Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT471 | Organism | Trypanosoma brucei brucei | Trypanosoma brucei brucei | IC50 | > | 100000 | nM | 22290833 |
NPT839 | Cell Line | L6 | Rattus norvegicus | IC50 | = | 70 | nM | DrugMatrix in vivo data: Pathology |
NPT2 | Others | Unspecified | Ratio IC50 | = | 1.8 | 15387655 | ||
NPT580 | Organism | Trypanosoma cruzi | Trypanosoma cruzi | IC50 | = | 40 | nM | 10579864 |
NPT844 | Organism | Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | IC50 | = | 45800 | nM | PubChem BioAssay data set |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC472167 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
0.9149 | High Similarity | NPC472162 |
0.9149 | High Similarity | NPC472166 |
0.8889 | High Similarity | NPC472136 |
0.8085 | Intermediate Similarity | NPC472161 |
0.7917 | Intermediate Similarity | NPC116231 |
0.7692 | Intermediate Similarity | NPC472165 |
0.6752 | Remote Similarity | NPC472164 |
0.6724 | Remote Similarity | NPC5485 |
0.661 | Remote Similarity | NPC7905 |
0.661 | Remote Similarity | NPC315652 |
0.6555 | Remote Similarity | NPC59751 |
0.6555 | Remote Similarity | NPC271621 |
0.6555 | Remote Similarity | NPC27413 |
0.65 | Remote Similarity | NPC296361 |
0.6476 | Remote Similarity | NPC280833 |
0.6449 | Remote Similarity | NPC248193 |
0.6415 | Remote Similarity | NPC113393 |
0.6393 | Remote Similarity | NPC473808 |
0.6381 | Remote Similarity | NPC307298 |
0.6355 | Remote Similarity | NPC166110 |
0.6341 | Remote Similarity | NPC315915 |
0.6316 | Remote Similarity | NPC133420 |
0.6311 | Remote Similarity | NPC474359 |
0.6271 | Remote Similarity | NPC44733 |
0.6226 | Remote Similarity | NPC143025 |
0.6226 | Remote Similarity | NPC53454 |
0.6214 | Remote Similarity | NPC8091 |
0.62 | Remote Similarity | NPC23778 |
0.619 | Remote Similarity | NPC220478 |
0.6168 | Remote Similarity | NPC142159 |
0.6168 | Remote Similarity | NPC95364 |
0.6154 | Remote Similarity | NPC60951 |
0.6147 | Remote Similarity | NPC476597 |
0.6147 | Remote Similarity | NPC476598 |
0.6147 | Remote Similarity | NPC271652 |
0.6139 | Remote Similarity | NPC475681 |
0.6106 | Remote Similarity | NPC316730 |
0.61 | Remote Similarity | NPC471225 |
0.61 | Remote Similarity | NPC283087 |
0.6095 | Remote Similarity | NPC475614 |
0.6091 | Remote Similarity | NPC476596 |
0.6075 | Remote Similarity | NPC478261 |
0.6075 | Remote Similarity | NPC478260 |
0.6075 | Remote Similarity | NPC478259 |
0.6068 | Remote Similarity | NPC176773 |
0.6058 | Remote Similarity | NPC222358 |
0.6058 | Remote Similarity | NPC288281 |
0.6055 | Remote Similarity | NPC32944 |
0.6055 | Remote Similarity | NPC193396 |
0.6034 | Remote Similarity | NPC75523 |
0.6034 | Remote Similarity | NPC87919 |
0.6019 | Remote Similarity | NPC474085 |
0.6 | Remote Similarity | NPC474619 |
0.5983 | Remote Similarity | NPC154601 |
0.5983 | Remote Similarity | NPC271269 |
0.5981 | Remote Similarity | NPC220930 |
0.5981 | Remote Similarity | NPC272039 |
0.598 | Remote Similarity | NPC471299 |
0.5963 | Remote Similarity | NPC471818 |
0.5962 | Remote Similarity | NPC10080 |
0.5962 | Remote Similarity | NPC123908 |
0.5957 | Remote Similarity | NPC98897 |
0.5954 | Remote Similarity | NPC307165 |
0.5943 | Remote Similarity | NPC133652 |
0.5943 | Remote Similarity | NPC241512 |
0.5943 | Remote Similarity | NPC8518 |
0.5943 | Remote Similarity | NPC132228 |
0.5943 | Remote Similarity | NPC90287 |
0.5943 | Remote Similarity | NPC6185 |
0.5943 | Remote Similarity | NPC263997 |
0.5941 | Remote Similarity | NPC187568 |
0.5941 | Remote Similarity | NPC41780 |
0.5938 | Remote Similarity | NPC146376 |
0.5938 | Remote Similarity | NPC125578 |
0.5938 | Remote Similarity | NPC263382 |
0.5932 | Remote Similarity | NPC251330 |
0.5926 | Remote Similarity | NPC185059 |
0.5926 | Remote Similarity | NPC475001 |
0.5923 | Remote Similarity | NPC478136 |
0.5918 | Remote Similarity | NPC474539 |
0.5913 | Remote Similarity | NPC471699 |
0.5913 | Remote Similarity | NPC77703 |
0.5913 | Remote Similarity | NPC469851 |
0.5909 | Remote Similarity | NPC190442 |
0.5909 | Remote Similarity | NPC248913 |
0.5905 | Remote Similarity | NPC193198 |
0.5905 | Remote Similarity | NPC474703 |
0.5897 | Remote Similarity | NPC472616 |
0.5895 | Remote Similarity | NPC16119 |
0.5893 | Remote Similarity | NPC470978 |
0.5893 | Remote Similarity | NPC295347 |
0.5893 | Remote Similarity | NPC470974 |
0.5893 | Remote Similarity | NPC91408 |
0.5888 | Remote Similarity | NPC203795 |
0.5887 | Remote Similarity | NPC316325 |
0.5882 | Remote Similarity | NPC471220 |
0.5882 | Remote Similarity | NPC470072 |
0.5882 | Remote Similarity | NPC315765 |
0.5878 | Remote Similarity | NPC97861 |
0.5877 | Remote Similarity | NPC270813 |
0.5877 | Remote Similarity | NPC166770 |
0.5876 | Remote Similarity | NPC94488 |
0.5873 | Remote Similarity | NPC477140 |
0.5873 | Remote Similarity | NPC477143 |
0.5873 | Remote Similarity | NPC13351 |
0.5872 | Remote Similarity | NPC284561 |
0.5865 | Remote Similarity | NPC471325 |
0.5862 | Remote Similarity | NPC80781 |
0.5856 | Remote Similarity | NPC229976 |
0.5851 | Remote Similarity | NPC474400 |
0.5851 | Remote Similarity | NPC34622 |
0.5847 | Remote Similarity | NPC185929 |
0.5847 | Remote Similarity | NPC472615 |
0.5846 | Remote Similarity | NPC96010 |
0.5846 | Remote Similarity | NPC317654 |
0.5833 | Remote Similarity | NPC218602 |
0.5833 | Remote Similarity | NPC103743 |
0.5833 | Remote Similarity | NPC243272 |
0.5833 | Remote Similarity | NPC113370 |
0.5833 | Remote Similarity | NPC215507 |
0.5833 | Remote Similarity | NPC476079 |
0.5826 | Remote Similarity | NPC215253 |
0.5826 | Remote Similarity | NPC185253 |
0.5825 | Remote Similarity | NPC276647 |
0.5825 | Remote Similarity | NPC268502 |
0.5825 | Remote Similarity | NPC254996 |
0.5825 | Remote Similarity | NPC622 |
0.5818 | Remote Similarity | NPC475823 |
0.5818 | Remote Similarity | NPC253177 |
0.5818 | Remote Similarity | NPC212679 |
0.5818 | Remote Similarity | NPC223093 |
0.5818 | Remote Similarity | NPC220454 |
0.5818 | Remote Similarity | NPC474209 |
0.5818 | Remote Similarity | NPC280592 |
0.5818 | Remote Similarity | NPC213636 |
0.5818 | Remote Similarity | NPC469595 |
0.5818 | Remote Similarity | NPC471399 |
0.5816 | Remote Similarity | NPC291062 |
0.5816 | Remote Similarity | NPC94743 |
0.5816 | Remote Similarity | NPC173321 |
0.5812 | Remote Similarity | NPC473144 |
0.5812 | Remote Similarity | NPC271059 |
0.5812 | Remote Similarity | NPC297281 |
0.5812 | Remote Similarity | NPC320154 |
0.5812 | Remote Similarity | NPC25666 |
0.5804 | Remote Similarity | NPC474882 |
0.5804 | Remote Similarity | NPC212812 |
0.5804 | Remote Similarity | NPC148463 |
0.58 | Remote Similarity | NPC264178 |
0.5794 | Remote Similarity | NPC471060 |
0.5794 | Remote Similarity | NPC2640 |
0.5794 | Remote Similarity | NPC96621 |
0.5794 | Remote Similarity | NPC189311 |
0.5794 | Remote Similarity | NPC476678 |
0.5789 | Remote Similarity | NPC134083 |
0.5789 | Remote Similarity | NPC208094 |
0.5789 | Remote Similarity | NPC241426 |
0.5784 | Remote Similarity | NPC316324 |
0.5784 | Remote Similarity | NPC473536 |
0.578 | Remote Similarity | NPC26078 |
0.578 | Remote Similarity | NPC473658 |
0.5778 | Remote Similarity | NPC239252 |
0.5778 | Remote Similarity | NPC473703 |
0.5776 | Remote Similarity | NPC472643 |
0.5776 | Remote Similarity | NPC34193 |
0.5776 | Remote Similarity | NPC314792 |
0.5773 | Remote Similarity | NPC134385 |
0.5766 | Remote Similarity | NPC471329 |
0.5766 | Remote Similarity | NPC296114 |
0.5766 | Remote Similarity | NPC473944 |
0.5763 | Remote Similarity | NPC470073 |
0.5755 | Remote Similarity | NPC470047 |
0.5755 | Remote Similarity | NPC470046 |
0.5752 | Remote Similarity | NPC150041 |
0.575 | Remote Similarity | NPC476276 |
0.575 | Remote Similarity | NPC220730 |
0.5748 | Remote Similarity | NPC11379 |
0.5746 | Remote Similarity | NPC133089 |
0.5745 | Remote Similarity | NPC57463 |
0.5745 | Remote Similarity | NPC151728 |
0.5743 | Remote Similarity | NPC244166 |
0.5743 | Remote Similarity | NPC175079 |
0.5741 | Remote Similarity | NPC472863 |
0.5741 | Remote Similarity | NPC38576 |
0.5741 | Remote Similarity | NPC186332 |
0.5741 | Remote Similarity | NPC47220 |
0.5741 | Remote Similarity | NPC279859 |
0.5741 | Remote Similarity | NPC472009 |
0.5741 | Remote Similarity | NPC261721 |
0.5739 | Remote Similarity | NPC264378 |
0.5728 | Remote Similarity | NPC478122 |
0.5728 | Remote Similarity | NPC128276 |
0.5728 | Remote Similarity | NPC475994 |
0.5728 | Remote Similarity | NPC30321 |
0.5728 | Remote Similarity | NPC231739 |
0.5727 | Remote Similarity | NPC307092 |
0.5727 | Remote Similarity | NPC210216 |
0.5727 | Remote Similarity | NPC51358 |
0.5726 | Remote Similarity | NPC251884 |
0.5726 | Remote Similarity | NPC469598 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC472167 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
0.6667 | Remote Similarity | NPD7299 | Clinical (unspecified phase) |
0.6134 | Remote Similarity | NPD7116 | Clinical (unspecified phase) |
0.6064 | Remote Similarity | NPD3704 | Approved |
0.5952 | Remote Similarity | NPD7739 | Clinical (unspecified phase) |
0.5906 | Remote Similarity | NPD7623 | Phase 3 |
0.5906 | Remote Similarity | NPD7624 | Clinical (unspecified phase) |
0.5895 | Remote Similarity | NPD6108 | Clinical (unspecified phase) |
0.5887 | Remote Similarity | NPD7500 | Approved |
0.5772 | Remote Similarity | NPD1376 | Discontinued |
0.5746 | Remote Similarity | NPD6845 | Suspended |
0.5725 | Remote Similarity | NPD7746 | Phase 1 |
0.5725 | Remote Similarity | NPD7747 | Phase 1 |
0.5672 | Remote Similarity | NPD2101 | Approved |
0.5659 | Remote Similarity | NPD8080 | Discontinued |
0.5636 | Remote Similarity | NPD5737 | Approved |
0.5636 | Remote Similarity | NPD6672 | Approved |
0.5631 | Remote Similarity | NPD4756 | Discovery |
0.5619 | Remote Similarity | NPD4695 | Discontinued |
PubChem CID   | |
ChEMBL   | CHEMBL3342754 |
ZINC   |
Molecular Weight:   | 365.26 |
ALogP:   | -2.3769 |
MLogP:   | 3.22 |
XLogP:   | 5.252 |
# Rotatable Bonds:   | 15 |
Polar Surface Area:   | 48 |
# H-Bond Aceptor:   | 3 |
# H-Bond Donor:   | 0 |
# Rings:   | 2 |
# Heavy Atoms:   | 26 |