Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[532298] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[532299] |
NPT6452 |
Individual Protein |
MAP kinase p38 alpha |
Mus musculus |
Kd |
= |
20.0 |
nM |
PMID[532301] |
NPT6452 |
Individual Protein |
MAP kinase p38 alpha |
Mus musculus |
Tm |
= |
46.6 |
degrees C |
PMID[532301] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
25.0 |
nM |
PMID[532303] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532303] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
160.0 |
nM |
PMID[532303] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Inhibition |
= |
55.0 |
% |
PMID[532303] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Inhibition |
= |
54.0 |
% |
PMID[532303] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Inhibition |
= |
22.0 |
% |
PMID[532303] |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
> |
5000.0 |
nM |
PMID[532303] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
IC50 |
= |
30000.0 |
nM |
PMID[532304] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
38.0 |
nM |
PMID[532305] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
IC50 |
= |
330.0 |
nM |
PMID[532306] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[532306] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
1900.0 |
nM |
PMID[532306] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
IC50 |
= |
3450.0 |
nM |
PMID[532306] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
IC50 |
= |
96000.0 |
nM |
PMID[532306] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
Inhibition |
= |
61.0 |
% |
PMID[532307] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Inhibition |
= |
75.0 |
% |
PMID[532307] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Inhibition |
= |
85.0 |
% |
PMID[532307] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
67.0 |
% |
PMID[532307] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
61.0 |
% |
PMID[532307] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
39.0 |
nM |
PMID[532308] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
78.0 |
nM |
PMID[532308] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Inhibition |
= |
46.0 |
% |
PMID[532308] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
IC50 |
= |
370.0 |
nM |
PMID[532308] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Inhibition |
= |
50.0 |
% |
PMID[532308] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
280.0 |
nM |
PMID[532308] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
1920.0 |
nM |
PMID[532308] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532309] |
NPT3089 |
Cell Line |
SW1353 |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532309] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532311] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532312] |
NPT3089 |
Cell Line |
SW1353 |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532312] |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
80.0 |
nM |
PMID[532315] |
NPT183 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Rattus norvegicus |
IC50 |
= |
58000.0 |
nM |
PMID[532315] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
IC50 |
= |
6000.0 |
nM |
PMID[532316] |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532317] |
NPT1814 |
Individual Protein |
Glucagon receptor |
Homo sapiens |
Inhibition |
= |
18.0 |
% |
PMID[532318] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532319] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532320] |
NPT3089 |
Cell Line |
SW1353 |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532320] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
72000.0 |
nM |
PMID[532321] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
136000.0 |
nM |
PMID[532321] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532322] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
10.0 |
nM |
PMID[532323] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
IC50 |
> |
33000.0 |
nM |
PMID[532323] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[532325] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532325] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Kd |
= |
6800.0 |
nM |
PMID[532326] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
IC50 |
= |
7800.0 |
nM |
PMID[532326] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Inhibition |
= |
86.5 |
% |
PMID[532326] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
16.0 |
nM |
PMID[532327] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
IC50 |
= |
135.0 |
nM |
PMID[532327] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
IC50 |
= |
124.0 |
nM |
PMID[532327] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532327] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
11000.0 |
nM |
PMID[532327] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50 |
= |
5000.0 |
nM |
PMID[532327] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
38.0 |
nM |
PMID[532327] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[532327] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[532329] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
= |
4400.0 |
nM |
PMID[532330] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
= |
45.0 |
nM |
PMID[532330] |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
= |
860.0 |
nM |
PMID[532330] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
= |
9000.0 |
nM |
PMID[532330] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
= |
95.0 |
nM |
PMID[532330] |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
= |
4600.0 |
nM |
PMID[532330] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
= |
2100.0 |
nM |
PMID[532330] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
= |
39.0 |
nM |
PMID[532330] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2900.0 |
nM |
PMID[532330] |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
= |
1500.0 |
nM |
PMID[532330] |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
220.0 |
nM |
PMID[532330] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
= |
1200.0 |
nM |
PMID[532330] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532330] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
= |
250.0 |
nM |
PMID[532330] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
17.0 |
nM |
PMID[532330] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[532331] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[532332] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Inhibition |
= |
92.0 |
% |
PMID[532333] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
73.0 |
% |
PMID[532333] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
77.0 |
% |
PMID[532333] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
68.0 |
nM |
PMID[532333] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
30.0 |
nM |
PMID[532334] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
IC50 |
= |
790.0 |
nM |
PMID[532334] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
462.0 |
nM |
PMID[532335] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
Inhibition |
= |
61.0 |
% |
PMID[532335] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Inhibition |
= |
75.0 |
% |
PMID[532335] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Inhibition |
= |
85.0 |
% |
PMID[532335] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
67.0 |
% |
PMID[532335] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
61.0 |
% |
PMID[532335] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
IC50 |
= |
20000.0 |
nM |
PMID[532337] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Ki |
= |
18.0 |
nM |
PMID[532340] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Ki |
= |
90.0 |
nM |
PMID[532340] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
16.0 |
nM |
PMID[532341] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
39.0 |
nM |
PMID[532341] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
6000.0 |
nM |
PMID[532341] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
IC50 |
= |
330.0 |
nM |
PMID[532342] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532343] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
45.0 |
nM |
PMID[532344] |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
FC |
= |
4.3 |
n.a. |
PMID[532346] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
62.0 |
nM |
PMID[532347] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Inhibition |
= |
85.0 |
% |
PMID[532347] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
15.0 |
% |
PMID[532347] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Inhibition |
= |
0.0 |
% |
PMID[532347] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Inhibition |
= |
32.0 |
% |
PMID[532347] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Inhibition |
= |
86.0 |
% |
PMID[532347] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
98.0 |
% |
PMID[532347] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Inhibition |
= |
90.0 |
% |
PMID[532347] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Inhibition |
= |
4.0 |
% |
PMID[532347] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Inhibition |
= |
7.0 |
% |
PMID[532347] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Inhibition |
= |
11.0 |
% |
PMID[532347] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Inhibition |
= |
34.0 |
% |
PMID[532347] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
23.0 |
% |
PMID[532347] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Inhibition |
= |
68.0 |
% |
PMID[532347] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
Inhibition |
= |
38.0 |
% |
PMID[532347] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Inhibition |
= |
87.0 |
% |
PMID[532347] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Inhibition |
= |
92.0 |
% |
PMID[532347] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
73.0 |
% |
PMID[532347] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Inhibition |
= |
77.0 |
% |
PMID[532347] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532349] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
7000.0 |
nM |
PMID[532350] |
NPT6239 |
Individual Protein |
Mitogen-activated protein kinase 1 |
Toxoplasma gondii |
IC50 |
= |
100.0 |
nM |
PMID[532350] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
= |
1500.0 |
nM |
PMID[532352] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3250 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3251 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3252 |
Individual Protein |
Serine/threonine-protein kinase PFTAIRE-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3224 |
Individual Protein |
Phosphorylase kinase gamma subunit 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3253 |
Individual Protein |
Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
= |
250.0 |
nM |
PMID[532352] |
NPT3255 |
Individual Protein |
Myosin light chain kinase family member 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3256 |
Individual Protein |
Serine/threonine-protein kinase WEE1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3257 |
Individual Protein |
Serine/threonine-protein kinase 32C |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1717 |
Individual Protein |
Serine/threonine-protein kinase 25 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3258 |
Individual Protein |
Mixed lineage kinase 7 |
Homo sapiens |
Kd |
= |
4400.0 |
nM |
PMID[532352] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Activity |
= |
73.0 |
% |
PMID[532353] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Activity |
= |
52.0 |
% |
PMID[532353] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Activity |
= |
13.0 |
% |
PMID[532353] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Activity |
= |
107.0 |
% |
PMID[532353] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Activity |
= |
104.0 |
% |
PMID[532353] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT3260 |
Individual Protein |
Phosphatidylinositol-5-phosphate 4-kinase type-2 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3261 |
Individual Protein |
cAMP-dependent protein kinase beta-1 catalytic subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3265 |
Individual Protein |
Casein kinase I isoform alpha-like |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532352] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Kd |
= |
37.0 |
nM |
PMID[532352] |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
100.0 |
nM |
PMID[532352] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Selectivity |
= |
0.0242 |
n.a. |
PMID[532352] |
NPT3356 |
Individual Protein |
Tyrosine-protein kinase receptor Tie-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3268 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
= |
820.0 |
nM |
PMID[532352] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3238 |
Individual Protein |
Dual specificity protein kinase TTK |
Homo sapiens |
Kd |
= |
2500.0 |
nM |
PMID[532352] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Activity |
= |
89.0 |
% |
PMID[532353] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Activity |
= |
83.0 |
% |
PMID[532353] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Activity |
= |
81.0 |
% |
PMID[532353] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Activity |
= |
82.0 |
% |
PMID[532353] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1598 |
Individual Protein |
Casein kinase II alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3230 |
Individual Protein |
Serine/threonine-protein kinase 17B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532352] |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Kd |
= |
4500.0 |
nM |
PMID[532352] |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Activity |
= |
97.0 |
% |
PMID[532353] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Activity |
= |
81.0 |
% |
PMID[532353] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Activity |
= |
89.0 |
% |
PMID[532353] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Activity |
= |
90.0 |
% |
PMID[532353] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
= |
1100.0 |
nM |
PMID[532352] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
= |
130.0 |
nM |
PMID[532352] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3278 |
Individual Protein |
LIM domain kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Kd |
= |
9600.0 |
nM |
PMID[532352] |
NPT3281 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Activity |
= |
89.0 |
% |
PMID[532353] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Activity |
= |
78.0 |
% |
PMID[532353] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Activity |
= |
91.0 |
% |
PMID[532353] |
NPT3228 |
Individual Protein |
Adaptor-associated kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Kd |
= |
25.0 |
nM |
PMID[532352] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
12.0 |
nM |
PMID[532352] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
= |
70.0 |
nM |
PMID[532352] |
NPT3301 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Activity |
= |
93.0 |
% |
PMID[532353] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Activity |
= |
80.0 |
% |
PMID[532353] |
NPT3288 |
Individual Protein |
Interleukin-1 receptor-associated kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
= |
35.0 |
nM |
PMID[532352] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3264 |
Individual Protein |
Serine/threonine-protein kinase RIO1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3289 |
Individual Protein |
Serine/threonine-protein kinase RIO3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Activity |
= |
91.0 |
% |
PMID[532353] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Activity |
= |
85.0 |
% |
PMID[532353] |
NPT3813 |
Individual Protein |
Tyrosine-protein kinase SRC |
Gallus gallus |
Activity |
= |
73.0 |
% |
PMID[532353] |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Kd |
= |
3000.0 |
nM |
PMID[532352] |
NPT3294 |
Individual Protein |
Activin receptor type-2A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3295 |
Individual Protein |
Activin receptor type-2B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3297 |
Individual Protein |
Non-receptor tyrosine-protein kinase TNK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3298 |
Individual Protein |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
Kd |
= |
3500.0 |
nM |
PMID[532352] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3300 |
Individual Protein |
Serine/threonine-protein kinase 32B |
Homo sapiens |
Kd |
= |
2100.0 |
nM |
PMID[532352] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
= |
19.0 |
nM |
PMID[532352] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1671 |
Individual Protein |
AMP-activated protein kinase, alpha-2 subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3342 |
Individual Protein |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
Kd |
= |
1000.0 |
nM |
PMID[532352] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Kd |
= |
5000.0 |
nM |
PMID[532352] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3304 |
Individual Protein |
Serine/threonine-protein kinase receptor R3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3305 |
Individual Protein |
Chaperone activity of bc1 complex-like, mitochondrial |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3307 |
Individual Protein |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3308 |
Individual Protein |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Kd |
= |
2800.0 |
nM |
PMID[532352] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3209 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Activity |
= |
85.0 |
% |
PMID[532353] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Activity |
= |
92.0 |
% |
PMID[532353] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT3306 |
Individual Protein |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
Kd |
= |
400.0 |
nM |
PMID[532352] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
340.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
710.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1300.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1600.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1500.0 |
nM |
PMID[532352] |
NPT3302 |
Individual Protein |
Ankyrin repeat and protein kinase domain-containing protein 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3310 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3311 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Activity |
= |
106.0 |
% |
PMID[532353] |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Activity |
= |
99.0 |
% |
PMID[532353] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Activity |
= |
66.0 |
% |
PMID[532353] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Activity |
= |
92.0 |
% |
PMID[532353] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3210 |
Individual Protein |
BMP-2-inducible protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3313 |
Individual Protein |
Bone morphogenetic protein receptor type-1A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3314 |
Individual Protein |
Bone morphogenetic protein receptor type-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
710.0 |
nM |
PMID[532352] |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
530.0 |
nM |
PMID[532352] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1673 |
Individual Protein |
CaM kinase I gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Kd |
= |
3700.0 |
nM |
PMID[532352] |
NPT3109 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3319 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Activity |
= |
8.0 |
% |
PMID[532353] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Activity |
= |
69.0 |
% |
PMID[532353] |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Activity |
= |
84.0 |
% |
PMID[532353] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Activity |
= |
97.0 |
% |
PMID[532353] |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3321 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3322 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3323 |
Individual Protein |
Cell division cycle 2-like protein kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3325 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Gallus gallus |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3328 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 11 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Kd |
= |
6200.0 |
nM |
PMID[532352] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Kd |
= |
2700.0 |
nM |
PMID[532352] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3460 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 3 |
Homo sapiens |
Activity |
= |
112.0 |
% |
PMID[532353] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Activity |
= |
98.0 |
% |
PMID[532353] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Activity |
= |
89.0 |
% |
PMID[532353] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Activity |
= |
83.0 |
% |
PMID[532353] |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Activity |
= |
93.0 |
% |
PMID[532353] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Activity |
= |
25.0 |
% |
PMID[532353] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3334 |
Individual Protein |
Citron Rho-interacting kinase |
Homo sapiens |
Kd |
= |
420.0 |
nM |
PMID[532352] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3335 |
Individual Protein |
Serine/threonine-protein kinase DCLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3337 |
Individual Protein |
Serine/threonine-protein kinase DCLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3243 |
Individual Protein |
myosin light chain kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3338 |
Individual Protein |
Myosin IIIA |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3339 |
Individual Protein |
Myosin-IIIB |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3233 |
Individual Protein |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3340 |
Individual Protein |
Serine/threonine-protein kinase Nek1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3341 |
Individual Protein |
Serine/threonine-protein kinase Nek5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3241 |
Individual Protein |
Serine/threonine-protein kinase NEK9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3120 |
Individual Protein |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Activity |
= |
81.0 |
% |
PMID[532353] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Activity |
= |
98.0 |
% |
PMID[532353] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Activity |
= |
96.0 |
% |
PMID[532353] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Activity |
= |
9.0 |
% |
PMID[532353] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
= |
1800.0 |
nM |
PMID[532352] |
NPT3343 |
Individual Protein |
Uncharacterized aarF domain-containing protein kinase 4 |
Homo sapiens |
Kd |
= |
3100.0 |
nM |
PMID[532352] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3345 |
Individual Protein |
Cyclin-dependent kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
= |
3700.0 |
nM |
PMID[532352] |
NPT3348 |
Individual Protein |
NUAK family SNF1-like kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Kd |
= |
5300.0 |
nM |
PMID[532352] |
NPT3350 |
Individual Protein |
Tyrosine-protein kinase Srms |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1708 |
Individual Protein |
Serine/threonine-protein kinase 16 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
= |
1300.0 |
nM |
PMID[532352] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3352 |
Individual Protein |
Dual specificity testis-specific protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Kd |
= |
7100.0 |
nM |
PMID[532352] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Activity |
= |
34.0 |
% |
PMID[532353] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Activity |
= |
86.0 |
% |
PMID[532353] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Activity |
= |
96.0 |
% |
PMID[532353] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Activity |
= |
95.0 |
% |
PMID[532353] |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1900.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
3200.0 |
nM |
PMID[532352] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2000.0 |
nM |
PMID[532352] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3220 |
Individual Protein |
Ephrin type-A receptor 6 |
Homo sapiens |
Kd |
= |
1200.0 |
nM |
PMID[532352] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3355 |
Individual Protein |
TGF-beta receptor type II |
Homo sapiens |
Kd |
= |
1800.0 |
nM |
PMID[532352] |
NPT3249 |
Individual Protein |
Tyrosine- and threonine-specific cdc2-inhibitory kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1656 |
Individual Protein |
Protein kinase N1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Activity |
= |
60.0 |
% |
PMID[532353] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Activity |
= |
72.0 |
% |
PMID[532353] |
NPT3815 |
Individual Protein |
Tyrosine-protein kinase LCK |
Mus musculus |
Activity |
= |
56.0 |
% |
PMID[532353] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Activity |
= |
84.0 |
% |
PMID[532353] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Activity |
= |
120.0 |
% |
PMID[532353] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3360 |
Individual Protein |
Tubulin alpha-1 chain |
Rattus norvegicus |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1692 |
Individual Protein |
Mitogen-activated protein kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3361 |
Individual Protein |
Mitogen-activated protein kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3362 |
Individual Protein |
Mitogen-activated protein kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3368 |
Individual Protein |
cGMP-dependent protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3369 |
Individual Protein |
Interferon-induced, double-stranded RNA-activated protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
= |
3900.0 |
nM |
PMID[532352] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Kd |
= |
980.0 |
nM |
PMID[532352] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Activity |
= |
98.0 |
% |
PMID[532353] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Activity |
= |
83.0 |
% |
PMID[532353] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Activity |
= |
85.0 |
% |
PMID[532353] |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Activity |
= |
109.0 |
% |
PMID[532353] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Activity |
= |
107.0 |
% |
PMID[532353] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3371 |
Individual Protein |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
= |
24.0 |
nM |
PMID[532352] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
= |
320.0 |
nM |
PMID[532352] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Activity |
= |
91.0 |
% |
PMID[532353] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Activity |
= |
96.0 |
% |
PMID[532353] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Activity |
= |
95.0 |
% |
PMID[532353] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Activity |
= |
7.0 |
% |
PMID[532353] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[532354] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Inhibition |
= |
78.0 |
% |
PMID[532355] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
IC50 |
= |
120.0 |
nM |
PMID[532356] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Inhibition |
= |
92.0 |
% |
PMID[532356] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
40.0 |
nM |
PMID[532356] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532357] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
70.0 |
nM |
PMID[532358] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
= |
320.0 |
nM |
PMID[532358] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532359] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
44.0 |
nM |
PMID[532360] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
39.0 |
nM |
PMID[532361] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
6000.0 |
nM |
PMID[532361] |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
FC |
= |
0.721 |
n.a. |
PMID[532363] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Inhibition |
= |
95.0 |
% |
PMID[532364] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Inhibition |
= |
32.0 |
% |
PMID[532364] |
NPT1610 |
Individual Protein |
Rho-associated protein kinase 2 |
Rattus norvegicus |
Inhibition |
= |
77.0 |
% |
PMID[532364] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Inhibition |
= |
66.0 |
% |
PMID[532364] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Inhibition |
= |
87.0 |
% |
PMID[532364] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Inhibition |
= |
83.0 |
% |
PMID[532364] |
NPT1443 |
Individual Protein |
Pyruvate dehydrogenase kinase isoform 1 |
Homo sapiens |
Inhibition |
= |
89.0 |
% |
PMID[532364] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Inhibition |
= |
89.0 |
% |
PMID[532364] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Inhibition |
= |
112.0 |
% |
PMID[532364] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Inhibition |
= |
86.0 |
% |
PMID[532364] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Inhibition |
= |
93.0 |
% |
PMID[532364] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Inhibition |
= |
93.0 |
% |
PMID[532364] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Inhibition |
= |
96.0 |
% |
PMID[532364] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Inhibition |
= |
10.0 |
% |
PMID[532364] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Inhibition |
= |
2.0 |
% |
PMID[532364] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Inhibition |
= |
101.0 |
% |
PMID[532364] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Inhibition |
= |
85.0 |
% |
PMID[532364] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Ki |
= |
57.0 |
nM |
PMID[532365] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
4.1 |
nM |
PMID[532365] |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PMID[532369] |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PMID[532368] |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PMID[532369] |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PMID[532368] |
NPT210 |
Individual Protein |
Thyroid stimulating hormone receptor |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PMID[532369] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
Potency |
= |
39.8 |
nM |
PMID[532369] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PMID[532369] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
12589.3 |
nM |
PMID[532368] |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
12589.3 |
nM |
PMID[532368] |
NPT150 |
Individual Protein |
Anthrax lethal factor |
Bacillus anthracis |
Potency |
= |
31622.8 |
nM |
PMID[532369] |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PMID[532368] |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PMID[532369] |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PMID[532369] |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PMID[532368] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
501.2 |
nM |
PMID[532368] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PMID[532369] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
1258.9 |
nM |
PMID[532369] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
Potency |
= |
1995.3 |
nM |
PMID[532369] |
NPT1139 |
Individual Protein |
Arachidonate 15-lipoxygenase, type II |
Homo sapiens |
Potency |
n.a. |
25118.9 |
nM |
PMID[532369] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
AC50 |
= |
39810.72 |
nM |
PMID[532369] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
AC50 |
= |
1995.26 |
nM |
PMID[532369] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
AC50 |
= |
501.19 |
nM |
PMID[532368] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
630.96 |
nM |
PMID[532368] |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
AC50 |
= |
1258.93 |
nM |
PMID[532369] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
AC50 |
= |
3981.07 |
nM |
PMID[532369] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
AC50 |
= |
39.81 |
nM |
PMID[532369] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
15.0 |
nM |
PMID[532372] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
1230.0 |
nM |
PMID[532372] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532373] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
55.0 |
nM |
PMID[532374] |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
n.a. |
70794.6 |
nM |
PMID[532369] |
NPT199 |
Individual Protein |
DNA polymerase kappa |
Homo sapiens |
Potency |
n.a. |
7943.3 |
nM |
PMID[532369] |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
n.a. |
56234.1 |
nM |
PMID[532369] |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Kd |
= |
1500.0 |
nM |
PMID[532375] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3378 |
Individual Protein |
Serine/threonine-protein kinase SIK3 |
Homo sapiens |
Kd |
= |
3900.0 |
nM |
PMID[532375] |
NPT1708 |
Individual Protein |
Serine/threonine-protein kinase 16 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3250 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Kd |
= |
5000.0 |
nM |
PMID[532375] |
NPT3304 |
Individual Protein |
Serine/threonine-protein kinase receptor R3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2213 |
Individual Protein |
Cyclin-dependent kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Kd |
= |
7900.0 |
nM |
PMID[532375] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3379 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 15 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3255 |
Individual Protein |
Myosin light chain kinase family member 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3301 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3380 |
Individual Protein |
Serine/threonine-protein kinase SBK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Kd |
= |
4800.0 |
nM |
PMID[532375] |
NPT3310 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3220 |
Individual Protein |
Ephrin type-A receptor 6 |
Homo sapiens |
Kd |
= |
1200.0 |
nM |
PMID[532375] |
NPT3339 |
Individual Protein |
Myosin-IIIB |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3295 |
Individual Protein |
Activin receptor type-2B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3383 |
Individual Protein |
Serine/threonine-protein kinase 32A |
Homo sapiens |
Kd |
= |
1300.0 |
nM |
PMID[532375] |
NPT3384 |
Individual Protein |
Cyclin-dependent kinase-like 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3283 |
Individual Protein |
MAP kinase-interacting serine/threonine-protein kinase MNK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3253 |
Individual Protein |
Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3385 |
Individual Protein |
Bone morphogenetic protein receptor type-1B |
Homo sapiens |
Kd |
= |
3300.0 |
nM |
PMID[532375] |
NPT3314 |
Individual Protein |
Bone morphogenetic protein receptor type-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3345 |
Individual Protein |
Cyclin-dependent kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1890 |
Individual Protein |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3294 |
Individual Protein |
Activin receptor type-2A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3168 |
Individual Protein |
Casein kinase I alpha |
Homo sapiens |
Kd |
= |
75.0 |
nM |
PMID[532375] |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
Kd |
= |
100.0 |
nM |
PMID[532375] |
NPT1598 |
Individual Protein |
Casein kinase II alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3342 |
Individual Protein |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
Kd |
= |
1000.0 |
nM |
PMID[532375] |
NPT3387 |
Individual Protein |
Receptor tyrosine-protein kinase erbB-3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Kd |
= |
1800.0 |
nM |
PMID[532375] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532375] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3388 |
Individual Protein |
Tyrosine-protein kinase CTK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3389 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3328 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 11 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3120 |
Individual Protein |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3251 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3392 |
Individual Protein |
Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1445 |
Individual Protein |
PI3-kinase p110-gamma subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3393 |
Individual Protein |
PI4-kinase beta subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3261 |
Individual Protein |
cAMP-dependent protein kinase beta-1 catalytic subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3361 |
Individual Protein |
Mitogen-activated protein kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1692 |
Individual Protein |
Mitogen-activated protein kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3362 |
Individual Protein |
Mitogen-activated protein kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Kd |
= |
1100.0 |
nM |
PMID[532375] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Kd |
= |
70.0 |
nM |
PMID[532375] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Kd |
= |
35.0 |
nM |
PMID[532375] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3281 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3369 |
Individual Protein |
Interferon-induced, double-stranded RNA-activated protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Kd |
= |
980.0 |
nM |
PMID[532375] |
NPT3395 |
Individual Protein |
Rhodopsin kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Kd |
= |
320.0 |
nM |
PMID[532375] |
NPT3319 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3396 |
Individual Protein |
Serine/threonine-protein kinase Nek4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3397 |
Individual Protein |
Cyclin-dependent kinase-like 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3355 |
Individual Protein |
TGF-beta receptor type II |
Homo sapiens |
Kd |
= |
1800.0 |
nM |
PMID[532375] |
NPT3238 |
Individual Protein |
Dual specificity protein kinase TTK |
Homo sapiens |
Kd |
= |
2500.0 |
nM |
PMID[532375] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Kd |
= |
4500.0 |
nM |
PMID[532375] |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Kd |
= |
2000.0 |
nM |
PMID[532375] |
NPT3256 |
Individual Protein |
Serine/threonine-protein kinase WEE1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3260 |
Individual Protein |
Phosphatidylinositol-5-phosphate 4-kinase type-2 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3398 |
Individual Protein |
Serine/threonine-protein kinase ULK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Kd |
= |
6200.0 |
nM |
PMID[532375] |
NPT3311 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3400 |
Individual Protein |
Peripheral plasma membrane protein CASK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3401 |
Individual Protein |
Cyclin-dependent kinase 13 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3371 |
Individual Protein |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Kd |
= |
24.0 |
nM |
PMID[532375] |
NPT3289 |
Individual Protein |
Serine/threonine-protein kinase RIO3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3402 |
Individual Protein |
Serine/threonine-protein kinase PRP4 homolog |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3403 |
Individual Protein |
Cyclin-dependent kinase-like 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3297 |
Individual Protein |
Non-receptor tyrosine-protein kinase TNK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1679 |
Individual Protein |
Cyclin-dependent kinase-like 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3230 |
Individual Protein |
Serine/threonine-protein kinase 17B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Kd |
= |
3000.0 |
nM |
PMID[532375] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3313 |
Individual Protein |
Bone morphogenetic protein receptor type-1A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
710.0 |
nM |
PMID[532375] |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
Kd |
= |
530.0 |
nM |
PMID[532375] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3404 |
Individual Protein |
Ephrin type-B receptor 6 |
Homo sapiens |
Kd |
= |
3100.0 |
nM |
PMID[532375] |
NPT3405 |
Individual Protein |
Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Kd |
= |
7100.0 |
nM |
PMID[532375] |
NPT3407 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3307 |
Individual Protein |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3408 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 13 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3335 |
Individual Protein |
Serine/threonine-protein kinase DCLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1446 |
Individual Protein |
PI3-kinase p110-delta subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1694 |
Individual Protein |
Serine/threonine-protein kinase OSR1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
= |
2600.0 |
nM |
PMID[532375] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Kd |
= |
3900.0 |
nM |
PMID[532375] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
340.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
710.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1300.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1600.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1500.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
1900.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
3200.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2000.0 |
nM |
PMID[532375] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Kd |
= |
2500.0 |
nM |
PMID[532375] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
Kd |
= |
19.0 |
nM |
PMID[532375] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Kd |
= |
2800.0 |
nM |
PMID[532375] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Kd |
= |
5300.0 |
nM |
PMID[532375] |
NPT3356 |
Individual Protein |
Tyrosine-protein kinase receptor Tie-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3278 |
Individual Protein |
LIM domain kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3410 |
Individual Protein |
Serine/threonine-protein kinase MAK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3411 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3209 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Kd |
= |
3900.0 |
nM |
PMID[532375] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Kd |
= |
2700.0 |
nM |
PMID[532375] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3224 |
Individual Protein |
Phosphorylase kinase gamma subunit 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1444 |
Individual Protein |
PI3-kinase p110-alpha subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3376 |
Individual Protein |
PI3-kinase p110-beta subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1671 |
Individual Protein |
AMP-activated protein kinase, alpha-2 subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3368 |
Individual Protein |
cGMP-dependent protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3352 |
Individual Protein |
Dual specificity testis-specific protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3412 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 12 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1717 |
Individual Protein |
Serine/threonine-protein kinase 25 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3109 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3413 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3334 |
Individual Protein |
Citron Rho-interacting kinase |
Homo sapiens |
Kd |
= |
420.0 |
nM |
PMID[532375] |
NPT3288 |
Individual Protein |
Interleukin-1 receptor-associated kinase 3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1710 |
Individual Protein |
Serine/threonine-protein kinase 38 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3340 |
Individual Protein |
Serine/threonine-protein kinase Nek1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3268 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3252 |
Individual Protein |
Serine/threonine-protein kinase PFTAIRE-1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3415 |
Individual Protein |
Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma |
Homo sapiens |
Kd |
= |
2600.0 |
nM |
PMID[532375] |
NPT3416 |
Individual Protein |
STE20/SPS1-related proline-alanine-rich protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3420 |
Individual Protein |
Eukaryotic translation initiation factor 2-alpha kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Kd |
= |
250.0 |
nM |
PMID[532375] |
NPT3308 |
Individual Protein |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3421 |
Individual Protein |
Hormonally up-regulated neu tumor-associated kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
= |
3700.0 |
nM |
PMID[532375] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3228 |
Individual Protein |
Adaptor-associated kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3423 |
Individual Protein |
Serine/threonine-protein kinase ICK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3424 |
Individual Protein |
Microtubule-associated serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3233 |
Individual Protein |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Kd |
= |
820.0 |
nM |
PMID[532375] |
NPT3323 |
Individual Protein |
Cell division cycle 2-like protein kinase 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
Kd |
= |
1300.0 |
nM |
PMID[532375] |
NPT3298 |
Individual Protein |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
Kd |
= |
3500.0 |
nM |
PMID[532375] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Kd |
= |
25.0 |
nM |
PMID[532375] |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3338 |
Individual Protein |
Myosin IIIA |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3306 |
Individual Protein |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
Kd |
= |
400.0 |
nM |
PMID[532375] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3210 |
Individual Protein |
BMP-2-inducible protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3428 |
Individual Protein |
Transient receptor potential cation channel subfamily M member 6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3429 |
Individual Protein |
SNF-related serine/threonine-protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1704 |
Individual Protein |
Serine/threonine-protein kinase RIO2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3300 |
Individual Protein |
Serine/threonine-protein kinase 32B |
Homo sapiens |
Kd |
= |
2100.0 |
nM |
PMID[532375] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3305 |
Individual Protein |
Chaperone activity of bc1 complex-like, mitochondrial |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1673 |
Individual Protein |
CaM kinase I gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3430 |
Individual Protein |
Receptor-interacting serine/threonine-protein kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3322 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3433 |
Individual Protein |
Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3343 |
Individual Protein |
Uncharacterized aarF domain-containing protein kinase 4 |
Homo sapiens |
Kd |
= |
3100.0 |
nM |
PMID[532375] |
NPT3434 |
Individual Protein |
SPS1/STE20-related protein kinase YSK4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Kd |
= |
9600.0 |
nM |
PMID[532375] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3348 |
Individual Protein |
NUAK family SNF1-like kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3264 |
Individual Protein |
Serine/threonine-protein kinase RIO1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3248 |
Individual Protein |
CaM-kinase kinase alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3241 |
Individual Protein |
Serine/threonine-protein kinase NEK9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3243 |
Individual Protein |
myosin light chain kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3337 |
Individual Protein |
Serine/threonine-protein kinase DCLK3 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3435 |
Individual Protein |
Serine/threonine-protein kinase pknB |
Mycobacterium tuberculosis |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3321 |
Individual Protein |
PITSLRE serine/threonine-protein kinase CDC2L1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3350 |
Individual Protein |
Tyrosine-protein kinase Srms |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3436 |
Individual Protein |
Serine/threonine-protein kinase 35 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3258 |
Individual Protein |
Mixed lineage kinase 7 |
Homo sapiens |
Kd |
= |
4400.0 |
nM |
PMID[532375] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
12.0 |
nM |
PMID[532375] |
NPT3363 |
Individual Protein |
Mitogen-activated protein kinase 15 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Kd |
= |
37.0 |
nM |
PMID[532375] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Kd |
= |
130.0 |
nM |
PMID[532375] |
NPT3437 |
Individual Protein |
Serine/threonine-protein kinase PFTAIRE-2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3439 |
Individual Protein |
Homeodomain-interacting protein kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3440 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 5 |
Homo sapiens |
Kd |
= |
1400.0 |
nM |
PMID[532375] |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3265 |
Individual Protein |
Casein kinase I isoform alpha-like |
Homo sapiens |
Kd |
= |
1700.0 |
nM |
PMID[532375] |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Kd |
= |
3700.0 |
nM |
PMID[532375] |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3445 |
Individual Protein |
Serine/threonine-protein kinase NIM1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3257 |
Individual Protein |
Serine/threonine-protein kinase 32C |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3302 |
Individual Protein |
Ankyrin repeat and protein kinase domain-containing protein 1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3446 |
Individual Protein |
Myosin light chain kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3249 |
Individual Protein |
Tyrosine- and threonine-specific cdc2-inhibitory kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3447 |
Individual Protein |
G protein-coupled receptor kinase 4 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3448 |
Individual Protein |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3341 |
Individual Protein |
Serine/threonine-protein kinase Nek5 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT1656 |
Individual Protein |
Protein kinase N1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3449 |
Individual Protein |
Wee1-like protein kinase 2 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3450 |
Individual Protein |
Putative uncharacterized serine/threonine-protein kinase SgK110 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3451 |
Individual Protein |
Dual serine/threonine and tyrosine protein kinase |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT3452 |
Individual Protein |
Calcium-dependent protein kinase 1 |
Plasmodium falciparum (isolate 3D7) |
Kd |
= |
850.0 |
nM |
PMID[532375] |
NPT3453 |
Individual Protein |
Cell division control protein 2 homolog |
Plasmodium falciparum (isolate 3D7) |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT216 |
Individual Protein |
Adenosine A1 receptor |
Homo sapiens |
IC50 |
= |
2950.0 |
nM |
PMID[532376] |
NPT216 |
Individual Protein |
Adenosine A1 receptor |
Homo sapiens |
Ki |
= |
1721.0 |
nM |
PMID[532376] |
NPT217 |
Individual Protein |
Adenosine A2a receptor |
Homo sapiens |
IC50 |
= |
6068.0 |
nM |
PMID[532376] |
NPT217 |
Individual Protein |
Adenosine A2a receptor |
Homo sapiens |
Ki |
= |
3407.0 |
nM |
PMID[532376] |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532376] |
NPT213 |
Individual Protein |
Cytochrome P450 2C19 |
Homo sapiens |
IC50 |
= |
800.0 |
nM |
PMID[532376] |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
IC50 |
= |
1000.0 |
nM |
PMID[532376] |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532376] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
10666.0 |
nM |
PMID[532376] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ki |
= |
2569.0 |
nM |
PMID[532376] |
NPT273 |
Individual Protein |
Phosphodiesterase 5A |
Homo sapiens |
IC50 |
= |
11476.0 |
nM |
PMID[532376] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
159.0 |
nM |
PMID[532376] |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
IC50 |
= |
18896.0 |
nM |
PMID[532376] |
NPT293 |
Individual Protein |
Serotonin 4 (5-HT4) receptor |
Cavia porcellus |
IC50 |
= |
10553.0 |
nM |
PMID[532376] |
NPT293 |
Individual Protein |
Serotonin 4 (5-HT4) receptor |
Cavia porcellus |
Ki |
= |
1759.0 |
nM |
PMID[532376] |
NPT300 |
Individual Protein |
Thromboxane-A synthase |
Homo sapiens |
IC50 |
= |
494.0 |
nM |
PMID[532376] |
NPT3275 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase epsilon subunit |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Ki |
= |
25.12 |
nM |
PMID[532379] |
NPT3327 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 10 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3318 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 4 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3309 |
Individual Protein |
Leukocyte tyrosine kinase receptor |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3271 |
Individual Protein |
NT-3 growth factor receptor |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3388 |
Individual Protein |
Tyrosine-protein kinase CTK |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3222 |
Individual Protein |
AMP-activated protein kinase, alpha-1 subunit |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1713 |
Individual Protein |
PDZ-binding kinase |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Ki |
= |
19.95 |
nM |
PMID[532379] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Ki |
= |
251.19 |
nM |
PMID[532379] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3368 |
Individual Protein |
cGMP-dependent protein kinase 2 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Ki |
= |
6309.57 |
nM |
PMID[532379] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3316 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
Ki |
= |
398.11 |
nM |
PMID[532379] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3114 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 1A |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3274 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3448 |
Individual Protein |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3280 |
Individual Protein |
Serine/threonine-protein kinase c-TAK1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3350 |
Individual Protein |
Tyrosine-protein kinase Srms |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3258 |
Individual Protein |
Mixed lineage kinase 7 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Ki |
= |
5011.87 |
nM |
PMID[532379] |
NPT1598 |
Individual Protein |
Casein kinase II alpha |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Ki |
= |
39.81 |
nM |
PMID[532379] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3290 |
Individual Protein |
Serine/threonine-protein kinase SIK2 |
Homo sapiens |
Ki |
= |
1000.0 |
nM |
PMID[532379] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Ki |
= |
199.53 |
nM |
PMID[532379] |
NPT3276 |
Individual Protein |
Tyrosine-protein kinase TYK2 |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT3240 |
Individual Protein |
Cyclin-dependent kinase 5 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Ki |
= |
2511.89 |
nM |
PMID[532379] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Ki |
> |
1258.93 |
nM |
PMID[532379] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3396 |
Individual Protein |
Serine/threonine-protein kinase Nek4 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Ki |
= |
1258.93 |
nM |
PMID[532379] |
NPT3168 |
Individual Protein |
Casein kinase I alpha |
Homo sapiens |
Ki |
= |
316.23 |
nM |
PMID[532379] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT286 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-2 |
Homo sapiens |
Ki |
> |
1258.93 |
nM |
PMID[532379] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3366 |
Individual Protein |
Protein kinase C nu |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3458 |
Individual Protein |
Cell division cycle 7-related protein kinase |
Homo sapiens |
Ki |
> |
1258.93 |
nM |
PMID[532379] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3287 |
Individual Protein |
Activin receptor type-1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3120 |
Individual Protein |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT3460 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 3 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3459 |
Individual Protein |
Dual specificity tyrosine-phosphorylation-regulated kinase 4 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Ki |
> |
5011.87 |
nM |
PMID[532379] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Ki |
= |
6309.57 |
nM |
PMID[532379] |
NPT3439 |
Individual Protein |
Homeodomain-interacting protein kinase 4 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3324 |
Individual Protein |
Cell division protein kinase 8 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3346 |
Individual Protein |
Cyclin-dependent kinase 7 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1423 |
Individual Protein |
Cyclin-dependent kinase 1 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Ki |
= |
1584.89 |
nM |
PMID[532379] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3347 |
Individual Protein |
Cyclin-dependent kinase 9 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Ki |
> |
1584.89 |
nM |
PMID[532379] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Ki |
= |
1995.26 |
nM |
PMID[532379] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT3109 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 5 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT3335 |
Individual Protein |
Serine/threonine-protein kinase DCLK1 |
Homo sapiens |
Ki |
> |
10000.0 |
nM |
PMID[532379] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Ki |
> |
1995.26 |
nM |
PMID[532379] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT3231 |
Individual Protein |
Dual specificity protein kinase CLK4 |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
100.0 |
nM |
PMID[532380] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
430.0 |
nM |
PMID[532380] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
22.4 |
% |
PMID[532382] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
50500.0 |
nM |
PMID[532382] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
50.6 |
% |
PMID[532382] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
52200.0 |
nM |
PMID[532382] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
0.0 |
% |
PMID[532382] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
40.0 |
nM |
PMID[532383] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532383] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
37.0 |
nM |
PMID[532384] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3317 |
Individual Protein |
Serine/threonine-protein kinase MARK1 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[532385] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[532385] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
11.0 |
% |
PMID[532385] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[532385] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[532385] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[532385] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
76.0 |
% |
PMID[532385] |
NPT14 |
Individual Protein |
Tyrosine-protein kinase FYN |
Homo sapiens |
Residual Activity |
= |
35.0 |
% |
PMID[532385] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
61.0 |
% |
PMID[532385] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
20.0 |
% |
PMID[532385] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[532385] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT3419 |
Individual Protein |
Serine/threonine-protein kinase SRPK3 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3284 |
Individual Protein |
Serine/threonine-protein kinase NEK7 |
Homo sapiens |
Residual Activity |
= |
116.0 |
% |
PMID[532385] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[532385] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT1432 |
Individual Protein |
Serine/threonine-protein kinase Aurora-A |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[532385] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[532385] |
NPT1721 |
Individual Protein |
Death-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[532385] |
NPT3219 |
Individual Protein |
Ephrin type-A receptor 5 |
Homo sapiens |
Residual Activity |
= |
48.0 |
% |
PMID[532385] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3372 |
Individual Protein |
Fibroblast growth factor receptor 4 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT491 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[532385] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT3236 |
Individual Protein |
Death-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3211 |
Individual Protein |
Ephrin type-A receptor 7 |
Homo sapiens |
Residual Activity |
= |
65.0 |
% |
PMID[532385] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT3406 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase kinase 2 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT1478 |
Individual Protein |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
60.0 |
% |
PMID[532385] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3282 |
Individual Protein |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[532385] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT3331 |
Individual Protein |
Serine/threonine-protein kinase MST2 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT1442 |
Individual Protein |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT1433 |
Individual Protein |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[532385] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
122.0 |
% |
PMID[532385] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
132.0 |
% |
PMID[532385] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[532385] |
NPT3457 |
Individual Protein |
G protein-coupled receptor kinase 5 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
129.0 |
% |
PMID[532385] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3242 |
Individual Protein |
LIM domain kinase 1 |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[532385] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT3381 |
Individual Protein |
Misshapen-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
63.0 |
% |
PMID[532385] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT3206 |
Individual Protein |
Serine/threonine-protein kinase Aurora-C |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3273 |
Individual Protein |
Casein kinase II alpha (prime) |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT3336 |
Individual Protein |
Serine/threonine-protein kinase DCLK2 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3216 |
Individual Protein |
Ephrin type-A receptor 8 |
Homo sapiens |
Residual Activity |
= |
43.0 |
% |
PMID[532385] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT4088 |
Individual Protein |
G protein-coupled receptor kinase 6 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT2574 |
Individual Protein |
Insulin receptor |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3279 |
Individual Protein |
Serine/threonine-protein kinase 11 |
Homo sapiens |
Residual Activity |
= |
85.0 |
% |
PMID[532385] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
43.0 |
% |
PMID[532385] |
NPT3332 |
Individual Protein |
Serine/threonine-protein kinase 24 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
122.0 |
% |
PMID[532385] |
NPT1659 |
Individual Protein |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3303 |
Individual Protein |
Discoidin domain-containing receptor 2 |
Homo sapiens |
Residual Activity |
= |
46.0 |
% |
PMID[532385] |
NPT3212 |
Individual Protein |
Ephrin type-B receptor 1 |
Homo sapiens |
Residual Activity |
= |
56.0 |
% |
PMID[532385] |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3386 |
Individual Protein |
Interleukin-1 receptor-associated kinase 1 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[532385] |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT3320 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase MER |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3245 |
Individual Protein |
Tyrosine kinase non-receptor protein 2 |
Homo sapiens |
Residual Activity |
= |
39.0 |
% |
PMID[532385] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
122.0 |
% |
PMID[532385] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
59.0 |
% |
PMID[532385] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
122.0 |
% |
PMID[532385] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT2941 |
Individual Protein |
Ephrin type-B receptor 2 |
Homo sapiens |
Residual Activity |
= |
61.0 |
% |
PMID[532385] |
NPT3438 |
Individual Protein |
G protein-coupled receptor kinase 7 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT3441 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[532385] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
123.0 |
% |
PMID[532385] |
NPT1337 |
Individual Protein |
Hepatocyte growth factor receptor |
Homo sapiens |
Residual Activity |
= |
68.0 |
% |
PMID[532385] |
NPT1661 |
Individual Protein |
ALK tyrosine kinase receptor |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[532385] |
NPT3215 |
Individual Protein |
Tyrosine-protein kinase BRK |
Homo sapiens |
Residual Activity |
= |
7.0 |
% |
PMID[532385] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
123.0 |
% |
PMID[532385] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT3244 |
Individual Protein |
Tyrosine-protein kinase FER |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3425 |
Individual Protein |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
27.0 |
% |
PMID[532385] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[532385] |
NPT2626 |
Individual Protein |
Myosin light chain kinase, smooth muscle |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3293 |
Individual Protein |
Activin receptor type-1B |
Homo sapiens |
Residual Activity |
= |
23.0 |
% |
PMID[532385] |
NPT3113 |
Individual Protein |
Tyrosine-protein kinase CSK |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT3359 |
Individual Protein |
Ephrin type-B receptor 3 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT1437 |
Individual Protein |
Tyrosine-protein kinase FES |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Residual Activity |
= |
34.0 |
% |
PMID[532385] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3286 |
Individual Protein |
Insulin receptor-related protein |
Homo sapiens |
Residual Activity |
= |
56.0 |
% |
PMID[532385] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[532385] |
NPT13 |
Individual Protein |
Tyrosine-protein kinase LCK |
Homo sapiens |
Residual Activity |
= |
32.0 |
% |
PMID[532385] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3213 |
Individual Protein |
MAP kinase signal-integrating kinase 2 |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[532385] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
143.0 |
% |
PMID[532385] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3312 |
Individual Protein |
Tyrosine-protein kinase BLK |
Homo sapiens |
Residual Activity |
= |
55.0 |
% |
PMID[532385] |
NPT3232 |
Individual Protein |
CaM kinase I alpha |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[532385] |
NPT3399 |
Individual Protein |
Dual-specificity tyrosine-phosphorylation regulated kinase 2 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT2572 |
Individual Protein |
Ephrin type-B receptor 4 |
Homo sapiens |
Residual Activity |
= |
41.0 |
% |
PMID[532385] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[532385] |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
47.0 |
% |
PMID[532385] |
NPT3326 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 9 |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[532385] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT3333 |
Individual Protein |
Muscle, skeletal receptor tyrosine protein kinase |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[532385] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[532385] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1608 |
Individual Protein |
Serine/threonine-protein kinase Chk1 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
1.0 |
% |
PMID[532385] |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
Residual Activity |
= |
-1.0 |
% |
PMID[532385] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT1435 |
Individual Protein |
Receptor protein-tyrosine kinase erbB-4 |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[532385] |
NPT3112 |
Individual Protein |
Tyrosine-protein kinase FGR |
Homo sapiens |
Residual Activity |
= |
51.0 |
% |
PMID[532385] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3444 |
Individual Protein |
Homeodomain-interacting protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT1439 |
Individual Protein |
Tyrosine-protein kinase ITK/TSK |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT3111 |
Individual Protein |
Tyrosine-protein kinase Lyn |
Homo sapiens |
Residual Activity |
= |
13.0 |
% |
PMID[532385] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
124.0 |
% |
PMID[532385] |
NPT3329 |
Individual Protein |
Serine/threonine-protein kinase MRCK-A |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT3443 |
Individual Protein |
Serine/threonine-protein kinase Nek11 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT2750 |
Individual Protein |
Tyrosine-protein kinase BMX |
Homo sapiens |
Residual Activity |
= |
36.0 |
% |
PMID[532385] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
125.0 |
% |
PMID[532385] |
NPT301 |
Individual Protein |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
39.0 |
% |
PMID[532385] |
NPT3432 |
Individual Protein |
Homeodomain-interacting protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3246 |
Individual Protein |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT1660 |
Individual Protein |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3315 |
Individual Protein |
BR serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[532385] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3354 |
Individual Protein |
Ephrin type-A receptor 1 |
Homo sapiens |
Residual Activity |
= |
26.0 |
% |
PMID[532385] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[532385] |
NPT1436 |
Individual Protein |
Focal adhesion kinase 1 |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[532385] |
NPT1650 |
Individual Protein |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
Residual Activity |
= |
82.0 |
% |
PMID[532385] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3409 |
Individual Protein |
Homeodomain-interacting protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1440 |
Individual Protein |
Tyrosine-protein kinase JAK3 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[532385] |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[532385] |
NPT3330 |
Individual Protein |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[532385] |
NPT3391 |
Individual Protein |
Serine/threonine-protein kinase Nek3 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
138.0 |
% |
PMID[532385] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3344 |
Individual Protein |
BR serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Residual Activity |
= |
61.0 |
% |
PMID[532385] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT3225 |
Individual Protein |
Ephrin type-A receptor 2 |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[532385] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
142.0 |
% |
PMID[532385] |
NPT1480 |
Individual Protein |
Fibroblast growth factor receptor 1 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
88.0 |
% |
PMID[532385] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1613 |
Individual Protein |
Ribosomal protein S6 kinase alpha 5 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
120.0 |
% |
PMID[532385] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[532385] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3217 |
Individual Protein |
Ephrin type-A receptor 3 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[532385] |
NPT2573 |
Individual Protein |
Vascular endothelial growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[532385] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT4093 |
Individual Protein |
Serine/threonine-protein kinase haspin |
Homo sapiens |
Residual Activity |
= |
35.0 |
% |
PMID[532385] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT1426 |
Individual Protein |
c-Jun N-terminal kinase 1 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[532385] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[532385] |
NPT1441 |
Individual Protein |
MAP kinase-activated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
133.0 |
% |
PMID[532385] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT3374 |
Individual Protein |
Ribosomal protein S6 kinase alpha 4 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[532385] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT2729 |
Individual Protein |
Tyrosine-protein kinase ABL |
Homo sapiens |
Residual Activity |
= |
72.0 |
% |
PMID[532385] |
NPT3214 |
Individual Protein |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Residual Activity |
= |
125.0 |
% |
PMID[532385] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Residual Activity |
= |
138.0 |
% |
PMID[532385] |
NPT3218 |
Individual Protein |
Ephrin type-A receptor 4 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT1481 |
Individual Protein |
Fibroblast growth factor receptor 2 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[532385] |
NPT3227 |
Individual Protein |
Fibroblast growth factor receptor 3 |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT3267 |
Individual Protein |
Macrophage colony stimulating factor receptor |
Homo sapiens |
Residual Activity |
= |
52.0 |
% |
PMID[532385] |
NPT3205 |
Individual Protein |
Tyrosine-protein kinase HCK |
Homo sapiens |
Residual Activity |
= |
52.0 |
% |
PMID[532385] |
NPT1438 |
Individual Protein |
Insulin-like growth factor I receptor |
Homo sapiens |
Residual Activity |
= |
122.0 |
% |
PMID[532385] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
Residual Activity |
= |
30.0 |
% |
PMID[532385] |
NPT3461 |
Individual Protein |
MAP kinase-activated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[532385] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[532385] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
95.0 |
% |
PMID[532385] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
132.0 |
% |
PMID[532385] |
NPT3349 |
Individual Protein |
Serine/threonine-protein kinase SIK1 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT3269 |
Individual Protein |
Serine/threonine-protein kinase tousled-like 2 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT4094 |
Individual Protein |
Serine/threonine-protein kinase WNK3 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT4094 |
Individual Protein |
Serine/threonine-protein kinase WNK3 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[532385] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT3106 |
Individual Protein |
Ribosomal protein S6 kinase alpha 1 |
Homo sapiens |
Residual Activity |
= |
80.0 |
% |
PMID[532385] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3394 |
Individual Protein |
Protein kinase C iota |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3291 |
Individual Protein |
Serine/threonine-protein kinase SRPK1 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT3299 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Residual Activity |
= |
45.0 |
% |
PMID[532385] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
124.0 |
% |
PMID[532385] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
123.0 |
% |
PMID[532385] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT3292 |
Individual Protein |
Serine/threonine-protein kinase SRPK2 |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT3462 |
Individual Protein |
Testis-specific serine/threonine-protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3259 |
Individual Protein |
Tyrosine-protein kinase ZAP-70 |
Homo sapiens |
Residual Activity |
= |
130.0 |
% |
PMID[532385] |
NPT1430 |
Individual Protein |
Serine/threonine-protein kinase AKT2 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT3364 |
Individual Protein |
Protein kinase C mu |
Homo sapiens |
Residual Activity |
= |
66.0 |
% |
PMID[532385] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3358 |
Individual Protein |
Serine/threonine-protein kinase PLK3 |
Homo sapiens |
Residual Activity |
= |
92.0 |
% |
PMID[532385] |
NPT3234 |
Individual Protein |
Ribosomal protein S6 kinase alpha 2 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT3296 |
Individual Protein |
Serine/threonine-protein kinase 33 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3351 |
Individual Protein |
Tyrosine-protein kinase TEC |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT3247 |
Individual Protein |
Serine/threonine-protein kinase PAK 3 |
Homo sapiens |
Residual Activity |
= |
78.0 |
% |
PMID[532385] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT2546 |
Individual Protein |
Serine/threonine-protein kinase AKT3 |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[532385] |
NPT3365 |
Individual Protein |
Serine/threonine-protein kinase D2 |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT3262 |
Individual Protein |
Serine/threonine-protein kinase PRKX |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT3254 |
Individual Protein |
Ribosomal protein S6 kinase alpha 6 |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
116.0 |
% |
PMID[532385] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
17.0 |
% |
PMID[532385] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT182 |
Individual Protein |
Protein kinase C alpha |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[532385] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
5.0 |
% |
PMID[532385] |
NPT3414 |
Individual Protein |
Serine/threonine-protein kinase PLK2 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT2576 |
Individual Protein |
Tyrosine-protein kinase TIE-2 |
Homo sapiens |
Residual Activity |
= |
62.0 |
% |
PMID[532385] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Residual Activity |
= |
121.0 |
% |
PMID[532385] |
NPT1424 |
Individual Protein |
Serine/threonine-protein kinase RAF |
Homo sapiens |
Residual Activity |
= |
3.0 |
% |
PMID[532385] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
125.0 |
% |
PMID[532385] |
NPT3263 |
Individual Protein |
Protein tyrosine kinase 2 beta |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[532385] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[532385] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
24.0 |
% |
PMID[532385] |
NPT1449 |
Individual Protein |
Tyrosine-protein kinase SYK |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3239 |
Individual Protein |
Nerve growth factor receptor Trk-A |
Homo sapiens |
Residual Activity |
= |
115.0 |
% |
PMID[532385] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT1479 |
Individual Protein |
Stem cell growth factor receptor |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3367 |
Individual Protein |
cGMP-dependent protein kinase 1 beta |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
145.0 |
% |
PMID[532385] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Residual Activity |
= |
21.0 |
% |
PMID[532385] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Residual Activity |
= |
2.0 |
% |
PMID[532385] |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT3442 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT3270 |
Individual Protein |
Neurotrophic tyrosine kinase receptor type 2 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
112.0 |
% |
PMID[532385] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT1612 |
Individual Protein |
MAP kinase-activated protein kinase 5 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[532385] |
NPT592 |
Individual Protein |
Rho-associated protein kinase 1 |
Homo sapiens |
Residual Activity |
= |
74.0 |
% |
PMID[532385] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT1615 |
Individual Protein |
MAP kinase p38 gamma |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[532385] |
NPT36 |
Individual Protein |
Tyrosine-protein kinase SRC |
Homo sapiens |
Residual Activity |
= |
65.0 |
% |
PMID[532385] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3235 |
Individual Protein |
MAP/microtubule affinity-regulating kinase 2 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
119.0 |
% |
PMID[532385] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3431 |
Individual Protein |
Serine/threonine-protein kinase TAO1 |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[532385] |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3272 |
Individual Protein |
Tyrosine-protein kinase TXK |
Homo sapiens |
Residual Activity |
= |
42.0 |
% |
PMID[532385] |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
120.0 |
% |
PMID[532385] |
NPT1344 |
Individual Protein |
Serine/threonine-protein kinase EEF2K |
Homo sapiens |
Residual Activity |
= |
91.0 |
% |
PMID[532385] |
NPT3454 |
Individual Protein |
PAS domain-containing serine/threonine-protein kinase |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT3357 |
Individual Protein |
Protein kinase N2 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
71.0 |
% |
PMID[532385] |
NPT3107 |
Individual Protein |
Rho-associated protein kinase 2 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT3426 |
Individual Protein |
Serine/threonine-protein kinase TAO2 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT3422 |
Individual Protein |
Serine/threonine-protein kinase ULK2 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3204 |
Individual Protein |
Tyrosine-protein kinase FRK |
Homo sapiens |
Residual Activity |
= |
17.0 |
% |
PMID[532385] |
NPT3370 |
Individual Protein |
Tyrosine-protein kinase receptor RET |
Homo sapiens |
Residual Activity |
= |
46.0 |
% |
PMID[532385] |
NPT1448 |
Individual Protein |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
Residual Activity |
= |
124.0 |
% |
PMID[532385] |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3427 |
Individual Protein |
Serine/threonine-protein kinase TAO3 |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT3382 |
Individual Protein |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT3020 |
Individual Protein |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3223 |
Individual Protein |
Phosphorylase kinase gamma subunit 2 |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT3390 |
Individual Protein |
Macrophage-stimulating protein receptor |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
124.0 |
% |
PMID[532385] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
114.0 |
% |
PMID[532385] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT2575 |
Individual Protein |
Platelet-derived growth factor receptor beta |
Homo sapiens |
Residual Activity |
= |
120.0 |
% |
PMID[532385] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT3455 |
Individual Protein |
Protein kinase C zeta |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
84.0 |
% |
PMID[532385] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT3456 |
Individual Protein |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
Residual Activity |
= |
81.0 |
% |
PMID[532385] |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
120.0 |
% |
PMID[532385] |
NPT3417 |
Individual Protein |
Serine/threonine-protein kinase TBK1 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
130.0 |
% |
PMID[532385] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT1611 |
Individual Protein |
Ribosomal protein S6 kinase 1 |
Homo sapiens |
Residual Activity |
= |
87.0 |
% |
PMID[532385] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT3124 |
Individual Protein |
Protein kinase C eta |
Homo sapiens |
Residual Activity |
= |
79.0 |
% |
PMID[532385] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Residual Activity |
= |
97.0 |
% |
PMID[532385] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Residual Activity |
= |
125.0 |
% |
PMID[532385] |
NPT3373 |
Individual Protein |
Proto-oncogene tyrosine-protein kinase ROS |
Homo sapiens |
Residual Activity |
= |
110.0 |
% |
PMID[532385] |
NPT3277 |
Individual Protein |
Tyrosine-protein kinase receptor TYRO3 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT3418 |
Individual Protein |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT3353 |
Individual Protein |
TGF-beta receptor type I |
Homo sapiens |
Residual Activity |
= |
77.0 |
% |
PMID[532385] |
NPT4096 |
Individual Protein |
Serine/threonine-protein kinase WNK2 |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
273.0 |
nM |
PMID[532386] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532386] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Inhibition |
< |
40.0 |
% |
PMID[532387] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
Inhibition |
= |
80.0 |
% |
PMID[532387] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
> |
10000.0 |
nM |
PMID[532387] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
340.0 |
nM |
PMID[532387] |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
1000.0 |
nM |
PMID[532387] |
NPT3464 |
Individual Protein |
Myelin transcription factor 1 |
Homo sapiens |
Activity |
< |
5.0 |
% |
PMID[532391] |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
n.a. |
33498.3 |
nM |
PMID[532369] |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
n.a. |
14963.1 |
nM |
PMID[532368] |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
n.a. |
29855.4 |
nM |
PMID[532368] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
25.0 |
nM |
PMID[532393] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
68.1 |
% |
PMID[532394] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
8600.0 |
nM |
PMID[532394] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Inhibition |
= |
8.4 |
% |
PMID[532394] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
52200.0 |
nM |
PMID[532394] |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
Activity |
= |
0.0 |
% |
PMID[532394] |
NPT1814 |
Individual Protein |
Glucagon receptor |
Homo sapiens |
IC50 |
= |
37.07 |
nM |
PMID[532398] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
723.0 |
nM |
PMID[532399] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532399] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
40.0 |
nM |
PMID[532400] |
NPT1663 |
Individual Protein |
Tyrosine-protein kinase YES |
Homo sapiens |
Potency |
n.a. |
10909.6 |
nM |
PMID[532368] |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
n.a. |
12589.3 |
nM |
PMID[532368] |
NPT49 |
Individual Protein |
DNA-(apurinic or apyrimidinic site) lyase |
Homo sapiens |
Potency |
n.a. |
39810.7 |
nM |
PMID[532370] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
19.0 |
nM |
PMID[532402] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
35.0 |
nM |
PMID[532403] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
IC50 |
= |
105.0 |
nM |
PMID[532406] |
NPT1699 |
Individual Protein |
3-phosphoinositide dependent protein kinase-1 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1265 |
Individual Protein |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
Thermal melting change |
= |
-2.1 |
degrees C |
PMID[532343] |
NPT1700 |
Individual Protein |
Serine/threonine-protein kinase PIM2 |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1701 |
Individual Protein |
Serine/threonine-protein kinase PIM3 |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1702 |
Individual Protein |
Serine/threonine-protein kinase PLK4 |
Homo sapiens |
Thermal melting change |
= |
0.7 |
degrees C |
PMID[532343] |
NPT1703 |
Individual Protein |
cAMP-dependent protein kinase alpha-catalytic subunit |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1704 |
Individual Protein |
Serine/threonine-protein kinase RIO2 |
Homo sapiens |
Thermal melting change |
= |
-0.2 |
degrees C |
PMID[532343] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Thermal melting change |
= |
0.3 |
degrees C |
PMID[532343] |
NPT1705 |
Individual Protein |
Ribosomal protein S6 kinase alpha 3 |
Homo sapiens |
Thermal melting change |
= |
-0.2 |
degrees C |
PMID[532343] |
NPT1706 |
Individual Protein |
Serine/threonine-protein kinase 2 |
Homo sapiens |
Thermal melting change |
= |
3.9 |
degrees C |
PMID[532343] |
NPT1707 |
Individual Protein |
Serine/threonine-protein kinase 10 |
Homo sapiens |
Thermal melting change |
= |
2.7 |
degrees C |
PMID[532343] |
NPT1708 |
Individual Protein |
Serine/threonine-protein kinase 16 |
Homo sapiens |
Thermal melting change |
= |
0.4 |
degrees C |
PMID[532343] |
NPT1709 |
Individual Protein |
Serine/threonine-protein kinase 17A |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1710 |
Individual Protein |
Serine/threonine-protein kinase 38 |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Thermal melting change |
= |
-0.4 |
degrees C |
PMID[532343] |
NPT1711 |
Individual Protein |
Serine/threonine-protein kinase MST1 |
Homo sapiens |
Thermal melting change |
= |
1.0 |
degrees C |
PMID[532343] |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
Thermal melting change |
= |
2.0 |
degrees C |
PMID[532343] |
NPT1713 |
Individual Protein |
PDZ-binding kinase |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT1715 |
Individual Protein |
Serine/threonine-protein kinase VRK2 |
Homo sapiens |
Thermal melting change |
= |
0.6 |
degrees C |
PMID[532343] |
NPT1717 |
Individual Protein |
Serine/threonine-protein kinase 25 |
Homo sapiens |
Thermal melting change |
= |
0.9 |
degrees C |
PMID[532343] |
NPT1671 |
Individual Protein |
AMP-activated protein kinase, alpha-2 subunit |
Homo sapiens |
Thermal melting change |
= |
-0.9 |
degrees C |
PMID[532343] |
NPT1672 |
Individual Protein |
CaM kinase I delta |
Homo sapiens |
Thermal melting change |
= |
-0.2 |
degrees C |
PMID[532343] |
NPT1673 |
Individual Protein |
CaM kinase I gamma |
Homo sapiens |
Thermal melting change |
= |
-0.2 |
degrees C |
PMID[532343] |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
Thermal melting change |
= |
0.3 |
degrees C |
PMID[532343] |
NPT1630 |
Individual Protein |
CaM kinase II beta |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1675 |
Individual Protein |
CaM kinase II delta |
Homo sapiens |
Thermal melting change |
= |
-0.3 |
degrees C |
PMID[532343] |
NPT1676 |
Individual Protein |
CaM kinase II gamma |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1677 |
Individual Protein |
CaM kinase IV |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1678 |
Individual Protein |
CaM-kinase kinase beta |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1371 |
Individual Protein |
Cyclin-dependent kinase 2 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1571 |
Individual Protein |
Cyclin-dependent kinase 6 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1679 |
Individual Protein |
Cyclin-dependent kinase-like 1 |
Homo sapiens |
Thermal melting change |
= |
-0.4 |
degrees C |
PMID[532343] |
NPT1680 |
Individual Protein |
Serine/threonine-protein kinase Chk2 |
Homo sapiens |
Thermal melting change |
= |
-0.5 |
degrees C |
PMID[532343] |
NPT1681 |
Individual Protein |
Dual specificty protein kinase CLK1 |
Homo sapiens |
Thermal melting change |
= |
-0.3 |
degrees C |
PMID[532343] |
NPT1682 |
Individual Protein |
Dual specificity protein kinase CLK2 |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT1683 |
Individual Protein |
Dual specificity protein kinase CLK3 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1684 |
Individual Protein |
Casein kinase I gamma 1 |
Homo sapiens |
Thermal melting change |
= |
0.8 |
degrees C |
PMID[532343] |
NPT1685 |
Individual Protein |
Casein kinase I gamma 2 |
Homo sapiens |
Thermal melting change |
= |
0.7 |
degrees C |
PMID[532343] |
NPT1686 |
Individual Protein |
Casein kinase I isoform gamma-3 |
Homo sapiens |
Thermal melting change |
= |
0.4 |
degrees C |
PMID[532343] |
NPT1687 |
Individual Protein |
Death-associated protein kinase 3 |
Homo sapiens |
Thermal melting change |
= |
-0.4 |
degrees C |
PMID[532343] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
Thermal melting change |
= |
0.1 |
degrees C |
PMID[532343] |
NPT591 |
Individual Protein |
Glycogen synthase kinase-3 beta |
Homo sapiens |
Thermal melting change |
= |
3.5 |
degrees C |
PMID[532343] |
NPT1689 |
Individual Protein |
Tyrosine-protein kinase JAK1 |
Homo sapiens |
Thermal melting change |
= |
2.3 |
degrees C |
PMID[532343] |
NPT1690 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 2 |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT1691 |
Individual Protein |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1431 |
Individual Protein |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
Thermal melting change |
= |
0.3 |
degrees C |
PMID[532343] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
Thermal melting change |
= |
9.6 |
degrees C |
PMID[532343] |
NPT281 |
Individual Protein |
MAP kinase ERK1 |
Homo sapiens |
Thermal melting change |
= |
0.1 |
degrees C |
PMID[532343] |
NPT1692 |
Individual Protein |
Mitogen-activated protein kinase 6 |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1693 |
Individual Protein |
Serine/threonine-protein kinase MST4 |
Homo sapiens |
Thermal melting change |
= |
-0.5 |
degrees C |
PMID[532343] |
NPT1658 |
Individual Protein |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
Thermal melting change |
= |
0.3 |
degrees C |
PMID[532343] |
NPT1657 |
Individual Protein |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT1694 |
Individual Protein |
Serine/threonine-protein kinase OSR1 |
Homo sapiens |
Thermal melting change |
= |
-0.2 |
degrees C |
PMID[532343] |
NPT1695 |
Individual Protein |
Serine/threonine-protein kinase PAK 4 |
Homo sapiens |
Thermal melting change |
= |
0.1 |
degrees C |
PMID[532343] |
NPT1696 |
Individual Protein |
Serine/threonine-protein kinase PAK7 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT1697 |
Individual Protein |
Serine/threonine-protein kinase PAK6 |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT1698 |
Individual Protein |
Serine/threonine-protein kinase PCTAIRE-1 |
Homo sapiens |
Thermal melting change |
= |
-0.8 |
degrees C |
PMID[532343] |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
53.0 |
% |
PMID[532407] |
NPT6603 |
Individual Protein |
P2X purinoceptor 7 |
Rattus norvegicus |
IC50 |
> |
30000.0 |
nM |
PMID[532408] |
NPT2654 |
Individual Protein |
P2X purinoceptor 7 |
Homo sapiens |
IC50 |
= |
5000.0 |
nM |
PMID[532408] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
T1/2 |
= |
0.006667 |
hr |
PMID[532409] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
K |
= |
0.0317 |
/s |
PMID[532409] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
10.0 |
nM |
PMID[532409] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
200.0 |
nM |
PMID[532409] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
251.19 |
nM |
PMID[532412] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
250.0 |
nM |
PMID[532412] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
= |
6310.0 |
nM |
PMID[532412] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
Ratio IC50 |
= |
25.0 |
n.a. |
PMID[532412] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
25.0 |
nM |
PMID[532413] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
= |
12.0 |
nM |
PMID[532413] |
NPT2816 |
Individual Protein |
Bromodomain-containing protein 4 |
Homo sapiens |
Delta Tm |
= |
1.3 |
degrees C |
PMID[532413] |
NPT1614 |
Individual Protein |
MAP kinase p38 delta |
Homo sapiens |
IC50 |
= |
87600000.0 |
nM |
PMID[532414] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
21.7 |
nM |
PMID[532417] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
T1/2 |
= |
0.0008889 |
hr |
PMID[532417] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
TIME |
= |
0.001278 |
hr |
PMID[532417] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Kd |
= |
2.18 |
10'-1/s |
PMID[532417] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Ka |
= |
1.0 |
10'7/M.s |
PMID[532417] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
EC50 |
= |
60.0 |
nM |
PMID[532422] |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
20.0 |
nM |
PMID[532422] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
35.0 |
nM |
PMID[532424] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
41.0 |
nM |
PMID[532425] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
65.0 |
nM |
PMID[532425] |
NPT2739 |
Individual Protein |
Tyrosinase |
Mus musculus |
IC50 |
= |
34.0 |
nM |
PMID[532426] |
NPT1616 |
Individual Protein |
MAP kinase p38 beta |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3266 |
Individual Protein |
Casein kinase I delta |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT1427 |
Individual Protein |
c-Jun N-terminal kinase 2 |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3207 |
Individual Protein |
c-Jun N-terminal kinase 3 |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT1712 |
Individual Protein |
TRAF2- and NCK-interacting kinase |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT1434 |
Individual Protein |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3334 |
Individual Protein |
Citron Rho-interacting kinase |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3226 |
Individual Protein |
Casein kinase I epsilon |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT1688 |
Individual Protein |
Myotonin-protein kinase |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3221 |
Individual Protein |
Serine/threonine-protein kinase GAK |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3285 |
Individual Protein |
Serine/threonine protein kinase NLK |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT1447 |
Individual Protein |
Serine/threonine-protein kinase RIPK2 |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT3208 |
Individual Protein |
Serine/threonine-protein kinase 36 |
Homo sapiens |
IC50 |
< |
1000.0 |
nM |
PMID[532432] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Delta Tm |
= |
6.8 |
degrees C |
PMID[532434] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Tm |
= |
56.8 |
degrees C |
PMID[532434] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
Activity |
= |
75.0 |
% |
PMID[532434] |
NPT2615 |
Cell Line |
HEK-293T |
Homo sapiens |
Cell Viability |
= |
0.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
16.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
9.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
0.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
5.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
38.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
0.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
3.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
2.0 |
n.a. |
PMID[532435] |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Cell Viability |
= |
1.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
4.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
1.0 |
n.a. |
PMID[532435] |
NPT4909 |
Cell Line |
Fibroblasts |
|
Cell Viability |
= |
2.0 |
n.a. |
PMID[532435] |
NPT283 |
Individual Protein |
MAP kinase p38 alpha |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[532436] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
590.0 |
nM |
PMID[532298] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
37.0 |
nM |
PMID[532298] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
940.0 |
nM |
PMID[532298] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
350.0 |
nM |
PMID[532298] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
72.0 |
nM |
PMID[532300] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
25.0 |
nM |
PMID[532302] |
NPT321 |
Protein Family |
cAMP-dependent protein kinase (PKA) |
Homo sapiens |
Inhibition |
= |
0.0 |
% |
PMID[532303] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
83.0 |
% |
PMID[532303] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
33.0 |
% |
PMID[532303] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
39.0 |
nM |
PMID[532306] |
NPT4148 |
Protein Family |
Dual specificity mitogen-activated protein kinase kinase; MEK1/2 |
Homo sapiens |
IC50 |
= |
61000.0 |
nM |
PMID[532306] |
NPT321 |
Protein Family |
cAMP-dependent protein kinase (PKA) |
Homo sapiens |
IC50 |
= |
50000.0 |
nM |
PMID[532306] |
NPT316 |
Protein Family |
Protein kinase C (PKC) |
Homo sapiens |
IC50 |
= |
75000.0 |
nM |
PMID[532306] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
1000.0 |
nM |
PMID[532306] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
290.0 |
nM |
PMID[532307] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
590.0 |
nM |
PMID[532307] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
37.0 |
nM |
PMID[532307] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
940.0 |
nM |
PMID[532307] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
350.0 |
nM |
PMID[532307] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ID50 |
= |
80.0 |
mg kg-1 day-1 |
PMID[532308] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
74.0 |
% |
PMID[532308] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
83.0 |
nM |
PMID[532308] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
360.0 |
nM |
PMID[532310] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
940.0 |
nM |
PMID[532310] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
350.0 |
nM |
PMID[532310] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
590.0 |
nM |
PMID[532310] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
37.0 |
nM |
PMID[532310] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
80.0 |
% |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
-1.4 |
% |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
< |
65.4 |
% |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.0 |
n.a. |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
IC |
= |
0.63 |
n.a. |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
IO |
= |
0.25 |
n.a. |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
38.0 |
ng ml-1 |
PMID[532311] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
13.0 |
ng ml-1 |
PMID[532311] |
NPT35 |
Others |
n.a. |
|
CLogP |
= |
3.6 |
n.a. |
PMID[532312] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
42.0 |
nM |
PMID[532313] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Change |
= |
-83.0 |
% |
PMID[532313] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
Kd |
= |
10.0 |
nM |
PMID[532314] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
EC50 |
= |
60.0 |
nM |
PMID[532314] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
42.0 |
nM |
PMID[532316] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
48.0 |
nM |
PMID[532316] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
50.0 |
nM |
PMID[532317] |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
400000.0 |
nM |
PMID[532317] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37.0 |
nM |
PMID[532318] |
NPT27 |
Others |
Unspecified |
|
IC50 |
= |
190.0 |
nM |
PMID[532322] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
4200.0 |
nM |
PMID[532322] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
50.0 |
% |
PMID[532322] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
47.0 |
% |
PMID[532322] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
0.0 |
% |
PMID[532322] |
NPT605 |
Organism |
Homo sapiens |
Homo sapiens |
IC50 |
= |
2000.0 |
nM |
PMID[532323] |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
6800.0 |
nM |
PMID[532324] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7800.0 |
nM |
PMID[532324] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
290.0 |
nM |
PMID[532328] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
70.0 |
nM |
PMID[532328] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
136.0 |
nM |
PMID[532329] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
136.0 |
nM |
PMID[532332] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
2640.0 |
nM |
PMID[532335] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
1117.0 |
nM |
PMID[532335] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
56.0 |
nM |
PMID[532336] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
42.0 |
nM |
PMID[532337] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
34.0 |
nM |
PMID[532343] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
600.0 |
nM |
PMID[532343] |
NPT20967 |
CELL-LINE |
Platelet |
n.a. |
IC50 |
= |
200.0 |
nM |
PMID[532343] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
2300.0 |
nM |
PMID[532347] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
1980.0 |
nM |
PMID[532347] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0.0 |
% |
PMID[532347] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
4.0 |
% |
PMID[532347] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Inhibition |
= |
38.0 |
% |
PMID[532347] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
100.0 |
nM |
PMID[532348] |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
IC50 |
= |
8500.0 |
nM |
PMID[532350] |
NPT486 |
Organism |
Toxoplasma gondii |
Toxoplasma gondii |
IC50 |
= |
2500.0 |
nM |
PMID[532350] |
NPT2255 |
Organism |
Toxoplasma gondii RH |
Toxoplasma gondii RH |
Activity |
= |
30.0 |
day |
PMID[532350] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
6400.0 |
nM |
PMID[532351] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ID50 |
= |
27.9 |
mg.kg-1 |
PMID[532351] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
104.0 |
% |
PMID[532353] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Activity |
= |
89.0 |
% |
PMID[532353] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
80.0 |
% |
PMID[532353] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Activity |
= |
104.0 |
% |
PMID[532353] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Activity |
= |
98.0 |
% |
PMID[532353] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Activity |
= |
95.0 |
% |
PMID[532353] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532352] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Activity |
= |
97.0 |
% |
PMID[532353] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
1760.0 |
nM |
PMID[532360] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
104.0 |
% |
PMID[532364] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Inhibition |
= |
97.0 |
% |
PMID[532364] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
96.0 |
% |
PMID[532364] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Inhibition |
= |
62.0 |
% |
PMID[532364] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
83.0 |
% |
PMID[532364] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
99.0 |
% |
PMID[532364] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Inhibition |
= |
84.3 |
% |
PMID[532366] |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PMID[532368] |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PMID[532369] |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PMID[532368] |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PMID[532370] |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PMID[532368] |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
7079.5 |
nM |
PMID[532368] |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
12589.3 |
nM |
PMID[532369] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
190.0 |
nM |
PMID[532374] |
NPT698 |
Individual Protein |
Regulator of G-protein signaling 4 |
Homo sapiens |
Potency |
n.a. |
2993.5 |
nM |
PMID[532370] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Kd |
> |
10000.0 |
nM |
PMID[532375] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5923.0 |
nM |
PMID[532376] |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
2026.0 |
nM |
PMID[532376] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11590.0 |
nM |
PMID[532376] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
Inhibition |
= |
62.0 |
% |
PMID[532377] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
73.0 |
% |
PMID[532377] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
7240.0 |
nM |
PMID[532378] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3530.0 |
nM |
PMID[532378] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5020.0 |
nM |
PMID[532378] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Ki |
> |
3162.28 |
nM |
PMID[532379] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Ki |
> |
2511.89 |
nM |
PMID[532379] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Ki |
> |
3981.07 |
nM |
PMID[532379] |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Ki |
> |
6309.57 |
nM |
PMID[532379] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Ki |
> |
7943.28 |
nM |
PMID[532379] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
220.0 |
nM |
PMID[532381] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
4685.9 |
nM |
PMID[532369] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
2.6 |
nM |
PMID[532369] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
2093.1 |
nM |
PMID[532369] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT2544 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin E |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT981 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase beta subunit |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT1609 |
Protein Complex |
Casein kinase II |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT4087 |
Protein Complex |
CDK3/cyclin E |
Homo sapiens |
Residual Activity |
= |
93.0 |
% |
PMID[532385] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
121.0 |
% |
PMID[532385] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
120.0 |
% |
PMID[532385] |
NPT1509 |
Protein Complex |
Cyclin-dependent kinase 5/CDK5 activator 1 |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
116.0 |
% |
PMID[532385] |
NPT4089 |
Protein Complex |
CDK6/cyclin D3 |
Homo sapiens |
Residual Activity |
= |
111.0 |
% |
PMID[532385] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
118.0 |
% |
PMID[532385] |
NPT676 |
Individual Protein |
Glycogen synthase kinase-3 alpha |
Homo sapiens |
Residual Activity |
= |
49.0 |
% |
PMID[532385] |
NPT833 |
Individual Protein |
Tyrosine-protein kinase BTK |
Homo sapiens |
Residual Activity |
= |
73.0 |
% |
PMID[532385] |
NPT4090 |
Protein Complex |
Cyclin-dependent kinase 7/ cyclin H |
Homo sapiens |
Residual Activity |
= |
100.0 |
% |
PMID[532385] |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
98.0 |
% |
PMID[532385] |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
109.0 |
% |
PMID[532385] |
NPT4091 |
Protein Complex |
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 |
Homo sapiens |
Residual Activity |
= |
94.0 |
% |
PMID[532385] |
NPT4092 |
Protein Complex |
CDK9/cyclin T1 |
Homo sapiens |
Residual Activity |
= |
108.0 |
% |
PMID[532385] |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT1767 |
Protein Complex |
AMP-activated protein kinase, AMPK |
Homo sapiens |
Residual Activity |
= |
90.0 |
% |
PMID[532385] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Residual Activity |
= |
107.0 |
% |
PMID[532385] |
NPT1561 |
Protein Complex |
Cyclin-dependent kinase 1/cyclin B1 |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT3814 |
Protein Complex |
Cyclin-dependent kinase 2/cyclin A |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT982 |
Individual Protein |
Inhibitor of nuclear factor kappa B kinase alpha subunit |
Homo sapiens |
Residual Activity |
= |
113.0 |
% |
PMID[532385] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
102.0 |
% |
PMID[532385] |
NPT728 |
Individual Protein |
Serine/threonine-protein kinase AKT |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
117.0 |
% |
PMID[532385] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Residual Activity |
= |
99.0 |
% |
PMID[532385] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
101.0 |
% |
PMID[532385] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
70.0 |
% |
PMID[532385] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT760 |
Individual Protein |
Protein kinase C beta |
Homo sapiens |
Residual Activity |
= |
75.0 |
% |
PMID[532385] |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
104.0 |
% |
PMID[532385] |
NPT880 |
Individual Protein |
Protein kinase C gamma |
Homo sapiens |
Residual Activity |
= |
103.0 |
% |
PMID[532385] |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
106.0 |
% |
PMID[532385] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
89.0 |
% |
PMID[532385] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
125.0 |
% |
PMID[532385] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
86.0 |
% |
PMID[532385] |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
Residual Activity |
= |
105.0 |
% |
PMID[532385] |
NPT940 |
Individual Protein |
Serine/threonine-protein kinase mTOR |
Homo sapiens |
Residual Activity |
= |
96.0 |
% |
PMID[532385] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
7370.0 |
nM |
PMID[532388] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3560.0 |
nM |
PMID[532388] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5670.0 |
nM |
PMID[532388] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5000.0 |
nM |
PMID[532389] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
7530.0 |
nM |
PMID[532390] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5210.0 |
nM |
PMID[532390] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3450.0 |
nM |
PMID[532390] |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
70.0 |
% |
PMID[532392] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
6.0 |
n.a. |
PMID[532393] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
7500.0 |
nM |
PMID[532396] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
5000.0 |
nM |
PMID[532396] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
IC50 |
= |
3500.0 |
nM |
PMID[532396] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
23485.0 |
nM |
PMID[532369] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
14950.2 |
nM |
PMID[532369] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
29565.9 |
nM |
PMID[532369] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
6853.0 |
nM |
PMID[532401] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
19952.6 |
nM |
PMID[532370] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
8912.5 |
nM |
PMID[532368] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
25118.9 |
nM |
PMID[532369] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
18821.2 |
nM |
PMID[532369] |
NPT35 |
Others |
n.a. |
|
LogD7.4 |
n.a. |
3.34 |
n.a. |
PMID[532404] |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Thermal melting change |
= |
0.2 |
degrees C |
PMID[532343] |
NPT22960 |
SINGLE PROTEIN |
Serine/threonine-protein kinase VRK1 |
Homo sapiens |
Thermal melting change |
= |
-0.1 |
degrees C |
PMID[532343] |
NPT22961 |
SINGLE PROTEIN |
Inactive serine/threonine-protein kinase VRK3 |
Homo sapiens |
Thermal melting change |
= |
0.0 |
degrees C |
PMID[532343] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
16626.1 |
nM |
PMID[532369] |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2.5 |
n.a. |
PMID[532410] |
NPT25835 |
SINGLE PROTEIN |
Bromodomain testis-specific protein |
Homo sapiens |
Delta Tm |
= |
0.85 |
degrees C |
PMID[532413] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3500.0 |
nM |
PMID[532415] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5000.0 |
nM |
PMID[532415] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7200.0 |
nM |
PMID[532415] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[532416] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
37.0 |
% |
PMID[532418] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
220.0 |
nM |
PMID[532419] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
-0.92 |
% |
PMID[532420] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
3018.0 |
nM |
PMID[532423] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
Inhibition |
= |
76.5 |
% |
PMID[532423] |
NPT1308 |
Tissue |
Blood |
Homo sapiens |
IC50 |
= |
3202.0 |
nM |
PMID[532425] |
NPT207 |
Protein Family |
MAP kinase p38 |
Homo sapiens |
IC50 |
= |
500.0 |
nM |
PMID[532427] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
24.88 |
% |
PMID[532428] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
9.655 |
% |
PMID[532429] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
0.28 |
% |
PMID[532430] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
0.02 |
% |
PMID[532431] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
IC50 |
> |
20000.0 |
nM |
PMID[532433] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
IC50 |
> |
19952.62 |
nM |
PMID[532433] |