Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT420 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Cavia porcellus |
pD2 |
= |
6.5 |
n.a. |
PMID[466203] |
NPT420 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Cavia porcellus |
Efficiency |
= |
100.0 |
% |
PMID[466203] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Inhibition |
= |
13.0 |
% |
PMID[466205] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ki |
= |
14.0 |
nM |
PMID[466205] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki |
= |
40.0 |
nM |
PMID[466205] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
inhibition (at 100uM) |
= |
42.0 |
% |
PMID[466205] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki |
= |
2400.0 |
nM |
PMID[466205] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki |
= |
26.0 |
nM |
PMID[466205] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
Inhibition |
= |
99.4 |
% |
PMID[466206] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
Ki |
= |
3.33 |
nM |
PMID[466206] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
Inhibition |
= |
101.0 |
% |
PMID[466206] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
Ki |
= |
5.45 |
nM |
PMID[466206] |
NPT1296 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Mus musculus |
Inhibition |
= |
65.0 |
% |
PMID[466206] |
NPT1296 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Mus musculus |
Km |
= |
2.4 |
nM |
PMID[466206] |
NPT1296 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Mus musculus |
Inhibition |
= |
35.0 |
% |
PMID[466206] |
NPT1296 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Mus musculus |
KL |
= |
0.56 |
nM |
PMID[466206] |
NPT1297 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Mus musculus |
Inhibition |
= |
100.0 |
% |
PMID[466206] |
NPT1297 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Mus musculus |
KL |
= |
0.87 |
nM |
PMID[466206] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
EC50 |
= |
27000.0 |
nM |
PMID[466206] |
NPT1295 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Mus musculus |
Smax |
= |
180.0 |
% |
PMID[466206] |
NPT1297 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Mus musculus |
EC50 |
= |
12000.0 |
nM |
PMID[466206] |
NPT1297 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Mus musculus |
Smax |
= |
96.0 |
% |
PMID[466206] |
NPT1298 |
Cell Line |
A9 |
Mus musculus |
IC50 |
= |
1200.0 |
nM |
PMID[466206] |
NPT1298 |
Cell Line |
A9 |
Mus musculus |
Inhibition |
= |
12.0 |
% |
PMID[466206] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
115500.0 |
nM |
PMID[466208] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
115.0 |
nM |
PMID[466208] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ratio |
= |
1001.62 |
n.a. |
PMID[466208] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
EC50 |
= |
83.0 |
nM |
PMID[466210] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
EC50 |
= |
3200.0 |
nM |
PMID[466215] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
EC50 |
= |
25.0 |
nM |
PMID[466215] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
EC50 |
= |
340.0 |
nM |
PMID[466215] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
EC50 |
= |
130.0 |
nM |
PMID[466215] |
NPT266 |
Individual Protein |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
EC50 |
= |
600.0 |
nM |
PMID[466215] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Max PI |
= |
25.0 |
% |
PMID[466216] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Max PI |
= |
51.0 |
% |
PMID[466216] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
EC50 |
= |
5603.0 |
nM |
PMID[466216] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Max cAMP |
= |
119.0 |
% |
PMID[466216] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
EC50 |
= |
10000.0 |
nM |
PMID[466216] |
NPT1301 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Rattus norvegicus |
IC50 |
= |
11000.0 |
nM |
PMID[466218] |
NPT1301 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Rattus norvegicus |
IC50 |
= |
590.0 |
nM |
PMID[466218] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
EC50 |
= |
100.0 |
nM |
PMID[466219] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ki |
= |
29000.0 |
nM |
PMID[466220] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki |
= |
2400.0 |
nM |
PMID[466220] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
Ki |
= |
43000.0 |
nM |
PMID[466220] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki |
= |
60000.0 |
nM |
PMID[466220] |
NPT266 |
Individual Protein |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
Ki |
= |
56000.0 |
nM |
PMID[466220] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
65000.0 |
nM |
PMID[466228] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
IC50 |
= |
1800.0 |
nM |
PMID[466228] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
IC50 |
= |
11000.0 |
nM |
PMID[466228] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
IC50 |
= |
13500.0 |
nM |
PMID[466228] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ratio |
= |
165.0 |
n.a. |
PMID[466228] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Max |
= |
95.0 |
% |
PMID[466231] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
545.0 |
nM |
PMID[466231] |
NPT1298 |
Cell Line |
A9 |
Mus musculus |
Max |
= |
73.0 |
% |
PMID[466232] |
NPT1298 |
Cell Line |
A9 |
Mus musculus |
EC50 |
= |
3080000.0 |
nM |
PMID[466232] |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
PI turnover |
= |
69.0 |
% |
PMID[466233] |
NPT1301 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Rattus norvegicus |
IC50 |
= |
9150.0 |
nM |
PMID[466233] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ratio |
= |
0.8 |
n.a. |
PMID[466233] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
IC50 |
= |
145000.0 |
nM |
PMID[466235] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
IC50 |
= |
4500.0 |
nM |
PMID[466235] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
IC50 |
= |
58000.0 |
nM |
PMID[466235] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
IC50 |
= |
47500.0 |
nM |
PMID[466235] |
NPT266 |
Individual Protein |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
IC50 |
= |
62500.0 |
nM |
PMID[466235] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Inhibition |
= |
13.0 |
% |
PMID[466236] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki |
= |
40.0 |
nM |
PMID[466236] |
NPT264 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Homo sapiens |
Ki |
= |
5700.0 |
nM |
PMID[466236] |
NPT265 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Homo sapiens |
Ki |
= |
2400.0 |
nM |
PMID[466236] |
NPT1301 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Rattus norvegicus |
Ki |
= |
40.0 |
nM |
PMID[466237] |
NPT1303 |
Individual Protein |
Muscarinic acetylcholine receptor M3 |
Rattus norvegicus |
Ki |
= |
5700.0 |
nM |
PMID[466237] |
NPT432 |
Individual Protein |
Muscarinic acetylcholine receptor M4 |
Rattus norvegicus |
Ki |
= |
2400.0 |
nM |
PMID[466237] |
NPT262 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Homo sapiens |
Ki |
= |
29512.09 |
nM |
PMID[466242] |
NPT263 |
Individual Protein |
Muscarinic acetylcholine receptor M2 |
Homo sapiens |
Ki |
= |
2454.71 |
nM |
PMID[466242] |
NPT266 |
Individual Protein |
Muscarinic acetylcholine receptor M5 |
Homo sapiens |
Ki |
= |
56234.13 |
nM |
PMID[466242] |
NPT483 |
Individual Protein |
Prelamin-A/C |
Homo sapiens |
Potency |
= |
1000.0 |
nM |
PMID[466247] |
NPT46 |
Individual Protein |
Thyroid hormone receptor beta-1 |
Homo sapiens |
Potency |
= |
35.5 |
nM |
PMID[466247] |
NPT583 |
Individual Protein |
Inositol monophosphatase 1 |
Rattus norvegicus |
Potency |
= |
3548.1 |
nM |
PMID[466248] |
NPT442 |
Individual Protein |
Ferritin light chain |
Equus caballus |
Potency |
= |
316.2 |
nM |
PMID[466247] |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
n.a. |
40533.4 |
nM |
PMID[466250] |
NPT1304 |
Individual Protein |
Nicotinic acetylcholine receptor alpha 5 subunit |
Musca domestica |
Ki |
= |
516000.0 |
nM |
PMID[466252] |
NPT1305 |
Individual Protein |
Voltage-dependent L-type calcium channel subunit alpha-1C |
Cavia porcellus |
IC50 |
= |
33730.0 |
nM |
PMID[466256] |
NPT153 |
Individual Protein |
Androgen Receptor |
Homo sapiens |
Potency |
n.a. |
33491.5 |
nM |
PubChem BioAssay data set |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
pD2 |
= |
6.6 |
n.a. |
PMID[466203] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Efficiency |
= |
80.0 |
% |
PMID[466203] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Efficiency |
= |
100.0 |
% |
PMID[466203] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
20.0 |
nM |
PMID[466203] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1740.0 |
nM |
PMID[466203] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Ratio |
= |
87.0 |
n.a. |
PMID[466203] |
NPT413 |
Protein Complex |
Neuronal acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
224.0 |
nM |
PMID[466204] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
40.0 |
nM |
PMID[466204] |
NPT2 |
Others |
Unspecified |
|
Selectivity |
= |
0.18 |
n.a. |
PMID[466204] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Inhibition |
= |
43.0 |
% |
PMID[466205] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
31.0 |
nM |
PMID[466205] |
NPT2 |
Others |
Unspecified |
|
Ratio |
> |
3000.0 |
n.a. |
PMID[466205] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
1900.0 |
nM |
PMID[466205] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
5.3 |
nM |
PMID[466205] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
360.0 |
n.a. |
PMID[466205] |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1000.0 |
nM |
PMID[466206] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Activity |
= |
110.0 |
% |
PMID[466206] |
NPT27 |
Others |
Unspecified |
|
Binding energy |
= |
7.2 |
kCal mol-1 |
PMID[466207] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466209] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466209] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
560.0 |
n.a. |
PMID[466209] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
EC50 |
>= |
220.0 |
nM |
PMID[466210] |
NPT1299 |
Others |
Muscarinic acetylcholine receptors; M2 & M3 |
Homo sapiens |
EC50 |
= |
140.0 |
nM |
PMID[466210] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
1000.0 |
nM |
PMID[466211] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PI metabolism |
= |
110.0 |
% |
PMID[466211] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.0000016 |
M |
PMID[466212] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
2.2 |
M |
PMID[466213] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
77.0 |
nM |
PMID[466214] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1300.0 |
nM |
PMID[466214] |
NPT419 |
Organism |
Oryctolagus cuniculus |
Oryctolagus cuniculus |
IC50 |
= |
545.0 |
nM |
PMID[466214] |
NPT419 |
Organism |
Oryctolagus cuniculus |
Oryctolagus cuniculus |
Inhibition |
= |
95.0 |
% |
PMID[466214] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
IC50 |
= |
600.0 |
nM |
PMID[466214] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
Inhibition |
= |
100.0 |
% |
PMID[466214] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
28000.0 |
nM |
PMID[466215] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
1700.0 |
nM |
PMID[466215] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
2100.0 |
nM |
PMID[466215] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
16.0 |
nM |
PMID[466215] |
NPT1300 |
Others |
Muscarinic acetylcholine receptors; M1 & M2 |
Homo sapiens |
M2/M1 index |
= |
0.1 |
n.a. |
PMID[466215] |
NPT2 |
Others |
Unspecified |
|
Agonist index |
= |
280.0 |
n.a. |
PMID[466215] |
NPT1300 |
Others |
Muscarinic acetylcholine receptors; M1 & M2 |
Homo sapiens |
Ratio |
= |
0.078 |
n.a. |
PMID[466215] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
24.0 |
nM |
PMID[466216] |
NPT2 |
Others |
Unspecified |
|
Potency ratio |
= |
2.0 |
n.a. |
PMID[466216] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
115.0 |
nM |
PMID[466217] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
25400.0 |
nM |
PMID[466217] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
222.0 |
n.a. |
PMID[466217] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1100.0 |
nM |
PMID[466218] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
1.9 |
nM |
PMID[466218] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
EC50 |
= |
150.0 |
nM |
PMID[466218] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
IC50 |
> |
1000.0 |
nM |
PMID[466218] |
NPT2 |
Others |
Unspecified |
|
M-agonist index |
= |
938.0 |
n.a. |
PMID[466218] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
0.07 |
n.a. |
PMID[466218] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
5600.0 |
nM |
PMID[466219] |
NPT35 |
Others |
n.a. |
|
pKa |
= |
7.8 |
n.a. |
PMID[466219] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
pD2 |
= |
6.5 |
n.a. |
PMID[466221] |
NPT938 |
Organism |
Cavia porcellus |
Cavia porcellus |
Efficacy |
= |
100.0 |
% |
PMID[466221] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
pD2 |
= |
6.6 |
n.a. |
PMID[466221] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Efficacy |
= |
80.0 |
% |
PMID[466221] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
pD2 |
= |
6.1 |
n.a. |
PMID[466221] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Efficacy |
= |
100.0 |
% |
PMID[466221] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1737.8 |
nM |
PMID[466221] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466222] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466222] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
560.0 |
n.a. |
PMID[466222] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466223] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466223] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
560.0 |
n.a. |
PMID[466223] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
77.0 |
nM |
PMID[466225] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1300.0 |
nM |
PMID[466225] |
NPT419 |
Organism |
Oryctolagus cuniculus |
Oryctolagus cuniculus |
IC50 |
= |
545.0 |
nM |
PMID[466225] |
NPT419 |
Organism |
Oryctolagus cuniculus |
Oryctolagus cuniculus |
Inhibition |
= |
95.0 |
% |
PMID[466225] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
1000.0 |
nM |
PMID[466226] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466227] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466227] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
560.0 |
n.a. |
PMID[466227] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
115.0 |
nM |
PMID[466228] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
19000.0 |
nM |
PMID[466228] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED Arec |
= |
0.32 |
mg kg-1 |
PMID[466228] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.022 |
mg.kg-1 |
PMID[466228] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
ED50 |
= |
0.024 |
mg.kg-1 |
PMID[466228] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Ratio |
= |
0.07 |
n.a. |
PMID[466228] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Ratio |
= |
0.075 |
n.a. |
PMID[466228] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
115.0 |
nM |
PMID[466229] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
25400.0 |
nM |
PMID[466229] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
222.0 |
n.a. |
PMID[466229] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ki |
= |
7120.0 |
nM |
PMID[466230] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Max stimulation |
= |
28.0 |
% |
PMID[466230] |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
7.4 |
nM |
PMID[466230] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
960.0 |
n.a. |
PMID[466230] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
77.0 |
nM |
PMID[466231] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1300.0 |
nM |
PMID[466231] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
77.0 |
nM |
PMID[466232] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
1300.0 |
nM |
PMID[466232] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Score |
= |
0.0 |
n.a. |
PMID[466232] |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
604.0 |
n.a. |
PMID[466233] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
11920.0 |
nM |
PMID[466233] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
77.0 |
nM |
PMID[466234] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
106000.0 |
nM |
PMID[466234] |
NPT1302 |
Protein Family |
Muscarinic acetylcholine receptor |
Homo sapiens |
EC50 |
= |
73.0 |
nM |
PMID[466234] |
NPT1302 |
Protein Family |
Muscarinic acetylcholine receptor |
Homo sapiens |
Max contraction |
= |
100.0 |
% |
PMID[466234] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Muscarinic agonist index |
= |
223.0 |
n.a. |
PMID[466234] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
62.7 |
nM |
PMID[466235] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
16.0 |
mg.kg-1 |
PMID[466235] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
ED50 |
= |
15.0 |
mg.kg-1 |
PMID[466235] |
NPT412 |
Protein Complex |
Neuronal acetylcholine receptor; alpha4/beta2 |
Rattus norvegicus |
Ki |
= |
270.0 |
nM |
PMID[466236] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Inhibition |
= |
43.0 |
% |
PMID[466236] |
NPT412 |
Protein Complex |
Neuronal acetylcholine receptor; alpha4/beta2 |
Rattus norvegicus |
Ki |
= |
270.0 |
nM |
PMID[466237] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Inhibition |
= |
43.0 |
% |
PMID[466237] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Inhibition |
= |
13.0 |
% |
PMID[466237] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
1000.0 |
nM |
PMID[466238] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
PI |
= |
110.0 |
% |
PMID[466238] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466239] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466239] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
560.0 |
n.a. |
PMID[466239] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
120.0 |
nM |
PMID[466240] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
IC50 |
= |
25000.0 |
nM |
PMID[466240] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
n.a. |
210.0 |
n.a. |
PMID[466240] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
6.2 |
uM |
PMID[466241] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
K app |
= |
0.011 |
uM |
PMID[466241] |
NPT422 |
Protein Family |
Muscarinic acetylcholine receptor |
Rattus norvegicus |
Ratio |
= |
560.0 |
n.a. |
PMID[466241] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Ki |
= |
86000.0 |
nM |
PMID[466243] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
469000.0 |
nM |
PMID[466243] |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
64.0 |
% |
PMID[466244] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Ki |
= |
86000.0 |
nM |
PMID[466245] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
469000.0 |
nM |
PMID[466245] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
Ki |
= |
88000.0 |
nM |
PMID[466246] |
NPT95 |
Individual Protein |
Muscarinic acetylcholine receptor M1 |
Rattus norvegicus |
IC50 |
= |
460000.0 |
nM |
PMID[466246] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
TIME |
= |
0.002778 |
hr |
PMID[466246] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
TIME |
= |
0.001389 |
hr |
PMID[466246] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
TIME |
= |
0.01444 |
hr |
PMID[466246] |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
TIME |
= |
0.01 |
hr |
PMID[466246] |
NPT533 |
Protein-Protein Interaction |
Runt-related transcription factor 1/Core-binding factor subunit beta |
Homo sapiens |
Potency |
n.a. |
19952.6 |
nM |
PMID[466247] |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
n.a. |
16944.1 |
nM |
PMID[466250] |
NPT7 |
Individual Protein |
Thioredoxin reductase 1, cytoplasmic |
Rattus norvegicus |
Potency |
n.a. |
1000.0 |
nM |
PMID[466251] |
NPT698 |
Individual Protein |
Regulator of G-protein signaling 4 |
Homo sapiens |
Potency |
n.a. |
3358.7 |
nM |
PMID[466250] |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
240000.0 |
nM |
PMID[466252] |
NPT35 |
Others |
n.a. |
|
pKa |
n.a. |
7.64 |
n.a. |
PMID[466253] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
14950.2 |
nM |
PMID[466254] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
21.1 |
nM |
PMID[466254] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
13324.4 |
nM |
PMID[466254] |
NPT20529 |
NON-MOLECULAR |
NON-PROTEIN TARGET |
n.a. |
Potency |
n.a. |
94.3 |
nM |
PMID[466254] |
NPT2 |
Others |
Unspecified |
|
AC50 |
n.a. |
44668.4 |
nM |
PMID[466255] |
NPT2 |
Others |
Unspecified |
|
Ac50 |
n.a. |
44.67 |
uM |
PMID[466255] |
NPT713 |
Individual Protein |
Bile salt export pump |
Homo sapiens |
IC50 |
> |
1000000.0 |
nM |
PMID[466257] |
NPT20556 |
SINGLE PROTEIN |
Replicase polyprotein 1ab |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
17.68 |
% |
PMID[466258] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
Inhibition |
= |
0.3 |
% |
PMID[466259] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
IC50 |
> |
20000.0 |
nM |
PMID[466260] |
NPT20555 |
ORGANISM |
SARS-CoV-2 |
Severe acute respiratory syndrome coronavirus 2 |
IC50 |
> |
19952.62 |
nM |
PMID[466260] |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
26832.5 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
n.a. |
14960.1 |
nM |
PubChem BioAssay data set |
NPT74 |
Individual Protein |
Proto-oncogene c-JUN |
Homo sapiens |
Potency |
n.a. |
6740 |
nM |
PubChem BioAssay data set |