C PMID[532343]
NPT1689 Individual Protein Tyrosine-protein kinase JAK1 Homo sapiens Thermal melting change = 2.3 degrees C PMID[532343]
NPT1690 Individual Protein Dual specificity mitogen-activated protein kinase kinase 2 Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT1691 Individual Protein Dual specificity mitogen-activated protein kinase kinase 6 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1431 Individual Protein Mitogen-activated protein kinase kinase kinase 5 Homo sapiens Thermal melting change = 0.3 degrees C PMID[532343]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens Thermal melting change = 9.6 degrees C PMID[532343]
NPT281 Individual Protein MAP kinase ERK1 Homo sapiens Thermal melting change = 0.1 degrees C PMID[532343]
NPT1692 Individual Protein Mitogen-activated protein kinase 6 Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1693 Individual Protein Serine/threonine-protein kinase MST4 Homo sapiens Thermal melting change = -0.5 degrees C PMID[532343]
NPT1658 Individual Protein Serine/threonine-protein kinase NEK2 Homo sapiens Thermal melting change = 0.3 degrees C PMID[532343]
NPT1657 Individual Protein Serine/threonine-protein kinase NEK6 Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT1694 Individual Protein Serine/threonine-protein kinase OSR1 Homo sapiens Thermal melting change = -0.2 degrees C PMID[532343]
NPT1695 Individual Protein Serine/threonine-protein kinase PAK 4 Homo sapiens Thermal melting change = 0.1 degrees C PMID[532343]
NPT1696 Individual Protein Serine/threonine-protein kinase PAK7 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT1697 Individual Protein Serine/threonine-protein kinase PAK6 Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT1698 Individual Protein Serine/threonine-protein kinase PCTAIRE-1 Homo sapiens Thermal melting change = -0.8 degrees C PMID[532343]
NPT113 Cell Line RAW264.7 Mus musculus Inhibition = 53.0 % PMID[532407]
NPT6603 Individual Protein P2X purinoceptor 7 Rattus norvegicus IC50 > 30000.0 nM PMID[532408]
NPT2654 Individual Protein P2X purinoceptor 7 Homo sapiens IC50 = 5000.0 nM PMID[532408]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens T1/2 = 0.006667 hr PMID[532409]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens K = 0.0317 /s PMID[532409]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 10.0 nM PMID[532409]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 200.0 nM PMID[532409]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 251.19 nM PMID[532412]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 250.0 nM PMID[532412]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 = 6310.0 nM PMID[532412]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens Ratio IC50 = 25.0 n.a. PMID[532412]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 25.0 nM PMID[532413]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens IC50 = 12.0 nM PMID[532413]
NPT2816 Individual Protein Bromodomain-containing protein 4 Homo sapiens Delta Tm = 1.3 degrees C PMID[532413]
NPT1614 Individual Protein MAP kinase p38 delta Homo sapiens IC50 = 87600000.0 nM PMID[532414]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 21.7 nM PMID[532417]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens T1/2 = 0.0008889 hr PMID[532417]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens TIME = 0.001278 hr PMID[532417]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Kd = 2.18 10'-1/s PMID[532417]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Ka = 1.0 10'7/M.s PMID[532417]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens EC50 = 60.0 nM PMID[532422]
NPT1970 Cell Line THP-1 Homo sapiens IC50 = 20.0 nM PMID[532422]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 35.0 nM PMID[532424]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 41.0 nM PMID[532425]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 65.0 nM PMID[532425]
NPT2739 Individual Protein Tyrosinase Mus musculus IC50 = 34.0 nM PMID[532426]
NPT1616 Individual Protein MAP kinase p38 beta Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3266 Individual Protein Casein kinase I delta Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT1427 Individual Protein c-Jun N-terminal kinase 2 Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3207 Individual Protein c-Jun N-terminal kinase 3 Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT1712 Individual Protein TRAF2- and NCK-interacting kinase Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT1434 Individual Protein Serine/threonine-protein kinase B-raf Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3334 Individual Protein Citron Rho-interacting kinase Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3226 Individual Protein Casein kinase I epsilon Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT1688 Individual Protein Myotonin-protein kinase Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3221 Individual Protein Serine/threonine-protein kinase GAK Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3285 Individual Protein Serine/threonine protein kinase NLK Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT1447 Individual Protein Serine/threonine-protein kinase RIPK2 Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT3208 Individual Protein Serine/threonine-protein kinase 36 Homo sapiens IC50 < 1000.0 nM PMID[532432]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Delta Tm = 6.8 degrees C PMID[532434]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Tm = 56.8 degrees C PMID[532434]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens Activity = 75.0 % PMID[532434]
NPT2615 Cell Line HEK-293T Homo sapiens Cell Viability = 0.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 16.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 9.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 0.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 5.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 38.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 0.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 3.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 2.0 n.a. PMID[532435]
NPT1045 Cell Line U2OS Homo sapiens Cell Viability = 1.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 4.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 1.0 n.a. PMID[532435]
NPT4909 Cell Line Fibroblasts Cell Viability = 2.0 n.a. PMID[532435]
NPT283 Individual Protein MAP kinase p38 alpha Homo sapiens IC50 = 500.0 nM PMID[532436]
NPT27 Others Unspecified IC50 = 590.0 nM PMID[532298]
NPT27 Others Unspecified IC50 = 37.0 nM PMID[532298]
NPT605 Organism Homo sapiens Homo sapiens IC50 = 940.0 nM PMID[532298]
NPT605 Organism Homo sapiens Homo sapiens IC50 = 350.0 nM PMID[532298]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 72.0 nM PMID[532300]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 25.0 nM PMID[532302]
NPT321 Protein Family cAMP-dependent protein kinase (PKA) Homo sapiens Inhibition = 0.0 % PMID[532303]
NPT2 Others Unspecified Inhibition = 83.0 % PMID[532303]
NPT2 Others Unspecified Inhibition = 33.0 % PMID[532303]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 39.0 nM PMID[532306]
NPT4148 Protein Family Dual specificity mitogen-activated protein kinase kinase; MEK1/2 Homo sapiens IC50 = 61000.0 nM PMID[532306]
NPT321 Protein Family cAMP-dependent protein kinase (PKA) Homo sapiens IC50 = 50000.0 nM PMID[532306]
NPT316 Protein Family Protein kinase C (PKC) Homo sapiens IC50 = 75000.0 nM PMID[532306]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 1000.0 nM PMID[532306]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 290.0 nM PMID[532307]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 590.0 nM PMID[532307]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 37.0 nM PMID[532307]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 940.0 nM PMID[532307]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 350.0 nM PMID[532307]
NPT29 Organism Rattus norvegicus Rattus norvegicus ID50 = 80.0 mg kg-1 day-1 PMID[532308]
NPT29 Organism Rattus norvegicus Rattus norvegicus Inhibition = 74.0 % PMID[532308]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 83.0 nM PMID[532308]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 360.0 nM PMID[532310]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 940.0 nM PMID[532310]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 350.0 nM PMID[532310]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 590.0 nM PMID[532310]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 37.0 nM PMID[532310]
NPT32 Organism Mus musculus Mus musculus Inhibition = 80.0 % PMID[532311]
NPT32 Organism Mus musculus Mus musculus Inhibition = -1.4 % PMID[532311]
NPT32 Organism Mus musculus Mus musculus Inhibition < 65.4 % PMID[532311]
NPT32 Organism Mus musculus Mus musculus Activity = 1.0 n.a. PMID[532311]
NPT32 Organism Mus musculus Mus musculus IC = 0.63 n.a. PMID[532311]
NPT32 Organism Mus musculus Mus musculus IO = 0.25 n.a. PMID[532311]
NPT32 Organism Mus musculus Mus musculus Activity = 38.0 ng ml-1 PMID[532311]
NPT32 Organism Mus musculus Mus musculus Activity = 13.0 ng ml-1 PMID[532311]
NPT35 Others n.a. CLogP = 3.6 n.a. PMID[532312]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 42.0 nM PMID[532313]
NPT32 Organism Mus musculus Mus musculus Change = -83.0 % PMID[532313]
NPT207 Protein Family MAP kinase p38 Homo sapiens Kd = 10.0 nM PMID[532314]
NPT207 Protein Family MAP kinase p38 Homo sapiens EC50 = 60.0 nM PMID[532314]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 42.0 nM PMID[532316]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 48.0 nM PMID[532316]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 50.0 nM PMID[532317]
NPT2 Others Unspecified IC50 > 400000.0 nM PMID[532317]
NPT2 Others Unspecified IC50 = 37.0 nM PMID[532318]
NPT27 Others Unspecified IC50 = 190.0 nM PMID[532322]
NPT605 Organism Homo sapiens Homo sapiens IC50 = 4200.0 nM PMID[532322]
NPT32 Organism Mus musculus Mus musculus Inhibition = 50.0 % PMID[532322]
NPT32 Organism Mus musculus Mus musculus Inhibition = 47.0 % PMID[532322]
NPT32 Organism Mus musculus Mus musculus Inhibition = 0.0 % PMID[532322]
NPT605 Organism Homo sapiens Homo sapiens IC50 = 2000.0 nM PMID[532323]
NPT2 Others Unspecified Kd = 6800.0 nM PMID[532324]
NPT2 Others Unspecified IC50 = 7800.0 nM PMID[532324]
NPT2 Others Unspecified IC50 = 290.0 nM PMID[532328]
NPT2 Others Unspecified IC50 = 70.0 nM PMID[532328]
NPT2 Others Unspecified IC50 = 136.0 nM PMID[532329]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 136.0 nM PMID[532332]
NPT1308 Tissue Blood Homo sapiens IC50 = 2640.0 nM PMID[532335]
NPT1308 Tissue Blood Homo sapiens IC50 = 1117.0 nM PMID[532335]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 56.0 nM PMID[532336]
NPT2 Others Unspecified IC50 = 42.0 nM PMID[532337]
NPT2 Others Unspecified IC50 = 34.0 nM PMID[532343]
NPT2 Others Unspecified IC50 = 600.0 nM PMID[532343]
NPT20967 CELL-LINE Platelet n.a. IC50 = 200.0 nM PMID[532343]
NPT1308 Tissue Blood Homo sapiens IC50 = 2300.0 nM PMID[532347]
NPT1308 Tissue Blood Homo sapiens IC50 = 1980.0 nM PMID[532347]
NPT2 Others Unspecified Inhibition = 0.0 % PMID[532347]
NPT2 Others Unspecified Inhibition = 4.0 % PMID[532347]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Inhibition = 38.0 % PMID[532347]
NPT2 Others Unspecified IC50 = 100.0 nM PMID[532348]
NPT2255 Organism Toxoplasma gondii RH Toxoplasma gondii RH IC50 = 8500.0 nM PMID[532350]
NPT486 Organism Toxoplasma gondii Toxoplasma gondii IC50 = 2500.0 nM PMID[532350]
NPT2255 Organism Toxoplasma gondii RH Toxoplasma gondii RH Activity = 30.0 day PMID[532350]
NPT1308 Tissue Blood Homo sapiens IC50 = 6400.0 nM PMID[532351]
NPT32 Organism Mus musculus Mus musculus ID50 = 27.9 mg.kg-1 PMID[532351]
NPT2 Others Unspecified Activity = 104.0 % PMID[532353]
NPT676 Individual Protein Glycogen synthase kinase-3 alpha Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Activity = 89.0 % PMID[532353]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT2 Others Unspecified Activity = 80.0 % PMID[532353]
NPT3814 Protein Complex Cyclin-dependent kinase 2/cyclin A Homo sapiens Activity = 104.0 % PMID[532353]
NPT1609 Protein Complex Casein kinase II Homo sapiens Activity = 98.0 % PMID[532353]
NPT833 Individual Protein Tyrosine-protein kinase BTK Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT981 Individual Protein Inhibitor of nuclear factor kappa B kinase beta subunit Homo sapiens Activity = 95.0 % PMID[532353]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT881 Individual Protein Protein kinase C delta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT761 Individual Protein Protein kinase C epsilon Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT887 Individual Protein Protein kinase C theta Homo sapiens Kd > 10000.0 nM PMID[532352]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Activity = 97.0 % PMID[532353]
NPT1308 Tissue Blood Homo sapiens IC50 = 1760.0 nM PMID[532360]
NPT2 Others Unspecified Inhibition = 104.0 % PMID[532364]
NPT1609 Protein Complex Casein kinase II Homo sapiens Inhibition = 97.0 % PMID[532364]
NPT2 Others Unspecified Inhibition = 96.0 % PMID[532364]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Inhibition = 62.0 % PMID[532364]
NPT2 Others Unspecified Inhibition = 83.0 % PMID[532364]
NPT2 Others Unspecified Inhibition = 99.0 % PMID[532364]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. Inhibition = 84.3 % PMID[532366]
NPT197 Protein-Protein Interaction Menin/Histone-lysine N-methyltransferase MLL Homo sapiens Potency = 39810.7 nM PMID[532368]
NPT94 Individual Protein Aldehyde dehydrogenase 1A1 Homo sapiens Potency = 35481.3 nM PMID[532369]
NPT94 Individual Protein Aldehyde dehydrogenase 1A1 Homo sapiens Potency = 28183.8 nM PMID[532368]
NPT94 Individual Protein Aldehyde dehydrogenase 1A1 Homo sapiens Potency = 28183.8 nM PMID[532370]
NPT792 Individual Protein Arachidonate 15-lipoxygenase Homo sapiens Potency = 19952.6 nM PMID[532368]
NPT2 Others Unspecified Potency = 7079.5 nM PMID[532368]
NPT2 Others Unspecified Potency = 12589.3 nM PMID[532369]
NPT1308 Tissue Blood Homo sapiens IC50 = 190.0 nM PMID[532374]
NPT698 Individual Protein Regulator of G-protein signaling 4 Homo sapiens Potency n.a. 2993.5 nM PMID[532370]
NPT833 Individual Protein Tyrosine-protein kinase BTK Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT982 Individual Protein Inhibitor of nuclear factor kappa B kinase alpha subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT981 Individual Protein Inhibitor of nuclear factor kappa B kinase beta subunit Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT940 Individual Protein Serine/threonine-protein kinase mTOR Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT761 Individual Protein Protein kinase C epsilon Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT881 Individual Protein Protein kinase C delta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT887 Individual Protein Protein kinase C theta Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT676 Individual Protein Glycogen synthase kinase-3 alpha Homo sapiens Kd > 10000.0 nM PMID[532375]
NPT2 Others Unspecified IC50 = 5923.0 nM PMID[532376]
NPT2 Others Unspecified Ki = 2026.0 nM PMID[532376]
NPT2 Others Unspecified IC50 = 11590.0 nM PMID[532376]
NPT207 Protein Family MAP kinase p38 Homo sapiens Inhibition = 62.0 % PMID[532377]
NPT2 Others Unspecified Inhibition = 73.0 % PMID[532377]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 7240.0 nM PMID[532378]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 3530.0 nM PMID[532378]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 5020.0 nM PMID[532378]
NPT981 Individual Protein Inhibitor of nuclear factor kappa B kinase beta subunit Homo sapiens Ki > 3162.28 nM PMID[532379]
NPT887 Individual Protein Protein kinase C theta Homo sapiens Ki > 2511.89 nM PMID[532379]
NPT881 Individual Protein Protein kinase C delta Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT982 Individual Protein Inhibitor of nuclear factor kappa B kinase alpha subunit Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT676 Individual Protein Glycogen synthase kinase-3 alpha Homo sapiens Ki > 3981.07 nM PMID[532379]
NPT880 Individual Protein Protein kinase C gamma Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT833 Individual Protein Tyrosine-protein kinase BTK Homo sapiens Ki > 6309.57 nM PMID[532379]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Ki > 7943.28 nM PMID[532379]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 220.0 nM PMID[532381]
NPT2 Others Unspecified Potency n.a. 4685.9 nM PMID[532369]
NPT2 Others Unspecified Potency n.a. 2.6 nM PMID[532369]
NPT2 Others Unspecified Potency n.a. 2093.1 nM PMID[532369]
NPT3814 Protein Complex Cyclin-dependent kinase 2/cyclin A Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT982 Individual Protein Inhibitor of nuclear factor kappa B kinase alpha subunit Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT2544 Protein Complex Cyclin-dependent kinase 2/cyclin E Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT2544 Protein Complex Cyclin-dependent kinase 2/cyclin E Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT981 Individual Protein Inhibitor of nuclear factor kappa B kinase beta subunit Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT981 Individual Protein Inhibitor of nuclear factor kappa B kinase beta subunit Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT4087 Protein Complex CDK3/cyclin E Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT1609 Protein Complex Casein kinase II Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT1609 Protein Complex Casein kinase II Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT4087 Protein Complex CDK3/cyclin E Homo sapiens Residual Activity = 93.0 % PMID[532385]
NPT1509 Protein Complex Cyclin-dependent kinase 5/CDK5 activator 1 Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT1509 Protein Complex Cyclin-dependent kinase 5/CDK5 activator 1 Homo sapiens Residual Activity = 121.0 % PMID[532385]
NPT1509 Protein Complex Cyclin-dependent kinase 5/CDK5 activator 1 Homo sapiens Residual Activity = 120.0 % PMID[532385]
NPT1509 Protein Complex Cyclin-dependent kinase 5/CDK5 activator 1 Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT4089 Protein Complex CDK6/cyclin D3 Homo sapiens Residual Activity = 116.0 % PMID[532385]
NPT4089 Protein Complex CDK6/cyclin D3 Homo sapiens Residual Activity = 111.0 % PMID[532385]
NPT676 Individual Protein Glycogen synthase kinase-3 alpha Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT833 Individual Protein Tyrosine-protein kinase BTK Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT4090 Protein Complex Cyclin-dependent kinase 7/ cyclin H Homo sapiens Residual Activity = 118.0 % PMID[532385]
NPT676 Individual Protein Glycogen synthase kinase-3 alpha Homo sapiens Residual Activity = 49.0 % PMID[532385]
NPT833 Individual Protein Tyrosine-protein kinase BTK Homo sapiens Residual Activity = 73.0 % PMID[532385]
NPT4090 Protein Complex Cyclin-dependent kinase 7/ cyclin H Homo sapiens Residual Activity = 100.0 % PMID[532385]
NPT4092 Protein Complex CDK9/cyclin T1 Homo sapiens Residual Activity = 98.0 % PMID[532385]
NPT4091 Protein Complex AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 Homo sapiens Residual Activity = 109.0 % PMID[532385]
NPT4091 Protein Complex AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 Homo sapiens Residual Activity = 94.0 % PMID[532385]
NPT4092 Protein Complex CDK9/cyclin T1 Homo sapiens Residual Activity = 108.0 % PMID[532385]
NPT1767 Protein Complex AMP-activated protein kinase, AMPK Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT1767 Protein Complex AMP-activated protein kinase, AMPK Homo sapiens Residual Activity = 90.0 % PMID[532385]
NPT1561 Protein Complex Cyclin-dependent kinase 1/cyclin B1 Homo sapiens Residual Activity = 107.0 % PMID[532385]
NPT1561 Protein Complex Cyclin-dependent kinase 1/cyclin B1 Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT3814 Protein Complex Cyclin-dependent kinase 2/cyclin A Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT982 Individual Protein Inhibitor of nuclear factor kappa B kinase alpha subunit Homo sapiens Residual Activity = 113.0 % PMID[532385]
NPT887 Individual Protein Protein kinase C theta Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT887 Individual Protein Protein kinase C theta Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Residual Activity = 102.0 % PMID[532385]
NPT728 Individual Protein Serine/threonine-protein kinase AKT Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Residual Activity = 117.0 % PMID[532385]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Residual Activity = 99.0 % PMID[532385]
NPT760 Individual Protein Protein kinase C beta Homo sapiens Residual Activity = 101.0 % PMID[532385]
NPT760 Individual Protein Protein kinase C beta Homo sapiens Residual Activity = 70.0 % PMID[532385]
NPT760 Individual Protein Protein kinase C beta Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT760 Individual Protein Protein kinase C beta Homo sapiens Residual Activity = 75.0 % PMID[532385]
NPT880 Individual Protein Protein kinase C gamma Homo sapiens Residual Activity = 104.0 % PMID[532385]
NPT880 Individual Protein Protein kinase C gamma Homo sapiens Residual Activity = 103.0 % PMID[532385]
NPT881 Individual Protein Protein kinase C delta Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT940 Individual Protein Serine/threonine-protein kinase mTOR Homo sapiens Residual Activity = 106.0 % PMID[532385]
NPT940 Individual Protein Serine/threonine-protein kinase mTOR Homo sapiens Residual Activity = 89.0 % PMID[532385]
NPT761 Individual Protein Protein kinase C epsilon Homo sapiens Residual Activity = 125.0 % PMID[532385]
NPT940 Individual Protein Serine/threonine-protein kinase mTOR Homo sapiens Residual Activity = 86.0 % PMID[532385]
NPT761 Individual Protein Protein kinase C epsilon Homo sapiens Residual Activity = 105.0 % PMID[532385]
NPT940 Individual Protein Serine/threonine-protein kinase mTOR Homo sapiens Residual Activity = 96.0 % PMID[532385]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 7370.0 nM PMID[532388]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 3560.0 nM PMID[532388]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 5670.0 nM PMID[532388]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 5000.0 nM PMID[532389]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 7530.0 nM PMID[532390]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 5210.0 nM PMID[532390]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 3450.0 nM PMID[532390]
NPT2 Others Unspecified Inhibition = 70.0 % PMID[532392]
NPT2 Others Unspecified Ratio = 6.0 n.a. PMID[532393]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 7500.0 nM PMID[532396]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 5000.0 nM PMID[532396]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. IC50 = 3500.0 nM PMID[532396]
NPT2 Others Unspecified Potency n.a. 23485.0 nM PMID[532369]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. Potency n.a. 14950.2 nM PMID[532369]
NPT2 Others Unspecified Potency n.a. 29565.9 nM PMID[532369]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. Potency n.a. 6853.0 nM PMID[532401]
NPT2 Others Unspecified Potency n.a. 19952.6 nM PMID[532370]
NPT2 Others Unspecified Potency n.a. 8912.5 nM PMID[532368]
NPT2 Others Unspecified Potency n.a. 25118.9 nM PMID[532369]
NPT20529 NON-MOLECULAR NON-PROTEIN TARGET n.a. Potency n.a. 18821.2 nM PMID[532369]
NPT35 Others n.a. LogD7.4 n.a. 3.34 n.a. PMID[532404]
NPT831 Individual Protein Serine/threonine-protein kinase PLK1 Homo sapiens Thermal melting change = 0.2 degrees C PMID[532343]
NPT22960 SINGLE PROTEIN Serine/threonine-protein kinase VRK1 Homo sapiens Thermal melting change = -0.1 degrees C PMID[532343]
NPT22961 SINGLE PROTEIN Inactive serine/threonine-protein kinase VRK3 Homo sapiens Thermal melting change = 0.0 degrees C PMID[532343]
NPT2 Others Unspecified Potency n.a. 16626.1 nM PMID[532369]
NPT2 Others Unspecified FC = 2.5 n.a. PMID[532410]
NPT25835 SINGLE PROTEIN Bromodomain testis-specific protein Homo sapiens Delta Tm = 0.85 degrees C PMID[532413]
NPT2 Others Unspecified IC50 = 3500.0 nM PMID[532415]
NPT2 Others Unspecified IC50 = 5000.0 nM PMID[532415]
NPT2 Others Unspecified IC50 = 7200.0 nM PMID[532415]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 500.0 nM PMID[532416]
NPT29 Organism Rattus norvegicus Rattus norvegicus Inhibition = 37.0 % PMID[532418]
NPT2 Others Unspecified IC50 = 220.0 nM PMID[532419]
NPT20555 ORGANISM SARS-CoV-2 Severe acute respiratory syndrome coronavirus 2 Inhibition = -0.92 % PMID[532420]
NPT1308 Tissue Blood Homo sapiens IC50 = 3018.0 nM PMID[532423]
NPT1308 Tissue Blood Homo sapiens Inhibition = 76.5 % PMID[532423]
NPT1308 Tissue Blood Homo sapiens IC50 = 3202.0 nM PMID[532425]
NPT207 Protein Family MAP kinase p38 Homo sapiens IC50 = 500.0 nM PMID[532427]
NPT20556 SINGLE PROTEIN Replicase polyprotein 1ab Severe acute respiratory syndrome coronavirus 2 Inhibition = 24.88 % PMID[532428]
NPT20556 SINGLE PROTEIN Replicase polyprotein 1ab Severe acute respiratory syndrome coronavirus 2 Inhibition = 9.655 % PMID[532429]
NPT20555 ORGANISM SARS-CoV-2 Severe acute respiratory syndrome coronavirus 2 Inhibition = 0.28 % PMID[532430]
NPT20555 ORGANISM SARS-CoV-2 Severe acute respiratory syndrome coronavirus 2 Inhibition = 0.02 % PMID[532431]
NPT20555 ORGANISM SARS-CoV-2 Severe acute respiratory syndrome coronavirus 2 IC50 > 20000.0 nM PMID[532433]
NPT20555 ORGANISM SARS-CoV-2 Severe acute respiratory syndrome coronavirus 2 IC50 > 19952.62 nM PMID[532433]

☑ Note for Activity Records:
☉ The quantitative biological activities were primarily integrated from ChEMBL (Version-30) database and were also directly collected from PubMed literature. PubMed PMID was provided as the reference link for each activity record.

  Chemically structural similarity: I. Similar Active Natural Products in NPASS

Top-200 similar NPs were calculated against the active-NP-set (includes 4,3285 NPs with experimentally-derived bioactivity available in NPASS)

Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient

●  The left chart: Distribution of similarity level between NPC469308 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).

Similarity Score Similarity Level Natural Product ID
0.8054 Intermediate Similarity NPC317054
0.7767 Intermediate Similarity NPC471603
0.7717 Intermediate Similarity NPC470203
0.7663 Intermediate Similarity NPC470204
0.7486 Intermediate Similarity NPC325903
0.7473 Intermediate Similarity NPC122141
0.7459 Intermediate Similarity NPC114209
0.7363 Intermediate Similarity NPC201380
0.7363 Intermediate Similarity NPC179787
0.7337 Intermediate Similarity NPC470233
0.7322 Intermediate Similarity NPC321911
0.7308 Intermediate Similarity NPC63545
0.7268 Intermediate Similarity NPC469811
0.7249 Intermediate Similarity NPC225018
0.7211 Intermediate Similarity NPC317105
0.7208 Intermediate Similarity NPC307191
0.7181 Intermediate Similarity NPC236711
0.7143 Intermediate Similarity NPC300238
0.7092 Intermediate Similarity NPC280852
0.7075 Intermediate Similarity NPC116555
0.7074 Intermediate Similarity NPC39092
0.7074 Intermediate Similarity NPC476219
0.7062 Intermediate Similarity NPC91895
0.7005 Intermediate Similarity NPC53947
0.699 Remote Similarity NPC314557
0.6989 Remote Similarity NPC470111
0.6984 Remote Similarity NPC476297
0.6973 Remote Similarity NPC204141
0.6972 Remote Similarity NPC267811
0.6968 Remote Similarity NPC470823
0.6968 Remote Similarity NPC216713
0.6965 Remote Similarity NPC108011
0.6963 Remote Similarity NPC474791
0.6935 Remote Similarity NPC143872
0.6935 Remote Similarity NPC288838
0.6927 Remote Similarity NPC215584
0.6927 Remote Similarity NPC44773
0.6919 Remote Similarity NPC315715
0.6906 Remote Similarity NPC216159
0.6898 Remote Similarity NPC471957
0.6862 Remote Similarity NPC282531
0.6853 Remote Similarity NPC82331
0.6848 Remote Similarity NPC469761
0.6848 Remote Similarity NPC469779
0.6848 Remote Similarity NPC115611
0.6848 Remote Similarity NPC469780
0.6848 Remote Similarity NPC284635
0.6848 Remote Similarity NPC469767
0.6848 Remote Similarity NPC469783
0.6848 Remote Similarity NPC469768
0.6848 Remote Similarity NPC469784
0.6842 Remote Similarity NPC200214
0.6834 Remote Similarity NPC474958
0.6823 Remote Similarity NPC216643
0.6821 Remote Similarity NPC274229
0.6816 Remote Similarity NPC16659
0.6811 Remote Similarity NPC469766
0.6793 Remote Similarity NPC73767
0.6788 Remote Similarity NPC56765
0.6788 Remote Similarity NPC135141
0.6788 Remote Similarity NPC92796
0.6776 Remote Similarity NPC84911
0.6769 Remote Similarity NPC478182
0.6766 Remote Similarity NPC265710
0.6742 Remote Similarity NPC173344
0.6737 Remote Similarity NPC40070
0.6733 Remote Similarity NPC164228
0.6721 Remote Similarity NPC96102
0.6721 Remote Similarity NPC261195
0.6721 Remote Similarity NPC29886
0.6718 Remote Similarity NPC478185
0.6717 Remote Similarity NPC97343
0.6716 Remote Similarity NPC473380
0.6716 Remote Similarity NPC248454
0.6716 Remote Similarity NPC240088
0.6715 Remote Similarity NPC231536
0.6712 Remote Similarity NPC149014
0.6711 Remote Similarity NPC130570
0.6703 Remote Similarity NPC110126
0.6702 Remote Similarity NPC314372
0.6701 Remote Similarity NPC49217
0.67 Remote Similarity NPC471579
0.6697 Remote Similarity NPC147810
0.6685 Remote Similarity NPC251722
0.6685 Remote Similarity NPC314102
0.6685 Remote Similarity NPC105127
0.6684 Remote Similarity NPC190296
0.6684 Remote Similarity NPC478184
0.6667 Remote Similarity NPC198988
0.6652 Remote Similarity NPC77022
0.6649 Remote Similarity NPC24678
0.6649 Remote Similarity NPC148592
0.6649 Remote Similarity NPC286427
0.6649 Remote Similarity NPC105818
0.6649 Remote Similarity NPC469897
0.6632 Remote Similarity NPC120070
0.663 Remote Similarity NPC325252
0.6622 Remote Similarity NPC216221
0.6618 Remote Similarity NPC191415
0.6615 Remote Similarity NPC206819
0.6615 Remote Similarity NPC293487
0.6615 Remote Similarity NPC318065
0.6615 Remote Similarity NPC41257
0.6613 Remote Similarity NPC88097
0.6606 Remote Similarity NPC282247
0.6595 Remote Similarity NPC125746
0.6593 Remote Similarity NPC82295
0.6585 Remote Similarity NPC163055
0.6582 Remote Similarity NPC229173
0.658 Remote Similarity NPC935
0.658 Remote Similarity NPC469786
0.658 Remote Similarity NPC267078
0.658 Remote Similarity NPC25008
0.658 Remote Similarity NPC259644
0.658 Remote Similarity NPC469760
0.658 Remote Similarity NPC469763
0.658 Remote Similarity NPC73952
0.658 Remote Similarity NPC469765
0.6578 Remote Similarity NPC279081
0.6571 Remote Similarity NPC324149
0.6553 Remote Similarity NPC284678
0.6552 Remote Similarity NPC474357
0.6548 Remote Similarity NPC253687
0.6546 Remote Similarity NPC212376
0.6546 Remote Similarity NPC75540
0.6546 Remote Similarity NPC80597
0.6546 Remote Similarity NPC70922
0.6546 Remote Similarity NPC211572
0.654 Remote Similarity NPC326422
0.6537 Remote Similarity NPC470323
0.6533 Remote Similarity NPC478183
0.6531 Remote Similarity NPC477591
0.653 Remote Similarity NPC66699
0.6526 Remote Similarity NPC159856
0.6515 Remote Similarity NPC247987
0.6515 Remote Similarity NPC90723
0.6508 Remote Similarity NPC42483
0.6505 Remote Similarity NPC48938
0.6505 Remote Similarity NPC102755
0.6503 Remote Similarity NPC101165
0.65 Remote Similarity NPC63751
0.6489 Remote Similarity NPC230002
0.6489 Remote Similarity NPC2949
0.6489 Remote Similarity NPC59084
0.6486 Remote Similarity NPC31385
0.6486 Remote Similarity NPC110602
0.6486 Remote Similarity NPC75726
0.6484 Remote Similarity NPC175916
0.6482 Remote Similarity NPC280864
0.6482 Remote Similarity NPC17751
0.6471 Remote Similarity NPC59269
0.6468 Remote Similarity NPC194411
0.6455 Remote Similarity NPC63157
0.6455 Remote Similarity NPC473868
0.645 Remote Similarity NPC56233
0.6447 Remote Similarity NPC474880
0.6447 Remote Similarity NPC475990
0.6447 Remote Similarity NPC221786
0.6442 Remote Similarity NPC308931
0.6442 Remote Similarity NPC15102
0.6442 Remote Similarity NPC99939
0.6441 Remote Similarity NPC124636
0.6441 Remote Similarity NPC54981
0.644 Remote Similarity NPC285731
0.644 Remote Similarity NPC470440
0.6432 Remote Similarity NPC294693
0.6429 Remote Similarity NPC469785
0.6422 Remote Similarity NPC317701
0.6422 Remote Similarity NPC69843
0.6417 Remote Similarity NPC150259
0.6413 Remote Similarity NPC193370
0.6413 Remote Similarity NPC475450
0.6411 Remote Similarity NPC62749
0.6404 Remote Similarity NPC477611
0.6402 Remote Similarity NPC316756
0.6396 Remote Similarity NPC469762
0.6393 Remote Similarity NPC475070
0.6392 Remote Similarity NPC33421
0.6386 Remote Similarity NPC474897
0.6386 Remote Similarity NPC32534
0.6378 Remote Similarity NPC473930
0.6373 Remote Similarity NPC37423
0.6373 Remote Similarity NPC21605
0.6373 Remote Similarity NPC275305
0.6372 Remote Similarity NPC272483
0.6368 Remote Similarity NPC49954
0.6368 Remote Similarity NPC474561
0.6364 Remote Similarity NPC218268
0.6359 Remote Similarity NPC22079
0.6359 Remote Similarity NPC469975
0.6354 Remote Similarity NPC86288
0.6351 Remote Similarity NPC472289
0.635 Remote Similarity NPC311276
0.6343 Remote Similarity NPC265576
0.6337 Remote Similarity NPC201700
0.6335 Remote Similarity NPC20144
0.6333 Remote Similarity NPC46358
0.6333 Remote Similarity NPC135601
0.6333 Remote Similarity NPC141612
0.6333 Remote Similarity NPC17273

  Chemically structural similarity: II. Similar Clinical/Approved Drugs

Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.

●  The left chart: Distribution of similarity level between NPC469308 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).

Similarity Score Similarity Level Drug ID Developmental Stage
1.0 High Similarity NPD4318 Clinical (unspecified phase)
0.8907 High Similarity NPD2818 Discontinued
0.8343 Intermediate Similarity NPD1567 Clinical (unspecified phase)
0.8128 Intermediate Similarity NPD4649 Clinical (unspecified phase)
0.8118 Intermediate Similarity NPD2930 Clinical (unspecified phase)
0.8075 Intermediate Similarity NPD1873 Clinical (unspecified phase)
0.8053 Intermediate Similarity NPD2963 Phase 1
0.8033 Intermediate Similarity NPD2333 Discontinued
0.8021 Intermediate Similarity NPD3341 Clinical (unspecified phase)
0.7979 Intermediate Similarity NPD5962 Phase 2
0.7969 Intermediate Similarity NPD7884 Discontinued
0.7958 Intermediate Similarity NPD6721 Phase 1
0.7887 Intermediate Similarity NPD3419 Clinical (unspecified phase)
0.7865 Intermediate Similarity NPD3378 Clinical (unspecified phase)
0.7865 Intermediate Similarity NPD2793 Discontinued
0.7846 Intermediate Similarity NPD6577 Clinical (unspecified phase)
0.7842 Intermediate Similarity NPD1895 Discontinued
0.7801 Intermediate Similarity NPD3512 Clinical (unspecified phase)
0.7789 Intermediate Similarity NPD6264 Discontinued
0.7784 Intermediate Similarity NPD2478 Clinical (unspecified phase)
0.7732 Intermediate Similarity NPD5590 Clinical (unspecified phase)
0.7706 Intermediate Similarity NPD1259 Discontinued
0.7701 Intermediate Similarity NPD2875 Clinical (unspecified phase)
0.767 Intermediate Similarity NPD4990 Clinical (unspecified phase)
0.7662 Intermediate Similarity NPD6816 Phase 3
0.7635 Intermediate Similarity NPD2364 Suspended
0.7626 Intermediate Similarity NPD6265 Discontinued
0.7622 Intermediate Similarity NPD2385 Clinical (unspecified phase)
0.76 Intermediate Similarity NPD6224 Clinical (unspecified phase)
0.759 Intermediate Similarity NPD4902 Discontinued
0.7586 Intermediate Similarity NPD3015 Discontinued
0.7552 Intermediate Similarity NPD1327 Discontinued
0.755 Intermediate Similarity NPD6278 Clinical (unspecified phase)
0.7536 Intermediate Similarity NPD4471 Approved
0.7536 Intermediate Similarity NPD4472 Approved
0.7512 Intermediate Similarity NPD4473 Clinical (unspecified phase)
0.75 Intermediate Similarity NPD6171 Clinical (unspecified phase)
0.7488 Intermediate Similarity NPD2026 Approved
0.7487 Intermediate Similarity NPD3430 Approved
0.7487 Intermediate Similarity NPD3431 Approved
0.7476 Intermediate Similarity NPD4023 Clinical (unspecified phase)
0.7474 Intermediate Similarity NPD6827 Clinical (unspecified phase)
0.7474 Intermediate Similarity NPD5806 Clinical (unspecified phase)
0.7474 Intermediate Similarity NPD6828 Phase 2
0.7466 Intermediate Similarity NPD7052 Phase 1
0.7452 Intermediate Similarity NPD7409 Clinical (unspecified phase)
0.745 Intermediate Similarity NPD3485 Clinical (unspecified phase)
0.7449 Intermediate Similarity NPD2868 Clinical (unspecified phase)
0.7448 Intermediate Similarity NPD2406 Clinical (unspecified phase)
0.7447 Intermediate Similarity NPD1313 Approved
0.7447 Intermediate Similarity NPD1333 Phase 3
0.744 Intermediate Similarity NPD7445 Phase 1
0.7437 Intermediate Similarity NPD7709 Discontinued
0.7429 Intermediate Similarity NPD4352 Phase 1
0.7426 Intermediate Similarity NPD5462 Discontinued
0.7423 Intermediate Similarity NPD702 Clinical (unspecified phase)
0.7415 Intermediate Similarity NPD6129 Phase 2
0.7411 Intermediate Similarity NPD2409 Clinical (unspecified phase)
0.7409 Intermediate Similarity NPD2731 Phase 2
0.7405 Intermediate Similarity NPD2927 Phase 3
0.74 Intermediate Similarity NPD7127 Clinical (unspecified phase)
0.7396 Intermediate Similarity NPD3859 Clinical (unspecified phase)
0.7393 Intermediate Similarity NPD2847 Phase 2
0.7389 Intermediate Similarity NPD3287 Clinical (unspecified phase)
0.7385 Intermediate Similarity NPD412 Approved
0.7383 Intermediate Similarity NPD5270 Discontinued
0.7376 Intermediate Similarity NPD7023 Clinical (unspecified phase)
0.7371 Intermediate Similarity NPD1893 Phase 2
0.7371 Intermediate Similarity NPD1892 Phase 2
0.735 Intermediate Similarity NPD6626 Approved
0.7349 Intermediate Similarity NPD5884 Clinical (unspecified phase)
0.7347 Intermediate Similarity NPD5105 Approved
0.7347 Intermediate Similarity NPD4441 Phase 2
0.7347 Intermediate Similarity NPD5106 Approved
0.734 Intermediate Similarity NPD1015 Phase 2
0.734 Intermediate Similarity NPD1016 Phase 2
0.7333 Intermediate Similarity NPD3843 Clinical (unspecified phase)
0.7333 Intermediate Similarity NPD5508 Phase 1
0.7327 Intermediate Similarity NPD3284 Phase 3
0.7316 Intermediate Similarity NPD1215 Discontinued
0.7313 Intermediate Similarity NPD2839 Phase 2
0.7311 Intermediate Similarity NPD5679 Clinical (unspecified phase)
0.7308 Intermediate Similarity NPD2736 Phase 1
0.7306 Intermediate Similarity NPD7006 Approved
0.7304 Intermediate Similarity NPD6469 Phase 3
0.7304 Intermediate Similarity NPD6468 Clinical (unspecified phase)
0.7299 Intermediate Similarity NPD4863 Approved
0.7291 Intermediate Similarity NPD3362 Clinical (unspecified phase)
0.7285 Intermediate Similarity NPD2062 Phase 2
0.7285 Intermediate Similarity NPD8004 Discontinued
0.7282 Intermediate Similarity NPD5730 Phase 2
0.7282 Intermediate Similarity NPD40 Phase 2
0.7282 Intermediate Similarity NPD3831 Approved
0.7273 Intermediate Similarity NPD1869 Phase 2
0.7273 Intermediate Similarity NPD4298 Clinical (unspecified phase)
0.7273 Intermediate Similarity NPD5415 Approved
0.7273 Intermediate Similarity NPD5864 Phase 2
0.7273 Intermediate Similarity NPD2735 Clinical (unspecified phase)
0.7268 Intermediate Similarity NPD3348 Phase 2
0.7255 Intermediate Similarity NPD2880 Discontinued
0.725 Intermediate Similarity NPD2728 Approved
0.725 Intermediate Similarity NPD2730 Approved
0.725 Intermediate Similarity NPD2729 Approved
0.7245 Intermediate Similarity NPD7063 Clinical (unspecified phase)
0.7236 Intermediate Similarity NPD2872 Phase 2
0.7236 Intermediate Similarity NPD5642 Approved
0.7231 Intermediate Similarity NPD7111 Discontinued
0.7227 Intermediate Similarity NPD1911 Approved
0.7227 Intermediate Similarity NPD1910 Approved
0.7225 Intermediate Similarity NPD6794 Approved
0.7225 Intermediate Similarity NPD2392 Clinical (unspecified phase)
0.722 Intermediate Similarity NPD1982 Phase 1
0.7215 Intermediate Similarity NPD2955 Approved
0.7215 Intermediate Similarity NPD2954 Approved
0.7214 Intermediate Similarity NPD5145 Clinical (unspecified phase)
0.7206 Intermediate Similarity NPD2316 Clinical (unspecified phase)
0.7204 Intermediate Similarity NPD6545 Clinical (unspecified phase)
0.7204 Intermediate Similarity NPD2837 Discontinued
0.7194 Intermediate Similarity NPD2084 Discontinued
0.7192 Intermediate Similarity NPD2446 Approved
0.7192 Intermediate Similarity NPD2320 Discontinued
0.7192 Intermediate Similarity NPD2445 Approved
0.719 Intermediate Similarity NPD8410 Clinical (unspecified phase)
0.7188 Intermediate Similarity NPD8159 Discontinued
0.7184 Intermediate Similarity NPD5828 Phase 2
0.7183 Intermediate Similarity NPD8458 Clinical (unspecified phase)
0.7178 Intermediate Similarity NPD6761 Discontinued
0.7173 Intermediate Similarity NPD3889 Approved
0.7171 Intermediate Similarity NPD3830 Phase 1
0.7167 Intermediate Similarity NPD174 Discontinued
0.7163 Intermediate Similarity NPD1556 Clinical (unspecified phase)
0.7157 Intermediate Similarity NPD4294 Phase 2
0.7157 Intermediate Similarity NPD1928 Discontinued
0.7156 Intermediate Similarity NPD6520 Phase 3
0.7156 Intermediate Similarity NPD6521 Phase 3
0.7151 Intermediate Similarity NPD2103 Approved
0.7151 Intermediate Similarity NPD2524 Discontinued
0.715 Intermediate Similarity NPD8488 Clinical (unspecified phase)
0.715 Intermediate Similarity NPD7264 Clinical (unspecified phase)
0.7143 Intermediate Similarity NPD2849 Clinical (unspecified phase)
0.7143 Intermediate Similarity NPD7722 Suspended
0.7136 Intermediate Similarity NPD1258 Discontinued
0.7136 Intermediate Similarity NPD5463 Clinical (unspecified phase)
0.7136 Intermediate Similarity NPD5885 Approved
0.7128 Intermediate Similarity NPD1569 Phase 2
0.7128 Intermediate Similarity NPD3799 Suspended
0.7122 Intermediate Similarity NPD2960 Clinical (unspecified phase)
0.7113 Intermediate Similarity NPD3609 Approved
0.7113 Intermediate Similarity NPD3610 Approved
0.7113 Intermediate Similarity NPD3347 Clinical (unspecified phase)
0.7109 Intermediate Similarity NPD1506 Discontinued
0.7107 Intermediate Similarity NPD3409 Phase 1
0.7098 Intermediate Similarity NPD2640 Approved
0.7098 Intermediate Similarity NPD2641 Approved
0.7097 Intermediate Similarity NPD1029 Clinical (unspecified phase)
0.7097 Intermediate Similarity NPD1030 Approved
0.7097 Intermediate Similarity NPD703 Discontinued
0.7097 Intermediate Similarity NPD1027 Approved
0.7092 Intermediate Similarity NPD2751 Phase 1
0.7092 Intermediate Similarity NPD2771 Approved
0.7091 Intermediate Similarity NPD6849 Phase 2
0.7091 Intermediate Similarity NPD6850 Phase 2
0.7075 Intermediate Similarity NPD4612 Discontinued
0.7064 Intermediate Similarity NPD5198 Approved
0.7064 Intermediate Similarity NPD5199 Approved
0.7062 Intermediate Similarity NPD2008 Discontinued
0.7059 Intermediate Similarity NPD4615 Phase 2
0.7056 Intermediate Similarity NPD4181 Approved
0.7053 Intermediate Similarity NPD4470 Phase 2
0.7053 Intermediate Similarity NPD1042 Clinical (unspecified phase)
0.7051 Intermediate Similarity NPD8257 Approved
0.7051 Intermediate Similarity NPD8258 Clinical (unspecified phase)
0.7051 Intermediate Similarity NPD8256 Approved
0.7047 Intermediate Similarity NPD1589 Clinical (unspecified phase)
0.7043 Intermediate Similarity NPD2104 Approved
0.7043 Intermediate Similarity NPD2102 Approved
0.7042 Intermediate Similarity NPD2408 Discontinued
0.7039 Intermediate Similarity NPD2142 Approved
0.7039 Intermediate Similarity NPD2141 Approved
0.7039 Intermediate Similarity NPD2140 Approved
0.7037 Intermediate Similarity NPD1290 Phase 2
0.7037 Intermediate Similarity NPD3848 Phase 2
0.7035 Intermediate Similarity NPD1708 Approved
0.7035 Intermediate Similarity NPD1707 Approved
0.7033 Intermediate Similarity NPD6151 Phase 2
0.7028 Intermediate Similarity NPD3905 Phase 3
0.7024 Intermediate Similarity NPD460 Discontinued
0.7023 Intermediate Similarity NPD2411 Approved
0.7021 Intermediate Similarity NPD695 Discontinued
0.7018 Intermediate Similarity NPD6470 Phase 3
0.7014 Intermediate Similarity NPD4446 Approved
0.7013 Intermediate Similarity NPD5615 Phase 2
0.7011 Intermediate Similarity NPD4849 Approved
0.7011 Intermediate Similarity NPD5671 Approved
0.7009 Intermediate Similarity NPD6192 Phase 3
0.7005 Intermediate Similarity NPD3228 Phase 1
0.7005 Intermediate Similarity NPD5843 Discontinued
0.7 Intermediate Similarity NPD1332 Clinical (unspecified phase)
0.7 Intermediate Similarity NPD6308 Phase 1
0.6995 Remote Similarity NPD2443 Approved

  Bioactivity similarity: Similar Natural Products in NPASS

Bioactivity similarity was calculated based on bioactivity descriptors of compounds. The bioactivity descriptors were calculated by a recently developed AI algorithm Chemical Checker (CC) [Nature Biotechnology, 38:1087–1096, 2020; Nature Communications, 12:3932, 2021], which evaluated bioactivity similarities at five levels:
A: chemistry similarity;
B: biological targets similarity;
C: networks similarity;
D: cell-based bioactivity similarity;
E: similarity based on clinical data.

Those 5 categories of CC bioactivity descriptors were calculated and then subjected to manifold projection using UMAP algorithm, to project all NPs on a 2-Dimensional space. The current NP was highlighted with a small circle in the 2-D map. Below figures: left-to-right, A-to-E.

A: chemistry similarity
B: biological targets similarity
C: networks similarity
D: cell-based bioactivity similarity
E: similarity based on clinical data